atropine has been researched along with colforsin in 62 studies
Studies (atropine) | Trials (atropine) | Recent Studies (post-2010) (atropine) | Studies (colforsin) | Trials (colforsin) | Recent Studies (post-2010) (colforsin) |
---|---|---|---|---|---|
26,711 | 1,259 | 1,697 | 13,460 | 46 | 1,298 |
Protein | Taxonomy | atropine (IC50) | colforsin (IC50) |
---|---|---|---|
nuclear receptor subfamily 0 group B member 1 | Homo sapiens (human) | 1.729 | |
5-hydroxytryptamine receptor 1A | Homo sapiens (human) | 0.041 | |
Adenylate cyclase type 1 | Homo sapiens (human) | 0.0955 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (25.81) | 18.7374 |
1990's | 31 (50.00) | 18.2507 |
2000's | 11 (17.74) | 29.6817 |
2010's | 4 (6.45) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Nakagawa-Yagi, Y; Nakamura, H; Saito, Y; Takada, Y | 1 |
Gintzler, AR; Xu, H | 1 |
Knudsen, MA; Tøttrup, A | 1 |
Funakoshi, A; Kitayama, N; Matsuoka, Y; Tateishi, K | 1 |
Osborne, NN | 1 |
Malinowska, DH | 1 |
Nakagawa-Yagi, Y; Saito, Y; Takada, Y; Takayama, M | 1 |
Hescheler, J; Wallukat, G; Wobus, AM | 1 |
Diener, M; Rummel, W | 1 |
Bizzarri, C; Corda, D; D'Orazio, MC; Di Girolamo, M | 1 |
Burton, MD; Johnson, DC; Kazemi, H | 1 |
Kristersson, A; Mazzoni, L; Morley, J; Sanjar, S; Schaeublin, E | 1 |
Meyer, EM; Millard, WJ; Poulakos, JJ; Pruysers, CR | 1 |
Nezu, E; Yoneyama, T; Yoshimura, K | 1 |
Miledi, R; Woodward, RM | 1 |
Linden, J | 1 |
Alberts, P; Ogren, VR | 1 |
Seidler, U; Sewing, KF | 1 |
Fong, JC; Ho, LT; Wang, FF | 1 |
Renit-Soria, J; Stinnakre, J; Van Renterghem, C | 1 |
Hermansen, K | 1 |
Nathanson, NM; Subers, EM | 1 |
Ernst, SA; Lowy, RJ | 1 |
Fredholm, BB; Larsson, O | 1 |
Foreman, JC; Rising, TJ; Webber, SE | 1 |
Chiba, S; Horiuchi, A; Iwatsuki, K; Yamagishi, F | 1 |
Rasmussen, H; Takuwa, N; Takuwa, Y | 1 |
Chew, CS | 1 |
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ | 1 |
Kaur, H; Khuller, GK | 1 |
Chowdhury, P; Doi, R; Inoue, K; Kaji, H; Rayford, PL | 1 |
Biden, TJ; Browne, CL | 1 |
Morikawa, M; Sasaki, H; Sekizawa, K | 1 |
Beil, W; Bersimbaev, RI; Gandjour, A; Heim, HK; Sewing, KF | 1 |
Ellis, JL; Fernandes, LB; Undem, BJ | 1 |
Johnson, GL; Russell, M; Winitz, S | 1 |
Migeon, JC; Nathanson, NM | 1 |
Dunér-Engström, M; Fredholm, BB | 1 |
Fischmeister, R; Hanf, R; Li, Y; Szabo, G | 1 |
Nahorski, SR; Tobin, AB | 1 |
Goldstein, I; Moreland, RB; Palmer, MS; Traish, AM | 1 |
Barnes, PJ; Belvisi, MG; Giembycz, MA; Patel, HJ; Takahashi, T | 1 |
Best, JA; Chen, Y; Nagamoto, K; Tank, AW | 1 |
Dawson, JJ; Iannazzo, L; Majewski, H | 1 |
Login, IS | 1 |
Clancy-Keen, J; Emala, CW; Hirshman, CA | 1 |
Berul, CI; Gehrmann, J; Hammer, PE; Maguire, CT; Martins, DC; Meister, M; Mende, U; Neer, EJ | 1 |
Chen, ZY; Huang, Y; Ko, WH; Lau, CW; Law, VW; Yip, WC; Yue, GG | 1 |
Choi, S; Lee, CJ; Nam, RH; Park, EJ | 1 |
Crittenden, EL; García, DM; González, A | 1 |
Chaudhuri, A; Gorelick, FS; Kolodecik, TR | 1 |
Philbrick, W; Yamazaki, H; Zawalich, KC; Zawalich, WS | 1 |
Kawahara, K; Kokubo, A; Nishikitani, M; Saigenji, K; Yasuoka, Y | 1 |
Barak, D; Pittel, Z; Segall, Y | 1 |
Hashimoto, N; Iida-Tanaka, N; Ishimaru, S; Ito, M; Matsuda, T; Saito, T; Shigenobu, K; Tanaka, H; Tsuruoka, N; Tsuruzoe, N; Yamashita, T | 1 |
Cho, NJ; Kim, S; Park, YS; Shin, Y | 1 |
Li, YR; Matsunami, H | 1 |
Hasselmo, ME; Heys, JG | 1 |
Bloomquist, JR; Gross, AD | 1 |
1 review(s) available for atropine and colforsin
Article | Year |
---|---|
The role of receptor binding in drug discovery.
