Page last updated: 2024-09-05

atropine and colforsin

atropine has been researched along with colforsin in 62 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
26,7111,2591,69713,460461,298

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (62)

TimeframeStudies, this research(%)All Research%
pre-199016 (25.81)18.7374
1990's31 (50.00)18.2507
2000's11 (17.74)29.6817
2010's4 (6.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Nakagawa-Yagi, Y; Nakamura, H; Saito, Y; Takada, Y1
Gintzler, AR; Xu, H1
Knudsen, MA; Tøttrup, A1
Funakoshi, A; Kitayama, N; Matsuoka, Y; Tateishi, K1
Osborne, NN1
Malinowska, DH1
Nakagawa-Yagi, Y; Saito, Y; Takada, Y; Takayama, M1
Hescheler, J; Wallukat, G; Wobus, AM1
Diener, M; Rummel, W1
Bizzarri, C; Corda, D; D'Orazio, MC; Di Girolamo, M1
Burton, MD; Johnson, DC; Kazemi, H1
Kristersson, A; Mazzoni, L; Morley, J; Sanjar, S; Schaeublin, E1
Meyer, EM; Millard, WJ; Poulakos, JJ; Pruysers, CR1
Nezu, E; Yoneyama, T; Yoshimura, K1
Miledi, R; Woodward, RM1
Linden, J1
Alberts, P; Ogren, VR1
Seidler, U; Sewing, KF1
Fong, JC; Ho, LT; Wang, FF1
Renit-Soria, J; Stinnakre, J; Van Renterghem, C1
Hermansen, K1
Nathanson, NM; Subers, EM1
Ernst, SA; Lowy, RJ1
Fredholm, BB; Larsson, O1
Foreman, JC; Rising, TJ; Webber, SE1
Chiba, S; Horiuchi, A; Iwatsuki, K; Yamagishi, F1
Rasmussen, H; Takuwa, N; Takuwa, Y1
Chew, CS1
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ1
Kaur, H; Khuller, GK1
Chowdhury, P; Doi, R; Inoue, K; Kaji, H; Rayford, PL1
Biden, TJ; Browne, CL1
Morikawa, M; Sasaki, H; Sekizawa, K1
Beil, W; Bersimbaev, RI; Gandjour, A; Heim, HK; Sewing, KF1
Ellis, JL; Fernandes, LB; Undem, BJ1
Johnson, GL; Russell, M; Winitz, S1
Migeon, JC; Nathanson, NM1
Dunér-Engström, M; Fredholm, BB1
Fischmeister, R; Hanf, R; Li, Y; Szabo, G1
Nahorski, SR; Tobin, AB1
Goldstein, I; Moreland, RB; Palmer, MS; Traish, AM1
Barnes, PJ; Belvisi, MG; Giembycz, MA; Patel, HJ; Takahashi, T1
Best, JA; Chen, Y; Nagamoto, K; Tank, AW1
Dawson, JJ; Iannazzo, L; Majewski, H1
Login, IS1
Clancy-Keen, J; Emala, CW; Hirshman, CA1
Berul, CI; Gehrmann, J; Hammer, PE; Maguire, CT; Martins, DC; Meister, M; Mende, U; Neer, EJ1
Chen, ZY; Huang, Y; Ko, WH; Lau, CW; Law, VW; Yip, WC; Yue, GG1
Choi, S; Lee, CJ; Nam, RH; Park, EJ1
Crittenden, EL; García, DM; González, A1
Chaudhuri, A; Gorelick, FS; Kolodecik, TR1
Philbrick, W; Yamazaki, H; Zawalich, KC; Zawalich, WS1
Kawahara, K; Kokubo, A; Nishikitani, M; Saigenji, K; Yasuoka, Y1
Barak, D; Pittel, Z; Segall, Y1
Hashimoto, N; Iida-Tanaka, N; Ishimaru, S; Ito, M; Matsuda, T; Saito, T; Shigenobu, K; Tanaka, H; Tsuruoka, N; Tsuruzoe, N; Yamashita, T1
Cho, NJ; Kim, S; Park, YS; Shin, Y1
Li, YR; Matsunami, H1
Hasselmo, ME; Heys, JG1
Bloomquist, JR; Gross, AD1

