Page last updated: 2024-08-24

aromasil and formestane

aromasil has been researched along with formestane in 23 studies

Research

Studies (23)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	8 (34.78)	18.2507
2000's	9 (39.13)	29.6817
2010's	5 (21.74)	24.3611
2020's	1 (4.35)	2.80

Authors

Authors	Studies
An, J; Davies, HM; Egbuta, C; Ghosh, D; Griswold, J; Hubbell, S; Jiang, W; Lo, J; Morton, D; Valette, D; Xi, J	1
Barmade, MA; Murumkar, PR; Tamboli, RS; Yadav, MR	1
Alcaro, S; Amaral, C; Carvalho, RA; Correia-da-Silva, G; Costa, G; Costa, SC; Roleira, FM; Tavares-da-Silva, EJ; Teixeira, NA; Varela, CL	1
Alcaro, S; Amaral, C; Correia-da-Silva, G; Costa, G; Costa, SC; Moraca, F; Roleira, FMF; Tavares da Silva, EJ; Teixeira, NAA; Varela, C	1
Chen, JZ; Khan, MZI; Nazli, A; Uzair, M	1
Coombes, RC; di Salle, E; Evans, TR; Giudici, D; Lassus, M; Ornati, G	1
Briatico, G; D'Alessio, R; Di Salle, E; Giudici, D; Lombardi, P; Ornati, G; Villa, V	1
Briatico, G; di Salle, E; Giudici, D; Ornati, G	1
Lønning, PE	1
Anker, GB; Johannessen, DC; Lien, EA; Lonning, PE; Refsum, H; Ueland, PM	1
Blijham, GH; de Jong, PC	1
Bonneterre, J; Feutrie, ML	1
Harvey, HA; Santen, RJ	1
Bajetta, E; Bichisao, E; Pozzi, P; Toffolatti, L; Zilembo, N	1
Auvray, P; Bichat, F; Genne, P	1
de Crémoux, P	1
Kerbrat, P; Lefeuvre, C	1
Buzdar, A; Howell, A	1
Lombardi, P	1
Delozier, T; Khayat, D; Spano, JP	1
Chen, S; Wang, X	1
Dutta, U; Pant, K	1
Csákvári, E; Gyenes, A; Hoyk, Z; Kóti, J; Paragi, G; Párducz, A; Pfoh, R; Rühl, S; Szájli, A; Wölfling, J	1

