Page last updated: 2024-08-24

aripiprazole and quinpirole

aripiprazole has been researched along with quinpirole in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (11.11)18.2507
2000's3 (16.67)29.6817
2010's12 (66.67)24.3611
2020's1 (5.56)2.80

Authors

AuthorsStudies
Bearden, M; Cui, J; Luedtke, RR; Mach, RH; Taylor, M; Vangveravong, S; Wang, W; Xu, J; Zhang, Z1
Gmeiner, P; Hübner, H; Kling, RC; Leuner, K; Möller, D; Skultety, M1
Gmeiner, P; Hübner, H; Kling, RC; Möller, D; Salama, I1
Alzheimer, C; Banerjee, A; Bouvier, M; Friedland, K; Gmeiner, P; Hübner, H; Huth, T; Möller, D; Müller, CP; Plouffe, B; Skultety, M; Uzuneser, TC1
Dengler, D; Gmeiner, P; Hübner, H; Männel, B; Möller, D; Shonberg, J1
Gmeiner, P; Hübner, H; Männel, B; Möller, D1
Cheng, J; Fan, L; Liu, R; Tan, L; Wang, H; Wang, S; Yan, W; Yu, J1
Harano, M; Tanaka, M; Yamada, S; Yokoo, H1
Inoue, A; Kikuchi, T; Miki, S; Misu, Y; Morita, S; Nakata, Y; Seto, M; Ueda, H1
Mailman, RB; Urban, JD; Vargas, GA; von Zastrow, M1
Hashioka, S; Horikawa, H; Iwaki, T; Kanba, S; Kato, T; Mizoguchi, Y; Monji, A; Seki, Y; Suzuki, SO1
Abe, M; Egashira, N; Fujiwara, M; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Oishi, R; Okuno, R1
Charntikov, S; Crawford, CA; Der-Ghazarian, T; McDougall, SA; Varela, FA1
De Carolis, L; Milella, MS; Nencini, P; Schepisi, C1
Lowry, JP; O'Connor, JJ1
Ma, GF; Ortiz, J; Raivio, N; Sabrià, J1
Gao, J; Li, M; Qin, R1
Bye, CR; Ganella, DE; Kim, JH; Lawrence, AJ; Madsen, HB; Perry, CJ; Zbukvic, IC1

Other Studies

18 other study(ies) available for aripiprazole and quinpirole

ArticleYear
Synthesis and characterization of selective dopamine D₂ receptor ligands using aripiprazole as the lead compound.
    Bioorganic & medicinal chemistry, 2011, Jun-01, Volume: 19, Issue:11

    Topics: Aripiprazole; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ligands; Piperazines; Protein Binding; Quinolones; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, sigma

2011
Functionally selective dopamine D₂, D₃ receptor partial agonists.
    Journal of medicinal chemistry, 2014, Jun-12, Volume: 57, Issue:11

    Topics: Animals; Antipsychotic Agents; Arrestins; beta-Arrestin 2; beta-Arrestins; CHO Cells; Cricetulus; Drug Partial Agonism; GTP-Binding Protein alpha Subunits, Gi-Go; HEK293 Cells; Heterocyclic Compounds, 2-Ring; Humans; Mice; Molecular Docking Simulation; Oximes; Piperazines; Pyrazoles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereoisomerism; Structure-Activity Relationship; Swine

2014
1,4-Disubstituted aromatic piperazines with high 5-HT2A/D2 selectivity: Quantitative structure-selectivity investigations, docking, synthesis and biological evaluation.
    Bioorganic & medicinal chemistry, 2015, Sep-15, Volume: 23, Issue:18

    Topics: Antipsychotic Agents; Binding Sites; HEK293 Cells; Humans; Ligands; Molecular Docking Simulation; Piperazines; Protein Structure, Tertiary; Quantitative Structure-Activity Relationship; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2

2015
Discovery of G Protein-Biased Dopaminergics with a Pyrazolo[1,5-a]pyridine Substructure.
    Journal of medicinal chemistry, 2017, 04-13, Volume: 60, Issue:7

    Topics: Animals; Antipsychotic Agents; beta-Arrestins; Dopamine Agonists; Drug Discovery; GTP-Binding Proteins; Humans; Male; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Schizophrenia

2017
Hydroxy-Substituted Heteroarylpiperazines: Novel Scaffolds for β-Arrestin-Biased D
    Journal of medicinal chemistry, 2017, 06-08, Volume: 60, Issue:11

    Topics: Animals; beta-Arrestins; CHO Cells; Cricetulus; Dopamine Agonists; Humans; Piperazines; Receptors, Dopamine D2

2017
β-Arrestin biased dopamine D2 receptor partial agonists: Synthesis and pharmacological evaluation.
    Bioorganic & medicinal chemistry, 2017, 10-15, Volume: 25, Issue:20

    Topics: Antiparkinson Agents; Antipsychotic Agents; beta-Arrestins; Dopamine Agonists; Dose-Response Relationship, Drug; Humans; Ligands; Molecular Structure; Protein Binding; Receptors, Dopamine D2

