Page last updated: 2024-09-05

atropine and 4-diphenylacetoxy-1,1-dimethylpiperidinium

atropine has been researched along with 4-diphenylacetoxy-1,1-dimethylpiperidinium in 140 studies

Compound Research Comparison

Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010)
(atropine)
Studies
(4-diphenylacetoxy-1,1-dimethylpiperidinium)
Trials
(4-diphenylacetoxy-1,1-dimethylpiperidinium)
Recent Studies (post-2010) (4-diphenylacetoxy-1,1-dimethylpiperidinium)
26,7111,2591,697446152

Research

Studies (140)

TimeframeStudies, this research(%)All Research%
pre-199011 (7.86)18.7374
1990's81 (57.86)18.2507
2000's39 (27.86)29.6817
2010's9 (6.43)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kashihara, K; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1
Kashima, K; Kataoka, K; Kato, M; Kuriyama, K; Ohkuma, S1
Ishihara, H; Shimura, S1
Abdallah, EA; Eldefrawi, AT; Eldefrawi, ME; Jett, DA1
Cazzola, M; Constantino, M; De Santis, D; Matera, MG; Rossi, F1
Aguilar, JS; Ballesta, JJ; Criado, M; Palmero, M; Reig, JA; Viniegra, S1
Akerman, KE; Kukkonen, J1
Hendriks, MG; Pfaffendorf, M; Van Zwieten, PA2
Badini, I; Beani, L; Bianchi, C; Cintra, A; Fuxe, K; Siniscalchi, A1
Bloom, JW; Halonen, M; Mahesh, VK; Nunan, LM; Palmer, JD; Yamamura, HI1
Funakoshi, A; Jimi, A; Kono, A; Tateishi, K; Tsuru, M; Wakasugi, H1
Cheung, CL; De Boer, T; Tonnaer, JA1
Bindslev, N; Winding, B1
Donoff, B; Lad, R; Rangachari, PK1
Alonso, MJ; Arribas, S; Balfagón, G; Marín, J; Salaices, M1
Angeli, P; Brasili, L; Cingolani, ML; Marucci, G; Pigini, P; Tonnini, MC1
Aikawa, T; Itabashi, S; Ohrui, T; Sasaki, H; Sekizawa, K; Takishima, T1
Low, PA; Torres, NE; Zollman, PJ1
Freschi, JE1
Benedito, S; García-Sacristán, A; Hernández, M; Prieto, D; Rivera, L1
Ballabeni, V; Barocelli, E; Impicciatore, M; Lavezzo, A; Morini, G1
Chiba, S; Tsukada, M1
Arruebo, MP; Bueno, L; Liberge, M1
Yang, CM1
Davidson, A; Matus-Leibovitch, N; Mengod, G; Oron, Y1
Fleming, N; Laniyonu, A; Sliwinski-Lis, E1
Entzeroth, M; Mayer, N1
Akahane, K; Chiba, S; Furukawa, Y; Karasawa, Y1
Alonso, R; Didier, M; Soubrie, P1
De Boer, P; Horn, AS; Rollema, H; Westerink, BH; Zaagsma, J1
Cazzola, M; Cenicola, ML; D'Amato, G; De Santis, D; Lisa, M; Maione, S; Marmo, E; Matera, MG1
Chiba, S; Haruta, K; Homma, N; Horiuchi, A; Iwatsuki, K; Yonekura, H1
Ghataorre, AS; Lambert, DG; Nahorski, SR1
Dodds, WJ; Gilbert, RJ1
Hsu, CT; Hyman, PE; Jing, J; Snape, WJ; Tomomasa, T1
Choo, LK; Mitchelson, F1
Brezenoff, HE; Xiao, YF1
Davidesko, D; Doods, HN; Rinner, I; van Charldorp, KJ; van Zwieten, PA1
Bitar, KN; Grider, JR; Makhlouf, GM1
Eglen, RM; Whiting, RL1
Gilbert, R; Goyal, RK; Rattan, S1
Heilbronn, E; Järlebark, L; Lawoko, G1
Ernsberger, P; Evinger, MJ; Joh, TH; Regunathan, S; Reis, DJ1
Bai, D; Sattelle, DB1
Cooke, HJ; Javed, N; Reddix, R; Wang, YZ1
Francis, NJ; Grant, MP; Landis, SC1
Nakamura, K; Okuma, Y; Osumi, Y; Yokotani, K1
DeSautel, MG; Maher, JW; Sandler, AD; Schlegel, JF1
Fukui, H; Inagaki, N; Kondou, H1
Hayakawa, T; Kitagawa, M; Kondo, T; Naruse, S; Shibata, T; Tanikawa, M1
Howell, RE; Kovalsky, MP1
Brown, MC; Liberman, MC; Sewell, WF; Sridhar, TS1
Corrêa, FM; Peres-Polon, VL1
Imaizumi, Y; Tanaka, M; Watanabe, M; Yamahara, NS1
Ballabeni, V; Barocelli, E; Caretta, A; Chiavarini, M; Impicciatore, M; Molina, E1
Howell, RE; Kovalsky, MP; Laemont, KD1
DelValle, J; Park, J; Yamada, T; Yokotani, K1
Bissonnette, BM; Brasitus, TA; Khare, S; Sitrin, MD; Tien, XY; Wali, RK; Wilson, D1
Fehér, E; Matkó, I; Vizi, ES1
Deirmengiant, C; Maslanski, JA; Patelt, J; Powelt, R1
Bobbin, RP; Erostegui, C; Norris, CH1
Davenport, TA; Fukumoto, Y; Gousse, A; Kamai, T; Latifpour, J; Weiss, RM; Yoshida, M1
Dobbie, JW; Duffield, R; Hjelle, JT; Ho, AK; Steidley, KR1
Baghdoyan, HA; Carlson, BX; Roth, MT1
Chuang, DM; Fukamauchi, F; Hough, C; Saunders, PA1
Osumi, Y; Yokotani, K1
Cosentino, M; Crema, A; D'Angelo, L; de Ponti, F; Einaudi, A; Frigo, GM; Lecchini, S1
Manjeet, S; Sim, MK1
Shiraishi, K; Takayanagi, I1
Garssen, J; Gierveld, CM; Nijkamp, FP; Van der Vliet, H; Van Loveren, H1
Garland, CJ; Hillier, K; Kerr, PM; Wallis, RM1
Chang, B; Melvin, JE; Zhang, GH1
Tobin, G1
McCaffrey, TV; Yang, B1
Acs, Z; Makara, GB; Pintér, I1
Arana, R; Bacman, S; Borda, E; Camusso, JJ; Hubscher, O; Sterin-Borda, L1
Murayama, T; Nomura, Y; Yamada, T1
Koss, MC1
Levin, RJ; Przyborski, SA1
Semba, K; White, TD1
Komori, S; Nakayama, T; Ohashi, H; Unno, T1
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M1
Blumenthal, JA; Carey, HV; Onorato, JJ1
Bégos, A; Bizot, JC; Breton, P; Brochet, D; Tambuté, A; Trovero, F1
Wallis, RM1
Pagano, AP; Parkman, HP; Ryan, JP1
Bernardi, G; Bonci, A; Grillner, P; Mercuri, NB; Svensson, TH1
Goldie, RG; Preuss, JM1
Corrêa, FM; Crippa, GE; Kuboyama, RH; Peres-Polon, VL1
Acs, Z; Makara, GB; Némethy, Z1
Fitzgerald, ME; Reiner, A; Zagvazdin, Y1
Harada, A; Honda, K; Kamiya, H; Takano, Y1
Halayko, AJ; Kahraman, S; Mitchell, RW; Solway, J; Wylam, ME1
Iannazzo, L; Majewski, H1
Malomough, A; Naumenko, N; Nikolsky, E; Urazaev, A; Vyskocil, F1
Zhao, D; Zhou, ZJ1
Fushimi, T; Masuda, T; Saitoh, H; Shimura, S; Shirato, K1
Kwon, SC1
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD1
Franco, W; Leite, RS1
Avellar, MC; Guaze, EF; Maróstica, E; Porto, CS1
Gerthoffer, WT; Singer, CA; Vang, S1
Pérez Leirós, C; Rosignoli, F1
Kato, T; Ogasawara, M; Sato, K; Shimoda, N; Sugaya, K1
Benoit, JN; Cohen, MV; Downey, JM; Oldenburg, O; Qin, Q; Sharma, AR1
Addison, S; Evangelista, S; Greer, S; Hernon, J; Johns, N; Johnson, I; Lewis, M; Lindqvist, S; Mackay, J; Rhodes, M; Sharp, P; Speakman, C; Stebbings, W; Tighe, R; Watson, M; Williams, M1
Albuquerque, EX; Aracava, Y; Castro, NG; Fawcett, WP; Pereira, EF; Randall, WR; Santos, MD1
de Groat, WC; Rocha, JN; Smith, CP; Somogyi, GT; Yoshiyama, M; Zernova, GV1
Arredondo, J; Chernyavsky, AI; Grando, SA; Ndoye, A; Nguyen, VT; Wess, J; Zia, S1
Farnbauch, LJ; Robertson, KL; Rowland, NE1
Abe, K; Chikuma, T; Hojyo, H; Kato, M; Miyatake, T; Taguchi, K; Utsunomiya, I1
Bordi, F; Costa, LG; Dieguez-Acuña, FJ; Guizzetti, M; Madia, F; Vitalone, A; Woods, JS1
Crittenden, EL; García, DM; González, A1
Ehlert, FJ; Griffin, MT; Hsu, JC; Lee, AG; Leung, K; Shehnaz, D1
Chen, LB; Liu, CY; Liu, KJ; Wang, PS; Xie, DP; Zhang, CL1
Ando, S; Harasawa, I; Honda, K; Kamiya, HO; Koga, K; Takano, Y1
Beitz, AJ; Choi, SM; Han, HJ; Jeong, TO; Kim, HW; Kwon, YB; Lee, HJ; Lee, JH; Roh, DH; Ryu, YH; Yoon, SY1
Forrest, AS; Ordög, T; Sanders, KM1
Paulose, CS; Renuka, TR; Savitha, B1
Miyazu, M; Ohinata, H; Sugawara, R; Takai, A; Takai, Y; Yoshida, A1
Alves, FH; Corrêa, FM; Crestani, CC; Resstel, LB1
Hao, LY; Kameyama, M; Onoue, Y; Wang, JW; Yazawa, K1
Chan, SH; Chang, AY; Tsai, CY; Wu, CH1
Campo, P; Lataye, R; Maguin, K1
Eguchi, K; Ohtubo, Y; Yoshii, K1
Huang, TJ; Ko, WC; Lin, LH; Lin, YL; Wang, SH; Wu, SN1
Advenier, C; Chen, HZ; Cui, YY; Devillier, P; Wang, H; Zhu, L1
Boone, TB; Lai, HH; Munoz, A; Smith, CP; Somogyi, GT; Szigeti, GP1
Bae, H; Choi, SM; Kim, HN; Kim, SK; Koo, S; Min, BI; Park, JH; Sun, B1
Britton, FC; Koh, SD; O'Driscoll, K; Sanders, KM; Sung, IK; Sung, TS; Zheng, H; Zhu, MH1
Chess-Williams, R; Moro, C; Uchiyama, J1
Gao, WY; Hu, J; Huang, LQ; Liu, CX; Ma, L; Man, SL1
Chen, HZ; Cui, YY; Hou, LN; Xu, GN; Xu, ZP; Yang, K; Zhang, WH; Zhu, L1
Arrighi, N; Bodei, S; Cosciani Cunico, S; Michel, MC; Sigala, S; Simeone, C; Spano, P; Zani, D1
Deng, J; Li, L; Shi, C; Song, B; Wu, Y; Zhang, X1
Albuquerque, AA; Capellini, VK; Celotto, AC; de Carvalho, MT; de Nadai, TR; Evora, PR; Ferreira, LG; Silveira, AP1
Dhillon, ES; Ludwig, J; Sharma, N; Steidl, S1
Ashpole, NM; Carvalho, FS; Castro, CH; Costa, EA; Fajemiroye, JO; Franco, OL; Lião, LM; Menegatti, R; Mourão, AA; Oliveira-Silva, I; Pedrino, GR; Silva, ON; Verli, H; Villavicencio, B; Xavier, CH1