Reviews

1 review(s) available for atropine and colforsin

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

61 other study(ies) available for atropine and colforsin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Suppressive effect of carbachol on forskolin-stimulated neurite outgrowth in human neuroblastoma NB-OK1 cells.
    Biochemical and biophysical research communications, 1992, Jan-15, Volume: 182, Issue:1

    Topics: Atropine; Calcium; Calcium Channel Blockers; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Interactions; Egtazic Acid; Gallic Acid; Humans; Inositol; Inositol Phosphates; Kinetics; Neurites; Neuroblastoma; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide

1992
Opioid enhancement of evoked [Met5]enkephalin release requires activation of cholinergic receptors: possible involvement of intracellular calcium.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Mar-01, Volume: 89, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Calcimycin; Calcium; Colforsin; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Enkephalins; Evoked Potentials; Fentanyl; Guinea Pigs; Hexamethonium Compounds; In Vitro Techniques; Myenteric Plexus; Naloxone; Pyrrolidines; Receptors, Muscarinic; Receptors, Opioid; Sufentanil

1992
A possible role of the L-arginine-nitric oxide pathway in the modulation of cholinergic transmission in the guinea-pig taenia coli.
    British journal of pharmacology, 1992, Volume: 107, Issue:3

    Topics: Animals; Arginine; Atropine; Carbachol; Colforsin; Colon; Dinoprost; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Neural Pathways; Nitric Oxide; Nitroarginine; Nitroprusside; Parasympathetic Nervous System; Synaptic Transmission

1992
Interaction between phosphoinositide turnover system and cyclic AMP pathway for the secretion of pancreastatin and somatostatin from QGP-1N cells.
    Biochemical and biophysical research communications, 1992, Jun-30, Volume: 185, Issue:3

    Topics: Adenoma, Islet Cell; Atropine; Bucladesine; Calcimycin; Carbachol; Cell Line; Chromogranin A; Colforsin; Cyclic AMP; Drug Synergism; Humans; Kinetics; Pancreatic Hormones; Pancreatic Neoplasms; Phosphatidylinositols; Somatostatin; Tetradecanoylphorbol Acetate; Theophylline; Tumor Cells, Cultured

1992
Effects of GTP, forskolin, sodium fluoride, serotonin, dopamine, and carbachol on adenylate cyclase in Teleost retina.
    Neurochemical research, 1990, Volume: 15, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Atropine; Carbachol; Colforsin; Cyclic AMP; Dopamine; Drug Synergism; Fishes; GTP-Binding Proteins; Guanosine Triphosphate; Pertussis Toxin; Retina; Serotonin; Sodium Fluoride; Tetrahydronaphthalenes; Virulence Factors, Bordetella

1990
Cl- channel blockers inhibit acid secretion in rabbit parietal cells.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Anthracenes; Atropine; Carbachol; Chloride Channels; Cimetidine; Colforsin; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Ion Channels; Kinetics; Membrane Proteins; ortho-Aminobenzoates; Rabbits

1990
Carbachol enhances forskolin-stimulated cyclic AMP accumulation via activation of calmodulin system in human neuroblastoma SH-SY5Y cells.
    Biochemical and biophysical research communications, 1991, Jul-15, Volume: 178, Issue:1

    Topics: Adenosine; Alprostadil; Atropine; Calmodulin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Drug Synergism; Humans; Kinetics; Naphthalenes; Neuroblastoma; Pertussis Toxin; Polycyclic Compounds; Protein Kinase C; Trifluoperazine; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella

1991
Pluripotent mouse embryonic stem cells are able to differentiate into cardiomyocytes expressing chronotropic responses to adrenergic and cholinergic agents and Ca2+ channel blockers.
    Differentiation; research in biological diversity, 1991, Volume: 48, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Animals, Newborn; Atropine; Calcium Channel Blockers; Carbachol; Cell Differentiation; Cell Line; Colforsin; Dose-Response Relationship, Drug; Embryo, Mammalian; Embryo, Nonmammalian; Heart; Heart Rate; Isoproterenol; Membrane Potentials; Myocardium; Parasympathomimetics; Phenylephrine; Prazosin; Stem Cells; Sympathomimetics

1991
Phospholipase A2 and mediation of the activation of short-circuit current in the rat colonic mucosa.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:6

    Topics: Animals; Arachidonic Acid; Atropine; Bradykinin; Colforsin; Colon; Dose-Response Relationship, Drug; Drug Interactions; Female; Indomethacin; Intestinal Mucosa; Masoprocol; Melitten; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Tetrodotoxin

1991
Evidence that a guanine nucleotide-binding protein linked to a muscarinic receptor inhibits directly phospholipase C.
    Proceedings of the National Academy of Sciences of the United States of America, 1990, Volume: 87, Issue:12

    Topics: Alkaloids; Animals; Atropine; Calcimycin; Calcium; Carbachol; Cell Line; Cell Membrane Permeability; Colforsin; Cyclic AMP; Cytosol; GTP-Binding Proteins; Guanosine Triphosphate; Inositol Phosphates; Kinetics; Norepinephrine; Pertussis Toxin; Phosphatidylinositols; Pirenzepine; Receptors, Muscarinic; Staurosporine; Type C Phospholipases; Virulence Factors, Bordetella

1990
Adrenergic and cholinergic interaction in central ventilatory control.
    Journal of applied physiology (Bethesda, Md. : 1985), 1990, Volume: 68, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Cardiovascular Physiological Phenomena; Cardiovascular System; Clonidine; Colforsin; Cyclic AMP; Dogs; Isoproterenol; Medulla Oblongata; Propanolamines; Receptors, Adrenergic; Receptors, Cholinergic; Respiration; Respiratory Center; Second Messenger Systems; Yohimbine

1990
Increased airway reactivity in the guinea-pig follows exposure to intravenous isoprenaline.
    The Journal of physiology, 1990, Volume: 425

    Topics: Airway Resistance; Animals; Atropine; Blood Platelets; Bombesin; Bronchodilator Agents; Colforsin; Dopamine; Epinephrine; Guinea Pigs; Histamine; Injections, Intravenous; Isoproterenol; Male; Norepinephrine; Platelet Activating Factor; Propranolol; Rabbits; Vagotomy; Vagus Nerve

1990
Neuropeptide Y-cholinergic interactions in neocortical tissue.
    Annals of the New York Academy of Sciences, 1990, Volume: 611

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Cholinergic Fibers; Colforsin; Gene Expression; In Vitro Techniques; Membrane Potentials; Neuropeptide Y; Potassium; Rats; Receptors, Muscarinic; RNA, Messenger

1990
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
    The Japanese journal of physiology, 1985, Volume: 35, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains

1985
Hormonal activation of ionic currents in follicle-enclosed Xenopus oocytes.
    Proceedings of the National Academy of Sciences of the United States of America, 1987, Volume: 84, Issue:12

    Topics: Acetylcholine; Animals; Atropine; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Female; Follicle Stimulating Hormone; Ion Channels; Kinetics; Membrane Potentials; Norepinephrine; Oocytes; Ovarian Follicle; Theophylline; Xenopus laevis

1987
Enhanced cAMP accumulation after termination of cholinergic action in the heart.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1987, Volume: 1, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Heart; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Myocardial Contraction; Myocardium; Parasympathomimetics; Pindolol; Receptors, Muscarinic

1987
Interaction of forskolin with the effect of atropine on [3H]acetylcholine secretion in guinea-pig ileum myenteric plexus.
    The Journal of physiology, 1988, Volume: 395

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Aminopyridines; Animals; Atropine; Colforsin; Cyclic GMP; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Myenteric Plexus; Neuromuscular Junction