Topics: Animals; Drug Design; Humans; Receptors, Drug | 1993 |
61 other study(ies) available for atropine and colforsin
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Suppressive effect of carbachol on forskolin-stimulated neurite outgrowth in human neuroblastoma NB-OK1 cells.
Topics: Atropine; Calcium; Calcium Channel Blockers; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Egtazic Acid; Gallic Acid; Humans; Inositol; Inositol Phosphates; Kinetics; Neurites; Neuroblastoma; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide | 1992 |
Opioid enhancement of evoked [Met5]enkephalin release requires activation of cholinergic receptors: possible involvement of intracellular calcium.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Calcimycin; Calcium; Colforsin; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Enkephalins; Evoked Potentials; Fentanyl; Guinea Pigs; Hexamethonium Compounds; In Vitro Techniques; Myenteric Plexus; Naloxone; Pyrrolidines; Receptors, Muscarinic; Receptors, Opioid; Sufentanil | 1992 |
A possible role of the L-arginine-nitric oxide pathway in the modulation of cholinergic transmission in the guinea-pig taenia coli.
Topics: Animals; Arginine; Atropine; Carbachol; Colforsin; Colon; Dinoprost; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Neural Pathways; Nitric Oxide; Nitroarginine; Nitroprusside; Parasympathetic Nervous System; Synaptic Transmission | 1992 |
Interaction between phosphoinositide turnover system and cyclic AMP pathway for the secretion of pancreastatin and somatostatin from QGP-1N cells.
Topics: Adenoma, Islet Cell; Atropine; Bucladesine; Calcimycin; Carbachol; Cell Line; Chromogranin A; Colforsin; Cyclic AMP; Drug Synergism; Humans; Kinetics; Pancreatic Hormones; Pancreatic Neoplasms; Phosphatidylinositols; Somatostatin; Tetradecanoylphorbol Acetate; Theophylline; Tumor Cells, Cultured | 1992 |
Effects of GTP, forskolin, sodium fluoride, serotonin, dopamine, and carbachol on adenylate cyclase in Teleost retina.
Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Atropine; Carbachol; Colforsin; Cyclic AMP; Dopamine; Drug Synergism; Fishes; GTP-Binding Proteins; Guanosine Triphosphate; Pertussis Toxin; Retina; Serotonin; Sodium Fluoride; Tetrahydronaphthalenes; Virulence Factors, Bordetella | 1990 |
Cl- channel blockers inhibit acid secretion in rabbit parietal cells.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Anthracenes; Atropine; Carbachol; Chloride Channels; Cimetidine; Colforsin; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Ion Channels; Kinetics; Membrane Proteins; ortho-Aminobenzoates; Rabbits | 1990 |
Carbachol enhances forskolin-stimulated cyclic AMP accumulation via activation of calmodulin system in human neuroblastoma SH-SY5Y cells.