Trials

1 trial(s) available for atropine and 4-diphenylacetoxy-1,1-dimethylpiperidinium

ArticleYear
Pre-clinical and clinical pharmacology of selective muscarinic M3 receptor antagonists.
    Life sciences, 1995, Volume: 56, Issue:11-12

    Topics: Animals; Atrial Function; Atropine; Colon; Dicyclomine; Dioxoles; Dogs; Drug Evaluation, Preclinical; Gastrointestinal Motility; Guinea Pigs; Heart Atria; Humans; Ileum; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Rabbits; Receptor, Muscarinic M3; Receptors, Muscarinic; Salivary Glands; Trachea; Vas Deferens

1995

Other Studies

139 other study(ies) available for atropine and 4-diphenylacetoxy-1,1-dimethylpiperidinium

ArticleYear
Cloning of the rat M3, M4 and M5 muscarinic acetylcholine receptor genes by the polymerase chain reaction (PCR) and the pharmacological characterization of the expressed genes.
    Life sciences, 1992, Volume: 51, Issue:12

    Topics: Acetylcholine; Amino Acid Sequence; Animals; Base Sequence; Carbachol; Cell Line; Cloning, Molecular; Cyclic AMP; Fibroblasts; Gene Expression; Inositol Phosphates; Molecular Sequence Data; Parasympatholytics; Polymerase Chain Reaction; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Muscarinic; Transfection

1992
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998
Characterization of muscarinic receptor subtypes on rat pancreatic acini: pharmacological identification by secretory responses and binding studies.
    Digestion, 1992, Volume: 52, Issue:3-4

    Topics: Amylases; Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Male; Pancreas; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Sincalide

1992
[The role of muscarinic receptor subtypes in feline tracheal submucosal gland secretion].
    Nihon Kyobu Shikkan Gakkai zasshi, 1992, Volume: 30 Suppl

    Topics: Animals; Atropine; Calcium; Cats; Electrolytes; Glycoproteins; In Vitro Techniques; Mucous Membrane; Piperidines; Pirenzepine; Receptors, Muscarinic; Second Messenger Systems; Trachea

1992
Differential effects of paraoxon on the M3 muscarinic receptor and its effector system in rat submaxillary gland cells.
    Journal of biochemical toxicology, 1992,Summer, Volume: 7, Issue:2

    Topics: Animals; Atropine; Binding Sites; Carbachol; Cyclic AMP; Hydrolysis; Male; Paraoxon; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Regression Analysis; Submandibular Gland

1992
Responsiveness and sensitivity to cholinergic agonists and antagonists in bovine isolated bronchial muscle.
    Clinical and experimental pharmacology & physiology, 1992, Volume: 19, Issue:9

    Topics: Acetylcholine; Animals; Atropine; Bronchi; Cattle; Gallamine Triethiodide; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine

1992
Muscarinic receptor subtypes in bovine adrenal medulla.
    Neurochemical research, 1992, Volume: 17, Issue:12

    Topics: Adrenal Medulla; Animals; Atropine; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Dicyclomine; Muscarine; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic

1992
Apparent noncompetitive antagonism of muscarinic receptor mediated Ca2+ mobilization by some muscarinic antagonists.
    Biochemical and biophysical research communications, 1992, Dec-15, Volume: 189, Issue:2

    Topics: Atropine; Calcium; Fura-2; Humans; Kinetics; Muscarinic Antagonists; N-Methylscopolamine; Neuroblastoma; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Spectrometry, Fluorescence; Tumor Cells, Cultured

1992
Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation.
    Journal of autonomic pharmacology, 1992, Volume: 12, Issue:6

    Topics: Animals; Atropine; Benzodiazepinones; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Methacholine Chloride; Parasympatholytics; Perfusion; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Vasodilation

1992
Muscarinic modulation of acetylcholine release from slices of guinea pig nucleus basalis magnocellularis.
    Neuroscience letters, 1992, Jun-22, Volume: 140, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Calcium; Choline; Female; Guinea Pigs; Male; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Receptors, Muscarinic; Substantia Innominata; Tetrodotoxin

1992
A minority of muscarinic receptors mediate rabbit tracheal smooth muscle contraction.
    American journal of respiratory cell and molecular biology, 1992, Volume: 6, Issue:3

    Topics: Animals; Atropine; Female; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Radioligand Assay; Receptors, Muscarinic; Trachea

1992
Acetylcholine regulates pancreastatin secretion from the human pancreastatin-producing cell line (QGP-1N).
    The Journal of clinical endocrinology and metabolism, 1991, Volume: 73, Issue:1

    Topics: Acetylcholine; Adenoma, Islet Cell; Atropine; Calcimycin; Calcium; Carbachol; Chromogranin A; Gastrin-Releasing Peptide; Humans; Pancreatic Hormones; Pancreatic Neoplasms; Parasympatholytics; Peptides; Piperidines; Pirenzepine; Receptors, Muscarinic; Sincalide; Tumor Cells, Cultured

1991
cGMP formation and phosphoinositide turnover in rat brain slices are mediated by pharmacologically distinct muscarinic acetylcholine receptors.
    European journal of pharmacology, 1991, Jul-12, Volume: 207, Issue:3

    Topics: Animals; Atropine; Brain; Carbachol; Cyclic GMP; Guanylate Cyclase; Hippocampus; Inositol Phosphates; Male; Nitroprusside; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Succinimides

