Page last updated: 2024-08-25

artemether and artenimol

artemether has been researched along with artenimol in 133 studies

Research

Studies (133)

TimeframeStudies, this research(%)All Research%
pre-19907 (5.26)18.7374
1990's23 (17.29)18.2507
2000's35 (26.32)29.6817
2010's46 (34.59)24.3611
2020's22 (16.54)2.80

Authors

AuthorsStudies
Combrinck, J; de Kock, C; N'Da, DD; Smit, FJ; Smith, PJ; Zuma, NH1
Dong, G; Liu, N; Sheng, C; Wang, Y; Wu, S1
Emami, SA; Taleghani, A; Tayarani-Najaran, Z1
Brossi, A; Buchs, P; Dominguez Gerpe, L; Flippen-Anderson, JL; Luo, XD; Milhous, W; Peters, W; Venugopalan, B; Yeh, HJ1
el-Feraly, FS; Kampinga, HH; Konings, AW; Malingré, TM; Moskal, TA; Pras, N; Woerdenbag, HJ1
Kan, KW; Maggs, JL; O'Neill, PM; Park, BK; Raynes, K; Searle, NL; Storr, RC; Ward, SA1
Ager, AL; Andersen, SL; Dong, Y; Edwards, G; Fu, H; Gerena, L; Holme, AD; Kyle, DE; McLean, WG; Milhous, WK; Miller, RE; Vennerstrom, JL; Walters, SM; Wesche, DL; Wood, JK1
Bishop, LP; Hindley, S; Maggs, JL; Miller, A; O'Neill, PM; Park, BK; Posner, GH; Roberts, SM; Scheinmann, F; Stachulski, AV; Ward, SA1
Brun, R; Charman, SA; Charman, WN; Chiu, FC; Chollet, J; Dong, Y; Dorn, A; Karle, JM; Matile, H; Santo Tomas, J; Scheurer, C; Scorneaux, B; Snyder, C; Tang, Y; Urwyler, H; Vennerstrom, JL; Wang, X; Wittlin, S1
ElSohly, MA; Galal, AM; Jacob, M; Ross, SA1
Adagu, IS; Fivelman, QL; Warhurst, DC1
Dembitsky, VM1
Charman, SA; Charman, WN; Chiu, FC; Creek, DJ; Dong, Y; Prankerd, RJ; Vennerstrom, JL1
Gottstein, B; Hemphill, A; Keiser, J; Lany, C; Ortega-Mora, LM; Roethlisberger, C; Spicher, M; Stadelmann, B1
Chadwick, J; Cosstick, R; Mercer, AE; O'Neill, PM; Park, BK1
Baird, J; Bray, PG; Charidza, T; Cosstick, R; Davies, J; Janneh, O; Jones, M; Kennedy, ME; La Pensée, LJ; Mercer, AE; O'Neill, PM; Park, BK; Piantanida, I; Rawe, SL; Stocks, PA; Ward, SA1
Charman, SA; Charman, WN; Chiu, FC; Creek, DJ; Prankerd, RJ; Ryan, E; Vennerstrom, JL1
Chung, WY; Jung, M; Lee, Y; Moon, HI; Park, KK; Park, N1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Biamonte, MA; Le Roch, KG; Wanner, J1
Fidock, DA; Flannery, EL; Winzeler, EA1
Edwards, G; Thomas, CG; Ward, SA1
Song, ZY; Zhao, KC1
Gu, HM; Peters, W; Warhurst, DC3
Li, ZL; Peters, W; Robinson, BL; Warhurst, DC1
Gu, HM; Li, ZL; Peters, W; Warhurst, DC1
Asokan, M; Chin, LK; Mansor, SM; Mordi, MN; Nair, NK; Navaratnam, V1
Mberu, EK; Muhia, DK; Watkins, WM1
Ager, AL; Klayman, DL; Lin, AJ1
Edwards, G; Mberu, EK; Muhia, DK; Thomas, CG; Ward, SA; Watkins, WM1
Edwards, G; Karbwang, J; Na Bangchang, K; Sukontason, K; Thanavibul, A; Thomas, CG; Ward, SA1
Davis, TM; Johnston, WA; Manning, LS; Skinner, TS1
Banmairuroi, V; Congpuong, K; Karbwang, J; Molunto, P; Na-Bangchang, K1
Donker, M; Godbillon, J; Netter, C; Sandrenan, N; Sioufi, A; van Valkenburg, C1
Mansor, SM; Mordi, MN; Navaratnam, V; Wernsdorfer, WH1
Brewer, TG; Fleckenstein, LL; Heiffer, MH; Li, QG; Masonic, K; Peggins, JO1
Berens, RL; Curiel, TJ; Krug, EC; Nash, PB1
Congpuong, K; Karbwang, J; Molunto, P; Na-Bangchang, K; Thanavibul, A; Wattanakoon, Y1
Karbwang, J; Molunto, P; Na-Bangchang, K; Thanavibul, A1
Harinasuta, T; Karbwang, J; Na-Bangchang, K; Rimchala, W; Sukontason, K; Tin, T1
Li, Y; Wu, YL1
McLean, WG; Ward, SA1
Cheng-Qi, S; Mull, R; Qing, JX; van Agtmael, MA; van Boxtel, CJ1
Edwards, G; Haynes, RK; Khalid, SA; Mohamed, SS; Tang, HP; Wan, TS; Ward, SA; Zheng, M1
Gupta, V; van Agtmael, MA; van Boxtel, CJ; van der Graaf, CA1
Dodd, CC; Edwards, G; McLean, WG; Park, BK; Sadler, CJ; Smith, SL; Ward, SA1
MacDonald, RD1
Tu, Y1
Green, MD; Mount, DL; Wirtz, RA1
Gauducheau, N; Richard, F; Sandrenan, N; Souppart, C1
Chen, YG; Yu, BY1
Brittenham, GM; Chalermrut, K; Kano, S; Krudsood, S; Looareesuwan, S; Pengruksa, C; Silachamroon, U; Srivilairit, S; Treeprasertsuk, S1
Aarons, L; Edwards, G; Kokwaro, GO; Majid, O; Marsh, K; Mithwani, S; Mohamed, S; Muchohi, S; Watkins, W1
Gabriëls, M; Plaizier-Vercammen, J1
Shen, WJ; Thiero, M1
Keiser, J; Shu-Hua, X; Tanner, M; Utzinger, J1
Ashley, EA; La, Y; Lindegardh, N; McGready, R; Nosten, F; Singhasivanon, P; Stepniewska, K; White, NJ1
Atemnkeng, MA; De Cock, K; Plaizier-Vercammen, J1
Ayede, I; Dada-Adegbola, HO; Fadero, FF; Falade, AG; Falade, CO; Gbotosho, GO; Happi, CT; Oduola, AM; Salako, LA1
Davis, TM; Ilett, KF; Karunajeewa, HA; Manning, L; Mueller, I1
Bukirwa, H; Dorsey, G; Kamya, MR; Lugemwa, M; Rosenthal, PJ; Rwakimari, JB; Staedke, SG; Talisuna, A; Wabwire-Mangen, F; Yeka, A1
Christophel, E; Hu, XM; Lin, SG; Liu, J; Meng, F; Wang, GZ; Wang, SQ; Zeng, LH1
Hou, J; Wang, D; Wang, H; Zhang, R1
Davis, TM; Gomorrai, PS; Griffin, S; Ilett, KF; Karunajeewa, HA; Kotab, K; Lautu, D; Law, I; Lin, E; Mueller, I; Oa, O; Page-Sharp, M; Salman, S; Senn, M; Siba, P; Suano, P; Tarongka, N; Ura, A; Wong, R1
Dorsey, G; Nosten, F; Price, RN1
Aweeka, FT; Huang, L; Jayewardene, AL; Li, X; Lizak, PS; Marzan, F1
Bacchieri, A; Bassat, Q; Borrmann, S; Corsi, M; D'Alessandro, U; Menéndez, C; Mulenga, M; Nabasumba, C; Nambozi, M; Piola, P; Sasi, P; Talisuna, A; Tinto, H; Ubben, D; Valéa, I1
Arinaitwe, E; Bigira, V; Dorsey, G; Gasasira, A; Homsy, J; Kakuru, A; Kamya, MR; Katrak, S; Sandison, TG; Tappero, JW; Wanzira, H1
Dokomajilar, C; Greenhouse, B; Ouédraogo, JB; Rosenthal, PJ; Rouamba, N; Séré, YY; Somé, AF; Zongo, I1
Annerberg, A; Ashton, M; Björkman, A; Dahlström, S; Färnert, A; Gil, P; Hietala, SF; Lindegårdh, N; Mårtensson, A; Ngasala, B; Premji, Z1
Arinaitwe, E; Bigira, V; Creek, D; Dorsey, G; Kakuru, A; Kamya, MR; Sandison, TG; Tappero, J; Wanzira, H1
Ali, S; Lindegardh, N; Najmi, MH; Tarning, J1
Day, NP; Hanpithakpong, W; Kamanikom, B; Lindegardh, N; Singhasivanon, P; White, NJ1
Bai, KH; Liu, T; Wang, RL; Xing, J; Zhang, LF; Zhang, SQ1
Duthaler, U; Huwyler, J; Keiser, J1
Dai, JR; Li, HJ; Li, YZ; Liang, YS; Qu, GL; Tao, YH; Wang, W; Wei, JY; Xing, YT1
Faye, B; Faye, O; Kane, D; Kassi, KF; Kiki Barro, CP; Kone, M; Kuete, T; Menan, H; N'diaye, JL; Oga, AS; Same-Ekobo, A; Tine, R; Vicky, AM; Yavo, W1
Davis, TM; Hwaiwhanje, I; Karunajeewa, HA; Laman, M; Manning, L; Morep, N; Mueller, I; Page-Sharp, M; Salman, S; Siba, P1