1988
Ca2+-dependent and -independent secretagogue action on gastric mucus secretion in rabbit mucosal explants.
    The American journal of physiology, 1989, Volume: 256, Issue:4 Pt 1

    Topics: Acetylcholine; Acetylglucosamine; Animals; Atropine; Calcimycin; Calcium; Calmodulin; Colforsin; Dinoprostone; Gastric Fundus; Gastric Mucosa; Glycoproteins; Histamine; Male; Molecular Weight; Organ Culture Techniques; Pentagastrin; Pyloric Antrum; Rabbits; Sulfonamides; Tetradecanoylphorbol Acetate

1989
Forskolin stimulation of pepsinogen secretion from frog esophageal mucosa is partly mediated by intrinsic cholinergic neurons.
    Biochemistry international, 1989, Volume: 19, Issue:6

    Topics: Animals; Atropine; Bethanechol Compounds; Cholinergic Fibers; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Esophagus; Mucous Membrane; Pepsinogens; Rana catesbeiana; Tetrodotoxin; Time Factors

1989
beta-Adrenergic induced K+ current in Xenopus oocytes: role of cAMP, inhibition by muscarinic agents.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1985, Jan-22, Volume: 223, Issue:1232

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adenosine; Aminobenzoates; Aminopyridines; Animals; Atropine; Calcimycin; Colforsin; Cyclic AMP; Diterpenes; Female; Isoproterenol; Oocytes; Phosphodiesterase Inhibitors; Potassium; Receptors, Adrenergic, beta; Tetraethylammonium Compounds; Xenopus laevis

1985
Forskolin, an activator of adenylate cyclase, stimulates pancreatic insulin, glucagon, and somatostatin release in the dog: studies in vitro.
    Endocrinology, 1985, Volume: 116, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcium; Colforsin; Diterpenes; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Glucagon; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Pancreas; Phentolamine; Propranolol; Somatostatin

1985
Muscarinic acetylcholine receptor function in chick heart cells cultured in serum-free medium.
    Journal of molecular and cellular cardiology, 1988, Volume: 20, Issue:2

    Topics: Animals; Atropine; Blood; Carbachol; Cells, Cultured; Chick Embryo; Colforsin; Culture Media; Cyclic AMP; Myocardium; Phosphatidylinositols; Receptors, Muscarinic

1988
Beta-adrenergic stimulation of ion transport in primary cultures of avian salt glands.
    The American journal of physiology, 1987, Volume: 252, Issue:6 Pt 1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Atropine; Biological Transport, Active; Carbachol; Cells, Cultured; Colforsin; Cyclic GMP; Ducks; Epinephrine; Furosemide; Ions; Kinetics; Ouabain; Phentolamine; Propranolol; Salt Gland

1987
Carbachol stimulation of inositol phosphate accumulation in rat submandibular gland fragments is not modified by VIP.
    Acta physiologica Scandinavica, 1989, Volume: 135, Issue:3

    Topics: Animals; Atropine; Carbachol; Colforsin; Inositol Phosphates; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Submandibular Gland; Sugar Phosphates; Vasoactive Intestinal Peptide

1989
A study of the histamine H2-receptor mediating relaxation of the parenchymal lung strip preparation of the guinea-pig.
    British journal of pharmacology, 1985, Volume: 86, Issue:2

    Topics: Animals; Atropine; Colforsin; Dimaprit; Female; Guinea Pigs; In Vitro Techniques; Lung; Male; Muscle Relaxation; Muscle, Smooth; Propranolol; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1985
Effects of forskolin on pancreatic exocrine secretion and cyclic nucleotide concentrations of the dog pancreas.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 286, Issue:2

    Topics: Animals; Atropine; Cimetidine; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Female; Male; Nucleotides, Cyclic; Pancreatic Juice; Phentolamine; Propranolol; Sulpiride; Verapamil

1987
The effects of isoproterenol on intracellular calcium concentration.
    The Journal of biological chemistry, 1988, Jan-15, Volume: 263, Issue:2

