Page last updated: 2024-09-04

atazanavir sulfate and dolutegravir

atazanavir sulfate has been researched along with dolutegravir in 19 studies

Compound Research Comparison

Studies
(atazanavir sulfate)
Trials
(atazanavir sulfate)
Recent Studies (post-2010)
(atazanavir sulfate)
Studies
(dolutegravir)
Trials
(dolutegravir)
Recent Studies (post-2010) (dolutegravir)
1,1022465901,1281791,105

Protein Interaction Comparison

ProteinTaxonomyatazanavir sulfate (IC50)dolutegravir (IC50)
Chain A, PFV integraseHuman spumaretrovirus0.0517
Chain A, PFV integraseHuman spumaretrovirus0.0517
Chain A, PFV integraseHuman spumaretrovirus0.0517
Solute carrier family 22 member 2Homo sapiens (human)1.9
Integrase Human immunodeficiency virus 10.0414

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's12 (63.16)24.3611
2020's7 (36.84)2.80

Authors

AuthorsStudies
Borland, J; Chen, S; Lou, Y; Min, S; Peppercorn, A; Piscitelli, SC; Song, I; Wajima, T1
Amiel, C; Caseris, M; Charpentier, C; Descamps, D; Desnoyer, A; Farnoux, C; Lassel, L; Lê, MP; Pain, JB; Peytavin, G; Pialoux, G1
Jones, R; Levy, JB; Milburn, J1
Concia, E; Cucchetto, G; Lanzafame, M; Lattuada, E; Nicolè, S; Rigo, F; Vento, S1
Cattaneo, D; Clementi, E; Cozzi, V; Galli, M; Gervasoni, C; Meraviglia, P; Minisci, D; Riva, A1
Alnouti, Y; Bade, AN; Dash, PK; Edagwa, B; Gautam, N; Gelbard, HA; Gendelman, HE; Gnanadhas, DP; Gorantla, S; Lin, Z; McMillan, J; Mosley, RL; Palandri, DL; Sillman, B1
Ancona, G; Cannizzo, ES; Castagna, A; Galli, A; Galli, L; Gianotti, N; Marchetti, G; Merlini, E; Monforte, AD; Muccini, C; Tincati, C1
Baldin, G; Belmonti, S; Borghetti, A; Ciccullo, A; De Luca, A; Di Giambenedetto, S; Emiliozzi, A; Gagliardini, R; Lamonica, S; Lombardi, F; Montagnani, F; Moschese, D; Visconti, E1
Bonora, S; Carosella, S; Castagna, A; Cattelan, A; De Socio, GV; Di Giambenedetto, S; Galli, L; Gulminetti, R; Ladisa, N; Mazzola, G; Mena, M; Poli, A; Quiros-Roldan, ME; Riva, A; Rusconi, S1
Biasiotto, G; Bonito, A; Calza, S; Castelli, F; Quiros-Roldan, E; Vezzoli, M; Zanella, I1
Cenderello, G; Di Biagio, A; Magnasco, L; Rizzardini, G1
Castagna, A1
Atzori, C; Baldelli, S; Cattaneo, D; Cozzi, V; Filice, C; Fusi, M; Gervasoni, C; Micheli, V1
Cassola, G; Del Puente, F; Pontali, E; Torresin, A1
Auclair, M; Capeau, J; Fellahi, S; Garcia, M; Guénantin, AC1
Cazzaniga, A; Galli, M; Maier, J; Rusconi, S; Scrimieri, R1
Alimohamadi, Y; Fard, SR; Kalantari, S; Maleki, D; Minaeian, S; Taher, MT; Yassin, Z1
Brummel, SS; Chadwick, EG; Huo, Y; Jacobson, DL; Jao, J; Kacanek, D; Kahlert, CR; Patel, K; Powis, KM; Seage, GR; Shiau, S; Sultan-Beyer, L; Williams, PL; Yee, LM; Zash, R1
Bamford, A; Burger, DM; Bwakura-Dangarembizi, M; Chabala, C; Colbers, A; Denti, P; Doerholt, K; Gibb, DM; Griffiths, AL; Makumbi, S; McIlleron, HM; Monkiewicz, LN; Mulenga, V; Mumbiro, V; Musiime, V; Nangiya, J; Szubert, AJ; Waalewijn, H; Wasmann, RE; Wiesner, L1

Reviews

1 review(s) available for atazanavir sulfate and dolutegravir

ArticleYear
Renal effects of novel antiretroviral drugs.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 2017, 03-01, Volume: 32, Issue:3