Jessing, KK; Juhler, RK; Strobel, BW1
Du, F; Liu, T; Xing, J; Zhu, F1
Bashraheil, M; Bassat, Q; González, R; Kipkeu, C; Lefèvre, G; Lyimo, J; Machevo, S; Maiga, H; Mårtensson, A; Menéndez, C; Nahum, A; Nwaiwu, O; Ogutu, B; Ouma, P; Ubben, D; Walter, V1
Day, NP; Dhorda, M; Guerin, PJ; Kloprogge, F; Lindegardh, N; Muwanga, S; Nosten, F; Nuengchamnong, N; Piola, P; Tarning, J; Turyakira, E; White, NJ1
Ahnoff, M; Blessborn, D; Kaewkhao, K; Sköld, K; Sköld, O; Zeeberg, D1
Achan, J; D'Alessandro, U; Talisuna, AO; Tibenderana, J; Yeka, A1
Back, DJ; Byakika-Kibwika, P; Hanpithakpong, W; Khoo, SH; Lamorde, M; Lefèvre, G; Mayito, J; Merry, C; Nabukeera, L; Ryan, M1
Aweeka, FT; Gingrich, D; Huang, L; Olson, A1
Dhorda, M; Guerin, PJ; Jullien, V; Kloprogge, F; Nosten, F; Piola, P; Tarning, J; White, NJ1
Cui, L; Cui, Y; Wang, B; Wang, M; Yan, G; Zhou, G1
Burkholder, B; Bustos, MD; Delacollette, C; Wongsrichanalai, C1
Ashton, M; Ericsson, T; Hoffmann, KJ; Sundell, J; Torkelsson, A1
Li, GX; Wang, W; Wang, YH; Xu, FL; Zhang, XG; Zhao, SS1
de Vries, R; Hendriks, G; Hilhorst, MJ; Hillewaert, V; van de Merbel, NC; Verhaege, T1
Batty, KT; Senarathna, SM1
Wang, FY; Wang, YB; Wei, DD; Wei, YB; Yin, B; Yu, ZH; Zhang, BG; Zhao, GH1
Bertinaria, M; Carvalho, LJ; Frangos, JA; Fruttero, R; Gasco, A; Guglielmo, S; Hofer, A; Marini, E; Martins, YC; Orjuela-Sanchez, P; Zanini, GM1
Adedeji, WA; Adewole, IF; Akinyinka, OO; Aweeka, FT; Darin, KM; Fehintola, F; Huang, L; Morse, GD; Murphy, RL; Olson, A; Parikh, S; Scarsi, KK; Taiwo, BO1
Bonfill, M; Cusido, RM; Dilshad, E; Mirza, B; Ramirez Estrada, K1
Acheampong, PR; Antwi, GD; Bart Plange, C; Cairns, M; Chandramohan, D; Tagbor, H1
Achan, J; Aweeka, F; Huang, L; Kajubi, R; Kiconco, S; Mwebaza, N; Mwima, MW; Nguyen, VK; Nyunt, MM; Parikh, S; Ssebuliba, J1
Barnes, KI; Cohen, K; Kredo, T; Maartens, G; Mauff, K; Smith, PJ; Van der Walt, JS; Wiesner, L; Workman, L1
Chavchich, M; Diagana, TT; Edstein, MD; Rowcliffe, K; Van Breda, K1
Bélard, S; Damm, G; Kim, J; Kurth, F; Lingscheid, T; Mayer, B; Menner, N; Pongratz, P; Salama, A; Seehofer, D; Stegemann, MS; Steiner, F; Suttorp, N; von Bernuth, H; Zoller, T1
Iyengar, K; Roepe, PD; Siriwardana, A1
Kofoed, PE; Rodrigues, A; Rombo, L; Ursing, J1
Wang, S; Xu, Z1
Ali, S; Farhat, K; Jafery, N; Waheed, A1
Gao, H; Hou, S; Liu, H; Su, R; Sun, J; Yang, Y1
Agaba, S; de Vries, PJ; Dorlo, TPC; Kaligirwa, N; Karlsson, MO; Lohy Das, J; Mens, PF; Rulisa, S; Tarning, J1
Dai, R; Dai, T; Guo, Z; Jiang, W; Xie, Y1
Beavogui, AH; Borghini-Fuhrer, I; Djimdé, AA; Duparc, S; Felices, M; Funck-Brentano, C; Khan, Y; Ouedraogo, JB; Ouologuem, N; Sagara, I; Sirima, SB; Soulama, I; Voiriot, P1
Badjanga, BB; Day, NPJ; Fanello, C; Hoglund, RM; Jackson, NV; Kabedi, C; Kayembe, D; Lee, SJ; McGready, R; Nosten, F; Onyamboko, MA; Tarning, J; Turner, GDH; White, NJ1
Aweeka, F; Huang, L; Hughes, E; Kajubi, R; Mwebaza, N; Mwima, MW; Nguyen, V; Nyunt, MM; Orukan, F; Parikh, S1
Barbieri, D; Blaud, M; Clain, J; Duval, R; Grougnet, R; Hammad, K; Houzé, S; Lavazec, C; Leproux, P; Maciuk, A; Michel, S; Neveu, G; Rondepierre, L; Sissoko, A; Vásquez-Ocmín, P1
Gille, L; Machín, L; Monzote, L; Nápoles, R1
Deng, C; Liang, Y; Lu, C; Song, J; Tan, B; Wang, Q; Wu, W; Xu, Q; Zhang, H; Zhou, C1
Bancone, G; Carrara, VI; Chu, C; Duanguppama, J; Gilder, ME; Haohankhunnatham, W; Imwong, M; Konghahong, K; Lee, SJ; McGready, R; Min, AM; Nosten, F; Paw, MK; Phyo, AP; Pimanpanarak, M; Proux, S; Saito, M; Singhasivanon, P; Tun, NW; Turner, C; Viladpai-Nguen, J; White, NJ1
Baltzell, K; Benjamin-Chung, J; Bhangu, K; Dlamini, B; Dlamini, N; Dufour, MK; Gosling, R; Greenhouse, B; Helb, D; Hsiang, MS; Kalungero, M; Kunene, S; Malambe, C; Maphalala, G; Mngadi, N; Nhlabathi, N; Ntshalintshali, N; Pindolia, D; Prach, LM; Tesfa, G; Vilakati, S; Whittemore, B1
Assefa, DG; Makonnen, E; Yismaw, G1
Baraka, V; Kamugisha, E; Kapesa, A; Kidenya, B; Konje, E; Marwa, K; Mukonzo, J; Swedberg, G1
Grundmann, O; Hernandez Maldonado, J1
Buff, AM; Chebore, W; Desai, M; Kariuki, S; Otieno, K; Owidhi, M; Samuels, AM; Westercamp, N1
Abera, A; Alemayehu, BH; Anand, A; Assefa, A; Bekele, W; Dilu, D; Etana, K; Ezema, B; Girma, S; Haile, M; Hwang, J; Minta, AA; Mohammed, H; Moriarty, LF; Murphy, M; Sime, H; Solomon, H; Svigel, SS; Tadesse, M; Tadesse, Y; Tasew, G; Teka, H; Woyessa, A; Zhou, Z1
Abongo, G; Basara, BB; Baseke, J; Bongo, GS; Day, NJP; Dhorda, M; Dondorp, AM; Fanello, C; Kayembe, DK; Maitland, K; Muhindo, R; Mukaka, M; Namayanja, C; Ndjowo, PO; Okalebo, CB; Olupot-Olupot, P; Onyamboko, MA; Onyas, P; Peerawaranun, P; Tarning, J; Taya, C; Taylor, WR; Titin, H; Uyoga, S; Waithira, N; Weere, W; Williams, TN1
Chen, Y; Cheng, Y; Li, P; Liu, H; Lu, X; Ma, Y; Song, C; Wang, Y; Zhang, Z1
Adjei, GO; Ahorhorlu, SY; Alifrangis, M; Duah-Quashie, NO; Dzudzor, B; Hansson, H; Jensen, RW; Kudzi, W; Nartey, ET; Quashie, NB; Wang, CW; Zoiku, F1
Deng, YN; Guh, JH; Hsu, LC; Hsu, YF; Huang, TE; Kung, FL; Marchesi, E; Marchetti, P; Navacchia, ML; Perrone, D1
Akala, HM; Amwoma, JG; Andagalu, BM; Chemwor, GC; Cheruiyot, AC; Egbo, TE; Garges, EC; Juma, DW; Juma, JA; Kamau, E; Mwakio, EW; Ogutu, BR; Okoth, RO; Onyango, IA; Opot, BH; Roth, AL; Wakoli, DM; Watson, OJ; Yedah, RA1
Aina, O; Awolola, ST; Babatunde, S; David, AN; Ekama, SO; Happi, CT; Ijezie, SN; Mohammed, AB; Mokuolu, O; Musa, AZ; Ogbulafor, N; Oguche, S; Okafor, H; Olukosi, AY; Ozor, L; Salako, BL; Uhomoibhi, PE; Wammanda, R1
Chepngetich, J; Gachie, B; Gathirwa, J; Kiboi, D; Kimani, F; Magoma, G; Muriithi, B; Mwitari, P; Onchieku, N; Thiong'o, K1
D'Alessandro, U; Dabira, ED; Diakite, H; Djimde, M; Dorlo, TP; Erhart, A; González, R; Kabore, B; Kayentao, K; Keita, M; Macuacua, S; Menendez, C; Mens, P; Muhindo, HM; Piqueras, M; Sagara, I; Schallig, H; Sevene, E; Tinto, H; Traore, M; Tshiongo, JK; Vala, A1
Bamisaiye, A; Basara, BB; Baseke, J; Day, NPJ; Fanello, C; Kayembe, DK; Maitland, K; Muhindo, R; Mukaka, M; Namayanja, C; Ndjowo, PO; Okalebo, CB; Olupot-Olupot, P; Onyamboko, MA; Onyas, P; Taya, C; Taylor, WRJ; Titin, H; Uyoga, S; Were, W; Williams, TN1

