Page last updated: 2024-08-26

arsenic and pentamidine

arsenic has been researched along with pentamidine in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199011 (40.74)18.7374
1990's6 (22.22)18.2507
2000's7 (25.93)29.6817
2010's2 (7.41)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Duke, BO1
Jennings, FW1
Brun, R; Kunz, C1
Baeriswyl, S; Brun, R; Kunz, C1
Williamson, J2
Dukes, P1
Boa Yapo, F; Doua, F1
Berger, BJ; Carter, NS; Fairlamb, AH1
Baltz, T; Barrett, MP; Denise, H; Giroud, C; Zhang, ZQ1
Scott, AG; Tait, A; Turner, CM1
Barrett, MP; Fairlamb, AH1
De Koning, HP3
Legros, D; Ollivier, G1
NEUJEAN, G1
HAWKING, F; SEN, AB1
ROLLO, IM; WILLIAMSON, J1
Barrett, MP; Brun, R; Burchmore, RJ; de Koning, HP; Enyaru, JC; Geiser, F; Kaminsky, R; Mäser, P; Matovu, E; Seebeck, T; Stewart, ML; Wallace, LJ1
Ebert, SN; Katchman, AN; Koerner, J; Tosaka, T; Woosley, RL1
Bridges, DJ; Burchmore, RJ; de Koning, HP; Gould, MK; Mäser, P; Nerima, B1
Arafa, RK; Boykin, DW; Brun, R; Gillingwater, K; Ismail, MA; Kumar, A; Stephens, CE; Tidwell, RR1
HARDING, RD1
Castagné, V; Goineau, S1
Alghamdi, AH; Campagnaro, GD; de Koning, HP; Natto, MJ; Ungogo, MA1

Reviews

2 review(s) available for arsenic and pentamidine

ArticleYear
The biochemical basis of arsenical-diamidine crossresistance in African trypanosomes.
    Parasitology today (Personal ed.), 1999, Volume: 15, Issue:4

    Topics: Animals; Arsenicals; Cattle; Drug Resistance; Humans; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African; Trypanosomiasis, Bovine

1999
Transporters in African trypanosomes: role in drug action and resistance.
    International journal for parasitology, 2001, May-01, Volume: 31, Issue:5-6

    Topics: Africa South of the Sahara; Animals; Arsenicals; Biological Transport; Eflornithine; Humans; Nitroimidazoles; Pentamidine; Phenanthridines; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis, African

2001

Other Studies

25 other study(ies) available for arsenic and pentamidine

ArticleYear
The effects of some drugs--pentamidine, stibocaptate, Hoechst 33258, F 151, compound 'E' and Nifurtimox--on Onchocerca volvulus in chimpanzees.
    Tropenmedizin und Parasitologie, 1977, Volume: 28, Issue:4

    Topics: Animals; Anthelmintics; Antimony; Arsenicals; Bisbenzimidazole; Female; Male; Nifurtimox; Onchocerca; Onchocerciasis; Organometallic Compounds; Pan troglodytes; Pentamidine; Succimer; Succinates

1977
Chemotherapy of sleeping sickness.
    The Central African journal of medicine, 1979, Volume: 25, Issue:11

    Topics: Arsenicals; Humans; Melarsoprol; Pentamidine; Suramin; Trypanosomiasis, African

1979
Chemotherapy of CNS-trypanosomiasis: the combined use of diminazene aceturate or pentamidine with DL-alpha-difluoromethylornithine (DFMO).
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1992, Volume: 43, Issue:2

    Topics: Animals; Arsenicals; Central Nervous System Diseases; Diminazene; Drug Administration Schedule; Drug Therapy, Combination; Eflornithine; Female; Mice; Pentamidine; Treatment Outcome; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1992
In vitro drug sensitivity test for Trypanosoma brucei subgroup bloodstream trypomastigotes.
    Acta tropica, 1989, Volume: 46, Issue:5-6

    Topics: Animals; Arsenicals; Diminazene; Hypoxanthine; Hypoxanthines; Leucine; Pentamidine; Phenanthridines; Suramin; Thymidine; Trypanocidal Agents; Trypanosoma brucei brucei