1991
Characterization of a muscarinic receptor controlling Cl- secretion in hen trachea.
    The American journal of physiology, 1990, Volume: 258, Issue:6 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Bethanechol; Bethanechol Compounds; Bumetanide; Calcium Channels; Chickens; Chlorides; Dicyclomine; Female; In Vitro Techniques; Ion Channels; Kinetics; Mucous Membrane; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1990
Functional subtyping of muscarinic receptors on canine esophageal mucosa.
    The American journal of physiology, 1991, Volume: 261, Issue:3 Pt 1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Amiloride; Animals; Atropine; Carbachol; Chlorides; Dogs; Electric Conductivity; Esophagus; Female; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Mucous Membrane; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Sodium

1991
Presynaptic M2-muscarinic receptors on noradrenergic nerve endings and endothelium-derived M3 receptors in cat cerebral arteries.
    Brain research, 1991, Dec-13, Volume: 567, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Carbachol; Cats; Cerebral Arteries; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptors, Muscarinic; Vasodilation

1991
Pharmacological characterization of muscarinic receptor subtypes in rabbit isolated tissue preparations.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:5

    Topics: Animals; Aorta, Thoracic; Atropine; Diamines; Jejunum; Male; Muscarinic Antagonists; Muscle Contraction; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Vas Deferens; Vasodilation

1991
Pre- and postjunctional muscarinic receptor subtypes in dog airways.
    European journal of pharmacology, 1991, Nov-12, Volume: 204, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Bronchi; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1991
Characterization of muscarinic receptor subtype of rat eccrine sweat gland by autoradiography.
    Brain research, 1991, May-31, Volume: 550, Issue:1

    Topics: Animals; Atropine; Autoradiography; Binding, Competitive; Eccrine Glands; Kinetics; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium

1991
The effect of subtype-selective muscarinic receptor antagonists on the cholinergic current in motoneurons of the lobster cardiac ganglion.
    Brain research, 1991, Jun-21, Volume: 552, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Binding, Competitive; Ganglia; In Vitro Techniques; Mammals; Methacholine Chloride; Motor Neurons; Nephropidae; Parasympathomimetics; Piperidines; Pirenzepine; Receptors, Muscarinic

1991
Distribution and function of cholinergic receptors in the sheep detrusor muscle.
    Journal of the autonomic nervous system, 1991, Jun-15, Volume: 34, Issue:2-3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Carbachol; Cholinesterase Inhibitors; Ganglia, Parasympathetic; Male; Muscle Contraction; Muscle, Smooth; Nerve Tissue Proteins; Piperidines; Pirenzepine; Receptors, Muscarinic; Sheep; Tetraisopropylpyrophosphamide; Urinary Bladder

1991
Effects of two new pirenzepine analogs on the contractile response of the guinea-pig oesophageal muscularis mucosae to acetylcholine, bethanechol, histamine and high potassium.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Esophagus; Guinea Pigs; Histamine; Histamine Antagonists; Male; Muscle Contraction; Piperidines; Pirenzepine; Potassium; Pyrilamine; Receptors, Muscarinic

1990
Predominant acetylcholine-induced vasoconstriction in isolated, perfused simian facial veins.
    European journal of pharmacology, 1990, Dec-04, Volume: 191, Issue:3

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Blood Pressure; Diltiazem; Face; Female; In Vitro Techniques; Macaca; Male; Muscle, Smooth, Vascular; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Potassium Chloride; Quinazolines; Receptors, Muscarinic; Saponins; Vasoconstriction; Veins

1990
Role of hypothalamic cholecystokinin octapeptide in the colonic motor response to a meal in rats.
    Gastroenterology, 1991, Volume: 100, Issue:2

    Topics: Animals; Atropine; Benzodiazepinones; Cholecystokinin; Colon; Devazepide; Electromyography; Food; Gastrointestinal Motility; Hypothalamic Area, Lateral; Hypothalamus; Male; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Receptors, Muscarinic; Sincalide; Ventromedial Hypothalamic Nucleus

1991
Characterization of muscarinic receptors in dog tracheal smooth muscle cells.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:1

    Topics: Animals; Atropine; Carbachol; Diamines; Dogs; In Vitro Techniques; Kinetics; Muscle, Smooth; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Trachea

1991
Native Xenopus oocytes express two types of muscarinic receptors.
    FEBS letters, 1991, Jun-24, Volume: 284, Issue:2

    Topics: Animals; Atropine; Elapid Venoms; Female; Oligonucleotide Probes; Oligonucleotides, Antisense; Oocytes; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Xenopus laevis

1991
Muscarinic M3 receptors are coupled to two signal transduction pathways in rat submandibular cells.
    European journal of pharmacology, 1990, Mar-13, Volume: 188, Issue:2-3

    Topics: Animals; Atropine; Carbachol; Cyclic AMP; Parasympatholytics; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Signal Transduction; Submandibular Gland

1990
Labeling of rat heart muscarinic receptors using the new M2 selective antagonist [3H]AF-DX 384.
    Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7

    Topics: Affinity Labels; Animals; Atropine; Binding, Competitive; Male; Muscarinic Antagonists; Myocardium; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1990
Muscarinic receptor subtypes mediating negative chrono- and inotropic responses in isolated, blood-perfused dog right atria.
    Journal of autonomic pharmacology, 1990, Volume: 10, Issue:1

    Topics: Animals; Atropine; Carbachol; Cardiotonic Agents; Dogs; Electric Stimulation; Female; Heart Atria; Male; Myocardial Contraction; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Vagus Nerve

1990
[3H]N-methylscopolamine binding studies reveal M2 and M3 muscarinic receptor subtypes on cerebellar granule cells in primary culture.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: Animals; Atropine; Binding, Competitive; Cell Survival; Cells, Cultured; Cerebellum; Diamines; Granulocytes; N-Methylscopolamine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives; Tritium

1990
An M3-like muscarinic autoreceptor regulates the in vivo release of acetylcholine in rat striatum.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Acetylcholine; Animals; Atropine; Chromatography, High Pressure Liquid; Corpus Striatum; Dialysis; Dose-Response Relationship, Drug; Male; Neostigmine; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Time Factors

1990
Evidence of muscarinic receptor subtypes in airway smooth muscle of normal volunteers and of chronic obstructive pulmonary disease patients.
    International journal of clinical pharmacology research, 1989, Volume: 9, Issue:1

    Topics: Atropine; Forced Expiratory Volume; Humans; Lung Diseases, Obstructive; Muscle, Smooth; Piperidines; Pirenzepine; Receptors, Muscarinic; Respiratory Muscles

1989
Subtypes of muscarinic receptors in pancreatic exocrine secretion in anesthetized dog.
    Pancreas, 1989, Volume: 4, Issue:3

    Topics: Animals; Atropine; Bethanechol Compounds; Dogs; Female; Kinetics; Male; Pancreas; Pancreatic Juice; Parasympathomimetics; Piperidines; Pirenzepine; Receptors, Muscarinic; Reference Values

1989
Muscarinic receptor binding characteristics of a human neuroblastoma SK-N-SH and its clones SH-SY5Y and SH-EP1.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Arecoline; Atropine; Carbachol; Cell Membrane; Humans; Neuroblastoma; Piperidines; Pirenzepine; Receptors, Muscarinic; Tumor Cells, Cultured

1989
Effect of selective muscarinic antagonists on peristaltic contractions in opossum smooth muscle.
    The American journal of physiology, 1986, Volume: 250, Issue:1 Pt 1

    Topics: Animals; Atropine; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Female; Male; Manometry; Muscle Contraction; Muscle, Smooth; Opossums; Peristalsis; Piperidines; Pirenzepine; Receptors, Muscarinic; Vagus Nerve

1986
Development of the muscarinic receptor in rabbit gastric smooth muscle.
    The American journal of physiology, 1988, Volume: 254, Issue:5 Pt 1

    Topics: Animals; Animals, Newborn; Atropine; Bethanechol; Bethanechol Compounds; Dose-Response Relationship, Drug; Kinetics; Muscle Contraction; Muscle Development; Muscle, Smooth; N-Methylscopolamine; Phenethylamines; Piperidines; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Stomach

1988
Displacement of [3H]oxotremorine-M binding by muscarinic antagonists in guinea-pig atrial and ileal membrane homogenates.
    European journal of pharmacology, 1988, Jul-07, Volume: 151, Issue:2

    Topics: Animals; Atropine; Binding, Competitive; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Oxotremorine; Parasympatholytics; Piperidines

1988
The role of M2 muscarinic receptors in the posterior hypothalamus in the pressor response to intracerebroventricularly-injected neostigmine.
    Neuropharmacology, 1988, Volume: 27, Issue:10