    Topics: Adenine; Alanine; Anti-HIV Agents; Atazanavir Sulfate; Cobicistat; Creatinine; Disease Progression; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Oxazines; Piperazines; Proteinuria; Pyridones; Quinolones; Raltegravir Potassium; Renal Insufficiency, Chronic; Tenofovir

2017

Trials

3 trial(s) available for atazanavir sulfate and dolutegravir

ArticleYear
Effect of atazanavir and atazanavir/ritonavir on the pharmacokinetics of the next-generation HIV integrase inhibitor, S/GSK1349572.
    British journal of clinical pharmacology, 2011, Volume: 72, Issue:1

    Topics: Adolescent; Adult; Area Under Curve; Atazanavir Sulfate; Cross-Over Studies; Drug Administration Schedule; Drug Combinations; Drug Interactions; Female; Glucuronosyltransferase; Heterocyclic Compounds, 3-Ring; HIV Integrase Inhibitors; HIV Protease Inhibitors; Humans; Linear Models; Male; Middle Aged; Oligopeptides; Oxazines; Piperazines; Pyridines; Pyridones; Ritonavir; Young Adult

2011
Comparing the effectiveness of Atazanavir/Ritonavir/Dolutegravir/Hydroxychloroquine and Lopinavir/Ritonavir/Hydroxychloroquine treatment regimens in COVID-19 patients.
    Journal of medical virology, 2021, Volume: 93, Issue:12

    Topics: Antiviral Agents; Atazanavir Sulfate; COVID-19; COVID-19 Drug Treatment; Drug Combinations; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; Humans; Hydroxychloroquine; Lopinavir; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Ritonavir; Treatment Outcome

2021
First Pharmacokinetic Data of Tenofovir Alafenamide Fumarate and Tenofovir With Dolutegravir or Boosted Protease Inhibitors in African Children: A Substudy of the CHAPAS-4 Trial.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2023, 09-18, Volume: 77, Issue:6

    Topics: Adult; Anti-HIV Agents; Antiviral Agents; Atazanavir Sulfate; Child; Darunavir; Emtricitabine; Fumarates; HIV Infections; Humans; Lopinavir; Protease Inhibitors; Ritonavir; Tenofovir

2023

Other Studies

15 other study(ies) available for atazanavir sulfate and dolutegravir

ArticleYear
Pharmacokinetics of dolutegravir in a premature neonate after HIV treatment intensification during pregnancy.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:6

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Cytochrome P-450 CYP3A; Emtricitabine; Female; Glucuronosyltransferase; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Infant, Newborn; Male; Oxazines; Piperazines; Pregnancy; Pyridones; Ritonavir; Tenofovir

2015
Dolutegravir 50 mg thrice weekly plus atazanavir 400 mg daily in a long-term virologically suppressed HIV-infected patient.
    International journal of STD & AIDS, 2017, Volume: 28, Issue:7

    Topics: Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Middle Aged; Oxazines; Piperazines; Pyridones; Treatment Outcome; Viral Load

2017
Dolutegravir plasma concentrations according to companion antiretroviral drug: unwanted drug interaction or desirable boosting effect?
    Antiviral therapy, 2017, Volume: 22, Issue:4

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Biological Availability; CD4 Lymphocyte Count; Darunavir; Dideoxynucleosides; Drug Administration Schedule; Drug Combinations; Drug Dosage Calculations; Drug Interactions; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Lamivudine; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Retrospective Studies; Rilpivirine; Viral Load

2017
Autophagy facilitates macrophage depots of sustained-release nanoformulated antiretroviral drugs.
    The Journal of clinical investigation, 2017, Mar-01, Volume: 127, Issue:3

    Topics: Acquired Immunodeficiency Syndrome; Animals; Anti-Retroviral Agents; Atazanavir Sulfate; Autophagy; Basic Helix-Loop-Helix Leucine Zipper Transcription Factors; Female; Heterocyclic Compounds, 3-Ring; HIV-1; Humans; Macrophages; Male; Mice; Nanoparticles; Oxazines; Piperazines; Pyridines; Pyridones; Pyrroles

2017
Immune activation, inflammation and HIV DNA after 96 weeks of ATV/r monotherapy: a MODAt substudy.
    Antiviral therapy, 2018, Volume: 23, Issue:7

