Page last updated: 2024-09-05

asimadoline and naloxone

asimadoline has been researched along with naloxone in 5 studies

Compound Research Comparison

Studies
(asimadoline)
Trials
(asimadoline)
Recent Studies (post-2010)
(asimadoline)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
4391120,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomyasimadoline (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Binder, W; Walker, JS1
Gebhart, GF; Sengupta, JN; Snider, A; Su, X1
Gebhart, GF; Julia, V; Su, X1
Gebhart, GF; Ozaki, N; Sengupta, JN1
Ambriz-Tututi, M; Araiza-Saldaña, CI; Arreola-Espino, R; Bartoszyk, GD; Caram-Salas, NL; Cruz, SL; Granados-Soto, V; Reyes-García, G; Rocha-González, HI1

Other Studies

5 other study(ies) available for asimadoline and naloxone

ArticleYear
Effect of the peripherally selective kappa-opioid agonist, asimadoline, on adjuvant arthritis.
    British journal of pharmacology, 1998, Volume: 124, Issue:4

    Topics: Acetamides; Administration, Oral; Analgesics, Opioid; Animals; Arthritis, Experimental; Benzomorphans; Dose-Response Relationship, Drug; Male; Motor Activity; Naloxone; Narcotic Antagonists; Pain Measurement; Pyrrolidines; Quaternary Ammonium Compounds; Rats; Rats, Inbred Lew; Receptors, Opioid, kappa; Time Factors

1998
Effects of kappa opioids in the inflamed rat colon.
    Pain, 1999, Volume: 79, Issue:2-3

    Topics: Acetamides; Action Potentials; Analgesics, Opioid; Animals; Benzamides; Chronic Disease; Colitis; Colon; Electrophysiology; Male; Morphine; Naloxone; Narcotic Antagonists; Nerve Fibers; Neurons, Afferent; Pain Measurement; Piperazines; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Rectum; Trinitrobenzenesulfonic Acid

1999
Effects of intracolonic opioid receptor agonists on polymodal pelvic nerve afferent fibers in the rat.
    Journal of neurophysiology, 2000, Volume: 83, Issue:2

    Topics: Acetamides; Analgesics; Analgesics, Opioid; Animals; Benzamides; Colon; Fentanyl; Hot Temperature; Male; Naloxone; Narcotic Antagonists; Nerve Fibers; Neurons, Afferent; Peripheral Nerves; Physical Stimulation; Piperazines; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Spinal Nerve Roots

2000
Differential effects of mu-, delta-, and kappa-opioid receptor agonists on mechanosensitive gastric vagal afferent fibers in the rat.
    Journal of neurophysiology, 2000, Volume: 83, Issue:4

    Topics: Acetamides; Analgesics; Analgesics, Opioid; Animals; Benzamides; Catheterization; Electric Stimulation; Male; Mechanoreceptors; Morphine; Naloxone; Narcotic Antagonists; Nerve Fibers; Neurons, Afferent; Pain; Piperazines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stomach; Vagus Nerve

2000
Subcutaneous, intrathecal and periaqueductal grey administration of asimadoline and ICI-204448 reduces tactile allodynia in the rat.
    European journal of pharmacology, 2007, Nov-14, Volume: 573, Issue:1-3

    Topics: Acetamides; Animals; Dose-Response Relationship, Drug; Female; Injections, Spinal; Injections, Subcutaneous; Ligation; Lumbosacral Plexus; Male; Naloxone; Pain Threshold; Periaqueductal Gray; Peripheral Nervous System Diseases; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Somatosensory Disorders; Time Factors

2007