    Topics: Animals; Atropine; Blood Pressure; Heart Rate; Hypothalamus; Injections, Intraventricular; Male; Neostigmine; Parasympathomimetics; Piperidines; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Binding of muscarine receptor antagonists to pig coronary smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:2

    Topics: Animals; Atropine; Carbachol; Coronary Vessels; Heart Atria; In Vitro Techniques; Muscle, Smooth, Vascular; Piperazines; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine; Tritium

1988
Identification of muscarinic M2 receptors on single muscle cells of the human and guinea pig intestine.
    Gastroenterology, 1987, Volume: 93, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Guinea Pigs; Humans; Jejunum; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Receptors, Muscarinic

1987
Determination of the muscarinic receptor subtype mediating vasodilatation.
    British journal of pharmacology, 1985, Volume: 84, Issue:1

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Atropine; Benzodiazepinones; Carbachol; Dogs; Female; Femoral Artery; Gallamine Triethiodide; In Vitro Techniques; Male; Pancuronium; Parasympatholytics; Phenethylamines; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Vasodilation

1985
Pharmacologic identification, activation and antagonism of two muscarine receptor subtypes in the lower esophageal sphincter.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Atropine; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Esophagogastric Junction; Hexamethonium Compounds; Opossums; Piperidines; Pirenzepine; Receptors, Muscarinic; Tetrodotoxin; Vagus Nerve

1984
Ligand-binding properties of an unusual nicotinic acetylcholine receptor subtype on isolated outer hair cells from guinea pig cochlea.
    Neuroscience letters, 1995, Jul-28, Volume: 195, Issue:1

    Topics: Animals; Atropine; Binding, Competitive; Bungarotoxins; Cochlea; Female; Guinea Pigs; Hair Cells, Auditory, Outer; In Vitro Techniques; Ligands; Male; Muscarinic Antagonists; Nicotine; Parasympatholytics; Piperidines; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Nicotinic; Strychnine

1995
A single transmitter regulates gene expression through two separate mechanisms: cholinergic regulation of phenylethanolamine N-methyltransferase mRNA via nicotinic and muscarinic pathways.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Atropine; Binding, Competitive; Calcimycin; Calcium; Carbachol; Cattle; Cells, Cultured; Colforsin; Epinephrine; Gene Expression Regulation, Enzymologic; Hexamethonium; Hexamethonium Compounds; Kinetics; Muscarine; Nicotine; Phenylethanolamine N-Methyltransferase; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Receptors, Nicotinic; RNA, Messenger

1994
Muscarinic acetylcholine receptors on an identified motor neurone in the cockroach, Periplaneta americana.
    Neuroscience letters, 1994, Jul-04, Volume: 175, Issue:1-2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Arecoline; Atropine; Dose-Response Relationship, Drug; Evoked Potentials; Ganglia, Invertebrate; In Vitro Techniques; Male; Motor Neurons; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Periplaneta; Piperidines; Pirenzepine; Receptors, Muscarinic; Scopolamine; Vertebrates

1994
Cholinergic and VIP-ergic pathways mediate histamine H2 receptor-induced cyclical secretion in the guinea pig colon.
    The American journal of physiology, 1995, Volume: 268, Issue:3 Pt 1

    Topics: Acetylcholine; Amiloride; Animals; Atropine; Choline; Colon; Dimaprit; Electric Conductivity; Guinea Pigs; Histamine Release; Intestinal Mucosa; Male; ortho-Aminobenzoates; Piperidines; Pirenzepine; Receptors, Histamine H2; Vasoactive Intestinal Peptide

1995
The role of acetylcholine in regulating secretory responsiveness in rat sweat glands.
    Molecular and cellular neurosciences, 1995, Volume: 6, Issue:1

    Topics: Acetylcholine; Age Factors; Animals; Atropine; Parasympatholytics; Pilocarpine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Sweat Glands; Time Factors

1995
Release of endogenous acetylcholine from a vascularly perfused rat stomach in vitro; inhibition by M3 muscarinic autoreceptors and alpha-2 adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Calcium; Clonidine; Diamines; Drug Interactions; Electric Stimulation; Gastric Mucosa; Hexamethonium; Hexamethonium Compounds; Male; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Perfusion; Phenylephrine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Stomach; Sympathetic Nervous System; Tetrodotoxin; Vagus Nerve

1993
Neuroregulation of a chemosensitive afferent system in the canine distal esophagus.
    The Journal of surgical research, 1993, Volume: 55, Issue:4

    Topics: Afferent Pathways; Animals; Atropine; Blood Pressure; Capsaicin; Chemoreceptor Cells; Dogs; Esophagus; Hexamethonium; Hexamethonium Compounds; Mucous Membrane; Nociceptors; Piperidines; Pressure; Pulse; Respiration; Substance P; Tetrodotoxin; Vagotomy

1993
Formation of inositol phosphates mediated by M3 muscarinic receptors in type-1 and type-2 astrocytes from neonatal rat cerebral cortex.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Animals, Newborn; Astrocytes; Atropine; Carbachol; Cells, Cultured; Cerebral Cortex; Inositol Phosphates; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Signal Transduction; Tubocurarine

1994
Regulation of pancreatic polypeptide release is mediated through M3 muscarinic receptors.
    Digestion, 1994, Volume: 55, Issue:6

    Topics: Animals; Atropine; Cholecystokinin; Dogs; Female; Gastric Acid; Male; Pancreatic Juice; Pancreatic Polypeptide; Parasympatholytics; Piperidines; Pirenzepine; Proglumide; Receptors, Muscarinic; Vagus Nerve

1994
Hypotensive effect of an M2-selective muscarinic antagonist in anaesthetized guinea-pigs.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:1

    Topics: Animals; Atropine; Blood Pressure; Depression, Chemical; Diamines; Guinea Pigs; Heart Rate; Male; Muscarinic Antagonists; Norepinephrine; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic

1995
A novel cholinergic "slow effect" of efferent stimulation on cochlear potentials in the guinea pig.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:5 Pt 1

    Topics: Acoustic Stimulation; Animals; Atropine; Bicuculline; Cochlea; Decamethonium Compounds; Dose-Response Relationship, Drug; Efferent Pathways; Electric Stimulation; Guinea Pigs; Hair Cells, Auditory, Outer; Hexamethonium; Membrane Potentials; Models, Neurological; Nerve Fibers; Piperidines; Strychnine; Time Factors; Vestibulocochlear Nerve

1995
Pressor effects of acetylcholine injected into the lateral septal area of conscious rats.
    Neuropharmacology, 1994, Volume: 33, Issue:12

    Topics: Acetylcholine; Adrenal Glands; Animals; Atropine; Blood Pressure; Ganglionic Blockers; Injections, Intraventricular; Male; Parasympatholytics; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar; Septal Nuclei; Stimulation, Chemical; Vasopressins

1994
Pertussis toxin-sensitive muscarinic relaxation in the rat iris dilator muscle.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Diamines; Dose-Response Relationship, Drug; Furans; GTP-Binding Proteins; In Vitro Techniques; Iris; Male; Microinjections; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Pertussis Toxin; Phentolamine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Virulence Factors, Bordetella

1995
Regional differences in motor responsiveness to antimuscarinic drugs in rabbit isolated small and large intestine.
    Pharmacological research, 1995, Volume: 31, Issue:1

    Topics: Animals; Atropine; Benzodiazepinones; Diamines; Dose-Response Relationship, Drug; Gastrointestinal Motility; Intestine, Large; Intestine, Small; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic

1995
Methoctramine induces nonspecific airway hyperresponsiveness in vivo.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: Aerosols; Albuterol; Animals; Arachidonic Acid; Atropine; Bronchial Hyperreactivity; Bronchoconstriction; Diamines; Drug Synergism; Gallamine Triethiodide; Guinea Pigs; Histamine; Male; Muscarinic Antagonists; Ovalbumin; Parasympatholytics; Piperazines; Piperidines; Platelet Activating Factor; Propranolol; Receptors, Muscarinic

1994
Muscarinic M3 receptor-mediated release of gastrin from canine antral G cells in primary culture.
    Digestion, 1995, Volume: 56, Issue:1

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Enterochromaffin Cells; Gastrins; Muscarinic Antagonists; Parasympathetic Nervous System; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Receptor, Muscarinic M3; Receptors, Muscarinic; Stimulation, Chemical

1995
Vitamin D status modulates rat colonic M3 muscarinic receptor characteristics and coupling to guanylate cyclase.
    FEBS letters, 1994, Jun-20, Volume: 347, Issue:1

    Topics: Animals; Atropine; Colon; Diamines; Enzyme Activation; Guanylate Cyclase; Male; Muscarinic Antagonists; Nutritional Status; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Vitamin D

1994
Receptor mediated presynaptic modulation of the release of noradrenaline in human papillary muscle.
    Cardiovascular research, 1994, Volume: 28, Issue:5