Reviews

14 review(s) available for artemether and artenimol

ArticleYear
Tackling Fungal Resistance by Biofilm Inhibitors.
    Journal of medicinal chemistry, 2017, 03-23, Volume: 60, Issue:6

    Topics: Animals; Antifungal Agents; Biofilms; Drug Discovery; Drug Resistance, Fungal; Fungi; Humans; Models, Molecular; Mycoses; Small Molecule Libraries

2017
Artemisia: a promising plant for the treatment of cancer.
    Bioorganic & medicinal chemistry, 2020, 01-01, Volume: 28, Issue:1

    Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisia; Cell Proliferation; Humans; Molecular Structure; Neoplasms; Neoplasms, Experimental; Plant Extracts; Plants, Medicinal

2020
Bioactive peroxides as potential therapeutic agents.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:2

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Drug Screening Assays, Antitumor; Humans; Peroxides

2008
Recent advances in malaria drug discovery.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Liver; Liver Transplantation; Malaria; Molecular Structure

2013
Using genetic methods to define the targets of compounds with antimalarial activity.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum

2013
Studies of qinghaosu and its active derivatives in biological materials and their pharmacokinetics.
    Proceedings of the Chinese Academy of Medical Sciences and the Peking Union Medical College = Chung-kuo i hsueh k'o hsueh yuan, Chung-kuo hsieh ho i k'o ta hsueh hsueh pao, 1989, Volume: 4, Issue:4

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Sesquiterpenes; Structure-Activity Relationship

1989
How Chinese scientists discovered qinghaosu (artemisinin) and developed its derivatives? What are the future perspectives?
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Drug Evaluation; Drug Resistance; Forecasting; Humans; Malaria, Falciparum; Medicine, Chinese Traditional; Sesquiterpenes

1998
Rectal administration of artemisinin derivatives for the treatment of malaria.
    JAMA, 2007, Jun-06, Volume: 297, Issue:21

    Topics: Administration, Rectal; Area Under Curve; Artemether; Artemisinins; Artesunate; Humans; Malaria; Sesquiterpenes

2007
Monitoring antimalarial drug efficacy in the Greater Mekong Subregion: an overview of in vivo results from 2008 to 2010.
    The Southeast Asian journal of tropical medicine and public health, 2013, Volume: 44 Suppl 1

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Asia, Southeastern; Chloroquine; Directly Observed Therapy; Drug Resistance; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Parasitemia; Quinolines

2013
A review of dihydroartemisinin as another gift from traditional Chinese medicine not only for malaria control but also for schistosomiasis control.
    Parasitology research, 2014, Volume: 113, Issue:5

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Drugs, Chinese Herbal; Female; Malaria, Falciparum; Mice; Praziquantel; Schistosomiasis japonica; Schistosomicides

2014
Mini Review - Analysis of Artemether and Dihydroartemisinin by high performance high liquid chromatography in biological fluids-issues and solutions.
    Pakistan journal of pharmaceutical sciences, 2017, Volume: 30, Issue:4

    Topics: Antimalarials; Artemether; Artemisinins; Body Fluids; Chemistry Techniques, Analytical; Humans

2017
Comparative effect of dihydroartemisinin-piperaquine and artemether-lumefantrine on gametocyte clearance and haemoglobin recovery in children with uncomplicated Plasmodium falciparum malaria in Africa: a systematic review and meta-analysis of randomized c
    International journal of infectious diseases : IJID : official publication of the International Society for Infectious Diseases, 2021, Volume: 113

    Topics: Africa; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Child; Drug Combinations; Fluorenes; Hemoglobins; Humans; Malaria, Falciparum; Plasmodium falciparum; Quinolines; Randomized Controlled Trials as Topic

2021
Therapeutic efficacy of artemether-lumefantrine, artesunate-amodiaquine and dihydroartemisinin-piperaquine in the treatment of uncomplicated Plasmodium falciparum malaria in Sub-Saharan Africa: A systematic review and meta-analysis.
    PloS one, 2022, Volume: 17, Issue:3

    Topics: Africa South of the Sahara; Amodiaquine; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Drug Combinations; Ethanolamines; Humans; Malaria; Malaria, Falciparum; Piperazines; Plasmodium falciparum; Quinolines

2022
Drug-Drug Interactions of Artemisinin-Based Combination Therapies in Malaria Treatment: A Narrative Review of the Literature.
    Journal of clinical pharmacology, 2022, Volume: 62, Issue:10

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Drug Combinations; Drug Interactions; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum

2022

Trials

32 trial(s) available for artemether and artenimol

ArticleYear
Differential extraction of artemether and its metabolite dihydroartemisinin from plasma and determination by high-performance liquid chromatography.
    Journal of chromatography. B, Biomedical applications, 1994, Oct-03, Volume: 660, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Chromatography, High Pressure Liquid; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Sesquiterpenes; Spectrophotometry, Ultraviolet

1994
Single dose pharmacokinetics of oral artemether in healthy Malaysian volunteers.
    British journal of clinical pharmacology, 1997, Volume: 43, Issue:4

    Topics: Administration, Oral; Adult; Antimalarials; Artemether; Artemisinins; Blood Specimen Collection; Chromatography, High Pressure Liquid; Drug Stability; Humans; Malaysia; Male; Sesquiterpenes; Temperature

1997
Pharmacokinetics of oral artemether in Thai patients with uncomplicated falciparum malaria.
    Fundamental & clinical pharmacology, 1998, Volume: 12, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Antimalarials; Area Under Curve; Artemether; Artemisinins; Chromatography, High Pressure Liquid; Follow-Up Studies; Humans; Malaria, Falciparum; Sesquiterpenes; Thailand

1998
Plasma concentrations of artemether and its major plasma metabolite, dihydroartemisinin, following a 5-day regimen of oral artemether, in patients with uncomplicated falciparum malaria.
    Annals of tropical medicine and parasitology, 1998, Volume: 92, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Drug Resistance, Multiple; Follow-Up Studies; Humans; Malaria, Falciparum; Male; Middle Aged; Sesquiterpenes

1998
Pharmacokinetics of intramuscular artemether in patients with severe falciparum malaria with or without acute renal failure.
    British journal of clinical pharmacology, 1998, Volume: 45, Issue:6

    Topics: Acute Kidney Injury; Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Humans; Kidney; Malaria, Falciparum; Male; Metabolic Clearance Rate; Middle Aged; Sesquiterpenes; Treatment Outcome

1998
Multiple dose pharmacokinetics of artemether in Chinese patients with uncomplicated falciparum malaria.
    International journal of antimicrobial agents, 1999, Volume: 12, Issue:2

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; China; Double-Blind Method; Drug Evaluation; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Male; Middle Aged; Models, Chemical; Sesquiterpenes; Time Factors

1999
The effect of grapefruit juice on the time-dependent decline of artemether plasma levels in healthy subjects.
    Clinical pharmacology and therapeutics, 1999, Volume: 66, Issue:4

    Topics: Administration, Oral; Adult; Antifungal Agents; Antimalarials; Antiprotozoal Agents; Artemether; Artemisinins; Beverages; Biological Availability; Citrus; Cross-Over Studies; Food-Drug Interactions; Humans; Male; Reference Values; Sesquiterpenes; Time Factors

1999
Comparative clinical trial of two-fixed combinations dihydroartemisinin-napthoquine-trimethoprim (DNP) and artemether-lumefantrine (Coartem/Riamet) in the treatment of acute uncomplicated falciparum malaria in Thailand.
    The Southeast Asian journal of tropical medicine and public health, 2003, Volume: 34, Issue:2

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Male; Middle Aged; Sesquiterpenes; Thailand; Treatment Outcome; Trimethoprim

2003
The pharmacokinetics of artemether and lumefantrine in pregnant women with uncomplicated falciparum malaria.
    European journal of clinical pharmacology, 2006, Volume: 62, Issue:12

    Topics: Adolescent; Adult; Antimalarials; Area Under Curve; Artemether; Artemisinins; Drug Administration Schedule; Ethanolamines; Female; Fluorenes; Follow-Up Studies; Half-Life; Humans; Lumefantrine; Malaria, Falciparum; Male; Pregnancy; Pregnancy Outcome; Pregnancy Trimester, Second; Pregnancy Trimester, Third; Recurrence; Remission Induction; Sesquiterpenes; Tablets; Thailand