    Topics: Adult; Atazanavir Sulfate; DNA; Heterocyclic Compounds, 3-Ring; HIV; Humans; Inflammation; Oxazines; Piperazines; Pyridones

2018
Efficacy and tolerability of lamivudine plus dolutegravir compared with lamivudine plus boosted PIs in HIV-1 positive individuals with virologic suppression: a retrospective study from the clinical practice.
    BMC infectious diseases, 2019, Jan-17, Volume: 19, Issue:1

    Topics: Adult; Anti-HIV Agents; Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; Cohort Studies; Darunavir; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Seropositivity; HIV-1; Humans; Lamivudine; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Retrospective Studies; Ritonavir; Tenofovir; Treatment Outcome; Viral Load

2019
Switch to dolutegravir and unboosted atazanavir in HIV-1 infected patients with undetectable viral load and long exposure to antiretroviral therapy.
    AIDS (London, England), 2019, 06-01, Volume: 33, Issue:7

    Topics: Antiretroviral Therapy, Highly Active; Atazanavir Sulfate; CD4 Lymphocyte Count; Drug Substitution; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Kaplan-Meier Estimate; Male; Middle Aged; Oxazines; Piperazines; Pyridones; RNA, Viral; Treatment Outcome; Viral Load

2019
The impact of integrase inhibitor-based regimens on markers of inflammation among HIV naïve patients.
    Cytokine, 2020, Volume: 126

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Cytokines; Drug Therapy, Combination; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Inflammation; Male; Middle Aged; Oxazines; Piperazines; Pyridones; Quinolones; Raltegravir Potassium

2020
Response to letter to the editor: switch to dolutegravir and unboosted atazanavir.
    AIDS (London, England), 2019, 11-15, Volume: 33, Issue:14

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Viral Load

2019
Two-drug regimens with dolutegravir for maintaining viral suppression: looking at the right companion.
    AIDS (London, England), 2019, 11-15, Volume: 33, Issue:14

    Topics: Atazanavir Sulfate; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Viral Load

2019
Drug-Drug Interactions Between Antiretrovirals and Carbamazepine/Oxcarbazepine: A Real-Life Investigation.
    Therapeutic drug monitoring, 2020, Volume: 42, Issue:2

    Topics: Adult; Anti-Retroviral Agents; Anticonvulsants; Atazanavir Sulfate; Carbamazepine; Darunavir; Drug Interactions; Drug Monitoring; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Male; Middle Aged; Oxazines; Oxcarbazepine; Piperazines; Pyridones

2020
Long-term safety and efficacy of dolutegravir and unboosted atazanavir among experienced HIV-infected adults.
    AIDS (London, England), 2019, 12-01, Volume: 33, Issue:15

    Topics: Adult; Atazanavir Sulfate; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Oxazines; Piperazines; Pyridones; Viral Load

2019
HIV antiretroviral drugs, dolutegravir, maraviroc and ritonavir-boosted atazanavir use different pathways to affect inflammation, senescence and insulin sensitivity in human coronary endothelial cells.
    PloS one, 2020, Volume: 15, Issue:1

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Cells, Cultured; Comorbidity; Coronary Vessels; Endothelial Cells; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Insulin Resistance; Male; Maraviroc; NF-kappa B; Oxazines; Piperazines; Pyridones; Ritonavir; Signal Transduction; Sirtuin 1; Ubiquitin Thiolesterase

2020
Unveiling the basis of antiretroviral therapy-induced osteopenia: the effects of Dolutegravir, Darunavir and Atazanavir on osteogenesis.
    AIDS (London, England), 2021, 02-02, Volume: 35, Issue:2

    Topics: Anti-HIV Agents; Atazanavir Sulfate; Bone Diseases, Metabolic; Darunavir; Heterocyclic Compounds, 3-Ring; HIV Infections; Humans; Osteogenesis; Oxazines; Piperazines; Pyridones

2021
Dolutegravir in Pregnancy as Compared with Current HIV Regimens in the United States.
    The New England journal of medicine, 2022, 09-01, Volume: 387, Issue:9

    Topics: Adult; Anti-HIV Agents; Atazanavir Sulfate; Cobicistat; Cohort Studies; Darunavir; Female; Heterocyclic Compounds, 3-Ring; HIV Infections; HIV Protease Inhibitors; HIV-1; Humans; Infant, Newborn; Oxazines; Piperazines; Pregnancy; Premature Birth; Pyridones; Quinolones; Raltegravir Potassium; Rilpivirine; Ritonavir; United States

2022