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Atropine; Berberine; Chromatography, High Pressure Liquid; Culture Techniques; Dopamine beta-Hydroxylase; Electric Stimulation; Feedback; Female; Heart Atria; Humans; Immunohistochemistry; Male; Middle Aged; Norepinephrine; Oxotremorine; Pancuronium; Papillary Muscles; Piperidines; Presynaptic Terminals; Receptors, Muscarinic; Sympathetic Nervous System; Tritium; Xylazine

1994
Assessment of the muscarinic receptor subtypes involved in pilocarpine-induced seizures in mice.
    Neuroscience letters, 1994, Feb-28, Volume: 168, Issue:1-2

    Topics: Animals; Atropine; Cerebral Ventricles; Injections, Intraventricular; Male; Mice; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Seizures

1994
In vitro pharmacologic characterization of a cholinergic receptor on outer hair cells.
    Hearing research, 1994, Volume: 74, Issue:1-2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Azocines; Bungarotoxins; Carbachol; Choline; Cholinergic Antagonists; Curare; Dimethylphenylpiperazinium Iodide; Guinea Pigs; Hair Cells, Auditory, Outer; In Vitro Techniques; Membrane Potentials; Nicotine; Piperidines; Pirenzepine; Quinolizines; Receptors, Cholinergic; Strychnine; Trimethaphan

1994
Diabetes-induced alterations in the properties of muscarinic cholinergic receptors in rat vas deferens.
    The Journal of urology, 1994, Volume: 152, Issue:3

    Topics: Animals; Atropine; Binding, Competitive; Diabetes Mellitus, Experimental; Diamines; Insulin; Male; Parasympatholytics; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Up-Regulation; Vas Deferens

1994
Evidence of muscarinic acetylcholine receptors and GTP-binding proteins in peritoneal mesothelial cells in vitro.
    Advances in peritoneal dialysis. Conference on Peritoneal Dialysis, 1993, Volume: 9

    Topics: Animals; Atropine; Binding, Competitive; Cells, Cultured; Epithelium; GTP-Binding Proteins; Humans; Peritoneum; Piperidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic

1993
Characterization of the muscarinic receptors in the mesenteric vascular bed of spontaneously hypertensive rats.
    Journal of hypertension, 1993, Volume: 11, Issue:12

    Topics: Animals; Atropine; Benzodiazepinones; Endothelium, Vascular; Hypertension; Male; Mesenteric Artery, Superior; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Vasodilation

1993
Pharmacological characterization of muscarinic cholinergic receptors in cat pons and cortex. Preliminary study.
    Pharmacology, 1994, Volume: 48, Issue:2

    Topics: Animals; Atropine; Binding, Competitive; Cats; Cerebral Cortex; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pons; Receptors, Muscarinic

1994
Agonist-induced down-regulation and antagonist-induced up-regulation of m2- and m3-muscarinic acetylcholine receptor mRNA and protein in cultured cerebellar granule cells.
    Molecular pharmacology, 1993, Volume: 44, Issue:5

    Topics: Animals; Atropine; Carbachol; Cells, Cultured; Cerebellum; Down-Regulation; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; RNA, Messenger; Up-Regulation

1993
Cholinergic M2 muscarinic receptor-mediated inhibition of endogenous noradrenaline release from the isolated vascularly perfused rat stomach.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:1

    Topics: Animals; Arteries; Atrial Function; Atropine; Depression, Chemical; Diamines; Electric Stimulation; Ethylmaleimide; Heart Atria; Male; Myocardial Contraction; Nerve Endings; Norepinephrine; Oxotremorine; Parasympatholytics; Perfusion; Pertussis Toxin; Phentolamine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Stomach; Sympathetic Nervous System; Vagus Nerve; Virulence Factors, Bordetella

1993
Differential effects of antimuscarinic agents on intestinal motility in the conscious dog.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Animals; Atropine; Dogs; Female; Gastrointestinal Motility; Heart Rate; Male; Parasympatholytics; Piperidines; Pirenzepine; Pupil; Receptors, Muscarinic

1993
Muscarinic receptors in the aortae of normo- and hypertensive rats: a binding study.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 1993, Volume: 15, Issue:2

    Topics: Acetylcholine; Animals; Aorta; Atropine; Binding, Competitive; Endothelium, Vascular; Guanylyl Imidodiphosphate; Hypertension; In Vitro Techniques; Kinetics; Muscle, Smooth, Vascular; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Scopolamine; Tropanes

1993
Subtype of muscarinic receptors mediating relaxation and contraction in the rat iris dilator smooth muscle.
    General pharmacology, 1993, Volume: 24, Issue:1

    Topics: Alkaloids; Animals; Atropine; Carbachol; Furans; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic

1993
Functional characterization of muscarinic receptors in murine airways.
    British journal of pharmacology, 1993, Volume: 109, Issue:1

    Topics: Administration, Inhalation; Airway Resistance; Animals; Atropine; Bronchi; Electric Stimulation; In Vitro Techniques; Isometric Contraction; Lung Compliance; Male; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1993
Characterization of muscarinic receptors mediating contractions of circular and longitudinal muscle of human isolated colon.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Alkaloids; Atropine; Carbachol; Carcinoma; Colon; Colonic Neoplasms; Dose-Response Relationship, Drug; Furans; Humans; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthalenes; Piperidines; Pirenzepine

1995
Mediation of the depolarization-induced [Ca(2+)]i increase in rat sublingual acini by acetylcholine released from nerve terminals.
    Archives of oral biology, 1996, Volume: 41, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Cadmium; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Cytosol; Fluorescent Dyes; Fura-2; Gallic Acid; Inositol 1,4,5-Trisphosphate; Male; Muscarinic Antagonists; Nerve Endings; Nicotinic Antagonists; Piperidines; Pirenzepine; Potassium; Rats; Rats, Wistar; Receptors, Nicotinic; Sublingual Gland

1996
Muscarinic receptor subtypes in the submandibular gland and the urinary bladder of the rabbit: in vivo and in vitro functional comparisons of receptor antagonists.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:6

    Topics: Animals; Atropine; Carbachol; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Muscarinic Antagonists; Piperidines; Pirenzepine; Rabbits; Receptors, Muscarinic; Submandibular Gland; Urinary Bladder

1995
The roles of muscarinic receptor subtypes in modulation of nasal ciliary action.
    Rhinology, 1996, Volume: 34, Issue:3

    Topics: Atropine; Cilia; Gallamine Triethiodide; Humans; In Vitro Techniques; Methacholine Chloride; Mucociliary Clearance; Muscarinic Agonists; Muscarinic Antagonists; Nasal Mucosa; Piperidines; Pirenzepine; Receptors, Muscarinic

1996
Acetylcholine stimulates growth hormone secretion in the neonatal rat pituitary.
    Journal of neuroendocrinology, 1996, Volume: 8, Issue:12

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Animals, Newborn; Atropine; Diamines; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Muscarinic Agonists; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar

1996
Circulating antibodies against rat parotid gland M3 muscarinic receptors in primary Sjögren's syndrome.
    Clinical and experimental immunology, 1996, Volume: 104, Issue:3

    Topics: Adolescent; Adrenergic beta-Agonists; Adult; Animals; Antibodies, Blocking; Atropine; Carbachol; Carbamates; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Female; Humans; Immunoglobulin G; Isoproterenol; Muscarinic Antagonists; Parasympatholytics; Parotid Gland; Phenylcarbamates; Phosphatidylinositols; Piperidines; Pirenzepine; Protease Inhibitors; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Sjogren's Syndrome

1996
Muscarinic acetylcholine receptors on rat thymocytes: their possible involvement in DNA fragmentation.
    Japanese journal of pharmacology, 1997, Volume: 73, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Apoptosis; Atropine; Binding, Competitive; Carbachol; DNA Fragmentation; Electrophoresis, Agar Gel; Hydrocortisone; Injections, Subcutaneous; Isotope Labeling; Male; Muscarinic Agonists; Muscarinic Antagonists; Nucleosomes; Oxotremorine; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Thymus Gland

1997
Functional characterization of peripheral muscarinic subtypes in anesthetized cats.
    Life sciences, 1997, Volume: 61, Issue:2

    Topics: Animals; Atropine; Blood Pressure; Cats; Gallamine Triethiodide; Galvanic Skin Response; Heart Rate; Methacholine Chloride; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Superior Cervical Ganglion; Synaptic Transmission; Vagus Nerve; Vasodilation

1997
Cholinergic modulation of electrogenic ion transport in different regions of the rat small intestine.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analysis of Variance; Animals; Atropine; Bethanechol; Carbachol; Chlorides; Diamines; Duodenum; Ileum; Intestinal Mucosa; Ion Transport; Jejunum; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship; Tetrodotoxin