2006
Dihydroartemisinin suppository in moderately severe malaria: comparative efficacy of dihydroartemisinin suppository versus intramuscular artemeter followed by oral sulfadoxine-pyrimethamine in the management of moderately severe malaria in Nigerian childr
    The American journal of tropical medicine and hygiene, 2007, Volume: 76, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Drug Combinations; Humans; Infant; Injections, Intramuscular; Malaria, Falciparum; Nigeria; Pyrimethamine; Sesquiterpenes; Sulfadoxine; Suppositories

2007
Artemether-lumefantrine versus dihydroartemisinin-piperaquine for treating uncomplicated malaria: a randomized trial to guide policy in Uganda.
    PloS one, 2008, Jun-11, Volume: 3, Issue:6

    Topics: Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Drug Therapy, Combination; Ethanolamines; Fluorenes; Health Policy; Humans; Infant; Lumefantrine; Malaria, Falciparum; Quinolines; Uganda

2008
[Efficacy of dihydroartemisinin-piperaquine and artemether-lumefantrine in the treatment of uncomplicated falciparum malaria in Hainan, China].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 2008, Feb-28, Volume: 26, Issue:1

    Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; China; Dose-Response Relationship, Drug; Drug Combinations; Ethanolamines; Female; Fluorenes; Follow-Up Studies; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Middle Aged; Quinolines; Treatment Outcome; Young Adult

2008
A trial of combination antimalarial therapies in children from Papua New Guinea.
    The New England journal of medicine, 2008, Dec-11, Volume: 359, Issue:24

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Child, Preschool; Chloroquine; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Infant; Kaplan-Meier Estimate; Lumefantrine; Malaria, Falciparum; Malaria, Vivax; Male; Proportional Hazards Models; Pyrimethamine; Quinolines; Recurrence; Sulfadoxine

2008
Dihydroartemisinin-piperaquine and artemether-lumefantrine for treating uncomplicated malaria in African children: a randomised, non-inferiority trial.
    PloS one, 2009, Nov-17, Volume: 4, Issue:11

    Topics: Africa; Antiparasitic Agents; Artemether; Artemisinins; Child, Preschool; Drug Therapy, Combination; Ethanolamines; Fluorenes; Humans; Infant; Lumefantrine; Malaria; Malaria, Falciparum; Plasmodium falciparum; Polymerase Chain Reaction; Quinolines; Time Factors

2009
Safety and tolerability of artemether-lumefantrine versus dihydroartemisinin-piperaquine for malaria in young HIV-infected and uninfected children.
    Malaria journal, 2009, Nov-30, Volume: 8

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Follow-Up Studies; HIV Infections; Humans; Infant; Longitudinal Studies; Malaria, Falciparum; Male; Quinolines; Risk Factors; Treatment Outcome; Uganda

2009
Population pharmacokinetics and pharmacodynamics of artemether and lumefantrine during combination treatment in children with uncomplicated falciparum malaria in Tanzania.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:11

    Topics: Antimalarials; Artemether; Artemisinins; Body Temperature; Child; Child, Preschool; Ethanolamines; Female; Fluorenes; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Tanzania; Treatment Outcome

2010
Increased risk of early vomiting among infants and young children treated with dihydroartemisinin-piperaquine compared with artemether-lumefantrine for uncomplicated malaria.
    The American journal of tropical medicine and hygiene, 2010, Volume: 83, Issue:4

    Topics: Antimalarials; Artemether; Artemisinins; Child, Preschool; Ethanolamines; Fluorenes; Humans; Infant; Lumefantrine; Malaria; Quinolines; Risk; Uganda; Vomiting

2010
Comparative study of the efficacy and tolerability of dihydroartemisinin-piperaquine-trimethoprim versus artemether-lumefantrine in the treatment of uncomplicated Plasmodium falciparum malaria in Cameroon, Ivory Coast and Senegal.
    Malaria journal, 2011, Jul-08, Volume: 10

    Topics: Adolescent; Adult; Animals; Antimalarials; Artemether; Artemisinins; Cameroon; Child; Child, Preschool; Cote d'Ivoire; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Male; Middle Aged; Quinolines; Senegal; Treatment Outcome; Trimethoprim; Young Adult

2011
Similar efficacy and safety of artemether-lumefantrine (Coartem®) in African infants and children with uncomplicated falciparum malaria across different body weight ranges.
    Malaria journal, 2011, Dec-16, Volume: 10

    Topics: Age Factors; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Body Weight; Child; Child, Preschool; Drug Combinations; Ethanolamines; Female; Fluorenes; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Plasmodium falciparum; Polymerase Chain Reaction; Time Factors; Treatment Outcome

2011
Efficacy of quinine, artemether-lumefantrine and dihydroartemisinin-piperaquine as rescue treatment for uncomplicated malaria in Ugandan children.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Child, Preschool; Ethanolamines; Fluorenes; Humans; Infant; Lumefantrine; Malaria, Falciparum; Male; Quinine; Quinolines; Safety; Treatment Outcome; Uganda

2013
Seasonal malaria chemoprevention in an area of extended seasonal transmission in Ashanti, Ghana: an individually randomised clinical trial.
    Tropical medicine & international health : TM & IH, 2016, Volume: 21, Issue:2

    Topics: Amodiaquine; Antimalarials; Artemether; Artemisinins; Chemoprevention; Child, Preschool; Drug Combinations; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Ghana; Humans; Infant; Infant, Newborn; Lumefantrine; Malaria; Male; Pyrimethamine; Quinolines; Rain; Seasons; Sulfadoxine

2016
Artemether-Lumefantrine Pharmacokinetics and Clinical Response Are Minimally Altered in Pregnant Ugandan Women Treated for Uncomplicated Falciparum Malaria.
    Antimicrobial agents and chemotherapy, 2015, Dec-14, Volume: 60, Issue:3

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Cohort Studies; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Middle Aged; Pregnancy; Pregnancy Complications, Parasitic; Prospective Studies; Treatment Outcome; Uganda; Young Adult

2015
The interaction between artemether-lumefantrine and lopinavir/ritonavir-based antiretroviral therapy in HIV-1 infected patients.
    BMC infectious diseases, 2016, Jan-27, Volume: 16

    Topics: Adult; Anti-HIV Agents; Artemether; Artemisinins; Drug Interactions; Ethanolamines; Female; Fluorenes; HIV Infections; HIV-1; Humans; Lopinavir; Lumefantrine; Male; Ritonavir

2016
Artemether-Lumefantrine versus Dihydroartemisinin-Piperaquine for Treatment of Uncomplicated Plasmodium falciparum Malaria in Children Aged Less than 15 Years in Guinea-Bissau - An Open-Label Non-Inferiority Randomised Clinical Trial.
    PloS one, 2016, Volume: 11, Issue:9

    Topics: Antimalarials; Artemether; Artemisinins; Child; Ethanolamines; Fluorenes; Guinea-Bissau; Humans; Lumefantrine; Malaria, Falciparum; Quinolines; Treatment Outcome

2016
A Randomized Controlled Trial of Three- versus Five-Day Artemether-Lumefantrine Regimens for Treatment of Uncomplicated Plasmodium falciparum Malaria in Pregnancy in Africa.
    Antimicrobial agents and chemotherapy, 2020, 02-21, Volume: 64, Issue:3

    Topics: Adult; Africa; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Female; Humans; Malaria, Falciparum; Pregnancy; Young Adult

2020
A randomized controlled trial of dihydroartemisinin-piperaquine, artesunate-mefloquine and extended artemether-lumefantrine treatments for malaria in pregnancy on the Thailand-Myanmar border.
    BMC medicine, 2021, 06-10, Volume: 19, Issue:1

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Artesunate; Drug Therapy, Combination; Female; Humans; Infant, Newborn; Malaria; Malaria, Falciparum; Mefloquine; Myanmar; Pregnancy; Premature Birth; Quinolines; Thailand

2021
Effectiveness and safety of reactive focal mass drug administration (rfMDA) using dihydroartemisinin-piperaquine to reduce malaria transmission in the very low-endemic setting of Eswatini: a pragmatic cluster randomised controlled trial.
    BMJ global health, 2021, Volume: 6, Issue:6

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Eswatini; Humans; Malaria; Mass Drug Administration; Quinolines

2021
Therapeutic efficacies of artemether-lumefantrine and dihydroartemisinin-piperaquine for the treatment of uncomplicated Plasmodium falciparum and chloroquine and dihydroartemisinin-piperaquine for uncomplicated Plasmodium vivax infection in Ethiopia.
    Malaria journal, 2022, Dec-01, Volume: 21, Issue:1

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Chloroquine; Ethiopia; Humans; Malaria, Falciparum; Malaria, Vivax; Plasmodium falciparum; Plasmodium vivax

2022
Safety of age-dosed, single low-dose primaquine in children with glucose-6-phosphate dehydrogenase deficiency who are infected with Plasmodium falciparum in Uganda and the Democratic Republic of the Congo: a randomised, double-blind, placebo-controlled, n
    The Lancet. Infectious diseases, 2023, Volume: 23, Issue:4

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Child; Democratic Republic of the Congo; Female; Glucosephosphate Dehydrogenase; Glucosephosphate Dehydrogenase Deficiency; Hemoglobins; Humans; Infant; Malaria, Falciparum; Male; Plasmodium falciparum; Primaquine; Uganda; World Health Organization

2023
Therapeutic response to artemisinin combination therapies among individuals with Plasmodium falciparum single infection vs mixed Plasmodium species infections: a retrospective posthoc analysis in Kisumu County, western Kenya.
    International journal of infectious diseases : IJID : official publication of the International Society for Infectious Diseases, 2023, Volume: 132

