Page last updated: 2024-09-05

asimadoline and levodopa

asimadoline has been researched along with levodopa in 2 studies

Compound Research Comparison

Studies
(asimadoline)
Trials
(asimadoline)
Recent Studies (post-2010)
(asimadoline)
Studies
(levodopa)
Trials
(levodopa)
Recent Studies (post-2010) (levodopa)
4391117,7741,9004,946

Protein Interaction Comparison

ProteinTaxonomyasimadoline (IC50)levodopa (IC50)
integrase, partialHuman immunodeficiency virus 10.5939
lens epithelium-derived growth factor p75Homo sapiens (human)0.5939
Epidermal growth factor receptorHomo sapiens (human)2.88
Tyrosine-protein kinase LckHomo sapiens (human)3.729
Tyrosine-protein kinase FynHomo sapiens (human)2.146
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)2.258

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Barber, A; Bartoszyk, GD; Gottschlich, R; Seyfried, CA1

Other Studies

2 other study(ies) available for asimadoline and levodopa

ArticleYear
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
The peripherally acting kappa-opiate agonist EMD 61753 and analogues: opioid activity versus peripheral selectivity.
    Drugs under experimental and clinical research, 1995, Volume: 21, Issue:5

    Topics: Acetamides; Analgesics, Opioid; Animals; Cerebellum; Dopamine Antagonists; Guinea Pigs; Haloperidol; Levodopa; Male; Nucleus Accumbens; Peripheral Nervous System; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa

1995