Page last updated: 2024-09-05

atropine and cytisine

atropine has been researched along with cytisine in 14 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(cytisine)
Trials
(cytisine)
Recent Studies (post-2010) (cytisine)
26,7111,2591,69751919178

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)cytisine (IC50)
Neuronal acetylcholine receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0692
Neuronal acetylcholine receptor subunit beta-2Rattus norvegicus (Norway rat)0.0692
Neuronal acetylcholine receptor subunit beta-2Homo sapiens (human)0.05
Neuronal acetylcholine receptor subunit alpha-4Homo sapiens (human)0.05

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19903 (21.43)18.7374
1990's5 (35.71)18.2507
2000's2 (14.29)29.6817
2010's3 (21.43)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Curtis, MA; Lin, SX; Sperry, J1
Fujiwara, M; Kameyama, M; Shimohama, S; Taniguchi, T1
Demushkin, VP; Gerateks, A; Martinez-Soler, R; Mendez, R; Pliashkevich, IuG1
Holstad, SG; Hong, SE; Isenberg, KE; Mennerick, SJ; Wong, ET; Zorumski, CF1
Khan, IM; Taylor, P; Yaksh, TL1
Bobbin, RP; Erostegui, C; Norris, CH1
Changeux, JP; Léna, C1
de la Lande, IS; Marino, V; Parker, DA; Zisimopoulos, S1
Lee, DH; Wang, HY1
Bermudez, I; Groot-Kormelink, PJ; Smulders, CJ; van Kleef, RG; Vijverberg, HP; Zwart, R1
Freeling, J; Lacroix, C; Li, YF1
Blakely, RD; Cherian, AK; Mallory, CS; Miller, TR; Paolone, G; Sarter, M1
Kuryatov, A; Ley, CK; Lindstrom, JM; Wang, J1

Reviews

1 review(s) available for atropine and cytisine

ArticleYear
Pyridine alkaloids with activity in the central nervous system.
    Bioorganic & medicinal chemistry, 2020, 12-15, Volume: 28, Issue:24

    Topics: Alkaloids; Amphibians; Animals; Bacteria; Central Nervous System Diseases; Fungi; Nicotine; Plants; Pyridines; Receptors, Nicotinic

2020

Other Studies

13 other study(ies) available for atropine and cytisine

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Biochemical characterization of the nicotinic cholinergic receptors in human brain: binding of (-)-[3H]nicotine.
    Journal of neurochemistry, 1985, Volume: 45, Issue:2

    Topics: Acetylcholine; Aged; Alkaloids; Atropine; Azocines; Brain; Bungarotoxins; Carbachol; Cell Membrane; Female; Hexamethonium; Hexamethonium Compounds; Humans; Male; Nicotine; Quinolizines; Receptors, Cholinergic; Stereoisomerism; Thalamus; Tubocurarine

1985
[Pharmacological characteristics of the acetylcholine and L-glutamate receptors of the subpharyngeal ganglion neuron in the mollusk Zachrysia guanensis].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 98, Issue:9

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Ganglia; Glutamates; Mollusca; Neurons; Quinolizines; Receptors, Cholinergic; Receptors, Glutamate; Receptors, Neurotransmitter; Tubocurarine

1984
Pharmacological and physiological properties of a putative ganglionic nicotinic receptor, alpha 3 beta 4, expressed in transfected eucaryotic cells.
    Brain research. Molecular brain research, 1995, Volume: 28, Issue:1

    Topics: Acetylcholine; Alkaloids; Atropine; Azocines; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Kidney; Nicotine; Patch-Clamp Techniques; Quinolizines; Receptors, Nicotinic

1995
Cardiovascular and behavioral responses to nicotinic agents administered intrathecally.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:1

    Topics: Aconitine; Alkaloids; Animals; Atropine; Azocines; Behavior, Animal; Blood Pressure; Bungarotoxins; Cardiovascular System; Dihydro-beta-Erythroidine; Ganglionic Stimulants; Heart Rate; Injections, Spinal; Lobeline; Male; Mecamylamine; Nicotine; Nicotinic Antagonists; Nociceptors; Quinolizines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Sensitivity and Specificity; Spinal Cord; Trimethaphan

1994
In vitro pharmacologic characterization of a cholinergic receptor on outer hair cells.
    Hearing research, 1994, Volume: 74, Issue:1-2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Bungarotoxins; Carbachol; Choline; Cholinergic Antagonists; Curare; Dimethylphenylpiperazinium Iodide; Guinea Pigs; Hair Cells, Auditory, Outer; In Vitro Techniques; Membrane Potentials; Nicotine; Piperidines; Pirenzepine; Quinolizines; Receptors, Cholinergic; Strychnine; Trimethaphan