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Drug Combinations; Humans; Kenya; Malaria; Malaria, Falciparum; Plasmodium falciparum; Quinolines; Reinfection; Retrospective Studies

2023
Efficacy and safety of pyronaridine-artesunate (PYRAMAX) for the treatment of
    BMJ open, 2023, 10-09, Volume: 13, Issue:10

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Clinical Trials, Phase III as Topic; Drug Combinations; Female; Humans; Infant; Malaria; Malaria, Falciparum; Pregnancy; Pregnant Women; Randomized Controlled Trials as Topic; Sub-Saharan African People; Treatment Outcome

2023
Factors affecting haemoglobin dynamics in African children with acute uncomplicated Plasmodium falciparum malaria treated with single low-dose primaquine or placebo.
    BMC medicine, 2023, 10-20, Volume: 21, Issue:1

    Topics: alpha-Thalassemia; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Child; Child, Preschool; Female; Glucosephosphate Dehydrogenase Deficiency; Hemoglobins; Humans; Malaria, Falciparum; Male; Plasmodium falciparum; Primaquine

2023

Other Studies

87 other study(ies) available for artemether and artenimol

ArticleYear
Synthesis and biological evaluation of a series of non-hemiacetal ester derivatives of artemisinin.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: Animals; Antineoplastic Agents; Antiprotozoal Agents; Artemisinins; Cell Line, Tumor; Chemistry Techniques, Synthetic; CHO Cells; Cricetinae; Cricetulus; Drug Design; Esters; Humans; Plasmodium falciparum

2016
Arteether, a new antimalarial drug: synthesis and antimalarial properties.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Animals; Antimalarials; Artemisinins; Magnetic Resonance Spectroscopy; Malaria; Mice; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Sesquiterpenes

1988
Cytotoxicity of artemisinin-related endoperoxides to Ehrlich ascites tumor cells.
    Journal of natural products, 1993, Volume: 56, Issue:6

    Topics: Animals; Antineoplastic Agents, Phytogenic; Artemisinins; Carcinoma, Ehrlich Tumor; Cell Survival; Chemical Phenomena; Chemistry, Physical; Cisplatin; Doxorubicin; Peroxides; Sesquiterpenes; Structure-Activity Relationship; Tetrazolium Salts; Tumor Cells, Cultured

1993
Novel, potent, semisynthetic antimalarial carba analogues of the first-generation 1,2,4-trioxane artemether.
    Journal of medicinal chemistry, 1999, Dec-30, Volume: 42, Issue:26

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Plasmodium falciparum; Sesquiterpenes; Spectrophotometry, Infrared

1999
Synthesis and antimalarial activity of sixteen dispiro-1,2,4, 5-tetraoxanes: alkyl-substituted 7,8,15,16-tetraoxadispiro[5.2.5. 2]hexadecanes.
    Journal of medicinal chemistry, 2000, Jul-13, Volume: 43, Issue:14

    Topics: Alkanes; Animals; Antimalarials; Malaria; Mice; Neurites; Neuroblastoma; Plasmodium berghei; Plasmodium falciparum; Spiro Compounds; Structure-Activity Relationship; Tumor Cells, Cultured

2000
Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin.
    Journal of medicinal chemistry, 2001, Jan-04, Volume: 44, Issue:1

    Topics: Animals; Antimalarials; Artemisinins; Bile; Crystallography, X-Ray; Electron Spin Resonance Spectroscopy; Ferrous Compounds; Free Radicals; Malaria; Male; Mice; Phenyl Ethers; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Rats, Wistar; Sesquiterpenes; Stereoisomerism; Structure-Activity Relationship

2001
Spiro and dispiro-1,2,4-trioxolanes as antimalarial peroxides: charting a workable structure-activity relationship using simple prototypes.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Adamantane; Animals; Antimalarials; Cell Line, Tumor; Drug Resistance; Half-Life; Malaria; Malaria, Falciparum; Mice; Micronucleus Tests; Ozone; Peroxides; Plasmodium berghei; Rats; Spiro Compounds; Structure-Activity Relationship

2005
Antifungal activity of artemisinin derivatives.
    Journal of natural products, 2005, Volume: 68, Issue:8

    Topics: Antifungal Agents; Artemisinins; Candida albicans; Combinatorial Chemistry Techniques; Cryptococcus neoformans; Microbial Sensitivity Tests; Molecular Structure

2005
Effects of piperaquine, chloroquine, and amodiaquine on drug uptake and of these in combination with dihydroartemisinin against drug-sensitive and -resistant Plasmodium falciparum strains.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:6

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Chloroquine; Drug Antagonism; Drug Combinations; Drug Interactions; Drug Resistance; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Sesquiterpenes; Tritium

2007
Relationship between antimalarial activity and heme alkylation for spiro- and dispiro-1,2,4-trioxolane antimalarials.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:4

    Topics: Alkylation; Animals; Antimalarials; Artemisinins; Heme; Humans; Kinetics; Parasitic Sensitivity Tests; Plasmodium falciparum; Spiro Compounds; Structure-Activity Relationship

2008
In vitro and in vivo treatments of echinococcus protoscoleces and metacestodes with artemisinin and artemisinin derivatives.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:9

    Topics: Albendazole; Animals; Anti-Infective Agents; Antiparasitic Agents; Artemisinins; Drug Therapy, Combination; Echinococcosis; Echinococcus granulosus; Echinococcus multilocularis; Humans; Larva; Mice; Mice, Inbred BALB C; Nitro Compounds; Parasitic Sensitivity Tests; Thiazoles; Treatment Outcome

2008
Synthesis and biological evaluation of extraordinarily potent C-10 carba artemisinin dimers against P. falciparum malaria parasites and HL-60 cancer cells.
    Bioorganic & medicinal chemistry, 2009, Feb-01, Volume: 17, Issue:3

    Topics: Animals; Antimalarials; Antineoplastic Agents; Artemisinins; Cell Line, Tumor; Dimerization; HL-60 Cells; Humans; Plasmodium falciparum

2009
Antitumour and antimalarial activity of artemisinin-acridine hybrids.
    Bioorganic & medicinal chemistry letters, 2009, Apr-01, Volume: 19, Issue:7

    Topics: Acridines; Animals; Antimalarials; Antineoplastic Agents; Apoptosis; Artemisinins; Cell Cycle; Cell Line, Tumor; Erythrocytes; Flow Cytometry; G1 Phase; HL-60 Cells; Humans; Plasmodium falciparum

2009
Stability of peroxide antimalarials in the presence of human hemoglobin.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:8

    Topics: Antimalarials; Artemisinins; Drug Stability; Hemoglobins; Humans; Molecular Structure; Peroxides; Spectrophotometry

2009
Synthesis and anticancer activity of novel amide derivatives of non-acetal deoxoartemisinin.
    Bioorganic & medicinal chemistry letters, 2009, Nov-15, Volume: 19, Issue:22

    Topics: Acetals; Amides; Animals; Apoptosis; Artemisinins; Cell Proliferation; Drug Design; Drug Screening Assays, Antitumor; Endothelium, Vascular; Humans; Inhibitory Concentration 50; Mice; Mice, Nude; Neoplasm Transplantation; Structure-Activity Relationship

2009
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Selective determination, in plasma, of artemether and its major metabolite, dihydroartemisinin, by high-performance liquid chromatography with ultraviolet detection.
    Journal of chromatography, 1992, Nov-27, Volume: 583, Issue:1

    Topics: Artemether; Artemisinins; Chromatography, High Pressure Liquid; Humans; Schistosomicides; Sesquiterpenes; Spectrophotometry, Ultraviolet

1992
Hemolysis induced by artemisinin and its derivatives in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1986, Volume: 7, Issue:3

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Erythrocytes; Hemoglobins; Hemolysis; Humans; Pyrans; Sesquiterpenes

1986
The chemotherapy of rodent malaria, XL. The action of artemisinin and related sesquiterpenes.
    Annals of tropical medicine and parasitology, 1986, Volume: 80, Issue:5

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Drug Resistance; Malaria; Male; Mice; Pigments, Biological; Plasmodium berghei; Pyrans; Sesquiterpenes

1986
Rapid action of Qinghaosu and related drugs on incorporation of [3H]isoleucine by Plasmodium falciparum in vitro.
    Biochemical pharmacology, 1983, Sep-01, Volume: 32, Issue:17

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Isoleucine; Kinetics; Plasmodium falciparum; Protein Biosynthesis; Pyrans; Sesquiterpenes; Tritium

1983
Effects of qinghaosu and related compounds on incorporation of [G-3H] hypoxanthine by Plasmodium falciparum in vitro.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:4

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Hypoxanthine; Hypoxanthines; Plasmodium falciparum; Pyrans; Sesquiterpenes; Time Factors

1983
Uptake of [3H] dihydroartemisinine by erythrocytes infected with Plasmodium falciparum in vitro.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1984, Volume: 78, Issue:2

    Topics: Anisomycin; Antimalarials; Artemether; Artemisinins; Chloroquine; Erythrocytes; Humans; Plasmodium falciparum; Pyrans; Sesquiterpenes

1984
Determination of artemether and dihydroartemisinin in blood plasma by high-performance liquid chromatography for application in clinical pharmacological studies.
    Journal of chromatography. B, Biomedical applications, 1995, Jul-21, Volume: 669, Issue:2

