Page last updated: 2024-09-04

asenapine and ziprasidone

asenapine has been researched along with ziprasidone in 6 studies

Compound Research Comparison

Studies
(asenapine)
Trials
(asenapine)
Recent Studies (post-2010)
(asenapine)
Studies
(ziprasidone)
Trials
(ziprasidone)
Recent Studies (post-2010) (ziprasidone)
265502091,068254362

Protein Interaction Comparison

ProteinTaxonomyasenapine (IC50)ziprasidone (IC50)
D(2) dopamine receptorHomo sapiens (human)0.005
Aspartate aminotransferase, cytoplasmicHomo sapiens (human)5.39
DRattus norvegicus (Norway rat)0.1514
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.1514
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.1514
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.1514
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.1514
Alpha-1D adrenergic receptorHomo sapiens (human)0.011
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0004
Alpha-1A adrenergic receptorHomo sapiens (human)0.011
Alpha-1B adrenergic receptorHomo sapiens (human)0.011
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.2301

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (33.33)18.2507
2000's1 (16.67)29.6817
2010's2 (33.33)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
De Loore, K; Gommeren, W; Janssen, PF; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van Gompel, P1
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
Shahid, M; Walker, GB; Wong, EH; Zorn, SH1
Chennoufi, L; Cheour, M; Ouanes, S1
Morrissette, DA; Stahl, SM1
Cao, D; Hong, Y; Huang, W; Wang, L; Wei, H; Xu, J; Zhang, J1

Reviews

3 review(s) available for asenapine and ziprasidone

ArticleYear
An update on the treatment of mixed bipolar states: what is new in 2013?
    Journal of affective disorders, 2014, Volume: 158

    Topics: Antipsychotic Agents; Aripiprazole; Benzodiazepines; Bipolar Disorder; Calcitonin; Dibenzocycloheptenes; Heterocyclic Compounds, 4 or More Rings; Humans; Olanzapine; Piperazines; Quinolones; Randomized Controlled Trials as Topic; Thiazoles; Treatment Outcome

2014
Treating the violent patient with psychosis or impulsivity utilizing antipsychotic polypharmacy and high-dose monotherapy.
    CNS spectrums, 2014, Volume: 19, Issue:5

    Topics: Antipsychotic Agents; Aripiprazole; Benzodiazepines; Brain; Clozapine; Dibenzocycloheptenes; Drug Therapy, Combination; Heterocyclic Compounds, 4 or More Rings; Humans; Impulsive Behavior; Isoxazoles; Lurasidone Hydrochloride; Olanzapine; Paliperidone Palmitate; Piperazines; Piperidines; Polypharmacy; Psychotic Disorders; Quetiapine Fumarate; Receptors, Dopamine D2; Risperidone; Thiazoles; Violence

2014
A cumulative Bayesian network meta-analysis on the comparative efficacy of pharmacotherapies for mania over the last 40 years.
    Psychopharmacology, 2022, Volume: 239, Issue:10

    Topics: Adult; Antimanic Agents; Antipsychotic Agents; Aripiprazole; Benzodiazepines; Carbamazepine; Dibenzocycloheptenes; Haloperidol; Humans; Lithium; Mania; Network Meta-Analysis; Olanzapine; Paliperidone Palmitate; Pharmaceutical Preparations; Piperazines; Quetiapine Fumarate; Risperidone; Tamoxifen; Thiazoles; Valproic Acid

2022

Other Studies

3 other study(ies) available for asenapine and ziprasidone

ArticleYear
Risperidone compared with new and reference antipsychotic drugs: in vitro and in vivo receptor binding.
    Psychopharmacology, 1996, Volume: 124, Issue:1-2

    Topics: Animals; Antipsychotic Agents; Brain; Cells, Cultured; Clozapine; Haloperidol; Humans; Male; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Serotonin; Risperidone

1996
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
    European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3

    Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes

1998
Asenapine: a novel psychopharmacologic agent with a unique human receptor signature.
    Journal of psychopharmacology (Oxford, England), 2009, Volume: 23, Issue:1

    Topics: Benzodiazepines; Bipolar Disorder; Clinical Trials as Topic; Cloning, Molecular; Clozapine; Dibenzocycloheptenes; Heterocyclic Compounds, 4 or More Rings; Histamine Release; Humans; Inhibitory Concentration 50; Molecular Structure; Olanzapine; Psychotropic Drugs; Radioligand Assay; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, Serotonin; Schizophrenia; Substrate Specificity

2009