1997
M3 muscarinic receptor-mediated enhancement of NMDA-evoked adenosine release in rat cortical slices in vitro.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Atropine; Carbachol; Cerebral Cortex; Diamines; Drug Synergism; In Vitro Techniques; Kinetics; Magnesium; Male; Muscarinic Agonists; Muscarinic Antagonists; N-Methylaspartate; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Muscarinic

1997
M2 and M3 muscarinic receptors couple, respectively, with activation of nonselective cationic channels and potassium channels in intestinal smooth muscle cells.
    Japanese journal of pharmacology, 1998, Volume: 76, Issue:2

    Topics: Animals; Atropine; Calcium; Carbachol; Guinea Pigs; Male; Muscarinic Agonists; Muscle, Smooth; Piperidines; Pirenzepine; Potassium Channels; Receptors, Muscarinic

1998
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
    Experimental neurology, 1998, Volume: 151, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon

1998
Muscarinic inhibition of substance P induced ion secretion in piglet jejunum.
    Canadian journal of physiology and pharmacology, 1998, Volume: 76, Issue:2

    Topics: Animals; Atropine; Carbachol; Cholinergic Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Gallamine Triethiodide; Histamine; Ion Transport; Jejunum; Mecamylamine; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Substance P; Swine; Time Factors

1998
Pharmacological profile of CEB-1957 and atropine toward brain muscarinic receptors and comparative study of their efficacy against sarin poisoning.
    Toxicology and applied pharmacology, 1998, Volume: 150, Issue:2

    Topics: Animals; Atropine; Autoradiography; Binding, Competitive; Brain; Cholinesterase Inhibitors; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Poisoning; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Sarin; Thiophenes

1998
Subtypes of muscarinic receptors regulating gallbladder cholinergic contractions.
    The American journal of physiology, 1999, Volume: 276, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Diamines; Electric Stimulation; Gallbladder; Guinea Pigs; Hexamethonium; Muscarinic Antagonists; Muscle Contraction; Parasympatholytics; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Tetrodotoxin; Tropicamide

1999
Presynaptic muscarinic (M3) receptors reduce excitatory transmission in dopamine neurons of the rat mesencephalon.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Atropine; Carbachol; Diamines; Dicyclomine; Dopamine; Electric Stimulation; Excitatory Postsynaptic Potentials; Mesencephalon; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reaction Time; Receptor, Muscarinic M3; Receptors, Muscarinic; Synaptic Transmission; Tetrodotoxin

1999
Muscarinic cholinoceptor subtypes mediating tracheal smooth muscle contraction and inositol phosphate generation in guinea pig and rat.
    European journal of pharmacology, 1999, May-21, Volume: 372, Issue:3

    Topics: Animals; Atropine; Diamines; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Trachea

1999
Cardiovascular response to the injection of acetylcholine into the anterior cingulate region of the medial prefrontal cortex of unanesthetized rats.
    Cerebral cortex (New York, N.Y. : 1991), 1999, Volume: 9, Issue:4

    Topics: Acetylcholine; Animals; Atropine; Blood Pressure; Dose-Response Relationship, Drug; Gyrus Cinguli; Hemodynamics; Injections; Male; Muscarinic Antagonists; Occipital Lobe; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar

1999
Effect of cholinergic drugs on the concentration of intracellular free calcium of rat pituitary intermediate lobe cells.
    Brain research bulletin, 1999, Sep-01, Volume: 50, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Age Factors; Animals; Atropine; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Cytosol; Female; Male; Melanocytes; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nicotinic Agonists; Piperidines; Pirenzepine; Pituitary Gland; Rats; Rats, Wistar; Vasodilator Agents

1999
Role of muscarinic cholinergic transmission in Edinger-Westphal nucleus-induced choroidal vasodilation in pigeon.
    Experimental eye research, 2000, Volume: 70, Issue:3

    Topics: Alkaloids; Animals; Atropine; Blood Pressure; Choroid; Columbidae; Electric Stimulation; Furans; Heart Rate; Muscarinic Antagonists; Naphthalenes; Parasympatholytics; Piperidines; Receptors, Muscarinic; Regional Blood Flow; Vasodilation

2000
Involvement of M3 muscarinic receptors of the spinal cord in formalin-induced nociception in mice.
    Brain research, 2000, Mar-17, Volume: 859, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Cholinergic Agents; Cholinesterase Inhibitors; Formaldehyde; Hemicholinium 3; Male; Mice; Mice, Inbred Strains; Muscarinic Antagonists; Naloxone; Narcotic Antagonists; Neostigmine; Nociceptors; Pain; Pain Measurement; Piperidines; Receptor, Muscarinic M3; Receptors, Muscarinic; Spinal Cord

2000
Selective restoration of calcium coupling to muscarinic M(3) receptors in contractile cultured airway myocytes.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 278, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Blood Proteins; Blotting, Western; Bradykinin; Calcium; Calcium Channels; Cells, Cultured; Diamines; Dogs; Dose-Response Relationship, Drug; Fluorescent Dyes; Fura-2; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Muscarinic Antagonists; Muscle, Smooth; Oxazoles; Parasympatholytics; Phenotype; Piperidines; Pirenzepine; Receptor, Muscarinic M3; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Receptors, Muscarinic; Trachea; Vasodilator Agents

2000
M(2)/M(4)-muscarinic receptors mediate automodulation of acetylcholine outflow from mouse cortex.
    Neuroscience letters, 2000, Jun-23, Volume: 287, Issue:2

    Topics: Acetylcholine; Alkaloids; Animals; Atropine; Autoreceptors; Binding, Competitive; Cerebral Cortex; Furans; Male; Mice; Muscarinic Antagonists; Naphthalenes; Neostigmine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic

2000
Carbachol and acetylcholine delay the early postdenervation depolarization of muscle fibres through M1-cholinergic receptors.
    Neuroscience research, 2000, Volume: 37, Issue:4

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Carbachol; Culture Techniques; Diaphragm; Male; Membrane Potentials; Muscarinic Agonists; Muscarinic Antagonists; Muscle Denervation; Muscle Fibers, Skeletal; Oxotremorine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic

2000
Coordinated transitions in neurotransmitter systems for the initiation and propagation of spontaneous retinal waves.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Sep-01, Volume: 20, Issue:17

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; Animals; Animals, Newborn; Atropine; Bungarotoxins; Calcium; Curare; Dimethylphenylpiperazinium Iodide; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Fura-2; Hexamethonium; Membrane Potentials; Muscarine; Muscarinic Antagonists; Neurotransmitter Agents; Nicotinic Antagonists; Patch-Clamp Techniques; Piperidines; Rabbits; Retina; Retinal Ganglion Cells

2000
Secretion and gene expression of secretory leukocyte protease inhibitor by human airway submucosal glands.
    American journal of physiology. Lung cellular and molecular physiology, 2001, Volume: 280, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Atropine; Bronchi; Dexamethasone; Dose-Response Relationship, Drug; Exocrine Glands; Female; Gene Expression; Glucocorticoids; Humans; Leukocyte Elastase; Male; Methacholine Chloride; Middle Aged; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Proteinase Inhibitory Proteins, Secretory; Proteins; Respiratory Mucosa; RNA, Messenger; Secretory Leukocyte Peptidase Inhibitor; Trachea

2001
Mechanisms of acetylcholine-induced vasorelaxation in high K+-stimulated rabbit renal arteries.
    The Journal of veterinary medical science, 2001, Volume: 63, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Calcium; Calcium Channel Blockers; Cations, Monovalent; Endothelium, Vascular; Gadolinium; Imidazoles; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Rabbits; Renal Artery; Tropicamide; Vasoconstriction; Vasodilation

2001
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate

2001
Effects of cholinergic agents on the vasopressin-mediated water transport in the isolated toad bladder.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 129, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Arginine Vasopressin; Atropine; Biological Transport; Bufo marinus; Calcium; Calcium Channel Blockers; Carbachol; Cholinergic Agonists; Cholinergic Antagonists; In Vitro Techniques; Isotonic Solutions; Lanthanum; Osmolar Concentration; Piperidines; Pirenzepine; Urinary Bladder; Vasoconstrictor Agents; Water

2001
Characterization of muscarinic acetylcholine receptors in the rat epididymis.
    Biology of reproduction, 2001, Volume: 65, Issue:4

    Topics: Animals; Atropine; Cell Membrane; Diamines; Epididymis; Male; Muscarinic Antagonists; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tritium

2001
Coupling of M(2) muscarinic receptors to Src activation in cultured canine colonic smooth muscle cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:1

    Topics: Animals; Atropine; Cells, Cultured; Colon; Dogs; Female; Gene Expression Regulation, Enzymologic; Genistein; Male; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fyn; Pyrazoles; Pyrimidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; src-Family Kinases; Teprotide

2002
Activation of nitric oxide synthase through muscarinic receptors in rat parotid gland.
    European journal of pharmacology, 2002, Mar-29, Volume: 439, Issue:1-3