    Topics: Adult; Antimalarials; Artemether; Artemisinins; Chromatography, High Pressure Liquid; Electrochemistry; Humans; Isomerism; Male; Reference Values; Reproducibility of Results; Sesquiterpenes

1995
Antimalarial activity of dihydroartemisinin derivatives by transdermal application.
    The American journal of tropical medicine and hygiene, 1994, Volume: 50, Issue:6

    Topics: Administration, Cutaneous; Animals; Antimalarials; Artemether; Artemisinins; Gels; Malaria; Mice; Plasmodium berghei; Sesquiterpenes; Structure-Activity Relationship

1994
Ferriprotoporphyrin catalysed decomposition of artemether: analytical and pharmacological implications.
    Biochemical pharmacology, 1994, Aug-30, Volume: 48, Issue:5

    Topics: Antimalarials; Artemether; Artemisinins; Carbon Radioisotopes; Catalysis; Chromatography, High Pressure Liquid; Hemin; Hemoglobins; Hemolysis; Humans; In Vitro Techniques; Sesquiterpenes; Spectrophotometry, Ultraviolet

1994
Pharmacokinetics of artemether after oral administration to healthy Thai males and patients with acute, uncomplicated falciparum malaria.
    British journal of clinical pharmacology, 1994, Volume: 37, Issue:3

    Topics: Administration, Oral; Adult; Animals; Antimalarials; Artemether; Artemisinins; Humans; Malaria, Falciparum; Male; Plasmodium falciparum; Sesquiterpenes; Thailand

1994
In vitro stage-specific sensitivity of Plasmodium falciparum to quinine and artemisinin drugs.
    International journal for parasitology, 1996, Volume: 26, Issue:5

    Topics: Adult; Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Chloroquine; Drug Evaluation, Preclinical; Drug Resistance; Humans; In Vitro Techniques; Malaria, Falciparum; Male; Middle Aged; Plasmodium falciparum; Quinine; Sesquiterpenes

1996
Determination of artemether and its major metabolite, dihydroartemisinin, in plasma using high-performance liquid chromatography with electrochemical detection.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Mar-07, Volume: 690, Issue:1-2

    Topics: Adult; Antimalarials; Artemether; Artemisinins; Chromatography, High Pressure Liquid; Electrochemistry; Humans; Isomerism; Male; Sensitivity and Specificity; Sesquiterpenes

1997
Determination of artemether and its metabolite, dihydroartemisinin, in plasma by high-performance liquid chromatography and electrochemical detection in the reductive mode.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Mar-28, Volume: 691, Issue:1

    Topics: Acetates; Acetonitriles; Antimalarials; Artemether; Artemisinins; Autoanalysis; Chromatography, High Pressure Liquid; Drug Stability; Humans; Quality Control; Sensitivity and Specificity; Sesquiterpenes

1997
The pharmacokinetics and bioavailability of dihydroartemisinin, arteether, artemether, artesunic acid and artelinic acid in rats.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:2

    Topics: Absorption; Animals; Antimalarials; Area Under Curve; Artemether; Artemisinins; Biological Availability; Bridged Bicyclo Compounds, Heterocyclic; Male; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Succinates

1998
Selection and characterization of Toxoplasma gondii mutants resistant to artemisinin.
    The Journal of infectious diseases, 1998, Volume: 177, Issue:4

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Artemether; Artemisinins; Drug Resistance; Ethyl Methanesulfonate; Female; Humans; Methylnitronitrosoguanidine; Mice; Mice, Inbred ICR; Mutagenesis; Sesquiterpenes; Toxoplasma; Toxoplasmosis, Animal

1998
In vitro neurotoxicity of artemisinin derivatives.
    Medecine tropicale : revue du Corps de sante colonial, 1998, Volume: 58, Issue:3 Suppl

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Cell Differentiation; Central Nervous System Diseases; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Mice; Microscopy, Electron; Neuroblastoma; Neurons; Reproducibility of Results; Sesquiterpenes; Tumor Cells, Cultured

1998
Simultaneous determination of artemether and its major metabolite dihydroartemisinin in plasma by gas chromatography-mass spectrometry-selected ion monitoring.
    Journal of chromatography. B, Biomedical sciences and applications, 1999, Aug-20, Volume: 731, Issue:2

    Topics: Adult; Antimalarials; Artemether; Artemisinins; Calibration; Gas Chromatography-Mass Spectrometry; Humans; Male; Reference Standards; Reference Values; Reproducibility of Results; Sensitivity and Specificity; Sesquiterpenes

1999
The role of glutathione in the neurotoxicity of artemisinin derivatives in vitro.
    Biochemical pharmacology, 2001, Feb-15, Volume: 61, Issue:4

    Topics: Animals; Antimalarials; Antimetabolites; Antioxidants; Artemether; Artemisinins; Buthionine Sulfoximine; Drug Interactions; Glutathione; Hemin; Humans; Mice; Neurites; Sesquiterpenes; Tumor Cells, Cultured

2001
Ammunition against malaria.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 2001, Sep-04, Volume: 165, Issue:5

    Topics: Antimalarials; Artemether; Artemisinins; Canada; Humans; Malaria; Sesquiterpenes

2001
The development of new antimalarial drugs: qinghaosu and dihydro-qinghaosu.
    Chinese medical journal, 1999, Volume: 112, Issue:11

    Topics: Animals; Antimalarials; Artemether; Artemisia; Artemisinins; Artesunate; Drugs, Chinese Herbal; Humans; Sesquiterpenes

1999
Authentication of artemether, artesunate and dihydroartemisinin antimalarial tablets using a simple colorimetric method.
    Tropical medicine & international health : TM & IH, 2001, Volume: 6, Issue:12

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Colorimetry; Diazonium Compounds; Sesquiterpenes; Tablets

2001
Development and validation of a high-performance liquid chromatography-mass spectrometry assay for the determination of artemether and its metabolite dihydroartemisinin in human plasma.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2002, Jul-15, Volume: 774, Issue:2

    Topics: Antimalarials; Artemether; Artemisinins; Calibration; Chromatography, High Pressure Liquid; Humans; Mass Spectrometry; Reproducibility of Results; Sensitivity and Specificity; Sesquiterpenes

2002
[Pharmacokinetic studies on artemether under conditions simulated in vivo].
    Se pu = Chinese journal of chromatography, 2002, Volume: 20, Issue:1

    Topics: Artemether; Artemisinins; Biological Availability; Chromatography, High Pressure Liquid; Hydrogen-Ion Concentration; Patient Simulation; Sesquiterpenes

2002
Population pharmacokinetics of artemether and dihydroartemisinin following single intramuscular dosing of artemether in African children with severe falciparum malaria.
    British journal of clinical pharmacology, 2004, Volume: 57, Issue:2

    Topics: Acidosis, Respiratory; Antimalarials; Artemether; Artemisinins; Child; Child, Preschool; Female; Half-Life; Humans; Infant; Injections, Intramuscular; Malaria, Falciparum; Male; Respiratory Insufficiency; Sesquiterpenes

2004
Design of a dissolution system for the evaluation of the release rate characteristics of artemether and dihydroartemisinin from tablets.
    International journal of pharmaceutics, 2004, Apr-15, Volume: 274, Issue:1-2

    Topics: Artemether; Artemisinins; Calibration; Chromatography, High Pressure Liquid; Drug Evaluation, Preclinical; Rotation; Sesquiterpenes; Solubility; Solvents; Tablets

2004
[Effects of combined artemether and dihydroarteamisinin in treatment of children with falciparum malaria].
    Zhonghua er ke za zhi = Chinese journal of pediatrics, 2005, Volume: 43, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Child; Drug Therapy, Combination; Humans; Malaria, Falciparum

2005
Artesunate and artemether are effective fasciolicides in the rat model and in vitro.
    The Journal of antimicrobial chemotherapy, 2006, Volume: 57, Issue:6

    Topics: Animals; Antiplatyhelmintic Agents; Artemether; Artemisinins; Artesunate; Bile Ducts; Disease Models, Animal; Fasciola hepatica; Fascioliasis; Female; Microscopy, Electron, Scanning; Rats; Rats, Wistar; Sesquiterpenes

2006
Quality control of active ingredients in artemisinin-derivative antimalarials within Kenya and DR Congo.
    Tropical medicine & international health : TM & IH, 2007, Volume: 12, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Capsules; Chromatography, High Pressure Liquid; Democratic Republic of the Congo; Dosage Forms; Endemic Diseases; Humans; Kenya; Malaria, Falciparum; Quality Control; Sesquiterpenes; Tablets

2007
Experimental therapy of hepatoma with artemisinin and its derivatives: in vitro and in vivo activity, chemosensitization, and mechanisms of action.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2008, Sep-01, Volume: 14, Issue:17

    Topics: Animals; Antineoplastic Agents; Artemether; Artemisinins; Artesunate; Carcinoma, Hepatocellular; Cell Cycle; Cell Line, Tumor; Female; Gene Expression Regulation, Neoplastic; Humans; Liver; Liver Neoplasms; Mice; Mice, Nude; Xenograft Model Antitumor Assays

2008
Antimalarial therapies in children from Papua New Guinea.
    The New England journal of medicine, 2009, Mar-19, Volume: 360, Issue:12

    Topics: Antimalarials; Artemether; Artemisinins; Biological Availability; Drug Therapy, Combination; Ethanolamines; Fats; Fluorenes; Humans; Lumefantrine; Malaria; Quinolines; Treatment Failure