1994
Role of Ca2+ ions in nicotinic facilitation of GABA release in mouse thalamus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aconitine; Action Potentials; Alkaloids; Animals; Arousal; Atropine; Azocines; Bacterial Toxins; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Calcium Channel Blockers; Calcium Channels; Carbachol; Cations, Divalent; Cyanobacteria Toxins; Dihydro-beta-Erythroidine; Dimethylphenylpiperazinium Iodide; GABA Antagonists; gamma-Aminobutyric Acid; Ion Transport; Lobeline; Marine Toxins; Mice; Mice, Inbred C57BL; Mice, Knockout; Microcystins; Neurons, Afferent; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium; Pyridazines; Pyridines; Quinolizines; Receptors, GABA-A; Receptors, Nicotinic; Tetrodotoxin; Thalamic Nuclei

1997
Evidence for presynaptic cholinergic receptors in sympathetic nerves in human dental pulp.
    Archives of oral biology, 1998, Volume: 43, Issue:3

    Topics: Adolescent; Adult; Alkaloids; Atropine; Azocines; Carbachol; Dental Pulp; Electric Stimulation; Enzyme Inhibitors; Female; Hexamethonium; Humans; Isotonic Solutions; Male; Muscarinic Agonists; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Nitric Oxide; Nitric Oxide Synthase; Norepinephrine; Quinolizines; Radiopharmaceuticals; Receptors, Muscarinic; Receptors, Nicotinic; Receptors, Presynaptic; Sympathetic Nervous System; Sympathomimetics; Tritium

1998
Differential physiologic responses of alpha7 nicotinic acetylcholine receptors to beta-amyloid1-40 and beta-amyloid1-42.
    Journal of neurobiology, 2003, Volume: 55, Issue:1

    Topics: Acetylcholine; Alkaloids; Amyloid beta-Peptides; Animals; Atropine; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Calcium Channel Blockers; Conotoxins; Dose-Response Relationship, Drug; Frontal Lobe; In Vitro Techniques; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Peptide Fragments; Potassium; Pyridines; Quinolizines; Rats; Receptors, Nicotinic; Subcellular Fractions; Synaptosomes

2003
Cholinergic drugs potentiate human nicotinic alpha4beta2 acetylcholine receptors by a competitive mechanism.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Binding, Competitive; Cholinergic Agents; Cholinesterase Inhibitors; Dichlorvos; Dose-Response Relationship, Drug; Female; Galantamine; Humans; Membrane Potentials; Models, Biological; Nicotine; Oocytes; Phenylcarbamates; Physostigmine; Plasmids; Quinolizines; Receptors, Nicotinic; Rivastigmine; Scopolamine; Tacrine; Xenopus laevis

2005
Cytisine induces autonomic cardiovascular responses via activations of different nicotinic receptors.
    Autonomic neuroscience : basic & clinical, 2010, Apr-19, Volume: 154, Issue:1-2

    Topics: Aconitine; Adrenergic alpha-Antagonists; Alkaloids; Analysis of Variance; Animals; Atropine; Azocines; Blood Pressure; Bradycardia; Cardiovascular Physiological Phenomena; Dihydro-beta-Erythroidine; Heart Rate; Hexamethonium; Male; Mice; Muscarinic Antagonists; Nicotinic Agonists; Nicotinic Antagonists; Prazosin; Quinolizines; Receptors, Nicotinic

2010
Monitoring cholinergic activity during attentional performance in mice heterozygous for the choline transporter: a model of cholinergic capacity limits.
    Neuropharmacology, 2013, Volume: 75

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Attention; Azocines; Cholinergic Antagonists; Conditioning, Operant; Female; Humans; Male; Mecamylamine; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Protein Binding; Quinolizines; Sodium Channel Blockers; Tetrodotoxin; Tritium

2013
Efficient expression of functional (α6β2)2β3 AChRs in Xenopus oocytes from free subunits using slightly modified α6 subunits.
    PloS one, 2014, Volume: 9, Issue:7

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Cholinergic Agonists; Female; Gene Expression; Humans; Membrane Potentials; Nicotine; Nicotinic Agonists; Oocytes; Patch-Clamp Techniques; Quinolizines; Receptors, Nicotinic; Recombinant Fusion Proteins; Varenicline; Xenopus laevis

2014