Page last updated: 2024-08-25

artemether and sodium artesunate

artemether has been researched along with sodium artesunate in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19901 (9.09)18.7374
1990's2 (18.18)18.2507
2000's5 (45.45)29.6817
2010's2 (18.18)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Brossi, A; Buchs, P; Dominguez Gerpe, L; Flippen-Anderson, JL; Luo, XD; Milhous, W; Peters, W; Venugopalan, B; Yeh, HJ1
Asawamahasadka, W; Kumar, N; McGarvey, DJ; Meshnick, SR; Oh, CH; Posner, GH1
el-Feraly, FS; Kampinga, HH; Konings, AW; Malingré, TM; Moskal, TA; Pras, N; Woerdenbag, HJ1
Bishop, LP; Hindley, S; Maggs, JL; Miller, A; O'Neill, PM; Park, BK; Posner, GH; Roberts, SM; Scheinmann, F; Stachulski, AV; Ward, SA1
Bray, PG; Davies, J; Hindley, S; O'Neill, PM; Park, BK; Searle, NL; Storr, RC; Ward, SA1
Dembitsky, VM1
Amewu, R; Bongard, E; Charnaud, S; Davies, J; Ellis, GL; Gargallo, D; Gibbons, P; Hall, C; Jesús, M; Lozanom, S; O'Neill, PM; Rimmer, K; Sabbani, S; Shone, A; Stanford, D; Stocks, PA; Vivas, L; Ward, SA1
Chen, X; Hergenrother, PJ; Liu, JO; Posner, GH; Rosenthal, AS; Shapiro, TA; West, DC1
Arav-Boger, R; Chen, X; Civin, CI; Fox, JM; He, R; Mott, BT; Posner, GH1
Bertinaria, M; Carvalho, LJ; Frangos, JA; Fruttero, R; Gasco, A; Guglielmo, S; Hofer, A; Marini, E; Martins, YC; Orjuela-Sanchez, P; Zanini, GM1
Aucamp, J; N'Da, DD; Zuma, NH1

Reviews

1 review(s) available for artemether and sodium artesunate

ArticleYear
Bioactive peroxides as potential therapeutic agents.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:2

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Drug Screening Assays, Antitumor; Humans; Peroxides

2008

Other Studies

10 other study(ies) available for artemether and sodium artesunate

ArticleYear
Arteether, a new antimalarial drug: synthesis and antimalarial properties.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Animals; Antimalarials; Artemisinins; Magnetic Resonance Spectroscopy; Malaria; Mice; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes

1988
Structure-activity relationships of lactone ring-opened analogs of the antimalarial 1,2,4-trioxane artemisinin.
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Animals; Antimalarials; Artemisinins; Lactones; Mice; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes; Structure-Activity Relationship

1995
Cytotoxicity of artemisinin-related endoperoxides to Ehrlich ascites tumor cells.
    Journal of natural products, 1993, Volume: 56, Issue:6

    Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisinins; Carcinoma, Ehrlich Tumor; Cell Survival; Chemical Phenomena; Chemistry, Physical; Cisplatin; Doxorubicin; Peroxides; Sesquiterpenes; Structure-Activity Relationship; Tetrazolium Salts; Tumor Cells, Cultured

1993
Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin.
    Journal of medicinal chemistry, 2001, Jan-04, Volume: 44, Issue:1

    Topics: Animals; Antimalarials; Artemisinins; Bile; Crystallography, X-Ray; Electron Spin Resonance Spectroscopy; Ferrous Compounds; Free Radicals; Malaria; Male; Mice; Phenyl Ethers; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Rats, Wistar; Sesquiterpenes; Stereoisomerism; Structure-Activity Relationship

2001
Mechanism-based design of parasite-targeted artemisinin derivatives: synthesis and antimalarial activity of new diamine containing analogues.
    Journal of medicinal chemistry, 2002, Feb-28, Volume: 45, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Heterocyclic Compounds, 4 or More Rings; Malaria; Male; Mice; Piperazines; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes

2002
Two-step synthesis of achiral dispiro-1,2,4,5-tetraoxanes with outstanding antimalarial activity, low toxicity, and high-stability profiles.
    Journal of medicinal chemistry, 2008, Apr-10, Volume: 51, Issue:7

    Topics: Animals; Antimalarials; Chlorocebus aethiops; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Stability; Humans; Male; Mice; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Rats; Salmonella typhimurium; Spiro Compounds; Stereoisomerism; Structure-Activity Relationship; Tetraoxanes

2008
Malaria-infected mice are cured by a single oral dose of new dimeric trioxane sulfones which are also selectively and powerfully cytotoxic to cancer cells.
    Journal of medicinal chemistry, 2009, Feb-26, Volume: 52, Issue:4

    Topics: Administration, Oral; Animals; Antimalarials; Antineoplastic Agents; Artemisinins; Cell Line, Tumor; Drug Screening Assays, Antitumor; Drug Stability; Drug Therapy, Combination; Humans; Malaria; Mefloquine; Mice; Sulfones

2009
Artemisinin-derived dimer phosphate esters as potent anti-cytomegalovirus (anti-CMV) and anti-cancer agents: a structure-activity study.
    Bioorganic & medicinal chemistry, 2013, Jul-01, Volume: 21, Issue:13

    Topics: Antineoplastic Agents; Antiviral Agents; Artemisinins; Cytomegalovirus; Cytomegalovirus Infections; Dimerization; Esters; Humans; Jurkat Cells; Leukemia; Phosphates

2013
NO-Donor Dihydroartemisinin Derivatives as Multitarget Agents for the Treatment of Cerebral Malaria.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Chemistry Techniques, Synthetic; Malaria, Cerebral; Mice; Molecular Targeted Therapy; Muscle Relaxation; Nitric Oxide Donors; Plasmodium berghei; Rats; Vasodilator Agents

2015
In vitro efficacy of synthesized artemisinin derivatives against Leishmania promastigotes.
    Bioorganic & medicinal chemistry letters, 2020, 11-15, Volume: 30, Issue:22

    Topics: Antimalarials; Artemisinins; Dose-Response Relationship, Drug; Leishmania; Molecular Structure; Parasitic Sensitivity Tests; Structure-Activity Relationship

2020