Reviews

15 review(s) available for aromasil and formestane

Article	Year
Developing steroidal aromatase inhibitors-an effective armament to win the battle against breast cancer. European journal of medicinal chemistry, 2015, Nov-13, Volume: 105 Topics: Aromatase; Aromatase Inhibitors; Breast Neoplasms; Drug Design; Female; Humans; Models, Molecular; Molecular Structure	2015
An overview on Estrogen receptors signaling and its ligands in breast cancer. European journal of medicinal chemistry, 2022, Nov-05, Volume: 241 Topics: Breast Neoplasms; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogens; Female; Humans; Ligands; Male; Receptors, Estrogen	2022
Exemestane (FCE 24304), a new steroidal aromatase inhibitor. The Journal of steroid biochemistry and molecular biology, 1992, Volume: 43, Issue:1-3 Topics: 5-alpha Reductase Inhibitors; Androgens; Androstadienes; Androstenedione; Animals; Antineoplastic Agents; Aromatase Inhibitors; Humans; Lyases; Receptors, Steroid	1992
Pharmacological profiles of exemestane and formestane, steroidal aromatase inhibitors used for treatment of postmenopausal breast cancer. Breast cancer research and treatment, 1998, Volume: 49 Suppl 1 Topics: Androstadienes; Androstenedione; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Enzyme Inhibitors; Female; Humans; Neoplasms, Hormone-Dependent; Postmenopause	1998
New aromatase inhibitors for the treatment of advanced breast cancer in postmenopausal women. The Netherlands journal of medicine, 1999, Volume: 55, Issue:2 Topics: Aminoglutethimide; Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Chemotherapy, Adjuvant; Clinical Trials, Phase III as Topic; Female; Humans; Letrozole; Megestrol Acetate; Nitriles; Postmenopause; Triazoles	1999
[Aromatase inhibitors]. Bulletin du cancer, 1999, Volume: 86, Issue:10 Topics: Aminoglutethimide; Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents; Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Estrogen Antagonists; Estrone; Female; Humans; Letrozole; Nitriles; Triazoles	1999
Use of aromatase inhibitors in breast carcinoma. Endocrine-related cancer, 1999, Volume: 6, Issue:1 Topics: Adult; Aminoglutethimide; Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents, Hormonal; Aromatase; Aromatase Inhibitors; Breast Neoplasms; Drug Design; Drug Interactions; Drug Resistance, Neoplasm; Enzyme Inhibitors; Estrogens; Female; Humans; Letrozole; Middle Aged; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Nitriles; Postmenopause; Premenopause; Tamoxifen; Triazoles	1999
Steroidal aromatase inhibitors in elderly patients. Critical reviews in oncology/hematology, 2000, Volume: 33, Issue:2 Topics: Aged; Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Enzyme Inhibitors; Female; Humans; Letrozole; Nitriles; Triazoles	2000
[Preclinical evaluation of aromatase inhibitors antitumor activity]. Bulletin du cancer, 2000, Volume: 87 Spec No Topics: Aminoglutethimide; Anastrozole; Androstadienes; Androstenedione; Animals; Antineoplastic Agents, Hormonal; Aromatase; Aromatase Inhibitors; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fadrozole; Female; Humans; Letrozole; Models, Animal; Nitriles; Rats; Structure-Activity Relationship; Triazoles	2000
[Aromatase inhibitors: pharmacological aspects]. Bulletin du cancer, 2000, Volume: 87 Spec No Topics: Aminoglutethimide; Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Enzyme Inhibitors; Fadrozole; Female; Humans; Letrozole; Nitriles; Triazoles	2000
[Aromatase inhibitors: a review of clinical trials]. Bulletin du cancer, 2000, Volume: 87 Spec No Topics: Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Chemotherapy, Adjuvant; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Enzyme Inhibitors; Female; Humans; Letrozole; Nitriles; Randomized Controlled Trials as Topic; Triazoles	2000
Advances in aromatase inhibition: clinical efficacy and tolerability in the treatment of breast cancer. Clinical cancer research : an official journal of the American Association for Cancer Research, 2001, Volume: 7, Issue:9 Topics: Anastrozole; Androstadienes; Androstenedione; Aromatase Inhibitors; Breast Neoplasms; Enzyme Inhibitors; Fadrozole; Female; Headache; Humans; Letrozole; Nausea; Nitriles; Treatment Outcome; Triazoles; Vomiting	2001
Exemestane, a new steroidal aromatase inhibitor of clinical relevance. Biochimica et biophysica acta, 2002, Jul-18, Volume: 1587, Issue:2-3 Topics: Androstadienes; Androstenedione; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Enzyme Inhibitors; Estrogen Receptor Modulators; Estrogens; Female; Humans; Neoplasms, Hormone-Dependent	2002
[Aromatase inhibitors in adjuvant setting in breast cancer]. Bulletin du cancer, 2004, Dec-01, Volume: 91 Suppl 4 Topics: Anastrozole; Androstadienes; Androstenedione; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Chemotherapy, Adjuvant; Female; Humans; Letrozole; Menopause; Nitriles; Triazoles	2004
Aromatase inhibitors: past, present and future in breast cancer therapy. Medical oncology (Northwood, London, England), 2008, Volume: 25, Issue:2 Topics: Aminoglutethimide; Androstadienes; Androstenedione; Aromatase Inhibitors; Breast Neoplasms; Clinical Trials as Topic; Fadrozole; Female; Humans; Letrozole; Nitriles; Triazoles	2008