Topics: Adenosine; Alprostadil; Atropine; Calmodulin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Synergism; Humans; Kinetics; Naphthalenes; Neuroblastoma; Pertussis Toxin; Polycyclic Compounds; Protein Kinase C; Trifluoperazine; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1991 |
Pluripotent mouse embryonic stem cells are able to differentiate into cardiomyocytes expressing chronotropic responses to adrenergic and cholinergic agents and Ca2+ channel blockers.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Animals, Newborn; Atropine; Calcium Channel Blockers; Carbachol; Cell Differentiation; Cell Line; Colforsin; Dose-Response Relationship, Drug; Embryo, Mammalian; Embryo, Nonmammalian; Heart; Heart Rate; Isoproterenol; Membrane Potentials; Myocardium; Parasympathomimetics; Phenylephrine; Prazosin; Stem Cells; Sympathomimetics | 1991 |
Phospholipase A2 and mediation of the activation of short-circuit current in the rat colonic mucosa.
Topics: Animals; Arachidonic Acid; Atropine; Bradykinin; Colforsin; Colon; Dose-Response Relationship, Drug; Drug Interactions; Female; Indomethacin; Intestinal Mucosa; Masoprocol; Melitten; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Tetrodotoxin | 1991 |
Evidence that a guanine nucleotide-binding protein linked to a muscarinic receptor inhibits directly phospholipase C.
Topics: Alkaloids; Animals; Atropine; Calcimycin; Calcium; Carbachol; Cell Line; Cell Membrane Permeability; Colforsin; Cyclic AMP; Cytosol; GTP-Binding Proteins; Guanosine Triphosphate; Inositol Phosphates; Kinetics; Norepinephrine; Pertussis Toxin; Phosphatidylinositols; Pirenzepine; Receptors, Muscarinic; Staurosporine; Type C Phospholipases; Virulence Factors, Bordetella | 1990 |
Adrenergic and cholinergic interaction in central ventilatory control.
Topics: Acetylcholine; Animals; Atropine; Cardiovascular Physiological Phenomena; Cardiovascular System; Clonidine; Colforsin; Cyclic AMP; Dogs; Isoproterenol; Medulla Oblongata; Propanolamines; Receptors, Adrenergic; Receptors, Cholinergic; Respiration; Respiratory Center; Second Messenger Systems; Yohimbine | 1990 |
Increased airway reactivity in the guinea-pig follows exposure to intravenous isoprenaline.
Topics: Airway Resistance; Animals; Atropine; Blood Platelets; Bombesin; Bronchodilator Agents; Colforsin; Dopamine; Epinephrine; Guinea Pigs; Histamine; Injections, Intravenous; Isoproterenol; Male; Norepinephrine; Platelet Activating Factor; Propranolol; Rabbits; Vagotomy; Vagus Nerve | 1990 |
Neuropeptide Y-cholinergic interactions in neocortical tissue.
Topics: Animals; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Cholinergic Fibers; Colforsin; Gene Expression; In Vitro Techniques; Membrane Potentials; Neuropeptide Y; Potassium; Rats; Receptors, Muscarinic; RNA, Messenger | 1990 |
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains | 1985 |
Hormonal activation of ionic currents in follicle-enclosed Xenopus oocytes.
Topics: Acetylcholine; Animals; Atropine; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Female; Follicle Stimulating Hormone; Ion Channels; Kinetics; Membrane Potentials; Norepinephrine; Oocytes; Ovarian Follicle; Theophylline; Xenopus laevis | 1987 |
Enhanced cAMP accumulation after termination of cholinergic action in the heart.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Heart; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Myocardial Contraction; Myocardium; Parasympathomimetics; Pindolol; Receptors, Muscarinic | 1987 |
Interaction of forskolin with the effect of atropine on [3H]acetylcholine secretion in guinea-pig ileum myenteric plexus.
Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Aminopyridines; Animals; Atropine; Colforsin; Cyclic GMP; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Myenteric Plexus; Neuromuscular Junction | 1988 |
Ca2+-dependent and -independent secretagogue action on gastric mucus secretion in rabbit mucosal explants.
Topics: Acetylcholine; Acetylglucosamine; Animals; Atropine; Calcimycin; Calcium; Calmodulin; Colforsin; Dinoprostone; Gastric Fundus; Gastric Mucosa; Glycoproteins; Histamine; Male; Molecular Weight; Organ Culture Techniques; Pentagastrin; Pyloric Antrum; Rabbits; Sulfonamides; Tetradecanoylphorbol Acetate | 1989 |
Forskolin stimulation of pepsinogen secretion from frog esophageal mucosa is partly mediated by intrinsic cholinergic neurons.
