artemotil has been researched along with artenimol in 32 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (3.13) | 18.7374 |
1990's | 15 (46.88) | 18.2507 |
2000's | 11 (34.38) | 29.6817 |
2010's | 2 (6.25) | 24.3611 |
2020's | 3 (9.38) | 2.80 |
Authors | Studies |
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Emami, SA; Taleghani, A; Tayarani-Najaran, Z | 1 |
Brossi, A; Buchs, P; Dominguez Gerpe, L; Flippen-Anderson, JL; Luo, XD; Milhous, W; Peters, W; Venugopalan, B; Yeh, HJ | 1 |
Baker, JK; Ramu, K | 1 |
el-Feraly, FS; Kampinga, HH; Konings, AW; Malingré, TM; Moskal, TA; Pras, N; Woerdenbag, HJ | 1 |
Ager, AL; Andersen, SL; Dong, Y; Edwards, G; Fu, H; Gerena, L; Holme, AD; Kyle, DE; McLean, WG; Milhous, WK; Miller, RE; Vennerstrom, JL; Walters, SM; Wesche, DL; Wood, JK | 1 |
Jeong, IH; Lee, S; Oh, S; Shin, WS | 1 |
ElSohly, MA; Galal, AM; Jacob, M; Ross, SA | 1 |
Chung, WY; Jung, M; Park, KK; Tak, J | 1 |
Dembitsky, VM | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Leskovac, V; Peggins, JO | 1 |
Leskovac, V; Theoharides, AD | 1 |
Brewer, TG; Melendez, V; Peggins, JO; Theoharides, AD | 1 |
Ayalp, A; Bishop, SJ; el-Feraly, FS; Tawfik, AF | 1 |
Asawamahasakda, W; Ittarat, I; Meshnick, SR; Pu, YM; Ziffer, H | 1 |
Baker, JK; Chi, HT; McChesney, JD | 1 |
Hossler, P; Kamchonwongpaisan, S; McKeever, P; Meshnick, SR; Ziffer, H | 1 |
Aguilar, T; Brewer, TG; Grace, JM; Leo, KU; Li, Q; Mitchell, AL; Peggins, J | 1 |
Brewer, TG; Fleckenstein, LL; Heiffer, MH; Li, QG; Masonic, K; Peggins, JO | 1 |
Aguilar, AJ; Brewer, TG; Grace, JM; Peggins, JO; Trotman, KM | 1 |
Dong, Y; Huang, KG; Liao, MZ; Liu, DQ; Yang, HL; Yang, PF; Yang, YM; Zhang, CY | 1 |
McLean, WG; Ward, SA | 1 |
Looareesuwan, S; Wilairatana, P | 1 |
Brewer, TG; Genovese, RF; Newman, DB | 1 |
Gupta, RC; Madhusudanan, KP; Rajanikanth, M; Sabarinath, S | 1 |
Chalearmrult, K; Krudsood, S; Li, Q; Looareesuwan, S; Lugt, CB; Milhous, WK; Vannaphan, S; Wilairatana, P | 1 |
Gupta, RC; Madhusudanan, KP; Sabarinath, S | 1 |
Atemnkeng, MA; De Cock, K; Plaizier-Vercammen, J | 1 |
Chaudhary, S; Puri, SK; Singh, C | 1 |
Hubert, P; Marini, RD; Mbinze, JK; Memvanga, PB; Préat, V; Rozet, E | 1 |
Barbieri, D; Blaud, M; Clain, J; Duval, R; Grougnet, R; Hammad, K; Houzé, S; Lavazec, C; Leproux, P; Maciuk, A; Michel, S; Neveu, G; Rondepierre, L; Sissoko, A; Vásquez-Ocmín, P | 1 |
Chen, Y; Cheng, Y; Li, P; Liu, H; Lu, X; Ma, Y; Song, C; Wang, Y; Zhang, Z | 1 |
3 review(s) available for artemotil and artenimol
Article | Year |
---|---|
Artemisia: a promising plant for the treatment of cancer.
Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisia; Cell Proliferation; Humans; Molecular Structure; Neoplasms; Neoplasms, Experimental; Plant Extracts; Plants, Medicinal | 2020 |
Bioactive peroxides as potential therapeutic agents.
Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Drug Screening Assays, Antitumor; Humans; Peroxides | 2008 |
The rational use of qinghaosu and its derivatives: what is the future of new compounds?
Topics: Administration, Oral; Administration, Rectal; Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Drug and Narcotic Control; Drug Resistance; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Registries; Sesquiterpenes; Suppositories; Thailand | 1998 |
1 trial(s) available for artemotil and artenimol
Article | Year |
---|---|
Pharmacokinetic investigation on the therapeutic potential of artemotil (beta-arteether) in Thai patients with severe Plasmodium falciparum malaria.
