Page last updated: 2024-09-03

argiotoxin-636 and jstx-3

argiotoxin-636 has been researched along with jstx-3 in 2 studies

Compound Research Comparison

Studies
(argiotoxin-636)
Trials
(argiotoxin-636)
Recent Studies (post-2010)
(argiotoxin-636)
Studies
(jstx-3)
Trials
(jstx-3)
Recent Studies (post-2010) (jstx-3)
5307901

Protein Interaction Comparison

ProteinTaxonomyargiotoxin-636 (IC50)jstx-3 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.065
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.019
Glutamate receptor 1Homo sapiens (human)0.04
Glutamate receptor 3Homo sapiens (human)0.03
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)1.71

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
England, PM; Fleming, JJ1
Bach, TB; Barslund, AF; Kristensen, AS; Lucas, S; Nørager, NG; Poulsen, MH; Strømgaard, K1

Other Studies

2 other study(ies) available for argiotoxin-636 and jstx-3

ArticleYear
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
General synthesis of β-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Animals; Asparagine; beta-Alanine; Indoleacetic Acids; Molecular Structure; Polyamines; Receptors, Ionotropic Glutamate; Receptors, Kainic Acid; Spider Venoms; Spiders; Structure-Activity Relationship; Toxins, Biological

2012