Page last updated: 2024-08-26

artenimol and artesunate

artenimol has been researched along with artesunate in 40 studies

Research

Studies (40)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	2 (5.00)	18.2507
2000's	3 (7.50)	29.6817
2010's	28 (70.00)	24.3611
2020's	7 (17.50)	2.80

Authors

Authors	Studies
Kong, L; Li, Y; Liu, H; Liu, X; Wang, LL; Yuan, F; Zhang, L; Zhang, Y; Zuo, Z	1
Benedetti, P; Bizzarri, BM; Botta, L; Cesarini, S; Cirigliano, A; Filippi, S; Fiorucci, D; Negri, R; Paiardini, A; Rinaldi, T; Saladino, R; Zippilli, C	1
Avery, V; Derese, S; Deyou, T; Duffy, S; Erdélyi, M; Fitzpatrick, PA; Gruhonjic, A; Gumula, I; Heydenreich, M; Holleran, J; Landberg, G; Mumo, M; Pang, F; Rissanen, K; Yenesew, A	1
Combrinck, J; de Kock, C; N'Da, DD; Smit, FJ; Smith, PJ; Zuma, NH	1
Dong, G; Liu, N; Sheng, C; Wang, Y; Wu, S	1
Avery, VM; Carroll, AR; Duffy, S; Robertson, LP; Wang, D; Wang, Y	1
Çapcı Karagöz, A; Efferth, T; Friedrich, O; Gruber, L; Hahn, F; Hampel, F; Kappes, B; Klein, V; Leidenberger, M; Marschall, M; Reiter, C; Seo, EJ; Tsogoeva, SB	1
Friedrich, O; Hahn, F; Hampel, F; Kappes, B; Karagöz, AÇ; Leidenberger, M; Marschall, M; Tsogoeva, SB	1
Chang, L; Ding, C; Feng, LS; Gao, C; Wu, X; Xu, Z; Yan, XF; Zhao, F	1
Avery, VM; Butler, GS; Drinkwater, N; Duffy, S; Grin, PM; Kassiou, M; Lucantoni, L; Malcolm, TR; McGowan, S; Overall, CM; Scammells, PJ; Vinh, NB	1
Avery, VM; Baell, JB; Ban, K; Beveridge, JG; Blundell, S; Charman, SA; Chavchich, M; Chiu, FCK; Creek, D; Cuellar, ME; Dahlin, JL; Diab, S; Dingjan, T; Duffy, S; Edstein, MD; Ellis, K; Fletcher, S; Harjani, JR; Huang, F; Lucantoni, L; Marfurt, J; Noviyanti, R; Price, RN; Ralph, SA; Shi, DH; Strasser, JM; Teguh, S; Walters, MA; Wirjanata, G; Xue, L	1
Avery, VM; Carroll, AR; Duffy, S; Lucantoni, L; Robertson, LP	1
Das, D; Hong, J	1
Liu, Y; Xu, Z; Zhao, SJ	1
Emami, SA; Taleghani, A; Tayarani-Najaran, Z	1
Avery, VM; Duffy, S; Erdélyi, M; Lindblad, S; Maeda, G; Munissi, JJE; Nyandoro, SS; Pelletier, J	1
Avery, VM; Challis, MP; Creek, DJ; De Paoli, A; Devine, SM; Kigotho, JK; MacRaild, CA; Norton, RS; Scammells, PJ; Siddiqui, G	1
Brun, R; Charman, SA; Charman, WN; Chiu, FC; Chollet, J; Dong, Y; Dorn, A; Karle, JM; Matile, H; Santo Tomas, J; Scheurer, C; Scorneaux, B; Snyder, C; Tang, Y; Urwyler, H; Vennerstrom, JL; Wang, X; Wittlin, S	1
Charman, SA; Charman, WN; Chiu, FC; Creek, DJ; Dong, Y; Prankerd, RJ; Vennerstrom, JL	1
Gottstein, B; Hemphill, A; Keiser, J; Lany, C; Ortega-Mora, LM; Roethlisberger, C; Spicher, M; Stadelmann, B	1
Brun, R; Charman, SA; Charman, WN; Chollet, J; Creek, DJ; Dong, Y; Dorn, A; Koltun, M; Matile, H; Morizzi, J; Padmanilayam, M; Santo Tomas, J; Scheurer, C; Snyder, C; Sriraghavan, K; Tang, Y; Urwyler, H; Vennerstrom, JL; Wang, X; Wittlin, S	1
Charman, SA; Charman, WN; Chiu, FC; Chollet, J; Dong, Y; Dorn, A; Johnson, LM; Matile, H; Morizzi, J; Scheurer, C; Snyder, C; Tang, Y; Tomas, JS; Urwyler, H; Vennerstrom, JL; Wittlin, S; Zhou, L	1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ	1
Biagini, GA; Chandramohanadas, R; Darling, C; DeGrado, WF; Diamond, SL; Fisher, N; Greenbaum, DC; Jing, H; Jo, H; Lucumi, E; Napper, AD; Shone, AE; Ward, SA	1
Fidock, DA; Krishna, S; Scanfeld, D; Uhlemann, AC; Valderramos, SG	1
Biamonte, MA; Le Roch, KG; Wanner, J	1
Alvarez, M; Blazquez, AG; Efferth, T; Fernandez-Dolon, M; Gomez-San Miguel, AB; Jansen, H; Maestre, AD; Marin, JJ; Romero, MR; Sanchez-Vicente, L; Serrano, MA	1
Fidock, DA; Flannery, EL; Winzeler, EA	1
Avery, VM; Sykes, ML	1
Amewu, RK; Burrell-Saward, H; Chadwick, J; Hussain, A; Janneh, O; Miguel, C; O'Neill, PM; Panda, S; Rinki, R; Vivas, L; Ward, SA	1
Cloete, TT; de Kock, C; N'Da, DD; Smith, PJ	1
Bathurst, I; Burrows, JN; Charman, SA; Cross, RM; Flanigan, DL; Fronczek, FR; Guida, WC; Kyle, DE; LaCrue, AN; Maignan, JR; Manetsch, R; Monastyrskyi, A; Mutka, TS; Sáenz, FE; Shackleford, DM; White, KL; Wojtas, L	1
Birkholtz, LM; N'Da, DD; Smit, FJ; van Biljon, RA	1
Efferth, T; Friedrich, O; Fröhlich, T; Gruber, L; Hutterer, C; Kappes, B; Marschall, M; Reiter, C; Tsogoeva, SB; Voigtländer, C	1
Brewer, TG; Fleckenstein, LL; Heiffer, MH; Li, QG; Masonic, K; Peggins, JO	1
Abdullah, MN; Akbar, A; Mansor, SM; Mordi, MN; Navaratnam, V	1
Belmudes, L; Couté, Y; Friedrich, O; Fröhlich, T; Hahn, F; Kappes, B; Leidenberger, M; Marschall, M; Tsogoeva, SB	1
Boaventura, S; Cass, QB; Oliveira, ASS; Rath, S; Rodrigues, MVN; Rodrigues-Silva, C	1
Boaventura, S; Gadelha, FR; Garcia, VL; Grazzia, N; Miguel, DC	1
Baratto, MC; Bizzarri, BM; Botta, L; Cesarini, S; Filippi, S; Pogni, R; Saladino, R; Zippilli, C	1

