Page last updated: 2024-09-05

atropine and clonazepam

atropine has been researched along with clonazepam in 17 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(clonazepam)
Trials
(clonazepam)
Recent Studies (post-2010) (clonazepam)
26,7111,2591,6972,719239519

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)clonazepam (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0017
GABA theta subunitRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0017

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19907 (41.18)18.7374
1990's3 (17.65)18.2507
2000's3 (17.65)29.6817
2010's4 (23.53)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Lipp, JA1
Breimer, DD; de Boer, AG; van Hoogdalem, E1
Iwai, S; Shirakawa, J; Tanaka, C; Taniyama, K1
Karobath, M; Supavilai, P1
Bryere, P; Menini, C; Rektor, I; Silva-Barrat, C1
Bryére, P; Ménini, C; Naquet, R; Rektor, I; Silva-Barrat, C; Valin, A2
Dola, T; Lipp, J1
Kawaguchi, M; Okubo, M1
Bykov, VN; Chepur, SV; Nikiforov, AS; Subbotina, SN; Yudin, MA1
Hamada, H; Haraki, T; Kawamoto, M; Miyoshi, H; Nakamura, R; Yamaga, A; Yasuda, T1

Reviews

3 review(s) available for atropine and clonazepam

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Pharmacokinetics of rectal drug administration, Part I. General considerations and clinical applications of centrally acting drugs.
    Clinical pharmacokinetics, 1991, Volume: 21, Issue:1

    Topics: Administration, Rectal; Antiemetics; Atropine; Carbamazepine; Clonazepam; Delayed-Action Preparations; Diazepam; Flunitrazepam; Humans; Hydromorphone; Intestinal Absorption; Methadone; Methohexital; Midazolam; Morphine; Pharmacokinetics; Phenobarbital; Valproic Acid

1991

Other Studies

14 other study(ies) available for atropine and clonazepam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Effect of atropine upon the cardiovascular system during soman-induced respiratory depression.
    Archives internationales de pharmacodynamie et de therapie, 1976, Volume: 220, Issue:1

    Topics: Animals; Atropine; Blood Pressure; Clonazepam; Depression, Chemical; Doxapram; Electroencephalography; Female; Haplorhini; Heart Rate; Hemodynamics; Intracranial Pressure; Isoproterenol; Macaca mulatta; Male; Organophosphorus Compounds; Respiration; Soman

1976
Regulation of [3H]GABA release from strips of guinea pig urinary bladder.
    The American journal of physiology, 1988, Volume: 255, Issue:6 Pt 2

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Bicuculline; Clonazepam; Clonidine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylephrine; Pirenzepine; Potassium; Prazosin; Tritium; Urinary Bladder; Yohimbine

1988
Modulation of acetylcholine release from rat striatal slices by the GABA/benzodiazepine receptor complex.
    Life sciences, 1985, Feb-04, Volume: 36, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Benzodiazepinones; Clonazepam; Corpus Striatum; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Haloperidol; In Vitro Techniques; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Stimulus-sensitive myoclonus of the baboon Papio papio: pharmacological studies reveal interactions between benzodiazepines and the central cholinergic system.
    Experimental neurology, 1986, Volume: 91, Issue:1

    Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Clonazepam; Drug Interactions; Flumazenil; Myoclonus; Neostigmine; Papio; Parasympathetic Nervous System; Physostigmine; Quinuclidinyl Benzilate

1986
[Type B myoclonus in Papio papio: results of the central anticholinergic effect of benzodiazepines].
    Ceskoslovenska psychiatrie, 1987, Volume: 83, Issue:4-5

    Topics: Animals; Atropine; Benzodiazepines; Clonazepam; Electroencephalography; Myoclonus; Papio; Parasympathetic Nervous System; Parasympatholytics; Physostigmine

1987
Physostigmine antagonizes benzodiazepine-induced myoclonus in the baboon, Papio papio.
    Neuroscience letters, 1984, Nov-23, Volume: 52, Issue:1-2

    Topics: Animals; Atropine; Benzodiazepinones; Clonazepam; Drug Synergism; Myoclonus; Papio; Parasympatholytics; Physostigmine

1984
comparison of the efficacy of HS-6 versus HI-6 when combined with atropine, pyridostigmine and clonazepam for soman poisoning in the monkey.
    Archives internationales de pharmacodynamie et de therapie, 1980, Volume: 246, Issue:1

    Topics: Animals; Atropine; Cholinesterases; Clonazepam; Electroencephalography; Female; Heart Rate; Macaca mulatta; Male; Organophosphate Poisoning; Oximes; Pralidoxime Compounds; Pyridinium Compounds; Pyridostigmine Bromide; Respiration; Soman

1980
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A

1998
Prospects of using benzodiazepines in complex therapy of poisonings with anticholinesterase agents.
    Bulletin of experimental biology and medicine, 2013, Volume: 155, Issue:3

    Topics: Animals; Atropine; Benzodiazepines; Cholinesterase Inhibitors; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Injections, Intramuscular; Male; Mice; Midazolam; Oximes; Pyridinium Compounds; Statistics, Nonparametric; Toxicity Tests

2013
Transient symptomatic worsening by atropine in opsoclonus-myoclonus syndrome.
    Pediatrics international : official journal of the Japan Pediatric Society, 2017, Volume: 59, Issue:1

    Topics: Adjuvants, Anesthesia; Anticonvulsants; Atropine; Child, Preschool; Clonazepam; Deep Sedation; Drug Therapy, Combination; Female; Glucocorticoids; Humans; Infant; Magnetic Resonance Imaging; Opsoclonus-Myoclonus Syndrome; Prednisolone; Retrospective Studies; Tomography, X-Ray Computed

2017