    Topics: Amylases; Animals; Atropine; Binding, Competitive; Carbachol; Cell Membrane; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Parotid Gland; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic; Specific Pathogen-Free Organisms

2002
[The effects of the antagonists of muscarinic acetylcholine receptor subtypes in rat brain on urinary bladder contraction].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 2002, Volume: 93, Issue:3

    Topics: Animals; Atropine; Brain; Female; Muscarine; Muscarinic Antagonists; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder; Urination

2002
Acetylcholine leads to free radical production dependent on K(ATP) channels, G(i) proteins, phosphatidylinositol 3-kinase and tyrosine kinase.
    Cardiovascular research, 2002, Aug-15, Volume: 55, Issue:3

    Topics: Acetylcholine; Analysis of Variance; Androstadienes; Animals; Aorta; Atropine; Cell Line; Decanoic Acids; Diazoxide; Enzyme Inhibitors; Female; Free Radical Scavengers; Genistein; GTP-Binding Protein alpha Subunits, Gi-Go; Hydroxy Acids; Ionophores; Ischemic Preconditioning; Male; Methacholine Chloride; Microscopy, Fluorescence; Muscarinic Agonists; Muscle, Smooth, Vascular; Perfusion; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Potassium Channel Blockers; Potassium Channels; Protein-Tyrosine Kinases; Rabbits; Rats; Reactive Oxygen Species; Receptors, Cholinergic; Signal Transduction; Tiopronin; Valinomycin; Wortmannin

2002
The colon-selective spasmolytic otilonium bromide inhibits muscarinic M(3) receptor-coupled calcium signals in isolated human colonic crypts.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: Acetylcholine; Animals; Atropine; Calcium; Calcium Signaling; CHO Cells; Colon; Cricetinae; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M3; Receptors, Muscarinic; Time Factors; Vasodilator Agents

2002
Low concentrations of pyridostigmine prevent soman-induced inhibition of GABAergic transmission in the central nervous system: involvement of muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Animals; Atropine; Central Nervous System; Cholinesterase Inhibitors; Cholinesterases; Electric Stimulation; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Membrane Potentials; Muscarinic Antagonists; Neurons; Patch-Clamp Techniques; Piperidines; Pirenzepine; Pyramidal Cells; Pyridostigmine Bromide; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Receptors, Nicotinic; Soman; Synaptic Transmission

2003
Change in muscarinic modulation of transmitter release in the rat urinary bladder after spinal cord injury.
    Neurochemistry international, 2003, Volume: 43, Issue:1

    Topics: Animals; Atropine; Electric Stimulation; Female; Muscarinic Antagonists; Neurotransmitter Agents; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3; Receptors, Muscarinic; Spinal Cord Injuries; Urinary Bladder; Urinary Bladder, Neurogenic

2003
The M4 muscarinic receptor-selective effects on keratinocyte crawling locomotion.
    Life sciences, 2003, Mar-28, Volume: 72, Issue:18-19

    Topics: Animals; Atropine; Cell Movement; Humans; Infant, Newborn; Keratinocytes; Mice; Mice, Knockout; Muscarine; Muscarinic Agonists; Piperidines; Pirenzepine; Receptor, Muscarinic M4; Receptors, Muscarinic; Stimulation, Chemical

2003
Brain muscarinic receptor subtypes mediating water intake and Fos following cerebroventricular administration of bethanecol in rats.
    Psychopharmacology, 2003, Volume: 167, Issue:2

    Topics: Animals; Atropine; Bethanechol; Dose-Response Relationship, Drug; Drinking Behavior; Injections, Intraventricular; Male; Muscarinic Agonists; Muscarinic Antagonists; Piperidines; Pirenzepine; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Water

2003
Characterization of muscarinic receptor subtypes in the rostral ventrolateral medulla and effects on morphine-induced antinociception in rats.
    European journal of pharmacology, 2003, Apr-04, Volume: 465, Issue:3

    Topics: Analgesics, Opioid; Animals; Atropine; Diamines; Male; Mecamylamine; Medulla Oblongata; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Pain Measurement; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Time Factors

2003
Nuclear factor kappaB activation by muscarinic receptors in astroglial cells: effect of ethanol.
    Neuroscience, 2003, Volume: 120, Issue:4

    Topics: Astrocytes; Astrocytoma; Atropine; Blotting, Western; Carbachol; Cell Line; Cellular Structures; Central Nervous System Depressants; Chelating Agents; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Ethanol; Gallamine Triethiodide; Humans; Muscarinic Antagonists; NF-kappa B; Nicotinic Antagonists; Pertussis Toxin; Piperidines; Receptors, Muscarinic; Thymidine; Time Factors; Tritium

2003
Activation of muscarinic acetylcholine receptors elicits pigment granule dispersion in retinal pigment epithelium isolated from bluegill.
    BMC neuroscience, 2004, Jul-13, Volume: 5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Arecoline; Atropine; Carbachol; Colforsin; Cyclic AMP; Cytoplasmic Granules; Light; Muscarinic Agonists; Muscarinic Antagonists; Perciformes; Pigment Epithelium of Eye; Piperidines; Pirenzepine; Quaternary Ammonium Compounds; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Retinal Pigments; Second Messenger Systems; Tropicamide

2004
Comparison of the antimuscarinic action of p-fluorohexahydrosiladifenidol in ileal and tracheal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 312, Issue:2

    Topics: Animals; Atropine; Cattle; Guinea Pigs; Histamine Antagonists; Hydrolysis; Ileum; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Phosphatidylinositols; Piperidines; Receptor, Muscarinic M3; Trachea

2005
Arecoline excites the colonic smooth muscle motility via M3 receptor in rabbits.
    The Chinese journal of physiology, 2004, Jun-30, Volume: 47, Issue:2

    Topics: Animals; Arecoline; Atropine; Colon; Dose-Response Relationship, Drug; Female; Ganglionic Stimulants; Gastrointestinal Motility; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Piperidines; Rabbits; Receptor, Muscarinic M2; Receptor, Muscarinic M3

2004
Intrathecal clonidine inhibits mechanical allodynia via activation of the spinal muscarinic M1 receptor in streptozotocin-induced diabetic mice.
    European journal of pharmacology, 2004, Nov-28, Volume: 505, Issue:1-3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesics; Animals; Atropine; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Diamines; Injections, Spinal; Male; Mice; Motor Activity; Muscarinic Agonists; Muscarinic Antagonists; Pain; Pain Threshold; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Spinal Cord; Streptozocin; Stress, Mechanical; Time Factors

2004
The anti-inflammatory effect of peripheral bee venom stimulation is mediated by central muscarinic type 2 receptors and activation of sympathetic preganglionic neurons.
    Brain research, 2005, Jul-12, Volume: 1049, Issue:2

    Topics: Animals; Animals, Newborn; Anti-Inflammatory Agents; Atropine; Autonomic Fibers, Preganglionic; Bee Venoms; Catecholamines; Cell Count; Choline O-Acetyltransferase; Disease Models, Animal; Drug Interactions; Exudates and Transudates; Hexamethonium; Immunohistochemistry; Inflammation; Leukocytes; Male; Mice; Mice, Inbred ICR; Muscarinic Antagonists; Neurons; Nicotinic Antagonists; Oncogene Proteins v-fos; Oxidopamine; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Spinal Cord; Sympathectomy, Chemical

2005
Neural regulation of slow-wave frequency in the murine gastric antrum.
    American journal of physiology. Gastrointestinal and liver physiology, 2006, Volume: 290, Issue:3

    Topics: Acetylcholine; Androstenes; Animals; Atropine; Benzamides; Benzimidazoles; Carbachol; Electric Stimulation; Electrophysiology; Enteric Nervous System; Female; Gastric Emptying; Male; Mice; Mice, Inbred BALB C; Mice, Inbred Strains; Motor Neurons; Muscle Contraction; Myenteric Plexus; Neostigmine; Piperidines; Pyloric Antrum; Tetrodotoxin

2006
Muscarinic M1 and M3 receptor binding alterations in pancreas during pancreatic regeneration of young rats.
    Endocrine research, 2005, Volume: 31, Issue:4

    Topics: Animals; Atropine; Carbachol; Cholinergic Agonists; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Muscarinic Antagonists; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Regeneration

2005
Agonist and antagonist sensitivity of non-selective cation channel currents evoked by muscarinic receptor stimulation in bovine ciliary muscle cells.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:3

    Topics: Animals; Atropine; Barium; Carbachol; Cattle; Cells, Cultured; Ciliary Body; Dose-Response Relationship, Drug; Membrane Potentials; Microscopy, Fluorescence; Muscarinic Agonists; Muscarinic Antagonists; Muscle Cells; Patch-Clamp Techniques; Piperidines; Pirenzepine; Receptor, Muscarinic M3; TRPC Cation Channels