Topics: Adult; Antimalarials; Area Under Curve; Artemisinins; Half-Life; Humans; Injections, Intramuscular; Malaria, Falciparum; Sesquiterpenes | 2004 |
28 other study(ies) available for artemotil and artenimol
Article | Year |
---|---|
Arteether, a new antimalarial drug: synthesis and antimalarial properties.
Topics: Animals; Antimalarials; Artemisinins; Magnetic Resonance Spectroscopy; Malaria; Mice; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes | 1988 |
Synthesis, characterization, and antimalarial activity of the glucuronides of the hydroxylated metabolites of arteether.
Topics: Animals; Antimalarials; Artemisinins; Chromatography, High Pressure Liquid; Glucuronates; Hydrolysis; Hydroxylation; Microbial Sensitivity Tests; Models, Chemical; Plasmodium falciparum; Sesquiterpenes; Stereoisomerism | 1995 |
Cytotoxicity of artemisinin-related endoperoxides to Ehrlich ascites tumor cells.
Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisinins; Carcinoma, Ehrlich Tumor; Cell Survival; Chemical Phenomena; Chemistry, Physical; Cisplatin; Doxorubicin; Peroxides; Sesquiterpenes; Structure-Activity Relationship; Tetrazolium Salts; Tumor Cells, Cultured | 1993 |
Synthesis and antimalarial activity of sixteen dispiro-1,2,4, 5-tetraoxanes: alkyl-substituted 7,8,15,16-tetraoxadispiro[5.2.5. 2]hexadecanes.
Topics: Alkanes; Animals; Antimalarials; Malaria; Mice; Neurites; Neuroblastoma; Plasmodium berghei; Plasmodium falciparum; Spiro Compounds; Structure-Activity Relationship; Tumor Cells, Cultured | 2000 |
Growth inhibition activity of thioacetal artemisinin derivatives against human umbilical vein endothelial cells.
Topics: Acetals; Artemisinins; Cell Division; Colorimetry; Endothelial Cells; Female; Humans; Lactones; Pregnancy; Sesquiterpenes; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Umbilical Veins | 2003 |
Antifungal activity of artemisinin derivatives.
Topics: Antifungal Agents; Artemisinins; Candida albicans; Combinatorial Chemistry Techniques; Cryptococcus neoformans; Microbial Sensitivity Tests; Molecular Structure | 2005 |
Antiangiogenic activity of deoxoartemisinin derivatives on chorioallantoic membrane.
Topics: Acetals; Angiogenesis Inhibitors; Animals; Artemisinins; Chick Embryo; Chorioallantoic Membrane; Molecular Structure; Sesquiterpenes; Structure-Activity Relationship | 2006 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Hepatic metabolism of artemisinin drugs--III. Induction of hydrogen peroxide production in rat liver microsomes by artemisinin drugs.
Topics: Animals; Antimalarials; Artemisinins; Hydrogen Peroxide; Kinetics; Male; Microsomes, Liver; NADP; Rats; Rats, Inbred Strains; Sesquiterpenes | 1992 |
Hepatic metabolism of artemisinin drugs--I. Drug metabolism in rat liver microsomes.
Topics: Animals; Antimalarials; Artemisinins; Chromatography, High Pressure Liquid; Chromatography, Liquid; Kinetics; Liver; Male; Mass Spectrometry; Microsomes, Liver; Rats; Rats, Inbred Strains; Sesquiterpenes | 1991 |
Determination of the antimalarial arteether and its deethylated metabolite dihydroartemisinin in plasma by high-performance liquid chromatography with reductive electrochemical detection.
Topics: Animals; Antimalarials; Artemisinins; Biological Availability; Chromatography, High Pressure Liquid; Dogs; Electrochemistry; Oxidation-Reduction; Reproducibility of Results; Sesquiterpenes | 1991 |
Effects of artemisinin, dihydroartemisinin and arteether on immune responses of normal mice.
Topics: Animals; Antibody Formation; Antimalarials; Artemisinins; Carrageenan; Hemolytic Plaque Technique; Hypersensitivity, Delayed; Immunosuppressive Agents; Inflammation; Male; Mice; Sesquiterpenes | 1990 |
Reaction of antimalarial endoperoxides with specific parasite proteins.
Topics: Animals; Antimalarials; Artemisinins; Autoradiography; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Erythrocytes; Plasmodium falciparum; Protozoan Proteins; Sesquiterpenes; Styrenes | 1994 |
Decomposition of arteether in simulated stomach acid yielding compounds retaining antimalarial activity.
Topics: Animals; Antimalarials; Artemisinins; Chromatography, High Pressure Liquid; Gastric Acid; Half-Life; Magnetic Resonance Spectroscopy; Plasmodium falciparum; Sesquiterpenes | 1993 |
Artemisinin neurotoxicity: neuropathology in rats and mechanistic studies in vitro.
Topics: Alkylation; Animals; Antimalarials; Artemisinins; Blood Proteins; Brain; Detergents; Erythrocytes; Male; Mice; Molecular Weight; Nerve Tissue Proteins; Neuroblastoma; Neurons; Octoxynol; Plasmodium falciparum; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Tumor Cells, Cultured | 1997 |
Effects of Plasmodium berghei infection on arteether metabolism and disposition.