1989
In vitro drug sensitivity of Trypanosoma gambiense isolates.
    Acta tropica, 1989, Volume: 46, Issue:5-6

    Topics: Animals; Arsenicals; Cote d'Ivoire; Humans; Melarsoprol; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei gambiense; Trypanosomiasis, African

1989
Drug sensitivity of pleomorphic Trypanosoma rhodesiense.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:2

    Topics: Animals; Arsenicals; Drug Resistance, Microbial; Ethidium; Mice; Pentamidine; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis, African

1983
Arsenic and old taxa: subspeciation and drug sensitivity in Trypanosoma brucei.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1984, Volume: 78, Issue:6

    Topics: Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance, Microbial; Isoenzymes; Male; Melarsoprol; Mice; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1984
[Current therapy of trypanosomiasis].
    Bulletin de la Societe de pathologie exotique (1990), 1994, Volume: 87, Issue:5

    Topics: Adenosylmethionine Decarboxylase; Animals; Arsenicals; Deoxyadenosines; Drug Resistance; Eflornithine; Enzyme Inhibitors; Hospitalization; Humans; Melarsoprol; Pentamidine; Randomized Controlled Trials as Topic; Recurrence; Suramin; Triazines; Trypanocidal Agents; Trypanosomiasis, African

1994
Uptake of diamidine drugs by the P2 nucleoside transporter in melarsen-sensitive and -resistant Trypanosoma brucei brucei.
    The Journal of biological chemistry, 1995, Nov-24, Volume: 270, Issue:47

    Topics: Adenosine; Animals; Arsenicals; Biological Transport; Carrier Proteins; Drug Resistance; Kinetics; Pentamidine; Species Specificity; Structure-Activity Relationship; Trypanosoma brucei brucei

1995
A diamidine-resistant Trypanosoma equiperdum clone contains a P2 purine transporter with reduced substrate affinity.
    Molecular and biochemical parasitology, 1995, Volume: 73, Issue:1-2

    Topics: Adenosine; Animals; Arsenicals; Biological Transport, Active; Carrier Proteins; Diminazene; Drug Resistance; Kinetics; Pentamidine; Receptors, Purinergic P2; Trypanocidal Agents; Trypanosoma

1995
Trypanosoma brucei: lack of cross-resistance to melarsoprol in vitro by cymelarsan-resistant parasites.
    Experimental parasitology, 1997, Volume: 86, Issue:3

    Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Female; Inosine; Melarsoprol; Mice; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei

1997
Uptake of pentamidine in Trypanosoma brucei brucei is mediated by three distinct transporters: implications for cross-resistance with arsenicals.
    Molecular pharmacology, 2001, Volume: 59, Issue:3

    Topics: Animals; Arsenicals; Biological Transport; Drug Resistance; Pentamidine; Phosphoprotein Phosphatases; Tritium; Trypanocidal Agents; Trypanosoma brucei brucei

2001
[Human african trypanosomiasis: A history of its therapies and their failures].
    Tropical medicine & international health : TM & IH, 2001, Volume: 6, Issue:11

    Topics: Arsenicals; Drug Resistance; History, 20th Century; History, 21st Century; Humans; Melarsoprol; Pentamidine; Treatment Outcome; Trypanocidal Agents; Trypanosomiasis, African

2001
[Chemotherapy and chemoprophylaxis of sleeping sickness caused by Trypanosoma gambiense].
    Revue medicale de Liege, 1959, Jan-01, Volume: 14, Issue:1

    Topics: Animals; Arsenicals; Chemoprevention; Humans; Pentamidine; Suramin; Trypanosoma brucei gambiense; Trypanosomiasis; Trypanosomiasis, African

1959
The trypanocidal action of homidium, quinapyramine and suramin.
    British journal of pharmacology and chemotherapy, 1960, Volume: 15

    Topics: Animals; Arsenicals; Ethidium; Mice; Pentamidine; Quinolines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis

