Page last updated: 2024-09-05

atropine and amiloride

atropine has been researched along with amiloride in 29 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(amiloride)
Trials
(amiloride)
Recent Studies (post-2010) (amiloride)
26,7111,2591,6977,584339788

Protein Interaction Comparison

ProteinTaxonomyatropine (IC50)amiloride (IC50)
Urokinase-type plasminogen activatorHomo sapiens (human)4.7
Urokinase-type plasminogen activatorMus musculus (house mouse)2.3
Amine oxidase [flavin-containing] AHomo sapiens (human)3.909
Sodium/hydrogen exchanger 1Rattus norvegicus (Norway rat)1
Amiloride-sensitive sodium channel subunit alphaHomo sapiens (human)0.776
Sodium/hydrogen exchanger 2Oryctolagus cuniculus (rabbit)1
Acid-sensing ion channel 3Homo sapiens (human)4.4

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19907 (24.14)18.7374
1990's9 (31.03)18.2507
2000's7 (24.14)29.6817
2010's6 (20.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Blackard, WG; Kikuchi, M; Rabinovitch, A; Renold, AE1
Obara, K; Usuki, T; Yabu, H1
Donoff, B; Lad, R; Rangachari, PK1
Kindle, H; Kunkel, JG; Lanzrein, B1
Dissing, S; Nauntofte, B1
Beeker, TG; Muallem, S; Pandol, SJ1
Bowen, S; Condon, C; Cooke, HJ; Kuwahara, A; Wang, J1
Barrett, RJ; Kau, ST1
Matthews, EK; Petersen, OH1
Alberti, KG; Aynsley-Green, A1
Pon, DJ; Sen, AK; Stewart, DJ1
Mao, H; Wong, LB1
Cooke, HJ; Javed, N; Reddix, R; Wang, YZ1
Komazaki, S; Takada, M; Takayama-Arita, K; Yai, H1
Cox, TC1
Madison, DV; McQuiston, AR1
Chan, MH; Farley, JM1
Cox, T; Holbird, D; Jensik, P1
Chen, ZY; Huang, Y; Ko, WH; Lau, CW; Law, VW; Yip, WC; Yue, GG1
Dortch-Carnes, J; Fedan, JS; Johnston, RA; Kommineni, C; Millecchia, LL; Van Scott, MR1
Beil, M; Danhof, M; Fu, F; Luttringer, O; Ploeger, BA; Rigel, DF; Snelder, N; Stanski, DR1
Cho, HJ; Choi, JY; Joo, NS; Krouse, ME; Wine, JJ1

Reviews

1 review(s) available for atropine and amiloride

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

28 other study(ies) available for atropine and amiloride

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
An effect of hyposmolarity on insulin release in vitro.
    The American journal of physiology, 1975, Volume: 228, Issue:3

    Topics: Amiloride; Amylases; Animals; Atropine; Calcium; Choline; Colchicine; Diazoxide; Epinephrine; Glucagon; Glucose; Hypotonic Solutions; Imidazoles; In Vitro Techniques; Insulin; Insulin Secretion; Male; Osmolar Concentration; Ouabain; Pancreas; Phentolamine; Phenytoin; Propranolol; Rats; Sorbitol; Tolbutamide; Trypsin Inhibitors; Vinblastine

1975
Calcium and potassium channel regulation by protein phosphorylation in smooth muscle cells of guinea pig taenia coli.
    Advances in experimental medicine and biology, 1992, Volume: 311

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amiloride; Animals; Atropine; Calcium Channels; Carbachol; Colon; Guinea Pigs; In Vitro Techniques; Isoquinolines; Marine Toxins; Membrane Potentials; Models, Biological; Muscle, Smooth; Nifedipine; Oxazoles; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Piperazines; Potassium Channels; Protein Kinase C

1992
Functional subtyping of muscarinic receptors on canine esophageal mucosa.
    The American journal of physiology, 1991, Volume: 261, Issue:3 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Amiloride; Animals; Atropine; Carbachol; Chlorides; Dogs; Electric Conductivity; Esophagus; Female; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Mucous Membrane; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Sodium

1991
The effect of ions, ion channel blockers, and ionophores on uptake of vitellogenin into cockroach follicles.
    Developmental biology, 1990, Volume: 142, Issue:2