2017
2-Phenylcyclopropylmethylamine Derivatives as Dopamine D
    Journal of medicinal chemistry, 2021, 12-09, Volume: 64, Issue:23

    Topics: Animals; Cell Line, Tumor; Disease Models, Animal; Dopamine Agonists; Drug Design; Drug Evaluation, Preclinical; Half-Life; Humans; Mice; Mice, Inbred ICR; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship

2021
Antagonistic effects of OPC-14597, a novel antipsychotic drug, on quinpirole- and (-)-sulpiride-induced changes in evoked dopamine release in rat striatal slices.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:2

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Dopamine; Dopamine Agents; Electric Stimulation; In Vitro Techniques; Male; Neostriatum; Piperazines; Quinolones; Quinpirole; Rats; Rats, Wistar; Sulpiride

1997
Aripiprazole, a novel antipsychotic drug, inhibits quinpirole-evoked GTPase activity but does not up-regulate dopamine D2 receptor following repeated treatment in the rat striatum.
    European journal of pharmacology, 1997, Feb-19, Volume: 321, Issue:1

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Dopamine Agonists; GTP Phosphohydrolases; Haloperidol; Male; Membranes; Neostriatum; Oligonucleotides, Antisense; Piperazines; Quinolones; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Up-Regulation

1997
Aripiprazole has functionally selective actions at dopamine D2 receptor-mediated signaling pathways.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2007, Volume: 32, Issue:1

    Topics: Analysis of Variance; Animals; Arachidonic Acid; Aripiprazole; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Guanosine Triphosphate; Mitogen-Activated Protein Kinases; Piperazines; Quinolones; Quinpirole; Receptors, Dopamine D2; Signal Transduction

2007
Inhibitory effects of aripiprazole on interferon-gamma-induced microglial activation via intracellular Ca2+ regulation in vitro.
    Journal of neurochemistry, 2008, Volume: 106, Issue:2

    Topics: Analysis of Variance; Animals; Animals, Newborn; Antipsychotic Agents; Aripiprazole; Brain; Calcium; Cell Survival; Cells, Cultured; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Interferon-gamma; Mice; Microglia; Neurons; Nitric Oxide; Piperazines; Quinolones; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tumor Necrosis Factor-alpha

2008
Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Anxiety; Aripiprazole; Behavior, Animal; Benzodiazepines; Catalepsy; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Ketanserin; Male; Mice; Mice, Inbred ICR; Olanzapine; Piperazines; Piperidines; Postural Balance; Psychomotor Performance; Pyridines; Quinolones; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Effects of repeated and acute aripiprazole or haloperidol treatment on dopamine synthesis in the dorsal striatum of young rats: comparison to adult rats.
    Journal of neural transmission (Vienna, Austria : 1996), 2010, Volume: 117, Issue:5

    Topics: Aging; Animals; Animals, Newborn; Antipsychotic Agents; Aripiprazole; Autoreceptors; Brain Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Drug Administration Schedule; Drug Interactions; Female; Haloperidol; Male; Piperazines; Quinolones; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

2010
Clomipramine, but not haloperidol or aripiprazole, inhibits quinpirole-induced water contrafreeloading, a putative animal model of compulsive behavior.
    Psychopharmacology, 2011, Volume: 218, Issue:4

    Topics: Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Aripiprazole; Clomipramine; Compulsive Behavior; Conditioning, Operant; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking Behavior; Haloperidol; Male; Piperazines; Quinolones; Quinpirole; Rats; Rats, Sprague-Dawley

2011
A comparison of the effects of the dopamine partial agonists aripiprazole and (-)-3-PPP with quinpirole on stimulated dopamine release in the rat striatum: Studies using fast cyclic voltammetry in vitro.
    European journal of pharmacology, 2012, Jul-05, Volume: 686, Issue:1-3

    Topics: Animals; Aripiprazole; Corpus Striatum; Dopamine; Dopamine Agonists; Drug Partial Agonism; In Vitro Techniques; Male; Piperazines; Piperidines; Quinolones; Quinpirole; Rats; Rats, Wistar

2012
Agonist and antagonist effects of aripiprazole on D₂-like receptors controlling rat brain dopamine synthesis depend on the dopaminergic tone.
    The international journal of neuropsychopharmacology, 2014, Oct-31, Volume: 18, Issue:4

    Topics: Animals; Aripiprazole; Autoreceptors; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Piperidines; Potassium; Presynaptic Terminals; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2

2014
Repeated administration of aripiprazole produces a sensitization effect in the suppression of avoidance responding and phencyclidine-induced hyperlocomotion and increases D2 receptor-mediated behavioral function.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:4

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Avoidance Learning; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Hyperkinesis; Male; Phencyclidine; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

2015
Role of Dopamine 2 Receptor in Impaired Drug-Cue Extinction in Adolescent Rats.
    Cerebral cortex (New York, N.Y. : 1991), 2016, Volume: 26, Issue:6

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Agonists; Dopamine Uptake Inhibitors; Extinction, Psychological; Learning; Male; Motivation; Prefrontal Cortex; Quinpirole; Random Allocation; Rats, Sprague-Dawley; Receptors, Dopamine D2; Self Administration

2016