Topics: Animals; Atropine; Bethanechol Compounds; Cholinergic Fibers; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Esophagus; Mucous Membrane; Pepsinogens; Rana catesbeiana; Tetrodotoxin; Time Factors | 1989 |
beta-Adrenergic induced K+ current in Xenopus oocytes: role of cAMP, inhibition by muscarinic agents.
Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adenosine; Aminobenzoates; Aminopyridines; Animals; Atropine; Calcimycin; Colforsin; Cyclic AMP; Diterpenes; Female; Isoproterenol; Oocytes; Phosphodiesterase Inhibitors; Potassium; Receptors, Adrenergic, beta; Tetraethylammonium Compounds; Xenopus laevis | 1985 |
Forskolin, an activator of adenylate cyclase, stimulates pancreatic insulin, glucagon, and somatostatin release in the dog: studies in vitro.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcium; Colforsin; Diterpenes; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Glucagon; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Pancreas; Phentolamine; Propranolol; Somatostatin | 1985 |
Muscarinic acetylcholine receptor function in chick heart cells cultured in serum-free medium.
Topics: Animals; Atropine; Blood; Carbachol; Cells, Cultured; Chick Embryo; Colforsin; Culture Media; Cyclic AMP; Myocardium; Phosphatidylinositols; Receptors, Muscarinic | 1988 |
Beta-adrenergic stimulation of ion transport in primary cultures of avian salt glands.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Atropine; Biological Transport, Active; Carbachol; Cells, Cultured; Colforsin; Cyclic GMP; Ducks; Epinephrine; Furosemide; Ions; Kinetics; Ouabain; Phentolamine; Propranolol; Salt Gland | 1987 |
Carbachol stimulation of inositol phosphate accumulation in rat submandibular gland fragments is not modified by VIP.
Topics: Animals; Atropine; Carbachol; Colforsin; Inositol Phosphates; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Submandibular Gland; Sugar Phosphates; Vasoactive Intestinal Peptide | 1989 |
A study of the histamine H2-receptor mediating relaxation of the parenchymal lung strip preparation of the guinea-pig.
Topics: Animals; Atropine; Colforsin; Dimaprit; Female; Guinea Pigs; In Vitro Techniques; Lung; Male; Muscle Relaxation; Muscle, Smooth; Propranolol; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1985 |
Effects of forskolin on pancreatic exocrine secretion and cyclic nucleotide concentrations of the dog pancreas.
Topics: Animals; Atropine; Cimetidine; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Female; Male; Nucleotides, Cyclic; Pancreatic Juice; Phentolamine; Propranolol; Sulpiride; Verapamil | 1987 |
The effects of isoproterenol on intracellular calcium concentration.
Topics: Animals; Atropine; Calcium; Carbachol; Cattle; Colforsin; Isoproterenol; Muscle Contraction; Muscle, Smooth; Phorbol Esters; Propranolol; Trachea; Vasoactive Intestinal Peptide | 1988 |
Cholecystokinin, carbachol, gastrin, histamine, and forskolin increase [Ca2+]i in gastric glands.
Topics: Aminoquinolines; Animals; Atropine; Calcium; Carbachol; Colforsin; Dibutyryl Cyclic GMP; Fluorescent Dyes; Gastric Mucosa; Gastrins; Histamine; Male; Pepsinogens; Rabbits; Sincalide; Spectrometry, Fluorescence | 1986 |
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger | 1994 |
Role of cyclic adenosine monophosphate in phospholipid synthesis in Mycobacterium smegmatis ATCC 607.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Atropine; Colforsin; Cyclic AMP; Enzyme Activation; Mycobacterium; Phospholipids; Phosphorylation | 1995 |
Structural and functional changes of exocrine pancreas induced by FK506 in rats.