Reviews

8 review(s) available for artenimol and artesunate

Article	Year
Tackling Fungal Resistance by Biofilm Inhibitors. Journal of medicinal chemistry, 2017, 03-23, Volume: 60, Issue:6 Topics: Animals; Antifungal Agents; Biofilms; Drug Discovery; Drug Resistance, Fungal; Fungi; Humans; Models, Molecular; Mycoses; Small Molecule Libraries	2017
Recent advances of tetrazole derivatives as potential anti-tubercular and anti-malarial agents. European journal of medicinal chemistry, 2019, Feb-01, Volume: 163 Topics: Animals; Antimalarials; Antitubercular Agents; Humans; Structure-Activity Relationship; Tetrazoles	2019
Recent advancements of 4-aminoquinazoline derivatives as kinase inhibitors and their applications in medicinal chemistry. European journal of medicinal chemistry, 2019, May-15, Volume: 170 Topics: Animals; Antineoplastic Agents; Chemistry Techniques, Synthetic; Humans; Neoplasms; Protein Kinase Inhibitors; Quinazolines	2019
1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships. European journal of medicinal chemistry, 2019, Dec-01, Volume: 183 Topics: Antineoplastic Agents; Humans; Molecular Structure; Neoplasms; Structure-Activity Relationship; Triazoles	2019
Artemisia: a promising plant for the treatment of cancer. Bioorganic & medicinal chemistry, 2020, 01-01, Volume: 28, Issue:1 Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisia; Cell Proliferation; Humans; Molecular Structure; Neoplasms; Neoplasms, Experimental; Plant Extracts; Plants, Medicinal	2020
Recent advances in malaria drug discovery. Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10 Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure	2013
Using genetic methods to define the targets of compounds with antimalarial activity. Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20 Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum	2013
Approaches to protozoan drug discovery: phenotypic screening. Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20 Topics: Drug Discovery; Humans; Molecular Structure; Neglected Diseases; Phenotype; Plasmodium falciparum; Protozoan Infections; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma cruzi	2013