1960
Drug resistance in trapanososmes: cross-resitance analyses.
    British journal of pharmacology and chemotherapy, 1959, Volume: 14

    Topics: Aminoquinolines; Arsenicals; Drug Resistance; Humans; Pentamidine; Phenanthridines; Stilbamidines; Suramin; Trypanosoma; Trypanosoma brucei rhodesiense

1959
Drug resistance in trypanosomes: selective interference with trypanocidal action.
    British journal of pharmacology and chemotherapy, 1959, Volume: 14

    Topics: 4-Aminobenzoic Acid; Arsenicals; Drug Resistance; Pentamidine; Trypanosoma

1959
Mechanisms of arsenical and diamidine uptake and resistance in Trypanosoma brucei.
    Eukaryotic cell, 2003, Volume: 2, Issue:5

    Topics: Adenine; Adenosine; Animals; Arsenicals; Benzamidines; Cell Death; Cell Division; Diminazene; Drug Resistance; Female; Gene Silencing; Hypoxanthine; Inhibitory Concentration 50; Inosine; Melarsoprol; Mice; Mutation; Nucleoside Transport Proteins; Pentamidine; Stilbamidines; Trypanosoma brucei brucei

2003
Comparative evaluation of HERG currents and QT intervals following challenge with suspected torsadogenic and nontorsadogenic drugs.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 316, Issue:3

    Topics: Animals; Arsenic Trioxide; Arsenicals; Cells, Cultured; Electrocardiography; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Haloperidol; Humans; Loratadine; Lovastatin; Methadone; Oxides; Pentamidine; Potassium Channel Blockers; Rabbits; Terfenadine; Torsades de Pointes

2006
Loss of the high-affinity pentamidine transporter is responsible for high levels of cross-resistance between arsenical and diamidine drugs in African trypanosomes.
    Molecular pharmacology, 2007, Volume: 71, Issue:4

    Topics: Animals; Arsenicals; Carrier Proteins; Drug Resistance; Female; Nucleoside Transport Proteins; Pentamidine; Protozoan Proteins; Rats; Rats, Wistar; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2007
Ever-increasing complexities of diamidine and arsenical crossresistance in African trypanosomes.
    Trends in parasitology, 2008, Volume: 24, Issue:8

    Topics: Animals; Arsenicals; Drug Resistance; Humans; Molecular Structure; Pentamidine; Trypanocidal Agents; Trypanosoma brucei gambiense; Trypanosomiasis, African

2008
In vitro activity and preliminary toxicity of various diamidine compounds against Trypanosoma evansi.
    Veterinary parasitology, 2010, May-11, Volume: 169, Issue:3-4

    Topics: Amidines; Animals; Arsenicals; Cells, Cultured; Diminazene; Drug Resistance; Female; Inhibitory Concentration 50; Mice; Pentamidine; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2010
Late results of treatment of sleeping sickness in Sierra Leone by antrypol tryparsamide pentamidine and propamidine singly and in various combinations.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1945, Volume: 39, Issue:2

    Topics: Animals; Arsenicals; Benzamidines; Humans; Pentamidine; Sierra Leone; Trypanosomiasis, African

1945
Proarrhythmic risk assessment using conventional and new in vitro assays.
    Regulatory toxicology and pharmacology : RTP, 2017, Volume: 88

    Topics: Action Potentials; Anti-Arrhythmia Agents; Arsenic; Dose-Response Relationship, Drug; Drug Discovery; Drug Evaluation, Preclinical; Fluoroquinolones; Humans; In Vitro Techniques; Induced Pluripotent Stem Cells; Long QT Syndrome; Moxifloxacin; Myocytes, Cardiac; Pentamidine; Phenethylamines; Risk Assessment; Sulfonamides

2017
Differences in Transporters Rather than Drug Targets Are the Principal Determinants of the Different Innate Sensitivities of
    International journal of molecular sciences, 2022, Mar-05, Volume: 23, Issue:5

    Topics: Animals; Arsenicals; Membrane Transport Proteins; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosoma congolense

2022