Topics: Amylases; Analysis of Variance; Animals; Atropine; Body Weight; Calcimycin; Calcium; Carbachol; Cholecystokinin; Colforsin; Cytosol; Dose-Response Relationship, Drug; Feeding Behavior; Kinetics; Male; N-Methylscopolamine; Pancreas; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Reference Values; Scopolamine; Scopolamine Derivatives; Secretin; Sincalide; Tacrolimus; Tetradecanoylphorbol Acetate; Time Factors; Trypsinogen; Vasoactive Intestinal Peptide | 1993 |
Cross-talk between muscarinic- and adenosine-receptor signalling in the regulation of cytosolic free Ca2+ and insulin secretion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine; Atropine; Calcium; Calcium Channels; Carbachol; Cells, Cultured; Colforsin; Cytosol; Enzyme Activation; Glyceraldehyde; Insulin; Insulin Secretion; Ion Channel Gating; Muscarinic Antagonists; Receptors, Muscarinic; Receptors, Purinergic; Signal Transduction; Type C Phospholipases | 1993 |
Inhibitory actions of cyclic AMP on neurogenic plasma extravasation in rat airways.
Topics: Anesthesia; Animals; Atropine; Autonomic Nervous System; Bucladesine; Colforsin; Cyclic AMP; Electric Stimulation; Evans Blue; Fenoterol; Hemodynamics; Rats; Rats, Sprague-Dawley; Respiratory System; Substance P; Vagus Nerve | 1993 |
Effects of prostaglandins on [Ca2+]i and adenylate cyclase activity in isolated porcine gastric mucous cells.
Topics: Adenylyl Cyclases; Animals; Atropine; Bucladesine; Calcium; Carbachol; Cells, Cultured; Colforsin; Gastric Mucosa; Histamine; Prostaglandins; Proteins; Ranitidine; Swine | 1994 |
Potentiation of nonadrenergic noncholinergic relaxation of human isolated bronchus by selective inhibitors of phosphodiesterase isozymes.
Topics: Atropine; Bronchi; Colforsin; Electric Stimulation; Histamine; Humans; In Vitro Techniques; Indomethacin; Isoenzymes; Molsidomine; Muscle Relaxation; Nitroprusside; Phosphodiesterase Inhibitors; Propranolol; Purinones; Pyrrolidinones; Rolipram | 1994 |
Acetylcholine muscarinic m1 receptor regulation of cyclic AMP synthesis controls growth factor stimulation of Raf activity.
Topics: Adenylyl Cyclases; Animals; Atropine; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Epidermal Growth Factor; ErbB Receptors; Gene Expression; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Models, Biological; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Platelet-Derived Growth Factor; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Rats; Receptor Protein-Tyrosine Kinases; Receptors, Muscarinic; Receptors, Platelet-Derived Growth Factor; Transfection | 1994 |
Differential regulation of cAMP-mediated gene transcription by m1 and m4 muscarinic acetylcholine receptors. Preferential coupling of m4 receptors to Gi alpha-2.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atropine; beta-Galactosidase; Calcium; Cell Line; Chickens; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA; Gene Expression Regulation; GTP-Binding Proteins; Kinetics; Luciferases; Pertussis Toxin; Rats; Receptors, Muscarinic; Transcription, Genetic; Transfection; Virulence Factors, Bordetella | 1994 |
Breakdown of membrane choline-phospholipids induced by endogenous and exogenous muscarinic agonist is potentiated by VIP in rat submandibular gland.
Topics: Animals; Atropine; Carbachol; Colforsin; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Membranes; Parasympathomimetics; Perfusion; Phosphatidylcholines; Phospholipases; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Signal Transduction; Stimulation, Chemical; Submandibular Gland; Vasoactive Intestinal Peptide | 1993 |
Agonist-independent effects of muscarinic antagonists on Ca2+ and K+ currents in frog and rat cardiac cells.
Topics: Adenylyl Cyclases; Animals; Atropine; Calcium; Cells, Cultured; Colforsin; Electrophysiology; Guanylyl Imidodiphosphate; Heart Ventricles; In Vitro Techniques; Muscarinic Antagonists; Myocardium; Potassium; Rana esculenta; Rats; Rats, Wistar; Receptors, Muscarinic | 1993 |
Rapid agonist-mediated phosphorylation of m3-muscarinic receptors revealed by immunoprecipitation.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Atropine; Base Sequence; Carbachol; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Electrophoresis, Polyacrylamide Gel; Glutathione Transferase; Humans; Immune Sera; Immunoblotting; Ionomycin; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Parasympathomimetics; Phosphates; Phosphorylation; Plasmids; Polymerase Chain Reaction; Protein Kinases; Receptors, Muscarinic; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection | 1993 |
Expression of functional muscarinic acetylcholine receptor subtypes in human corpus cavernosum and in cultured smooth muscle cells.