    Topics: Animals; Atropine; Calcium; Carbachol; Cattle; Colforsin; Isoproterenol; Muscle Contraction; Muscle, Smooth; Phorbol Esters; Propranolol; Trachea; Vasoactive Intestinal Peptide

1988
Cholecystokinin, carbachol, gastrin, histamine, and forskolin increase [Ca2+]i in gastric glands.
    The American journal of physiology, 1986, Volume: 250, Issue:6 Pt 1

    Topics: Aminoquinolines; Animals; Atropine; Calcium; Carbachol; Colforsin; Dibutyryl Cyclic GMP; Fluorescent Dyes; Gastric Mucosa; Gastrins; Histamine; Male; Pepsinogens; Rabbits; Sincalide; Spectrometry, Fluorescence

1986
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger

1994
Role of cyclic adenosine monophosphate in phospholipid synthesis in Mycobacterium smegmatis ATCC 607.
    Lipids, 1995, Volume: 30, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Atropine; Colforsin; Cyclic AMP; Enzyme Activation; Mycobacterium; Phospholipids; Phosphorylation

1995
Structural and functional changes of exocrine pancreas induced by FK506 in rats.
    Gastroenterology, 1993, Volume: 104, Issue:4

    Topics: Amylases; Analysis of Variance; Animals; Atropine; Body Weight; Calcimycin; Calcium; Carbachol; Cholecystokinin; Colforsin; Cytosol; Dose-Response Relationship, Drug; Feeding Behavior; Kinetics; Male; N-Methylscopolamine; Pancreas; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Reference Values; Scopolamine; Scopolamine Derivatives; Secretin; Sincalide; Tacrolimus; Tetradecanoylphorbol Acetate; Time Factors; Trypsinogen; Vasoactive Intestinal Peptide

1993
Cross-talk between muscarinic- and adenosine-receptor signalling in the regulation of cytosolic free Ca2+ and insulin secretion.
    The Biochemical journal, 1993, Aug-01, Volume: 293 ( Pt 3)

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine; Atropine; Calcium; Calcium Channels; Carbachol; Cells, Cultured; Colforsin; Cytosol; Enzyme Activation; Glyceraldehyde; Insulin; Insulin Secretion; Ion Channel Gating; Muscarinic Antagonists; Receptors, Muscarinic; Receptors, Purinergic; Signal Transduction; Type C Phospholipases

1993
Inhibitory actions of cyclic AMP on neurogenic plasma extravasation in rat airways.
    European journal of pharmacology, 1993, Sep-07, Volume: 241, Issue:1

    Topics: Anesthesia; Animals; Atropine; Autonomic Nervous System; Bucladesine; Colforsin; Cyclic AMP; Electric Stimulation; Evans Blue; Fenoterol; Hemodynamics; Rats; Rats, Sprague-Dawley; Respiratory System; Substance P; Vagus Nerve

1993
Effects of prostaglandins on [Ca2+]i and adenylate cyclase activity in isolated porcine gastric mucous cells.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 1994, Volume: 45, Issue:2

    Topics: Adenylyl Cyclases; Animals; Atropine; Bucladesine; Calcium; Carbachol; Cells, Cultured; Colforsin; Gastric Mucosa; Histamine; Prostaglandins; Proteins; Ranitidine; Swine

1994
Potentiation of nonadrenergic noncholinergic relaxation of human isolated bronchus by selective inhibitors of phosphodiesterase isozymes.
    American journal of respiratory and critical care medicine, 1994, Volume: 150, Issue:5 Pt 1

    Topics: Atropine; Bronchi; Colforsin; Electric Stimulation; Histamine; Humans; In Vitro Techniques; Indomethacin; Isoenzymes; Molsidomine; Muscle Relaxation; Nitroprusside; Phosphodiesterase Inhibitors; Propranolol; Purinones; Pyrrolidinones; Rolipram

1994
Acetylcholine muscarinic m1 receptor regulation of cyclic AMP synthesis controls growth factor stimulation of Raf activity.
    Molecular and cellular biology, 1994, Volume: 14, Issue:4

