Page last updated: 2024-08-24

aripiprazole and raclopride

aripiprazole has been researched along with raclopride in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (54.55)29.6817
2010's4 (36.36)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Benjamin, PS; Schetz, JA; Sibley, DR1
Schetz, JA; Sibley, DR1
Biziere, K; Bramer, S; Dannals, RF; Dogan, AS; Gründer, G; Ravert, H; Stephane, M; Suri, A; Wong, DF; Yokoi, F1
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K1
Chen, R; Johnson, JL; Jordan, S; Kambayashi, J; Kikuchi, T; Kitagawa, H; McQuade, R; Regardie, K; Tadori, Y1
Graff, A; Kapur, S; Mamo, D; Mizrahi, R; Romeyer, F; Shammi, CM1
Arakawa, R; Fujiwara, H; Ito, H; Kato, M; Kimura, Y; Kodaka, F; Mimura, M; Nagashima, T; Nogami, T; Sasaki, T; Shimada, H; Suhara, T; Suzuki, M; Takahata, K; Takano, H1
Arakawa, R; Ito, H; Kodaka, F; Nogami, T; Suhara, T; Suzuki, M; Takahashi, H; Takahata, K; Takano, H1
Howes, OD; Jang, IJ; Jeong, JM; Kapur, S; Kim, BH; Kim, E; Kim, JW; Kwon, JS; Lee, JS; Shin, SG; Turkheimer, FE1
Howes, OD; Kim, E; Kim, S; Kwon, JS; Lee, JS; Seo, S; Shin, S1
Kim, E; Kim, S; Kwon, JS; Ock, EY1

Trials

3 trial(s) available for aripiprazole and raclopride

ArticleYear
Differential effects of aripiprazole on D(2), 5-HT(2), and 5-HT(1A) receptor occupancy in patients with schizophrenia: a triple tracer PET study.
    The American journal of psychiatry, 2007, Volume: 164, Issue:9

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Basal Ganglia; Basal Ganglia Diseases; Carbon Radioisotopes; Caudate Nucleus; Cerebral Cortex; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Piperazines; Positron-Emission Tomography; Psychotic Disorders; Putamen; Pyridines; Pyrimidinones; Quinolones; Raclopride; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine; Receptors, Dopamine D2; Schizophrenia; Serotonin 5-HT1 Receptor Agonists; Treatment Outcome

2007
Striatal and extrastriatal dopamine D₂ receptor occupancy by the partial agonist antipsychotic drug aripiprazole in the human brain: a positron emission tomography study with [¹¹C]raclopride and [¹¹C]FLB457.
    Psychopharmacology, 2012, Volume: 222, Issue:1

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Brain; Carbon Radioisotopes; Corpus Striatum; Humans; Male; Piperazines; Positron-Emission Tomography; Pyrrolidines; Quinolones; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Salicylamides; Young Adult

2012
The relationship between antipsychotic D2 occupancy and change in frontal metabolism and working memory : A dual [(11)C]raclopride and [(18) F]FDG imaging study with aripiprazole.
    Psychopharmacology, 2013, Volume: 227, Issue:2

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Carbon Radioisotopes; Cognition; Corpus Striatum; Fluorodeoxyglucose F18; Frontal Lobe; Humans; Male; Memory, Short-Term; Piperazines; Positron-Emission Tomography; Quinolones; Raclopride; Reaction Time; Receptors, Dopamine D2; Single-Blind Method; Young Adult

2013

Other Studies

8 other study(ies) available for aripiprazole and raclopride

ArticleYear
Nonconserved residues in the second transmembrane-spanning domain of the D(4) dopamine receptor are molecular determinants of D(4)-selective pharmacology.
    Molecular pharmacology, 2000, Volume: 57, Issue:1

    Topics: Animals; Binding Sites; COS Cells; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ligands; Membrane Proteins; Mutagenesis, Site-Directed; Protein Conformation; Pyridines; Pyrroles; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4; Structure-Activity Relationship; Transfection

2000
Tandem sulfur-containing amino acids are epicritical determinants of dopamine D(2) receptor pharmacology.
    European journal of pharmacology, 2000, Jan-28, Volume: 388, Issue:2

    Topics: Amino Acids, Sulfur; Animals; Aripiprazole; Aspartic Acid; Chlorocebus aethiops; COS Cells; Dopamine; Kinetics; Ligands; Piperazines; Point Mutation; Quinolones; Raclopride; Receptors, Dopamine D2

2000
Dopamine D2 and D3 receptor occupancy in normal humans treated with the antipsychotic drug aripiprazole (OPC 14597): a study using positron emission tomography and [11C]raclopride.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 27, Issue:2

    Topics: Administration, Oral; Adult; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Brain; Cerebellum; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Male; Neurons; Piperazines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Tomography, Emission-Computed

2002
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium

2005
In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:6

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Calcium Signaling; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Immunoblotting; Lisuride; MAP Kinase Signaling System; Microscopy, Confocal; Mitogen-Activated Protein Kinase 1; Phosphorylation; Piperazines; Piperidines; Quinolones; Raclopride; Receptors, Dopamine D2; Schizophrenia; Time Factors; Transfection

2007
Effects of dopamine D2 receptor partial agonist antipsychotic aripiprazole on dopamine synthesis in human brain measured by PET with L-[β-11C]DOPA.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Carbon Radioisotopes; Caudate Nucleus; Dopamine; Dopamine D2 Receptor Antagonists; Humans; Levodopa; Male; Neuroimaging; Piperazines; Positron-Emission Tomography; Putamen; Quinolones; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Tissue Distribution; Young Adult

2012
The relationship between dopamine receptor blockade and cognitive performance in schizophrenia: a [
    Translational psychiatry, 2018, 04-24, Volume: 8, Issue:1

    Topics: Adult; Aripiprazole; Cognition; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Humans; Male; Memory, Short-Term; Positron-Emission Tomography; Prospective Studies; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Schizophrenic Psychology

2018
Relationship between subjective well-being and aripiprazole: an [
    Scientific reports, 2022, 07-15, Volume: 12, Issue:1

    Topics: Antipsychotic Agents; Aripiprazole; Humans; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2

2022