Page last updated: 2024-09-04

atrasentan and rifampin

atrasentan has been researched along with rifampin in 2 studies

Compound Research Comparison

Studies
(atrasentan)
Trials
(atrasentan)
Recent Studies (post-2010)
(atrasentan)
Studies
(rifampin)
Trials
(rifampin)
Recent Studies (post-2010) (rifampin)
3584110820,4681,4996,552

Protein Interaction Comparison

ProteinTaxonomyatrasentan (IC50)rifampin (IC50)
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)2.949
Caspase-1Homo sapiens (human)8.319
Alpha-synucleinHomo sapiens (human)7.1
Enoyl-[acyl-carrier-protein] reductase [NADH]Mycobacterium tuberculosis H37Rv0.03
DNA-directed RNA polymerase subunit betaMycobacterium tuberculosis H37Rv0.01
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.5
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.5

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Achari, R; Carr, RA; Doan, TT; Jankowski, JR; Katz, DA; Locke, CS; Sleep, DJ; Wang, P; Xiong, H1
Gordi, T1

Trials

1 trial(s) available for atrasentan and rifampin

ArticleYear
Dual effects of rifampin on the pharmacokinetics of atrasentan.
    Journal of clinical pharmacology, 2007, Volume: 47, Issue:4

    Topics: Adult; Area Under Curve; Atrasentan; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Synergism; Endothelin A Receptor Antagonists; Enzyme Induction; Half-Life; Humans; Male; Metabolic Clearance Rate; Middle Aged; Pyrrolidines; Rifampin

2007

Other Studies

1 other study(ies) available for atrasentan and rifampin

ArticleYear
Comments on "Dual effects of rifampin on the pharmacokinetics of atrasentan".
    Journal of clinical pharmacology, 2007, Volume: 47, Issue:9

    Topics: Area Under Curve; Atrasentan; Drug Interactions; Half-Life; Humans; Protein Binding; Pyrrolidines; Rifampin; Tissue Distribution

2007