    Topics: Adenylyl Cyclases; Animals; Atropine; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Epidermal Growth Factor; ErbB Receptors; Gene Expression; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Models, Biological; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Platelet-Derived Growth Factor; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Rats; Receptor Protein-Tyrosine Kinases; Receptors, Muscarinic; Receptors, Platelet-Derived Growth Factor; Transfection

1994
Differential regulation of cAMP-mediated gene transcription by m1 and m4 muscarinic acetylcholine receptors. Preferential coupling of m4 receptors to Gi alpha-2.
    The Journal of biological chemistry, 1994, Apr-01, Volume: 269, Issue:13

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Atropine; beta-Galactosidase; Calcium; Cell Line; Chickens; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA; Gene Expression Regulation; GTP-Binding Proteins; Kinetics; Luciferases; Pertussis Toxin; Rats; Receptors, Muscarinic; Transcription, Genetic; Transfection; Virulence Factors, Bordetella

1994
Breakdown of membrane choline-phospholipids induced by endogenous and exogenous muscarinic agonist is potentiated by VIP in rat submandibular gland.
    Acta physiologica Scandinavica, 1993, Volume: 149, Issue:1

    Topics: Animals; Atropine; Carbachol; Colforsin; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Membranes; Parasympathomimetics; Perfusion; Phosphatidylcholines; Phospholipases; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Signal Transduction; Stimulation, Chemical; Submandibular Gland; Vasoactive Intestinal Peptide

1993
Agonist-independent effects of muscarinic antagonists on Ca2+ and K+ currents in frog and rat cardiac cells.
    The Journal of physiology, 1993, Volume: 461

    Topics: Adenylyl Cyclases; Animals; Atropine; Calcium; Cells, Cultured; Colforsin; Electrophysiology; Guanylyl Imidodiphosphate; Heart Ventricles; In Vitro Techniques; Muscarinic Antagonists; Myocardium; Potassium; Rana esculenta; Rats; Rats, Wistar; Receptors, Muscarinic

1993
Rapid agonist-mediated phosphorylation of m3-muscarinic receptors revealed by immunoprecipitation.
    The Journal of biological chemistry, 1993, May-05, Volume: 268, Issue:13

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Atropine; Base Sequence; Carbachol; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Electrophoresis, Polyacrylamide Gel; Glutathione Transferase; Humans; Immune Sera; Immunoblotting; Ionomycin; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Parasympathomimetics; Phosphates; Phosphorylation; Plasmids; Polymerase Chain Reaction; Protein Kinases; Receptors, Muscarinic; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection

1993
Expression of functional muscarinic acetylcholine receptor subtypes in human corpus cavernosum and in cultured smooth muscle cells.
    Receptor, 1995,Fall, Volume: 5, Issue:3

    Topics: Adenylyl Cyclases; Alprostadil; Atropine; Carbachol; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Humans; In Situ Hybridization; Isoproterenol; Kinetics; Male; Models, Biological; Muscle, Smooth; Penis; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Muscarinic; RNA, Messenger; Transcription, Genetic

1995
Paradoxical facilitation of acetylcholine release from parasympathetic nerves innervating guinea-pig trachea by isoprenaline.
    British journal of pharmacology, 1996, Volume: 117, Issue:7

    Topics: Acetylcholine; Adrenergic beta-Agonists; Animals; Atropine; Colforsin; Cyclic AMP; Dinoprostone; Electric Stimulation; Guinea Pigs; Humans; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth; Neuromuscular Junction; Parasympathetic Nervous System; Phosphodiesterase Inhibitors; Synaptic Transmission; Trachea

1996
Regulation of tyrosine hydroxylase gene expression by the m1 muscarinic acetylcholine receptor in rat pheochromocytoma cells.
    Brain research. Molecular brain research, 1996, Volume: 40, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenal Gland Neoplasms; Animals; Atropine; Calcium; Carbachol; Cell Membrane; Chloramphenicol O-Acetyltransferase; Colforsin; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Mice; Mutagenesis, Site-Directed; Pheochromocytoma; Phosphatidylinositols; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Recombinant Fusion Proteins; Transcription, Genetic; Tumor Cells, Cultured; Tyrosine 3-Monooxygenase