2009
Development and validation of a high-performance liquid chromatography/tandem mass spectrometry method for the determination of artemether and its active metabolite dihydroartemisinin in human plasma.
    Journal of pharmaceutical and biomedical analysis, 2009, Dec-05, Volume: 50, Issue:5

    Topics: Antimalarials; Artemether; Artemisinins; Calibration; Chromatography, High Pressure Liquid; Formates; HIV Infections; Humans; Malaria; Models, Chemical; Quality Control; Reproducibility of Results; Solid Phase Extraction; Tandem Mass Spectrometry; Time Factors

2009
Selection of known Plasmodium falciparum resistance-mediating polymorphisms by artemether-lumefantrine and amodiaquine-sulfadoxine-pyrimethamine but not dihydroartemisinin-piperaquine in Burkina Faso.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:5

    Topics: Amodiaquine; Antimalarials; Artemether; Artemisinins; Burkina Faso; Drug Combinations; Drug Resistance, Bacterial; Ethanolamines; Fluorenes; Genotype; Humans; Infant; Lumefantrine; Malaria, Falciparum; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Pyrimethamine; Quinolines; Randomized Controlled Trials as Topic; Recurrence; Sulfadoxine

2010
Pharmacokinetics of artemether and dihydroartemisinin in healthy Pakistani male volunteers treated with artemether-lumefantrine.
    Malaria journal, 2010, Oct-11, Volume: 9

    Topics: Administration, Oral; Adult; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Chromatography, Liquid; Drug Combinations; Ethanolamines; Fluorenes; Human Experimentation; Humans; Male; Middle Aged; Pakistan; Plasma; Tandem Mass Spectrometry; Time Factors

2010
A liquid chromatographic-tandem mass spectrometric method for determination of artemether and its metabolite dihydroartemisinin in human plasma.
    Bioanalysis, 2009, Volume: 1, Issue:1

    Topics: Antimalarials; Artemether; Artemisinins; Calibration; Chromatography, Liquid; Drug Therapy, Combination; Ethanolamines; Fluorenes; High-Throughput Screening Assays; Humans; Lumefantrine; Malaria, Falciparum; Reproducibility of Results; Solid Phase Extraction; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry

2009
The multiple-dosing pharmacokinetics of artemether, artesunate, and their metabolite dihydroartemisinin in rats.
    Xenobiotica; the fate of foreign compounds in biological systems, 2011, Volume: 41, Issue:3

    Topics: Administration, Oral; Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Male; Rats; Rats, Wistar

2011
Development and validation of a liquid chromatography and ion spray tandem mass spectrometry method for the quantification of artesunate, artemether and their major metabolites dihydroartemisinin and dihydroartemisinin-glucuronide in sheep plasma.
    Journal of mass spectrometry : JMS, 2011, Volume: 46, Issue:2

    Topics: Animals; Artemether; Artemisinins; Artesunate; Calibration; Chromatography, Liquid; Chromatography, Reverse-Phase; Glucuronides; Logistic Models; Reproducibility of Results; Sensitivity and Specificity; Sheep; Tandem Mass Spectrometry

2011
Effects of artemether, artesunate and dihydroartemisinin administered orally at multiple doses or combination in treatment of mice infected with Schistosoma japonicum.
    Parasitology research, 2011, Volume: 109, Issue:2

    Topics: Administration, Oral; Animals; Antiprotozoal Agents; Artemether; Artemisinins; Artesunate; Disease Models, Animal; Female; Mice; Rodent Diseases; Schistosoma japonicum; Schistosomiasis japonica; Treatment Outcome

2011
Meningeal inflammation increases artemether concentrations in cerebrospinal fluid in Papua New Guinean children treated with intramuscular artemether.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:11

    Topics: Artemether; Artemisinins; Child; Child, Preschool; Female; Humans; Infant; Injections, Intramuscular; Malaria, Falciparum; Male; Meninges; Papua New Guinea; Prospective Studies

2011
Monitoring of artemisinin, dihydroartemisinin, and artemether in environmental matrices using high-performance liquid chromatography-tandem mass spectrometry (LC-MS/MS).
    Journal of agricultural and food chemistry, 2011, Nov-09, Volume: 59, Issue:21

    Topics: Artemether; Artemisia annua; Artemisinins; Chromatography, High Pressure Liquid; Kenya; Plant Extracts; Soil; Tandem Mass Spectrometry

2011
Metabolite identification of artemether by data-dependent accurate mass spectrometric analysis using an LTQ-Orbitrap hybrid mass spectrometer in combination with the online hydrogen/deuterium exchange technique.
    Rapid communications in mass spectrometry : RCM, 2011, Nov-15, Volume: 25, Issue:21

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Bile; Chromatography, Liquid; Deuterium Exchange Measurement; Hydroxylation; Male; Mass Spectrometry; Methylation; Microsomes, Liver; Rats; Rats, Wistar; Tandem Mass Spectrometry

2011
Population pharmacokinetics of Artemether and dihydroartemisinin in pregnant women with uncomplicated Plasmodium falciparum malaria in Uganda.
    Malaria journal, 2012, Aug-22, Volume: 11

    Topics: Administration, Oral; Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Chromatography; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Mass Spectrometry; Models, Statistical; Plasma; Pregnancy; Pregnancy Complications, Infectious; Uganda; Young Adult

2012
Heat stabilization of blood spot samples for determination of metabolically unstable drug compounds.
    Bioanalysis, 2013, Volume: 5, Issue:1

    Topics: Amodiaquine; Analytic Sample Preparation Methods; Artemether; Artemisinins; Butyrylcholinesterase; Cefotaxime; Dried Blood Spot Testing; Drug Stability; Hot Temperature; Humans; Oseltamivir; Pharmaceutical Preparations

2013
Lower artemether, dihydroartemisinin and lumefantrine concentrations during rifampicin-based tuberculosis treatment.
    AIDS (London, England), 2013, Mar-27, Volume: 27, Issue:6

    Topics: Adult; Antimalarials; Antitubercular Agents; Artemether; Artemisinins; Drug Antagonism; Ethanolamines; Female; Fluorenes; HIV Infections; Humans; Longitudinal Studies; Lumefantrine; Male; Rifampin; Tuberculosis; Uganda

2013
Determination of artemether and dihydroartemisinin in human plasma with a new hydrogen peroxide stabilization method.
    Bioanalysis, 2013, Volume: 5, Issue:12

    Topics: Antimalarials; Artemether; Artemisinins; Chromatography, High Pressure Liquid; Humans; Hydrogen Peroxide; Isotope Labeling; Tandem Mass Spectrometry; Temperature

2013
Pharmacokinetic properties of artemether, dihydroartemisinin, lumefantrine, and quinine in pregnant women with uncomplicated plasmodium falciparum malaria in Uganda.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:10

    Topics: Adolescent; Adult; Artemether; Artemisinins; Ethanolamines; Female; Fluorenes; Humans; Lumefantrine; Malaria, Falciparum; Pregnancy; Quinine; Young Adult

2013
Validation of ELISA for quantitation of artemisinin-based antimalarial drugs.
    The American journal of tropical medicine and hygiene, 2013, Volume: 89, Issue:6

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Chromatography, High Pressure Liquid; Confidence Intervals; Counterfeit Drugs; Enzyme-Linked Immunosorbent Assay

2013
Effects of artemisinin antimalarials on Cytochrome P450 enzymes in vitro using recombinant enzymes and human liver microsomes: potential implications for combination therapies.
    Xenobiotica; the fate of foreign compounds in biological systems, 2014, Volume: 44, Issue:7

    Topics: Antimalarials; Artemether; Artemisinins; Artesunate; Cytochrome P-450 CYP1A2; Cytochrome P-450 CYP2C19; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Evaluation, Preclinical; Drug Interactions; Humans; Inhibitory Concentration 50; Microsomes, Liver; Recombinant Proteins; Tandem Mass Spectrometry

2014
A high-performance liquid chromatography-tandem mass spectrometry method for the determination of artemether and dihydroartemisinin in human plasma.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2014, Aug-15, Volume: 965

    Topics: Artemether; Artemisinins; Chromatography, High Pressure Liquid; Humans; Linear Models; Reproducibility of Results; Sensitivity and Specificity; Tandem Mass Spectrometry

2014
Interspecies allometric scaling of antimalarial drugs and potential application to pediatric dosing.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:10

    Topics: Age Factors; Antimalarials; Artemether; Artemisinins; Artesunate; Child; Child, Preschool; Female; Humans; Male; Models, Theoretical

2014
[Therapeutic effect of 138 imported falciparum malaria patients].
    Zhongguo xue xi chong bing fang zhi za zhi = Chinese journal of schistosomiasis control, 2014, Volume: 26, Issue:6

    Topics: Adult; Africa; Antimalarials; Artemether; Artemisinins; Artesunate; China; Diagnostic Errors; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Plasmodium falciparum; Retrospective Studies; Travel; Young Adult

2014
NO-Donor Dihydroartemisinin Derivatives as Multitarget Agents for the Treatment of Cerebral Malaria.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antimalarials; Artemether; Artemisinins; Artesunate; Chemistry Techniques, Synthetic; Malaria, Cerebral; Mice; Molecular Targeted Therapy; Muscle Relaxation; Nitric Oxide Donors; Plasmodium berghei; Rats; Vasodilator Agents

2015
Artemether-Lumefantrine Exposure in HIV-Infected Nigerian Subjects on Nevirapine-Containing Antiretroviral Therapy.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:12