Trials

1 trial(s) available for aromasil and formestane

Article	Year
Exemestane (FCE 24304), a new steroidal aromatase inhibitor. The Journal of steroid biochemistry and molecular biology, 1992, Volume: 43, Issue:1-3 Topics: 5-alpha Reductase Inhibitors; Androgens; Androstadienes; Androstenedione; Animals; Antineoplastic Agents; Aromatase Inhibitors; Humans; Lyases; Receptors, Steroid	1992

Other Studies

8 other study(ies) available for aromasil and formestane

Article	Year
Novel aromatase inhibitors by structure-guided design. Journal of medicinal chemistry, 2012, Oct-11, Volume: 55, Issue:19 Topics: Androstadienes; Antineoplastic Agents; Aromatase Inhibitors; Cell Line, Tumor; Crystallography, X-Ray; Drug Design; Drug Screening Assays, Antitumor; Female; Humans; Molecular Docking Simulation; Molecular Structure; Placenta; Pregnancy; Protein Binding; Stereoisomerism; Structure-Activity Relationship	2012
Exploring new chemical functionalities to improve aromatase inhibition of steroids. Bioorganic & medicinal chemistry, 2016, 06-15, Volume: 24, Issue:12 Topics: Androstanes; Androstenedione; Aromatase; Aromatase Inhibitors; Breast Neoplasms; Cell Line, Tumor; Female; Humans; Molecular Docking Simulation; Steroids; Structure-Activity Relationship	2016
C-6α- vs C-7α-Substituted Steroidal Aromatase Inhibitors: Which Is Better? Synthesis, Biochemical Evaluation, Docking Studies, and Structure-Activity Relationships. Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7 Topics: Aromatase Inhibitors; Humans; Molecular Docking Simulation; Steroids; Structure-Activity Relationship	2019
4-Aminoandrostenedione derivatives: a novel class of irreversible aromatase inhibitors. Comparison with FCE 24304 and 4-hydroxyandrostenedione. The Journal of steroid biochemistry and molecular biology, 1990, Nov-20, Volume: 37, Issue:3 Topics: Androstadienes; Androstenedione; Animals; Aromatase Inhibitors; Female; Male; Pregnancy; Rats; Rats, Inbred Strains	1990
Novel irreversible aromatase inhibitors. Annals of the New York Academy of Sciences, 1990, Volume: 595 Topics: Aminoglutethimide; Androstadienes; Androstenedione; Animals; Aromatase Inhibitors; Female; Gonadotropins, Equine; Humans; In Vitro Techniques; Kinetics; Microsomes; Ovary; Pargyline; Placenta; Rats; Rats, Inbred Strains	1990
Influence of aromatase inhibitors on plasma total homocysteine in postmenopausal breast cancer patients. Clinical chemistry, 1999, Volume: 45, Issue:2 Topics: Aminoglutethimide; Androstadienes; Androstenedione; Aromatase Inhibitors; Breast Neoplasms; Creatinine; Enzyme Inhibitors; Estrogen Antagonists; Homocysteine; Humans; Postmenopause; Vitamins	1999
Aromatase destabilizer: novel action of exemestane, a food and drug administration-approved aromatase inhibitor. Cancer research, 2006, Nov-01, Volume: 66, Issue:21 Topics: Androstadienes; Androstenedione; Aromatase; Aromatase Inhibitors; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Stability; Female; Humans; Proteasome Endopeptidase Complex	2006
Computer-aided structure analysis of an epimerized dehydroepiandrosterone derivative and its biological effect in a model of reactive gliosis. Steroids, 2010, Volume: 75, Issue:3 Topics: Androstadienes; Androstenedione; Animals; Aromatase; Aromatase Inhibitors; Crystallography, X-Ray; Dehydroepiandrosterone; Glial Fibrillary Acidic Protein; Gliosis; Male; Molecular Sequence Data; Molecular Structure; Rats; Rats, Wistar	2010