1996
Muscarinic autoinhibition of acetylcholine release in mouse atria is not transduced through cyclic AMP or protein kinase C.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adenylyl Cyclases; Animals; Atrial Function; Atropine; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Heart; Heart Atria; In Vitro Techniques; Male; Mice; Phorbol 12,13-Dibutyrate; Protein Kinase C; Receptors, Muscarinic; Second Messenger Systems; Staurosporine

1996
Carbachol inhibits basal and forskolin-evoked adult rat striatal acetylcholine release.
    Neuroreport, 1997, May-27, Volume: 8, Issue:8

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Atropine; Carbachol; Cholinergic Agonists; Cholinergic Antagonists; Colforsin; Depression, Chemical; In Vitro Techniques; Male; Neostriatum; Neurons; Rats

1997
Decreased adenylyl cyclase protein and function in airway smooth muscle by chronic carbachol pretreatment.
    American journal of physiology. Cell physiology, 2000, Volume: 279, Issue:4

    Topics: Adenylyl Cyclases; Aluminum; Animals; Atropine; Carbachol; Cattle; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Down-Regulation; Enzyme Activation; Erythrocytes; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Immunoblotting; Mice; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth; Radioligand Assay; Sodium Fluoride; Time; Trachea

2000
Impaired parasympathetic heart rate control in mice with a reduction of functional G protein betagamma-subunits.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Atropine; Cardiotonic Agents; Cell Membrane; Colforsin; Consciousness; Cyclic AMP; Cytosol; Electrocardiography; Electrophysiology; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Heart Rate; Heterotrimeric GTP-Binding Proteins; Isoproterenol; Mice; Mice, Transgenic; Parasympathetic Nervous System; Propranolol; Sinoatrial Node; Transgenes; Vagus Nerve; Vasodilator Agents

2002
Stimulation of chloride secretion by baicalein in isolated rat distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Animals; Atropine; Calcium; Carbachol; Chlorides; Colforsin; Colon; Cyclic AMP; Dinoprostone; Electric Conductivity; Female; Flavanones; Flavonoids; Indomethacin; Intestinal Mucosa; Male; Muscarinic Antagonists; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Thapsigargin

2002
Carbachol induces a form of long-term potentiation in lateral amygdala.
    Neuroreport, 2004, Jun-07, Volume: 15, Issue:8

    Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Afferent Pathways; Amygdala; Animals; Atropine; Carbachol; Cholinergic Agonists; Colforsin; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Long-Term Potentiation; Muscarinic Antagonists; Neurons; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Thalamus

2004
Activation of muscarinic acetylcholine receptors elicits pigment granule dispersion in retinal pigment epithelium isolated from bluegill.
    BMC neuroscience, 2004, Jul-13, Volume: 5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Arecoline; Atropine; Carbachol; Colforsin; Cyclic AMP; Cytoplasmic Granules; Light; Muscarinic Agonists; Muscarinic Antagonists; Perciformes; Pigment Epithelium of Eye; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Retinal Pigments; Second Messenger Systems; Tropicamide

2004
Effects of increased intracellular cAMP on carbachol-stimulated zymogen activation, secretion, and injury in the pancreatic acinar cell.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 288, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amylases; Animals; Atropine; Carbachol; Cholinergic Agonists; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Precursors; Gastrointestinal Agents; In Vitro Techniques; Male; Muscarinic Antagonists; Pancreas, Exocrine; Rats; Rats, Sprague-Dawley; Secretin

2005
Acute and chronic effects of glucose and carbachol on insulin secretion and phospholipase C activation: studies with diazoxide and atropine.
    American journal of physiology. Endocrinology and metabolism, 2006, Volume: 290, Issue:1

