Page last updated: 2024-09-04

atrasentan and arachidonic acid

atrasentan has been researched along with arachidonic acid in 2 studies

Compound Research Comparison

Studies
(atrasentan)
Trials
(atrasentan)
Recent Studies (post-2010)
(atrasentan)
Studies
(arachidonic acid)
Trials
(arachidonic acid)
Recent Studies (post-2010) (arachidonic acid)
3584110819,2954863,040

Protein Interaction Comparison

ProteinTaxonomyatrasentan (IC50)arachidonic acid (IC50)
60 kDa heat shock protein, mitochondrialHomo sapiens (human)4.5
Fatty acid-binding protein, adipocyteHomo sapiens (human)2.75
10 kDa heat shock protein, mitochondrialHomo sapiens (human)4.5
60 kDa chaperonin Escherichia coli7.3
10 kDa chaperonin Escherichia coli7.3
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.0715
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)0.6026

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adler, AL; Calzadilla, SV; Chiou, WJ; Dayton, BD; Dixon, DB; Gehrke, LJ; Hernandez, L; Magnuson, SR; Marsh, KC; Novosad, EI; Opgenorth, TJ; Von Geldern, TW; Wessale, JL; Winn, M; Wu-Wong, JR1
Chiou, WJ; Dixon, DB; Jae, HS; Liu, G; Opgenorth, TJ; Sorensen, BK; Tasker, A; von Geldern, TW; Winn, M; Wu-Wong, JR1

Other Studies

2 other study(ies) available for atrasentan and arachidonic acid

ArticleYear
Pharmacological characterization of A-127722: an orally active and highly potent ETA-selective receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Administration, Oral; Animals; Arachidonic Acid; Atrasentan; CHO Cells; Cricetinae; Dogs; Endothelin Receptor Antagonists; Female; Humans; Macaca fascicularis; Male; Phosphatidylinositols; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Stereoisomerism; Vasoconstriction

1996
Pharmacology of endothelin receptor antagonists ABT-627, ABT-546, A-182086 and A-192621: in vitro studies.
    Clinical science (London, England : 1979), 2002, Volume: 103 Suppl 48

    Topics: Animals; Arachidonic Acid; Atrasentan; Binding, Competitive; Cell Line; CHO Cells; Cricetinae; Endothelin Receptor Antagonists; Endothelin-1; Humans; Hydrolysis; Iodine Radioisotopes; Phosphatidylinositols; Pyrrolidines; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Sulfonamides; Transfection; Vasodilator Agents

2002