    Topics: Adult; Anti-HIV Agents; Antimalarials; Artemether; Artemisinins; Case-Control Studies; Coinfection; Drug Combinations; Drug Interactions; Ethanolamines; Female; Fluorenes; HIV Infections; HIV-1; Humans; Lumefantrine; Malaria, Falciparum; Male; Nevirapine; Nigeria; Plasmodium falciparum

2015
Genetic Transformation of Artemisia carvifolia Buch with rol Genes Enhances Artemisinin Accumulation.
    PloS one, 2015, Volume: 10, Issue:10

    Topics: Agrobacterium tumefaciens; Antimalarials; Artemether; Artemisia annua; Artemisinins; Artesunate; Base Sequence; Biosynthetic Pathways; Gene Expression Regulation, Plant; Molecular Sequence Data; Plant Proteins; Plants, Genetically Modified; Transformation, Genetic; Trichomes

2015
The Spiroindolone KAE609 Does Not Induce Dormant Ring Stages in Plasmodium falciparum Parasites.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:9

    Topics: Antimalarials; Artemether; Artemisinins; Drug Resistance; Erythrocytes; Ethanolamines; Fluorenes; Humans; Indoles; Inhibitory Concentration 50; Life Cycle Stages; Lumefantrine; Plasmodium falciparum; Rhodamine 123; Spiro Compounds

2016
Hemolysis after Oral Artemisinin Combination Therapy for Uncomplicated Plasmodium falciparum Malaria.
    Emerging infectious diseases, 2016, Volume: 22, Issue:8

    Topics: Administration, Oral; Adolescent; Adult; Anemia; Antimalarials; Artemether; Artemisinins; Child; Drug Therapy, Combination; Ethanolamines; Female; Fluorenes; Hemolysis; Humans; Lumefantrine; Malaria, Falciparum; Male; Prospective Studies; Quinolines

2016
Endoperoxide Drug Cross-Resistance Patterns for Plasmodium falciparum Exhibiting an Artemisinin Delayed-Clearance Phenotype.
    Antimicrobial agents and chemotherapy, 2016, Volume: 60, Issue:11

    Topics: Adamantane; Antimalarials; Artemether; Artemisinins; Dose-Response Relationship, Drug; Drug Resistance; Heterocyclic Compounds, 1-Ring; Inactivation, Metabolic; Lethal Dose 50; Microbial Sensitivity Tests; Peroxides; Plasmodium falciparum; Spiro Compounds

2016
Effects of Dihydroartemisinin and Artemether on the Growth, Chlorophyll Fluorescence, and Extracellular Alkaline Phosphatase Activity of the Cyanobacterium Microcystis aeruginosa.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alkaline Phosphatase; Artemether; Artemisinins; Bacterial Proteins; Chlorophyll; Chlorophyll A; Electron Transport; Malondialdehyde; Microcystis; Photosynthesis; Photosystem II Protein Complex; Spectrometry, Fluorescence

2016
A sensitive, high-throughput, and ecofriendly method for the determination of lumefantrine, artemether, and its active metabolite dihydroartemisinin by supercritical fluid chromatography and tandem mass spectrometry.
    Journal of separation science, 2018, Volume: 41, Issue:12

    Topics: Animals; Artemether; Artemisinins; Chromatography, Supercritical Fluid; Ethanolamines; Fluorenes; Lumefantrine; Male; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Tandem Mass Spectrometry

2018
Population Pharmacokinetics of Artemether, Dihydroartemisinin, and Lumefantrine in Rwandese Pregnant Women Treated for Uncomplicated Plasmodium falciparum Malaria.
    Antimicrobial agents and chemotherapy, 2018, Volume: 62, Issue:10

    Topics: Adolescent; Adult; Antimalarials; Artemether; Artemisinins; Female; Humans; Lumefantrine; Malaria, Falciparum; Pregnancy; Tandem Mass Spectrometry; Young Adult

2018
Comparison of in vitro/in vivo blood distribution and pharmacokinetics of artemisinin, artemether and dihydroartemisinin in rats.
    Journal of pharmaceutical and biomedical analysis, 2019, Jan-05, Volume: 162

    Topics: Administration, Oral; Animals; Antimalarials; Artemether; Artemisinins; Chromatography, Liquid; Drug Monitoring; Injections, Intravenous; Male; Rats, Sprague-Dawley; Tandem Mass Spectrometry; Tissue Distribution

2019
Evaluation of the effects on the QT-interval of 4 artemisinin-based combination therapies with a correction-free and heart rate-free method.
    Scientific reports, 2019, 01-29, Volume: 9, Issue:1

    Topics: Adolescent; Amodiaquine; Antimalarials; Arrhythmias, Cardiac; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Child; Child, Preschool; Drug Combinations; Ethanolamines; Female; Fluorenes; Heart Rate; Humans; Long QT Syndrome; Malaria; Malaria, Falciparum; Male; Quinolines; Young Adult

2019
Efavirenz-Based Antiretroviral Therapy Reduces Artemether-Lumefantrine Exposure for Malaria Treatment in HIV-Infected Pregnant Women.
    Journal of acquired immune deficiency syndromes (1999), 2020, 02-01, Volume: 83, Issue:2

    Topics: Adolescent; Adult; Alkynes; Anti-HIV Agents; Anti-Retroviral Agents; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Benzoxazines; Cyclopropanes; Drug Combinations; Drug Interactions; Female; HIV Infections; Humans; Lumefantrine; Malaria; Malaria, Falciparum; Pregnancy; Prospective Studies; Uganda; Young Adult

2020
A Chemically Stable Fluorescent Mimic of Dihydroartemisinin, Artemether, and Arteether with Conserved Bioactivity and Specificity Shows High Pharmacological Relevance to the Antimalarial Drugs.
    ACS infectious diseases, 2020, 07-10, Volume: 6, Issue:7

    Topics: Antimalarials; Artemether; Artemisinins

2020
Leishmania amazonensis response to artemisinin and derivatives.
    Parasitology international, 2021, Volume: 80

    Topics: Animals; Artemether; Artemisinins; Artesunate; Disease Models, Animal; Female; Leishmania mexicana; Mice; Mice, Inbred BALB C; Parasite Load; Trypanocidal Agents

2021
Electrocardiographic effect of artemisinin-piperaquine, dihydroartemisinin-piperaquine, and artemether-lumefantrine treatment in falciparum malaria patients.
    Revista da Sociedade Brasileira de Medicina Tropical, 2021, Volume: 54

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Drug Combinations; Electrocardiography; Humans; Malaria; Malaria, Falciparum; Quinolines

2021
Efficacy of Artemether-Lumefantrine and Dihydroartemisinin-Piperaquine for the Treatment of Uncomplicated Plasmodium falciparum Malaria among Children in Western Kenya, 2016 to 2017.
    Antimicrobial agents and chemotherapy, 2022, 09-20, Volume: 66, Issue:9

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Child; Drug Combinations; Ethanolamines; Fluorenes; Folic Acid Antagonists; Humans; Infant; Kenya; Malaria; Malaria, Falciparum; Piperazines; Plasmodium falciparum; Quinolines; Reinfection

2022
Exploring the Potential Mechanism of Artemisinin and Its Derivatives in the Treatment of Osteoporosis Based on Network Pharmacology and Molecular Docking.
    Computational and mathematical methods in medicine, 2022, Volume: 2022

    Topics: Artemether; Artemisinins; Artesunate; Caspase 3; Drugs, Chinese Herbal; ErbB Receptors; Humans; Interleukin-17; Mitogen-Activated Protein Kinase 14; Molecular Docking Simulation; Network Pharmacology; Osteoporosis; Prolactin

2022
Assessment of artemisinin tolerance in Plasmodium falciparum clinical isolates in children with uncomplicated malaria in Ghana.
    Malaria journal, 2023, Feb-19, Volume: 22, Issue:1

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Artemisinins; Child; Drug Combinations; Drug Tolerance; Ghana; Humans; Lumefantrine; Malaria; Malaria, Falciparum; Plasmodium falciparum

2023
Anticancer Activity and Molecular Mechanisms of an Ursodeoxycholic Acid Methyl Ester-Dihydroartemisinin Hybrid via a Triazole Linkage in Hepatocellular Carcinoma Cells.
    Molecules (Basel, Switzerland), 2023, Mar-03, Volume: 28, Issue:5

    Topics: Apoptosis; Artemether; Carcinoma, Hepatocellular; Cell Line, Tumor; Humans; Liver Neoplasms; Tandem Mass Spectrometry; Ursodeoxycholic Acid

2023
Design, Implementation, and Coordination of Malaria Therapeutic Efficacy Studies in Nigeria in 2018.
    The American journal of tropical medicine and hygiene, 2023, 06-07, Volume: 108, Issue:6

    Topics: Amodiaquine; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Child; Drug Combinations; Ethanolamines; Fluorenes; Humans; Malaria; Malaria, Falciparum; Nigeria

2023
Prevalence of mutations in the cysteine desulfurase IscS (Pfnfs1) gene in recurrent Plasmodium falciparum infections following artemether-lumefantrine (AL) and dihydroartemisinin-piperaquine (DP) treatment in Matayos, Western Kenya.
    Malaria journal, 2023, May-19, Volume: 22, Issue:1

    Topics: Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Drug Combinations; Humans; Kenya; Lumefantrine; Malaria; Malaria, Falciparum; Mutation; Plasmodium falciparum; Prevalence; Quinolines; Reinfection

2023