    Topics: Animals; Atropine; Carbachol; Colforsin; Diazoxide; Enzyme Activation; Glucose; Hyperglycemia; In Vitro Techniques; Inositol; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Sprague-Dawley; Type C Phospholipases

2006
Restoration by VIP of the carbachol-stimulated Cl- secretion in TTX-treated guinea pig distal colon.
    The Japanese journal of physiology, 2005, Volume: 55, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atropine; Carbachol; Chlorides; Cholinergic Agents; Cholinergic Fibers; Colforsin; Colon, Descending; Dose-Response Relationship, Drug; Electric Stimulation; Enteric Nervous System; Gastrointestinal Agents; Guinea Pigs; Intestinal Mucosa; Male; Membrane Potentials; Neuroepithelial Cells; Neurotransmitter Agents; Patch-Clamp Techniques; Poisons; Tetrodotoxin; Vasoactive Intestinal Peptide

2005
Function-specific blockage of M(1) and M(3) muscarinic acetylcholine receptors by VX and echothiophate.
    Brain research, 2006, Apr-26, Volume: 1085, Issue:1

    Topics: Animals; Atropine; CHO Cells; Cholinesterase Inhibitors; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Echothiophate Iodide; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Organothiophosphorus Compounds; Oxotremorine; Phosphatidylinositols; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Transfection; Tritium

2006
Blockade by NIP-142, an antiarrhythmic agent, of carbachol-induced atrial action potential shortening and GIRK1/4 channel.
    Journal of pharmacological sciences, 2006, Volume: 101, Issue:4

    Topics: Action Potentials; Adenosine; Animals; Anti-Arrhythmia Agents; Atrial Function; Atropine; Bee Venoms; Benzopyrans; Carbachol; Cell Line; Colforsin; Dose-Response Relationship, Drug; Ether-A-Go-Go Potassium Channels; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Guinea Pigs; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Patch-Clamp Techniques; Potassium Channel Blockers; Time Factors

2006
Regulation of ERK1/2 by the C. elegans muscarinic acetylcholine receptor GAR-3 in Chinese hamster ovary cells.
    Molecules and cells, 2008, Jun-30, Volume: 25, Issue:4

    Topics: Alternative Splicing; Animals; Atropine; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Carbachol; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Estrenes; Indoles; Isoquinolines; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscarinic Agonists; Muscarinic Antagonists; Protein Isoforms; Protein Kinase C; Pyrrolidinones; Receptors, Muscarinic; Recombinant Proteins; Signal Transduction; Sulfonamides; Transfection; Type C Phospholipases

2008
Activation state of the M3 muscarinic acetylcholine receptor modulates mammalian odorant receptor signaling.
    Science signaling, 2011, Jan-11, Volume: 4, Issue:155

    Topics: Atropine; Benzofurans; Carbachol; Cholinergic Agonists; Colforsin; Cyclic AMP; HEK293 Cells; Humans; Immunohistochemistry; Ionomycin; Ionophores; Membrane Transport Proteins; Muscarinic Antagonists; Olfactory Receptor Neurons; Protein Binding; Pyrrolidines; Receptor, Muscarinic M3; Receptors, G-Protein-Coupled; Receptors, Odorant; Signal Transduction; Transfection

2011
Neuromodulation of I(h) in layer II medial entorhinal cortex stellate cells: a voltage-clamp study.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Jun-27, Volume: 32, Issue:26

    Topics: Animals; Animals, Newborn; Anthracenes; Atropine; Biophysical Phenomena; Carbachol; Cardiotonic Agents; Cholinergic Antagonists; Colforsin; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Entorhinal Cortex; Female; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotransmitter Agents; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2012
Pharmacology of central octopaminergic and muscarinic pathways in Drosophila melanogaster larvae: Assessing the target potential of GPCRs.
    Pesticide biochemistry and physiology, 2018, Volume: 151

    Topics: Animals; Atropine; Central Nervous System; Colforsin; Cyclic CMP; Drosophila melanogaster; Electrophysiology; Larva; Octopamine; Phentolamine; Pilocarpine; Receptors, G-Protein-Coupled

2018