    Topics: Amiloride; Animals; Atropine; Calcium Channel Blockers; Cockroaches; Female; In Vitro Techniques; Ions; Ouabain; Ovarian Follicle; Tetraethylammonium Compounds; Valinomycin; Verapamil; Vitellogenins

1990
Na+ transport properties of isolated rat parotid acini.
    The American journal of physiology, 1990, Volume: 259, Issue:6 Pt 1

    Topics: Acetazolamide; Amiloride; Animals; Atropine; Biological Transport, Active; Bumetanide; Carbachol; Chlorides; Fluoresceins; Fluorescent Dyes; Furosemide; In Vitro Techniques; Kinetics; Male; Ouabain; Parotid Gland; Rats; Rats, Inbred Strains; Sodium

1990
Modulation of agonist-activated calcium influx by extracellular pH in rat pancreatic acini.
    The American journal of physiology, 1989, Volume: 257, Issue:6 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetates; Acetic Acid; Amiloride; Ammonium Chloride; Animals; Atropine; Calcium; Calcium Radioisotopes; Carbachol; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Lanthanum; Pancreas; Rats; Rats, Inbred Strains; Sincalide

1989
Epithelial responses evoked by stimulation of submucosal neurons in guinea pig distal colon.
    The American journal of physiology, 1987, Volume: 252, Issue:5 Pt 1

    Topics: Amiloride; Animals; Atropine; Bicarbonates; Colon; Electric Conductivity; Electric Stimulation; Epithelium; Evoked Potentials; Extracellular Space; Female; Guinea Pigs; Ions; Male; Neurons; Submucous Plexus; Tetrodotoxin

1987
Myocardial and vascular actions of amiloride in spontaneously hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Amiloride; Animals; Atropine; Blood Pressure; Cardiovascular System; Cimetidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Male; Nephrectomy; Pyrilamine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Stimulation, Chemical; Sulpiride

1986
Pancreatic acinar cells: ionic dependence of the membrane potential and acetycholine-induced depolarization.
    The Journal of physiology, 1973, Volume: 231, Issue:2

    Topics: Acetylcholine; Amiloride; Animals; Atropine; Calcium; Cell Membrane Permeability; Cholecystokinin; Cyclic AMP; Dinitrophenols; Epinephrine; In Vitro Techniques; Membrane Potentials; Mice; Pancreas; Potassium; Sodium; Strophanthins; Tetracaine

1973
In vivo stimulation of insulin secretion by guanidine derivatives in the rat.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1974, Volume: 6, Issue:2

    Topics: Acetates; Amiloride; Animals; Arginine; Atropine; Blood Glucose; Butyrates; Female; Guanidines; Insulin; Propionates; Rats; Structure-Activity Relationship; Time Factors

1974
Cholinergic stimulation of ouabain-sensitive respiration in rat submandibular gland.
    The American journal of physiology, 1983, Volume: 245, Issue:3

    Topics: Amiloride; Animals; Atropine; Calcimycin; Carbachol; Dose-Response Relationship, Drug; Kinetics; Male; Ouabain; Oxygen Consumption; Rats; Rats, Inbred Strains; Submandibular Gland

1983
Depolarization of cell membrane is associated with an increase in ciliary beat frequency (CBF).
    Biochemical and biophysical research communications, 1995, Oct-24, Volume: 215, Issue:3

    Topics: Amiloride; Animals; Atropine; Carbachol; Cell Membrane; Cells, Cultured; Cilia; Fluorescent Dyes; Ionomycin; Kinetics; Microscopy, Fluorescence; Muscarinic Agonists; Photons; Pyridinium Compounds; Receptors, Muscarinic; Scattering, Radiation; Sheep; Time Factors; Trachea; Verapamil

1995
Cholinergic and VIP-ergic pathways mediate histamine H2 receptor-induced cyclical secretion in the guinea pig colon.
    The American journal of physiology, 1995, Volume: 268, Issue:3 Pt 1

    Topics: Acetylcholine; Amiloride; Animals; Atropine; Choline; Colon; Dimaprit; Electric Conductivity; Guinea Pigs; Histamine Release; Intestinal Mucosa; Male; ortho-Aminobenzoates; Piperidines; Pirenzepine; Receptors, Histamine H2; Vasoactive Intestinal Peptide

1995
Prolactin enables normal development of ACh-stimulated current in cultured larval bullfrog skin.
    The American journal of physiology, 1996, Volume: 271, Issue:4 Pt 1

