Page last updated: 2024-09-04

atrasentan and sirolimus

atrasentan has been researched along with sirolimus in 1 studies

Compound Research Comparison

Studies
(atrasentan)
Trials
(atrasentan)
Recent Studies (post-2010)
(atrasentan)
Studies
(sirolimus)
Trials
(sirolimus)
Recent Studies (post-2010) (sirolimus)
3584110820,7112,36811,516

Protein Interaction Comparison

ProteinTaxonomyatrasentan (IC50)sirolimus (IC50)
Bile salt export pumpHomo sapiens (human)10
ATP-dependent translocase ABCB1Homo sapiens (human)1.25
Cytochrome P450 3A4Homo sapiens (human)2
Cytochrome P450 2C9 Homo sapiens (human)2
Peptidyl-prolyl cis-trans isomerase FKBP1AMus musculus (house mouse)0.001
Cytochrome P450 2C19Homo sapiens (human)4
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0897
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.0042
Regulatory-associated protein of mTORHomo sapiens (human)0.225
Target of rapamycin complex subunit LST8Homo sapiens (human)0.225
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.9
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.1

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Becker, M; Börgermann, C; Hess, J; Rübben, H; Schenck, M; Vom Dorp, F1

Other Studies

1 other study(ies) available for atrasentan and sirolimus

ArticleYear
[Value of targeted therapy for prostate cancer].
    Der Urologe. Ausg. A, 2008, Volume: 47, Issue:10

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Atrasentan; Calcitriol; Drug Delivery Systems; Humans; Male; Neoplasm Staging; Prostatic Neoplasms; Protein-Tyrosine Kinases; Pyrrolidines; Sirolimus; Survival Rate; Thionucleotides

2008