Other Studies

32 other study(ies) available for artenimol and artesunate

Article	Year
Design and synthesis of novel artemisinin derivatives with potent activities against colorectal cancer in vitro and in vivo. European journal of medicinal chemistry, 2019, Nov-15, Volume: 182 Topics: Animals; Antineoplastic Agents; Artemisinins; Cell Proliferation; Cell Survival; Colorectal Neoplasms; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Female; HCT116 Cells; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Molecular Structure; Neoplasms, Experimental; Structure-Activity Relationship; Tumor Cells, Cultured	2019
Artemisinin Derivatives with Antimelanoma Activity Show Inhibitory Effect against Human DNA Topoisomerase 1. ACS medicinal chemistry letters, 2020, May-14, Volume: 11, Issue:5 Topics:	2020
Rotenoids, Flavonoids, and Chalcones from the Root Bark of Millettia usaramensis. Journal of natural products, 2015, Dec-24, Volume: 78, Issue:12 Topics: Antimalarials; Chalcones; Chloroquine; Crystallography, X-Ray; Flavanones; Flavonoids; HEK293 Cells; Humans; Millettia; Molecular Conformation; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Plant Bark; Plant Extracts; Plasmodium falciparum	2015
Synthesis and biological evaluation of a series of non-hemiacetal ester derivatives of artemisinin. European journal of medicinal chemistry, 2016, Oct-21, Volume: 122 Topics: Animals; Antineoplastic Agents; Antiprotozoal Agents; Artemisinins; Cell Line, Tumor; Chemistry Techniques, Synthetic; CHO Cells; Cricetinae; Cricetulus; Drug Design; Esters; Humans; Plasmodium falciparum	2016
Pimentelamines A-C, Indole Alkaloids Isolated from the Leaves of the Australian Tree Flindersia pimenteliana. Journal of natural products, 2017, 12-22, Volume: 80, Issue:12 Topics: Antimalarials; Australia; Biological Products; Indole Alkaloids; Magnetic Resonance Spectroscopy; Plant Extracts; Plant Leaves; Plasmodium falciparum; Rutaceae; Trees	2017
Access to new highly potent antileukemia, antiviral and antimalarial agents via hybridization of natural products (homo)egonol, thymoquinone and artemisinin. Bioorganic & medicinal chemistry, 2018, 07-23, Volume: 26, Issue:12 Topics: Animals; Anisoles; Antimalarials; Antineoplastic Agents; Antiviral Agents; Artemisinins; Benzofurans; Benzoquinones; Biological Products; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; Cytomegalovirus; Humans; Molecular Conformation; Plasmodium falciparum	2018
Synthesis of new betulinic acid/betulin-derived dimers and hybrids with potent antimalarial and antiviral activities. Bioorganic & medicinal chemistry, 2019, 01-01, Volume: 27, Issue:1 Topics: Antimalarials; Antiviral Agents; Artemisinins; Cytomegalovirus; Ferrous Compounds; Fibroblasts; Humans; Parasitic Sensitivity Tests; Plasmodium falciparum; Triterpenes	2019
Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases. Journal of medicinal chemistry, 2019, 01-24, Volume: 62, Issue:2 Topics: Aminopeptidases; Antimalarials; Binding Sites; Catalytic Domain; Cell Survival; Drug Resistance; HEK293 Cells; Humans; Hydroxamic Acids; Molecular Docking Simulation; Plasmodium; Protease Inhibitors; Protozoan Proteins; Structure-Activity Relationship	2019
3,3'-Disubstituted 5,5'-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity. Journal of medicinal chemistry, 2019, 03-14, Volume: 62, Issue:5 Topics: Animals; Antimalarials; Chloroquine; Drug Resistance; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Mice; Molecular Structure; Plasmodium; Species Specificity; Structure-Activity Relationship; Triazines	2019
Acrotrione: An Oxidized Xanthene from the Roots of Acronychia pubescens. Journal of natural products, 2019, 04-26, Volume: 82, Issue:4 Topics: Oxidation-Reduction; Plant Roots; Rutaceae; Xanthenes	2019