2006
Cardiovascular effects of carbachol microinjected into the bed nucleus of the stria terminalis of the rat brain.
    Brain research, 2007, Apr-27, Volume: 1143

    Topics: Animals; Arginine Vasopressin; Atropine; Blood Pressure; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Heart Rate; Male; Microinjections; Muscarinic Antagonists; Nicotinic Antagonists; Pentolinium Tartrate; Piperidines; Rats; Rats, Wistar; Septal Nuclei

2007
Verrucotoxin inhibits KATP channels in cardiac myocytes through a muscarinic M3 receptor-PKC pathway.
    European journal of pharmacology, 2007, Jun-01, Volume: 563, Issue:1-3

    Topics: Adenosine Triphosphate; Alkaloids; Animals; Atropine; Benzophenanthridines; Dose-Response Relationship, Drug; Female; Fish Venoms; Glycoproteins; Guinea Pigs; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Membrane Potentials; Muscarinic Antagonists; Myocytes, Cardiac; Patch-Clamp Techniques; Pinacidil; Piperidines; Potassium Channel Blockers; Potassium Channels; Protein Kinase C; Protein Kinase Inhibitors; Receptor, Muscarinic M3; Signal Transduction; Time Factors

2007
Muscarinic receptor-independent activation of cyclic adenosine monophosphate-dependent protein kinase in rostral ventrolateral medulla underlies the sympathoexcitatory phase of cardiovascular responses during mevinphos intoxication in the rat.
    Shock (Augusta, Ga.), 2007, Volume: 27, Issue:5

    Topics: Animals; Atropine; Blotting, Western; Cardiovascular System; Cholinesterase Inhibitors; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Intracellular Signaling Peptides and Proteins; Male; Medulla Oblongata; Mevinphos; Muscarinic Antagonists; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Time Factors; Tropicamide

2007
Increase in cochlear microphonic potential after toluene administration.
    Hearing research, 2007, Volume: 230, Issue:1-2

    Topics: Acoustic Stimulation; Animals; Atropine; Cholinergic Antagonists; Cochlea; Cochlear Microphonic Potentials; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Gentamicins; Neurons, Efferent; Noise; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Reflex, Acoustic; Solvents; Toluene

2007
Functional expression of M3, a muscarinic acetylcholine receptor subtype, in taste bud cells of mouse fungiform papillae.
    Chemical senses, 2008, Volume: 33, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Calcium Signaling; Cells, Cultured; Diamines; Electrophysiology; Gene Expression; Inositol 1,4,5-Trisphosphate Receptors; Mice; Mice, Inbred Strains; Muscarinic Antagonists; Patch-Clamp Techniques; Phospholipase C beta; Piperidines; Pirenzepine; Receptor, Muscarinic M3; Receptors, Muscarinic; Reverse Transcriptase Polymerase Chain Reaction; Synaptosomal-Associated Protein 25; Taste Buds; Tropicamide; Vesicular Acetylcholine Transport Proteins

2008
Bronchodilatory effects of S-isopetasin, an antimuscarinic sesquiterpene of Petasites formosanus, on obstructive airway hyperresponsiveness.
    European journal of pharmacology, 2008, Apr-28, Volume: 584, Issue:2-3

    Topics: Acetylcholine; Animals; Atropine; Binding, Competitive; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Bronchodilator Agents; Cells, Cultured; Cholinesterase Inhibitors; Diamines; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Ipratropium; Male; Muscarinic Antagonists; Muscle, Smooth; N-Methylscopolamine; Neostigmine; Petasites; Piperidines; Protein Binding; Receptor, Muscarinic M3; Sesquiterpenes; Time Factors; Trachea

2008
Muscarinic receptors involved in airway vascular leakage induced by experimental gastro-oesophageal reflux.
    Life sciences, 2008, Apr-23, Volume: 82, Issue:17-18

    Topics: Animals; Atropine; Capillary Permeability; Diamines; Female; Ganglionic Blockers; Gastroesophageal Reflux; Guinea Pigs; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Receptors, Nicotinic; Regional Blood Flow; Respiratory System

2008
Activation of cholinergic receptors blocks non-adrenergic non-cholinergic contractions in the rat urinary bladder.
    Brain research bulletin, 2008, Dec-16, Volume: 77, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Antineoplastic Agents; Atropine; Calcium Channel Agonists; Carbachol; Cholinergic Agonists; Cholinesterase Inhibitors; Electric Stimulation; Female; In Vitro Techniques; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Physostigmine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Suramin; Urinary Bladder

2008
Spinal cholinergic mechanism of the relieving effects of electroacupuncture on cold and warm allodynia in a rat model of neuropathic pain.
    The journal of physiological sciences : JPS, 2009, Volume: 59, Issue:4

    Topics: Animals; Atropine; Cholinergic Agents; Cholinergic Fibers; Cold Temperature; Diamines; Disease Models, Animal; Electroacupuncture; Hot Temperature; Hyperesthesia; Male; Mecamylamine; Neuralgia; Pain Threshold; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Spinal Nerves

2009
Muscarinic activation of Ca2+-activated Cl- current in interstitial cells of Cajal.
    The Journal of physiology, 2011, Sep-15, Volume: 589, Issue:Pt 18

    Topics: Animals; Atropine; Carbachol; Chloride Channels; Green Fluorescent Proteins; Interstitial Cells of Cajal; Intestine, Small; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Models, Animal; Muscarinic Agonists; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Receptors, Muscarinic

2011
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
    Urology, 2011, Volume: 78, Issue:6

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium

2011
Activation of M3 muscarinic receptor and Ca²⁺ influx by crude fraction from Crotonis Fructus in isolated rabbit jejunum.
    Journal of ethnopharmacology, 2012, Jan-06, Volume: 139, Issue:1

    Topics: Animals; Atropine; Calcium; Calcium Channel Blockers; Croton; Female; Fruit; In Vitro Techniques; Jejunum; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Piperidines; Plant Extracts; Rabbits; Receptor, Muscarinic M3; Solvents; Verapamil

2012
Role of M3 mAChR in in vivo and in vitro models of LPS-induced inflammatory response.
    International immunopharmacology, 2012, Volume: 14, Issue:3

    Topics: Acute Lung Injury; Animals; Atropine; Cell Line; Lipopolysaccharides; Macrophages, Alveolar; Male; Mice; Muscarinic Antagonists; NF-kappa B; Piperidines; Pneumonia; Receptor, Muscarinic M3

2012
Different muscarinic receptor subtypes modulate proliferation of primary human detrusor smooth muscle cells via Akt/PI3K and map kinases.
    Pharmacological research, 2013, Volume: 74

    Topics: Aged; Atropine; Benzofurans; Carbachol; Cell Proliferation; Cells, Cultured; Cholinergic Agonists; Gene Expression; Humans; Male; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Myocytes, Smooth Muscle; Phosphatidylinositol 3-Kinases; Piperidines; Pirenzepine; Proto-Oncogene Proteins c-akt; Pyrrolidines; Receptors, Muscarinic; RNA, Messenger; Urinary Bladder

2013
Expression and function of muscarinic subtype receptors in bladder interstitial cells of cajal in rats.
    Urology journal, 2014, Jul-08, Volume: 11, Issue:3

    Topics: Action Potentials; Animals; Atropine; Calcium Channels; Carbachol; Cholinergic Agonists; Diamines; Interstitial Cells of Cajal; Male; Muscarinic Antagonists; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder

2014
In vitro effects of the organophosphorus pesticide malathion on the reactivity of rat aorta.
    Pharmacology, 2014, Volume: 94, Issue:3-4

    Topics: Animals; Aorta, Thoracic; Atropine; Endothelium, Vascular; Epoprostenol; Gallamine Triethiodide; In Vitro Techniques; Indomethacin; Malathion; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Pesticides; Phenylephrine; Piperidines; Pirenzepine; Rats, Wistar; Vasodilator Agents

2014
Muscarinic cholinergic receptor antagonists in the VTA and RMTg have opposite effects on morphine-induced locomotion in mice.
    Behavioural brain research, 2017, 04-14, Volume: 323

    Topics: Acetylcholine; Animals; Atropine; Locomotion; Mice; Mice, Inbred C57BL; Morphine; Muscarinic Antagonists; Piperidines; Receptor, Muscarinic M3; Receptor, Muscarinic M4; Tropicamide; Ventral Tegmental Area

2017
Novel choline analog 2-(4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazin-1-yl)ethan-1-ol produces sympathoinhibition, hypotension, and antihypertensive effects.
    Naunyn-Schmiedeberg's archives of pharmacology, 2019, Volume: 392, Issue:9

    Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Atropine; Blood Pressure; Heart Rate; Hypertension; Hypotension; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperazines; Piperidines; Pirenzepine; Pyrazoles; Rats, Inbred SHR; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M3

2019