Topics: Adenylyl Cyclases; Alprostadil; Atropine; Carbachol; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Humans; In Situ Hybridization; Isoproterenol; Kinetics; Male; Models, Biological; Muscle, Smooth; Penis; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Muscarinic; RNA, Messenger; Transcription, Genetic | 1995 |
Paradoxical facilitation of acetylcholine release from parasympathetic nerves innervating guinea-pig trachea by isoprenaline.
Topics: Acetylcholine; Adrenergic beta-Agonists; Animals; Atropine; Colforsin; Cyclic AMP; Dinoprostone; Electric Stimulation; Guinea Pigs; Humans; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Neuromuscular Junction; Parasympathetic Nervous System; Phosphodiesterase Inhibitors; Synaptic Transmission; Trachea | 1996 |
Regulation of tyrosine hydroxylase gene expression by the m1 muscarinic acetylcholine receptor in rat pheochromocytoma cells.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenal Gland Neoplasms; Animals; Atropine; Calcium; Carbachol; Cell Membrane; Chloramphenicol O-Acetyltransferase; Colforsin; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Mice; Mutagenesis, Site-Directed; Pheochromocytoma; Phosphatidylinositols; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Fusion Proteins; Transcription, Genetic; Tumor Cells, Cultured; Tyrosine 3-Monooxygenase | 1996 |
Muscarinic autoinhibition of acetylcholine release in mouse atria is not transduced through cyclic AMP or protein kinase C.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adenylyl Cyclases; Animals; Atrial Function; Atropine; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Heart; Heart Atria; In Vitro Techniques; Male; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Muscarinic; Second Messenger Systems; Staurosporine | 1996 |
Carbachol inhibits basal and forskolin-evoked adult rat striatal acetylcholine release.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Atropine; Carbachol; Cholinergic Agonists; Cholinergic Antagonists; Colforsin; Depression, Chemical; In Vitro Techniques; Male; Neostriatum; Neurons; Rats | 1997 |
Decreased adenylyl cyclase protein and function in airway smooth muscle by chronic carbachol pretreatment.
Topics: Adenylyl Cyclases; Aluminum; Animals; Atropine; Carbachol; Cattle; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Down-Regulation; Enzyme Activation; Erythrocytes; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Immunoblotting; Mice; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth; Radioligand Assay; Sodium Fluoride; Time; Trachea | 2000 |
Impaired parasympathetic heart rate control in mice with a reduction of functional G protein betagamma-subunits.
Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Atropine; Cardiotonic Agents; Cell Membrane; Colforsin; Consciousness; Cyclic AMP; Cytosol; Electrocardiography; Electrophysiology; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Heart Rate; Heterotrimeric GTP-Binding Proteins; Isoproterenol; Mice; Mice, Transgenic; Parasympathetic Nervous System; Propranolol; Sinoatrial Node; Transgenes; Vagus Nerve; Vasodilator Agents | 2002 |
Stimulation of chloride secretion by baicalein in isolated rat distal colon.
Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Animals; Atropine; Calcium; Carbachol; Chlorides; Colforsin; Colon; Cyclic AMP; Dinoprostone; Electric Conductivity; Female; Flavanones; Flavonoids; Indomethacin; Intestinal Mucosa; Male; Muscarinic Antagonists; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Thapsigargin | 2002 |
Carbachol induces a form of long-term potentiation in lateral amygdala.
Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Afferent Pathways; Amygdala; Animals; Atropine; Carbachol; Cholinergic Agonists; Colforsin; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Long-Term Potentiation; Muscarinic Antagonists; Neurons; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Thalamus | 2004 |
Activation of muscarinic acetylcholine receptors elicits pigment granule dispersion in retinal pigment epithelium isolated from bluegill.