    Topics: Acetylcholine; Age Factors; Aldosterone; Amiloride; Animals; Atropine; Cell Differentiation; Cell Separation; Cells, Cultured; Cholinesterase Inhibitors; Edetic Acid; Larva; Muscarinic Antagonists; Nicotinic Antagonists; Physostigmine; Prolactin; Rana catesbeiana; Skin Physiological Phenomena; Tubocurarine

1996
Apical regulation of nonselective cation channels by ATP in larval bullfrog skin.
    The Journal of experimental zoology, 1997, Oct-15, Volume: 279, Issue:3

    Topics: Acetylcholine; Adenosine Triphosphate; Amiloride; Animals; Atropine; Calcium; Calcium Channels; Diltiazem; Egtazic Acid; Electric Conductivity; In Vitro Techniques; Larva; Potassium Chloride; Rana catesbeiana; Receptors, Purinergic P2; Skin Physiological Phenomena; Sulfonamides; Suramin

1997
Muscarinic receptor activity induces an afterdepolarization in a subpopulation of hippocampal CA1 interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-15, Volume: 19, Issue:14

    Topics: Acetylcholine; Action Potentials; Amiloride; Animals; Atropine; Cadmium; Calcium; Hippocampus; In Vitro Techniques; Interneurons; Male; Muscarine; Muscarinic Agonists; Rats; Receptors, Muscarinic; Sodium; Tetrodotoxin

1999
Lidocaine-induced alterations in agonist-induced ion transport of cultured swine tracheal submucosal gland cells.
    Toxicology and applied pharmacology, 2000, Sep-15, Volume: 167, Issue:3

    Topics: Acetylcholine; Amiloride; Anesthetics, Local; Animals; Atropine; Biological Transport; Cell Survival; Cells, Cultured; Drug Interactions; Electrophysiology; Ions; Isoproterenol; Lidocaine; Male; Respiratory Mucosa; Swine; Trachea

2000
Aldosterone upregulates purinergic responses in larval amphibian skin epithelium.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2001, Volume: 171, Issue:5

    Topics: Acetylcholine; Adenosine Triphosphate; Aldosterone; Amiloride; Animals; Antineoplastic Agents; Atropine; Diuretics; Epithelial Cells; Gene Expression; Larva; Muscarinic Antagonists; Nicotinic Antagonists; Potassium; Purinergic P2 Receptor Antagonists; Rana catesbeiana; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Receptors, Purinergic P2X5; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Skin; Sodium; Sulfonamides; Suramin; Tubocurarine; Up-Regulation; Vasodilator Agents

2001
Stimulation of chloride secretion by baicalein in isolated rat distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Animals; Atropine; Calcium; Carbachol; Chlorides; Colforsin; Colon; Cyclic AMP; Dinoprostone; Electric Conductivity; Female; Flavanones; Flavonoids; Indomethacin; Intestinal Mucosa; Male; Muscarinic Antagonists; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Thapsigargin

2002
Hyperosmolar solution effects in guinea pig airways. IV. Lipopolysaccharide-induced alterations in airway reactivity and epithelial bioelectric responses to methacholine and hyperosmolarity.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 308, Issue:1

    Topics: Amiloride; Animals; Atropine; Bronchoconstrictor Agents; Diuretics; Drug Interactions; Electrophysiology; Enzyme Inhibitors; Epithelial Cells; Guinea Pigs; Indomethacin; Lipopolysaccharides; Male; Methacholine Chloride; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Nitroprusside; Osmolar Concentration; Perfusion; Respiratory Function Tests; Sodium Chloride; Trachea; Vasodilator Agents

2004
Drug effects on the CVS in conscious rats: separating cardiac output into heart rate and stroke volume using PKPD modelling.
    British journal of pharmacology, 2014, Volume: 171, Issue:22

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amiloride; Amlodipine; Animals; Atropine; Enalapril; Hemodynamics; Hydrochlorothiazide; Hypertension; Male; Models, Biological; Prazosin; Propranolol; Rats, Inbred SHR; Rats, Inbred WKY

2014
Inhibition of airway surface fluid absorption by cholinergic stimulation.
    Scientific reports, 2016, Feb-05, Volume: 6

    Topics: Amiloride; Animals; Atropine; Carbachol; Cells, Cultured; Epithelial Sodium Channels; Ferrets; Humans; Mucus; Rabbits; Respiratory Mucosa; Sheep; Swine; Trachea

2016