Page last updated: 2024-09-04

atazanavir and pepstatin

atazanavir has been researched along with pepstatin in 2 studies

Compound Research Comparison

Studies
(atazanavir)
Trials
(atazanavir)
Recent Studies (post-2010)
(atazanavir)
Studies
(pepstatin)
Trials
(pepstatin)
Recent Studies (post-2010) (pepstatin)
751376960125

Protein Interaction Comparison

ProteinTaxonomyatazanavir (IC50)pepstatin (IC50)
Pepsin ASus scrofa (pig)0.011
ReninHomo sapiens (human)1.9333
Cathepsin DHomo sapiens (human)0.3597
Procathepsin LHomo sapiens (human)0.8
Cathepsin BHomo sapiens (human)4.26
Candidapepsin-2Candida albicans0.09
Pepsin A-5Homo sapiens (human)0.059
Cathepsin EHomo sapiens (human)0.5558
Plasmepsin-1Plasmodium falciparum (malaria parasite P. falciparum)0.0009
Plasmepsin-2Plasmodium falciparum (malaria parasite P. falciparum)0.0005
Cathepsin D Bos taurus (cattle)0.0235
Disintegrin and metalloproteinase domain-containing protein 9Homo sapiens (human)0.0563
Plasmepsin 4 Plasmodium falciparum (malaria parasite P. falciparum)0.0003
Cysteine proteaseLeishmania donovani0.16
Protease Human immunodeficiency virus 10.947

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Abbenante, G; Fairlie, DP; Leung, D1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Reviews

1 review(s) available for atazanavir and pepstatin

ArticleYear
Protease inhibitors: current status and future prospects.
    Journal of medicinal chemistry, 2000, Feb-10, Volume: 43, Issue:3

    Topics: Animals; Aspartic Acid Endopeptidases; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Humans; Metalloendopeptidases; Models, Molecular; Protease Inhibitors; Serine Endopeptidases; Serine Proteinase Inhibitors

2000

Other Studies

1 other study(ies) available for atazanavir and pepstatin

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023