Page last updated: 2024-09-03

asi-222 and digoxin

asi-222 has been researched along with digoxin in 9 studies

Compound Research Comparison

Studies
(asi-222)
Trials
(asi-222)
Recent Studies (post-2010)
(asi-222)
Studies
(digoxin)
Trials
(digoxin)
Recent Studies (post-2010) (digoxin)
160111,4839581,289

Protein Interaction Comparison

ProteinTaxonomyasi-222 (IC50)digoxin (IC50)
STAT3, partialHomo sapiens (human)1.862
Sodium/potassium-transporting ATPase subunit alpha-1 Homo sapiens (human)0.32
Sodium/potassium-transporting ATPase subunit beta-1Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-2Rattus norvegicus (Norway rat)0.22
Sodium/potassium-transporting ATPase subunit alpha-3 Rattus norvegicus (Norway rat)0.22
Sodium/potassium-transporting ATPase subunit beta-1 Rattus norvegicus (Norway rat)0.0055
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 20.19
Sodium/potassium-transporting ATPase subunit alpha-3Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit beta-2Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-2Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-1Canis lupus familiaris (dog)0.5
Nuclear receptor ROR-gammaHomo sapiens (human)3.4798
Sodium/potassium-transporting ATPase subunit beta-3Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit gammaHomo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-4Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-4Rattus norvegicus (Norway rat)0.0055
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.2359

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19906 (66.67)18.7374
1990's3 (33.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Greenblatt, DJ; Lloyd, BL; Mudge, GH; Smith, TW1
Caldwell, RW; Cook, LS; Nash, CB1
Caldwell, RW; Rebagay, WR3
Caldwell, RW; Gunter, JL; Songu-Mize, E1
Caldwell, RW; Nash, CB1
Caldwell, RW; Elam, JT; Nash, CB; Songu-Mize, E1
Caldwell, RW; Cook, LS; Doherty, JE; Nash, CB; Straub, KD1

Other Studies

9 other study(ies) available for asi-222 and digoxin

ArticleYear
Inotropic and toxic effects of a polar cardiac glycoside derivative in the dog.
    Circulation research, 1978, Volume: 43, Issue:6

    Topics: Aminoglycosides; Animals; Blood-Brain Barrier; Brain; Digitoxigenin; Digoxin; Dogs; Dose-Response Relationship, Drug; Heart Conduction System; Injections, Intravenous; Male; Methods; Myocardial Contraction; Radioimmunoassay

1978
Comparison of the cardiac effects of ASI-222 HCl, an aminosugar cardiac glycoside, and digoxin.
    Archives internationales de pharmacodynamie et de therapie, 1977, Volume: 227, Issue:2

    Topics: Aminoglycosides; Animals; Blood Pressure; Cardiac Output; Central Venous Pressure; Digitalis Glycosides; Digitoxigenin; Digoxin; Dogs; Female; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Rabbits; Time Factors; Vagotomy

1977
Effects of sinoaortic denervation on the reflex actions of digoxin and a polar aminocardenolide.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:1

    Topics: Animals; Blood Pressure; Cardiac Glycosides; Denervation; Digitoxigenin; Digoxin; Dobutamine; Dogs; Heart Rate; Nerve Endings; Neurons, Afferent; Ouabain; Pressoreceptors; Reflex; Sinoatrial Node; Sympathetic Nervous System; Vagus Nerve

1992
Effect of transient vagal cold blockade upon reflex actions of a polar and nonpolar cardiac glycoside.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Atropine; Cold Temperature; Digitoxigenin; Digoxin; Dogs; Female; Hemodynamics; Infusions, Intravenous; Male; Nerve Block; Reflex; Sympathetic Nervous System; Vagus Nerve

1992
Different patterns of autonomic nerve activity produced by a polar vs. a neutral cardiac glycoside.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Animals; Autonomic Nervous System; Blood Pressure; Cardiac Glycosides; Digitoxigenin; Digoxin; Dogs; Female; Heart; Heart Rate; Male; Pressoreceptors; Reflex; Sympathetic Nervous System; Vagus Nerve

1990
Comparative ability of digoxin and an aminosugar cardiac glycoside to bind to and inhibit Na+,K+-adenosine triphosphatase. Effect of potassium.
    Biochemical pharmacology, 1989, Nov-01, Volume: 38, Issue:21

    Topics: Animals; Binding Sites; Binding, Competitive; Cardiac Glycosides; Digitoxigenin; Digoxin; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Kinetics; Myocardium; Potassium; Sodium-Potassium-Exchanging ATPase

1989
Effect of an aminocardenolide and digoxin upon atrioventricular refractory period in the dog.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Atrioventricular Node; Atropine; Digitoxigenin; Digoxin; Dogs; Female; Heart Conduction System; Male; Metoprolol; Neural Conduction; Pressoreceptors; Refractory Period, Electrophysiological; Sympathectomy

1985
Metabolism and cardiac actions of a polar aminocardenolide and digoxin in the conscious dog.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:1

    Topics: Animals; Blood Pressure; Digitoxigenin; Digoxin; Dogs; Feces; Female; Heart; Heart Rate; Kinetics; Male; Myocardial Contraction

1983
Adrenergic and cholinergic mechanisms in digitalis inotropy.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:3

    Topics: Animals; Blood Pressure; Digitalis Glycosides; Digitoxigenin; Digoxin; Dogs; Female; Heart; Heart Rate; Male; Myocardial Contraction; Parasympathetic Nervous System; Sympathetic Nervous System

1982