Topics: Animals; Antimalarials; Area Under Curve; Artemisinins; Bile; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Half-Life; Isotope Labeling; Liver; Malaria; Male; Microsomes, Liver; NADPH-Ferrihemoprotein Reductase; Perfusion; Plasmodium berghei; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Tissue Distribution | 1997 |
The pharmacokinetics and bioavailability of dihydroartemisinin, arteether, artemether, artesunic acid and artelinic acid in rats.
Topics: Absorption; Animals; Antimalarials; Area Under Curve; Artemether; Artemisinins; Biological Availability; Bridged Bicyclo Compounds, Heterocyclic; Male; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Succinates | 1998 |
Metabolism of beta-arteether to dihydroqinghaosu by human liver microsomes and recombinant cytochrome P450.
Topics: Antimalarials; Artemisinins; Cytochrome P-450 Enzyme System; Humans; Microsomes, Liver; Sesquiterpenes | 1998 |
In vitro sensitivity of Plasmodium falciparum to eight antimalarials in China-Myanmar and China-Lao PDR border areas.
Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Artesunate; China; Chloroquine; Drug Evaluation, Preclinical; Drug Resistance; Humans; Laos; Microbial Sensitivity Tests; Myanmar; Naphthyridines; Plasmodium falciparum; Quinine; Sesquiterpenes | 1997 |
In vitro neurotoxicity of artemisinin derivatives.
Topics: Animals; Antimalarials; Artemether; Artemisinins; Cell Differentiation; Central Nervous System Diseases; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Mice; Microscopy, Electron; Neuroblastoma; Neurons; Reproducibility of Results; Sesquiterpenes; Tumor Cells, Cultured | 1998 |
Behavioral and neural toxicity of the artemisinin antimalarial, arteether, but not artesunate and artelinate, in rats.
Topics: Animals; Antimalarials; Artemisinins; Artesunate; Behavior, Animal; Brain; Brain Stem; Discrimination Learning; Male; Rats; Rats, Sprague-Dawley; Sesquiterpenes | 2000 |
A sensitive and selective liquid chromatographic/electrospray ionization tandem mass spectrometric assay for the simultaneous quantification of alpha-,beta-arteether and its metabolite dihydroartemisinin in plasma, useful for pharmacokinetic studies.
Topics: Antimalarials; Artemisinins; Chromatography, High Pressure Liquid; Sensitivity and Specificity; Sesquiterpenes; Spectrometry, Mass, Electrospray Ionization | 2003 |
Pharmacokinetics of the diastereomers of arteether, a potent antimalarial drug, in rats.
Topics: Administration, Oral; Animals; Antimalarials; Area Under Curve; Artemisinins; Injections, Intramuscular; Injections, Intravenous; Male; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Stereoisomerism | 2005 |
Quality control of active ingredients in artemisinin-derivative antimalarials within Kenya and DR Congo.
Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Capsules; Chromatography, High Pressure Liquid; Democratic Republic of the Congo; Dosage Forms; Endemic Diseases; Humans; Kenya; Malaria, Falciparum; Quality Control; Sesquiterpenes; Tablets | 2007 |
Orally active esters of dihydroartemisinin: Synthesis and antimalarial activity against multidrug-resistant Plasmodium yoelii in mice.
Topics: Adamantane; Administration, Oral; Animals; Antimalarials; Artemisinins; Biphenyl Compounds; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Esters; Malaria; Mice; Models, Molecular; Plasmodium yoelii; Sesquiterpenes; Structure-Activity Relationship | 2008 |
Development of a liquid chromatographic method for the simultaneous quantification of curcumin, β-arteether, tetrahydrocurcumin and dihydroartemisinin. Application to lipid-based formulations.
Topics: Acetates; Algorithms; Antimalarials; Artemisinins; Calibration; Chemistry Techniques, Analytical; Chemistry, Pharmaceutical; Chromatography, Liquid; Curcumin; Hydrogen-Ion Concentration; Limit of Detection; Lipids; Methanol; Reproducibility of Results; Temperature | 2014 |
A Chemically Stable Fluorescent Mimic of Dihydroartemisinin, Artemether, and Arteether with Conserved Bioactivity and Specificity Shows High Pharmacological Relevance to the Antimalarial Drugs.
Topics: Antimalarials; Artemether; Artemisinins | 2020 |
Exploring the Potential Mechanism of Artemisinin and Its Derivatives in the Treatment of Osteoporosis Based on Network Pharmacology and Molecular Docking.
Topics: Artemether; Artemisinins; Artesunate; Caspase 3; Drugs, Chinese Herbal; ErbB Receptors; Humans; Interleukin-17; Mitogen-Activated Protein Kinase 14; Molecular Docking Simulation; Network Pharmacology; Osteoporosis; Prolactin | 2022 |