A Meroisoprenoid, Heptenolides, and Journal of natural products, 2020, 02-28, Volume: 83, Issue:2 Topics: Annonaceae; Antimalarials; Flavanones; Flavonoids; HEK293 Cells; Humans; Molecular Structure; Plant Extracts; Plant Leaves; Plasmodium berghei; Plasmodium falciparum	2020
Discovery and development of 2-aminobenzimidazoles as potent antimalarials. European journal of medicinal chemistry, 2021, Oct-05, Volume: 221 Topics: Antimalarials; Benzimidazoles; Dose-Response Relationship, Drug; Drug Discovery; HEK293 Cells; Humans; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship	2021
Spiro and dispiro-1,2,4-trioxolanes as antimalarial peroxides: charting a workable structure-activity relationship using simple prototypes. Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15 Topics: Adamantane; Animals; Antimalarials; Cell Line, Tumor; Drug Resistance; Half-Life; Malaria; Malaria, Falciparum; Mice; Micronucleus Tests; Ozone; Peroxides; Plasmodium berghei; Rats; Spiro Compounds; Structure-Activity Relationship	2005
Relationship between antimalarial activity and heme alkylation for spiro- and dispiro-1,2,4-trioxolane antimalarials. Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:4 Topics: Alkylation; Animals; Antimalarials; Artemisinins; Heme; Humans; Kinetics; Parasitic Sensitivity Tests; Plasmodium falciparum; Spiro Compounds; Structure-Activity Relationship	2008
In vitro and in vivo treatments of echinococcus protoscoleces and metacestodes with artemisinin and artemisinin derivatives. Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:9 Topics: Albendazole; Animals; Anti-Infective Agents; Antiparasitic Agents; Artemisinins; Drug Therapy, Combination; Echinococcosis; Echinococcus granulosus; Echinococcus multilocularis; Humans; Larva; Mice; Mice, Inbred BALB C; Nitro Compounds; Parasitic Sensitivity Tests; Thiazoles; Treatment Outcome	2008
The structure-activity relationship of the antimalarial ozonide arterolane (OZ277). Journal of medicinal chemistry, 2010, Jan-14, Volume: 53, Issue:1 Topics: Animals; Antimalarials; Heterocyclic Compounds, 1-Ring; Malaria, Falciparum; Mice; Molecular Conformation; Parasitic Sensitivity Tests; Peroxides; Plasmodium falciparum; Spiro Compounds; Stereoisomerism; Structure-Activity Relationship	2010
The comparative antimalarial properties of weak base and neutral synthetic ozonides. Bioorganic & medicinal chemistry letters, 2010, Jan-15, Volume: 20, Issue:2 Topics: Animals; Antimalarials; Heterocyclic Compounds; Mice; Plasmodium falciparum; Rats	2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species. Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6 Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics	2010
Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay. Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:9 Topics: Animals; Antimalarials; Drug Resistance, Multiple; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum	2010
Investigations into the role of the Plasmodium falciparum SERCA (PfATP6) L263E mutation in artemisinin action and resistance. Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:9 Topics: Animals; Antimalarials; Artemisinins; Inhibitory Concentration 50; Malaria, Falciparum; Mutation; Plasmodium falciparum; Reverse Transcriptase Polymerase Chain Reaction; Sarcoplasmic Reticulum Calcium-Transporting ATPases	2010
Novel artemisinin derivatives with potential usefulness against liver/colon cancer and viral hepatitis. Bioorganic & medicinal chemistry, 2013, Jul-15, Volume: 21, Issue:14 Topics: Animals; Artemisinins; Cell Line, Tumor; Cell Proliferation; Cell Survival; Colonic Neoplasms; Hepatitis, Viral, Human; Humans; Liver Neoplasms; Molecular Structure; Virus Replication	2013
Synthesis and evaluation of the antimalarial, anticancer, and caspase 3 activities of tetraoxane dimers. Bioorganic & medicinal chemistry, 2013, Dec-01, Volume: 21, Issue:23 Topics: Antimalarials; Antineoplastic Agents; Caspase 3; Cell Line, Tumor; Dimerization; Humans; Malaria, Falciparum; Neoplasms; Plasmodium falciparum; Tetraoxanes	2013