Topics: Adenylyl Cyclase Inhibitors; Animals; Arecoline; Atropine; Carbachol; Colforsin; Cyclic AMP; Cytoplasmic Granules; Light; Muscarinic Agonists; Muscarinic Antagonists; Perciformes; Pigment Epithelium of Eye; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Retinal Pigments; Second Messenger Systems; Tropicamide | 2004 |
Effects of increased intracellular cAMP on carbachol-stimulated zymogen activation, secretion, and injury in the pancreatic acinar cell.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amylases; Animals; Atropine; Carbachol; Cholinergic Agonists; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Precursors; Gastrointestinal Agents; In Vitro Techniques; Male; Muscarinic Antagonists; Pancreas, Exocrine; Rats; Rats, Sprague-Dawley; Secretin | 2005 |
Acute and chronic effects of glucose and carbachol on insulin secretion and phospholipase C activation: studies with diazoxide and atropine.
Topics: Animals; Atropine; Carbachol; Colforsin; Diazoxide; Enzyme Activation; Glucose; Hyperglycemia; In Vitro Techniques; Inositol; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Sprague-Dawley; Type C Phospholipases | 2006 |
Restoration by VIP of the carbachol-stimulated Cl- secretion in TTX-treated guinea pig distal colon.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atropine; Carbachol; Chlorides; Cholinergic Agents; Cholinergic Fibers; Colforsin; Colon, Descending; Dose-Response Relationship, Drug; Electric Stimulation; Enteric Nervous System; Gastrointestinal Agents; Guinea Pigs; Intestinal Mucosa; Male; Membrane Potentials; Neuroepithelial Cells; Neurotransmitter Agents; Patch-Clamp Techniques; Poisons; Tetrodotoxin; Vasoactive Intestinal Peptide | 2005 |
Function-specific blockage of M(1) and M(3) muscarinic acetylcholine receptors by VX and echothiophate.
Topics: Animals; Atropine; CHO Cells; Cholinesterase Inhibitors; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Echothiophate Iodide; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Organothiophosphorus Compounds; Oxotremorine; Phosphatidylinositols; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Transfection; Tritium | 2006 |
Blockade by NIP-142, an antiarrhythmic agent, of carbachol-induced atrial action potential shortening and GIRK1/4 channel.
Topics: Action Potentials; Adenosine; Animals; Anti-Arrhythmia Agents; Atrial Function; Atropine; Bee Venoms; Benzopyrans; Carbachol; Cell Line; Colforsin; Dose-Response Relationship, Drug; Ether-A-Go-Go Potassium Channels; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Guinea Pigs; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Patch-Clamp Techniques; Potassium Channel Blockers; Time Factors | 2006 |
Regulation of ERK1/2 by the C. elegans muscarinic acetylcholine receptor GAR-3 in Chinese hamster ovary cells.
Topics: Alternative Splicing; Animals; Atropine; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Carbachol; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Estrenes; Indoles; Isoquinolines; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscarinic Agonists; Muscarinic Antagonists; Protein Isoforms; Protein Kinase C; Pyrrolidinones; Receptors, Muscarinic; Recombinant Proteins; Signal Transduction; Sulfonamides; Transfection; Type C Phospholipases | 2008 |
Activation state of the M3 muscarinic acetylcholine receptor modulates mammalian odorant receptor signaling.
Topics: Atropine; Benzofurans; Carbachol; Cholinergic Agonists; Colforsin; Cyclic AMP; HEK293 Cells; Humans; Immunohistochemistry; Ionomycin; Ionophores; Membrane Transport Proteins; Muscarinic Antagonists; Olfactory Receptor Neurons; Protein Binding; Pyrrolidines; Receptor, Muscarinic M3; Receptors, G-Protein-Coupled; Receptors, Odorant; Signal Transduction; Transfection | 2011 |
Neuromodulation of I(h) in layer II medial entorhinal cortex stellate cells: a voltage-clamp study.
Topics: Animals; Animals, Newborn; Anthracenes; Atropine; Biophysical Phenomena; Carbachol; Cardiotonic Agents; Cholinergic Antagonists; Colforsin; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Entorhinal Cortex; Female; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotransmitter Agents; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Sodium Channel Blockers; Tetrodotoxin; Time Factors | 2012 |
Pharmacology of central octopaminergic and muscarinic pathways in Drosophila melanogaster larvae: Assessing the target potential of GPCRs.
Topics: Animals; Atropine; Central Nervous System; Colforsin; Cyclic CMP; Drosophila melanogaster; Electrophysiology; Larva; Octopamine; Phentolamine; Pilocarpine; Receptors, G-Protein-Coupled | 2018 |