Page last updated: 2024-09-03

as 35 and pyrimidinones

as 35 has been researched along with pyrimidinones in 9 studies

Compound Research Comparison

Studies
(as 35)
Trials
(as 35)
Recent Studies (post-2010)
(as 35)
Studies
(pyrimidinones)
Trials
(pyrimidinones)
Recent Studies (post-2010) (pyrimidinones)
9006,0596042,692

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (88.89)18.2507
2000's1 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Horiba, M; Inoue, K; Ohata, K; Ohkawa, E; Watanabe-Kohno, S; Yamamura, H; Yasui, K1
Kasai, H; Kawashima, T; Omura, S; Yanagihara, Y1
Kasai, H; Yanagihara, Y1
Bando, T; Fujimura, M; Matsuda, T; Mizuhashi, K1
Honma, M; Shibasaki, A; Takata, H; Takishima, T; Tamura, G1
Iwakaji, A; Iwamoto, I; Kawashima, T; Nagaki, S; Tomioka, H; Yoshida, S1
Bando, T; Fujimura, M; Kurashima, K; Matsuda, T; Nishi, K; Saito, M; Shintani, H1
Fujimura, M; Matsuda, T; Ogawa, H; Saito, M1
Hamasaki, Y; Hayasaki, R; Ichimaru, T; Kobayashi, I; Matsuo, M; Miyazaki, M; Miyazaki, S; Muro, E; Tsuji, K; Yamamoto, S; Zaitu, M1

Other Studies

9 other study(ies) available for as 35 and pyrimidinones

ArticleYear
Effect of AS-35 on agonist-induced contractions and the resting tonus of airway smooth muscles and the in vitro release of chemical mediators from passively sensitized lung fragments from humans and guinea pigs.
    Japanese journal of pharmacology, 1992, Volume: 59, Issue:2

    Topics: Animals; Chromones; Guinea Pigs; Histamine Release; Humans; In Vitro Techniques; Leukotrienes; Lung; Male; Muscle Contraction; Muscle, Smooth; Passive Cutaneous Anaphylaxis; Pyridines; Pyrimidinones; Respiratory Muscles; SRS-A; Tetrazoles

1992
Peptide leukotriene antagonistic activity of AS-35, a new antiallergic drug.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:4

    Topics: Animals; Bronchoconstriction; Capillary Permeability; Chromones; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Leukotriene Antagonists; Leukotrienes; Male; Muscle, Smooth; Pyridines; Pyrimidinones; Rats; Tetrazoles; Trachea

1992
Inhibition of radiolabeled leukotriene-binding by AS-35 in guinea pig lung membrane fraction.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:4

    Topics: Animals; Binding Sites; Chromatography, High Pressure Liquid; Guinea Pigs; In Vitro Techniques; Leukotrienes; Lung; Male; Membranes; Pyridines; Pyrimidinones; Radioligand Assay; Tetrazoles; Tritium

1992
Interaction of thromboxane A2 and leukotrienes in guinea pig airways in vivo.
    Prostaglandins, 1991, Volume: 42, Issue:4

    Topics: Administration, Inhalation; Animals; Asthma; Bridged Bicyclo Compounds; Bronchoconstriction; Dose-Response Relationship, Drug; Fatty Acids, Monounsaturated; Guinea Pigs; Histamine; Male; Pyridines; Pyrimidines; Pyrimidinones; Receptors, Immunologic; Receptors, Leukotriene; Receptors, Prostaglandin; Receptors, Thromboxane; SRS-A; Tetrazoles; Thromboxane A2

1991
[Effect of AS-35 aerosol on bronchoconstriction induced by specific antigens in macacus rhesus monkeys].
    Arerugi = [Allergy], 1993, Volume: 42, Issue:7

    Topics: Aerosols; Allergens; Animals; Bronchoconstriction; Bronchodilator Agents; Female; Histamine Release; Macaca mulatta; Pyridines; Pyrimidinones; Tetrazoles

1993
[Inhibitory effect of AS-35. a novel antiallergic drug, on chemical mediator release from human eosinophils].
    Arerugi = [Allergy], 1994, Volume: 43, Issue:11

    Topics: Cells, Cultured; Eosinophil Peroxidase; Eosinophils; Humans; Hypersensitivity; Leukotriene C4; Peroxidases; Pyridines; Pyrimidinones; Tetrazoles

1994
Inhibitory effect of aerosol administration of a sulfidopeptide leukotriene antagonist on bronchoconstriction induced by antigen inhalation in guinea pigs.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:6

    Topics: Administration, Inhalation; Aerosols; Animals; Antigens; Bronchoconstriction; Bronchodilator Agents; Guinea Pigs; Histamine Antagonists; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Ovalbumin; Pyridines; Pyrimidinones; Respiratory Hypersensitivity; Tetrazoles

1994
Role of leukotrienes and platelet activating factor in allergic bronchoconstriction and their interactions in guinea pig airway in vivo.
    Prostaglandins, leukotrienes, and essential fatty acids, 1993, Volume: 49, Issue:2

    Topics: Animals; Asthma; Azepines; Bronchoconstriction; Bronchodilator Agents; Guinea Pigs; Leukotriene Antagonists; Leukotrienes; Male; Platelet Activating Factor; Pyridines; Pyrimidinones; Respiratory Hypersensitivity; Tetrazoles; Triazoles

1993
(9-[4-acetyl-3-hydroxy-2-n-propylphenoxy) methyl]-3-(1H-tetrazol-5-yl)-4H-pyrido [1,2-a] pyrimidin-4-one), AS-35, inhibits leukotriene synthesis.
    International journal of immunopharmacology, 2000, Volume: 22, Issue:7

    Topics: Animals; Arachidonic Acid; beta-N-Acetylhexosaminidases; Cell-Free System; Cytosol; Leukotriene A4; Leukotriene Antagonists; Leukotriene B4; Leukotriene C4; Phospholipases A; Pyridines; Pyrimidinones; Rats; Substrate Specificity; Tetrazoles; Tumor Cells, Cultured

2000