Page last updated: 2024-09-03

argiotoxin-636 and kainic acid

argiotoxin-636 has been researched along with kainic acid in 8 studies

Compound Research Comparison

Studies
(argiotoxin-636)
Trials
(argiotoxin-636)
Recent Studies (post-2010)
(argiotoxin-636)
Studies
(kainic acid)
Trials
(kainic acid)
Recent Studies (post-2010) (kainic acid)
53079,54031,775

Protein Interaction Comparison

ProteinTaxonomyargiotoxin-636 (IC50)kainic acid (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 2Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 3Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 4Rattus norvegicus (Norway rat)4.2857
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 1Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 2Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 3Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 4Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.0126

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19902 (25.00)18.7374
1990's5 (62.50)18.2507
2000's0 (0.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
England, PM; Fleming, JJ1
Gapon, SA; Magazanik, LG1
Grishin, EV; Kiskin, NI; Kryshtal', OA; Tsyndrenko, AIa; Volkova, TM1
Kemp, JA; Priestley, T; Woodruff, GN1
Herlitze, S; Jahn, W; Monyer, H; Raditsch, M; Ruppersberg, JP; Schoepfer, R; Witzemann, V1
Bell, DR; Brackley, PT; Choi, SK; Nakanishi, K; Usherwood, PN1
Green, AC; Nakanishi, K; Usherwood, PN1
Dingledine, R; Numberger, M; Washburn, MS; Zhang, S1

Other Studies

8 other study(ies) available for argiotoxin-636 and kainic acid

ArticleYear
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
Different types of glutamate receptors in isolated and identified neurones of the mollusc Planorbarius corneus.
    The Journal of physiology, 1991, Volume: 439

    Topics: Animals; Glutamates; Guanosine 5'-O-(3-Thiotriphosphate); Kainic Acid; Membrane Potentials; Mollusca; Neurons; Oligopeptides; Pertussis Toxin; Polyamines; Potassium Channels; Quisqualic Acid; Receptors, Glutamate; Receptors, Neurotransmitter; Spider Venoms; Virulence Factors, Bordetella

1991
[Argiopine, argiopinines and pseudoargiopinines--blockers of the glutamate receptors in hippocampal neurons].
    Neirofiziologiia = Neurophysiology, 1989, Volume: 21, Issue:6

    Topics: Animals; Arthropod Venoms; Depression, Chemical; Dose-Response Relationship, Drug; Glutamates; Hippocampus; In Vitro Techniques; Ion Channels; Kainic Acid; Microelectrodes; Oligopeptides; Polyamines; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Spider Venoms

1989
Antagonism of responses to excitatory amino acids on rat cortical neurones by the spider toxin, argiotoxin636.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Cerebral Cortex; Electrophysiology; Ibotenic Acid; In Vitro Techniques; Indoleacetic Acids; Kainic Acid; Male; Membrane Potentials; Neurons; Phenylacetates; Polyamines; Rats; Rats, Inbred Strains

1989
Argiotoxin detects molecular differences in AMPA receptor channels.
    Neuron, 1993, Volume: 10, Issue:6

    Topics: Animals; Base Sequence; Cell Membrane; Evoked Potentials; Female; Indoleacetic Acids; Ion Channels; Kainic Acid; Macromolecular Substances; Molecular Sequence Data; Mutagenesis; Oligodeoxyribonucleotides; Oocytes; Phenylacetates; Polyamines; Protein Conformation; Receptors, AMPA; Receptors, Glutamate; Spider Venoms; Xenopus laevis

1993
Selective antagonism of native and cloned kainate and NMDA receptors by polyamine-containing toxins.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Animals; Arthropod Venoms; Cloning, Molecular; Excitatory Amino Acid Antagonists; Female; Indoleacetic Acids; Kainic Acid; Male; N-Methylaspartate; Oocytes; Phenols; Phenylacetates; Polyamines; Rats; Rats, Wistar; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; RNA; Spider Venoms; Transcription, Genetic; Xenopus

1993
Polyamine amides are neuroprotective in cerebellar granule cell cultures challenged with excitatory amino acids.
    Brain research, 1996, Apr-22, Volume: 717, Issue:1-2

    Topics: Amides; Animals; Arthropod Venoms; Calcium; Cells, Cultured; Cerebellum; Excitatory Amino Acid Agonists; Glutamic Acid; Indoleacetic Acids; Kainic Acid; N-Methylaspartate; Neurons; Neuroprotective Agents; Phenols; Phenylacetates; Polyamines; Potassium; Rats; Rats, Wistar; Spider Venoms

1996
Differential dependence on GluR2 expression of three characteristic features of AMPA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-15, Volume: 17, Issue:24

    Topics: Animals; Calcium; Excitatory Amino Acid Agonists; Hippocampus; Indoleacetic Acids; Interneurons; Kainic Acid; Male; Oocytes; Patch-Clamp Techniques; Phenotype; Phenylacetates; Polyamines; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Recombinant Proteins; RNA, Messenger; Spermine; Spider Venoms; Synapses; Xenopus

1997