Synthesis, in vitro antiplasmodial activity and cytotoxicity of a series of artemisinin-triazine hybrids and hybrid-dimers. European journal of medicinal chemistry, 2014, Apr-09, Volume: 76 Topics: Antimalarials; Artemisinins; Dimerization; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mass Spectrometry; Plasmodium falciparum; Spectrophotometry, Infrared; Triazines	2014
Orally bioavailable 6-chloro-7-methoxy-4(1H)-quinolones efficacious against multiple stages of Plasmodium. Journal of medicinal chemistry, 2014, Nov-13, Volume: 57, Issue:21 Topics: Animals; Antimalarials; Humans; Inhibitory Concentration 50; Malaria; Mice; Microsomes, Liver; Parasitemia; Plasmodium; Plasmodium berghei; Quinolones; Structure-Activity Relationship	2014
Synthesis and in vitro biological evaluation of dihydroartemisinyl-chalcone esters. European journal of medicinal chemistry, 2015, Jan-27, Volume: 90 Topics: Antimalarials; Antineoplastic Agents; Artemisinins; Cell Line, Tumor; Cell Proliferation; Chalcone; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Esters; Humans; MCF-7 Cells; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship	2015
Highly potent artemisinin-derived dimers and trimers: Synthesis and evaluation of their antimalarial, antileukemia and antiviral activities. Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17 Topics: Antimalarials; Antineoplastic Agents, Phytogenic; Antiviral Agents; Artemisinins; Humans; Molecular Structure	2015
The pharmacokinetics and bioavailability of dihydroartemisinin, arteether, artemether, artesunic acid and artelinic acid in rats. The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:2 Topics: Absorption; Animals; Antimalarials; Area Under Curve; Artemether; Artemisinins; Biological Availability; Bridged Bicyclo Compounds, Heterocyclic; Male; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Succinates	1998
Comparative pharmacokinetic study of oral and rectal formulations of artesunic acid in healthy volunteers. European journal of clinical pharmacology, 1998, Volume: 54, Issue:5 Topics: Administration, Oral; Administration, Rectal; Adult; Antimalarials; Artemisinins; Bridged Bicyclo Compounds, Heterocyclic; Cross-Over Studies; Humans; Male; Sesquiterpenes; Succinates	1998
Synthesis of Artemisinin-Derived Dimers, Trimers and Dendrimers: Investigation of Their Antimalarial and Antiviral Activities Including Putative Mechanisms of Action. Chemistry (Weinheim an der Bergstrasse, Germany), 2018, Jun-07, Volume: 24, Issue:32 Topics: Antimalarials; Antiviral Agents; Artemisinins; Cytomegalovirus; Dendrimers; Humans; Succinates	2018
On-Flow LC-MS/MS method for screening of xanthine oxidase inhibitors. Journal of pharmaceutical and biomedical analysis, 2020, Mar-20, Volume: 181 Topics: Artemisinins; Chromatography, High Pressure Liquid; Drug Discovery; Enzyme Inhibitors; Glycosides; High-Throughput Screening Assays; Pyrans; Succinates; Tandem Mass Spectrometry; Xanthine Oxidase	2020
Dihydroartemisinin, an active metabolite of artemisinin, interferes with Leishmania braziliensis mitochondrial bioenergetics and survival. Parasitology research, 2021, Volume: 120, Issue:2 Topics: Animals; Antiprotozoal Agents; Artemisinins; Energy Metabolism; Hydrogen Peroxide; Leishmania braziliensis; Macrophages; Mitochondria; Succinates	2021
Stereoselective Access to Antimelanoma Agents by Hybridization and Dimerization of Dihydroartemisinin and Artesunic acid. ChemMedChem, 2021, 07-20, Volume: 16, Issue:14 Topics: Antineoplastic Agents; Artemisinins; Cell Proliferation; Cell Survival; Cells, Cultured; Dimerization; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Melanoma; Molecular Structure; Stereoisomerism; Structure-Activity Relationship; Succinates	2021