arginine vasopressin has been researched along with relcovaptan in 48 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 31 (64.58) | 18.2507 |
2000's | 10 (20.83) | 29.6817 |
2010's | 7 (14.58) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Auzan, C; Berti-Mattera, L; Clauser, E; Madhun, Z; Thibonnier, M; Wilkins, P | 1 |
Berti-Mattera, LN; Dulin, N; Mattera, R; Preston, JA; Thibonnier, M; Wilkins, PL | 1 |
Barberis, C; Carnazzi, E; Cotte, N; Jard, S; Mahe, E; Mouillac, B; Phalipou, S; Seyer, R | 1 |
Ishii, N; Kusayama, T; Saito, M; Sugimoto, T; Tahara, A; Tanaka, A; Tomura, Y; Tsukada, J; Uchida, W; Wada, K; Yatsu, T | 1 |
Akerlund, M; Bossmar, T; Brouard, R; Kostrzewska, A; Laudanski, T; Lemancewicz, A; Serradeil-Le Gal, C; Steinwall, M | 1 |
Aumelas, A; Balestre, MN; Barberis, C; Cotte, N; Durroux, T; Hibert, M; Mahé, E; Manning, M; Morin, D; Mouillac, B; Phalipou, S | 1 |
Double-Cazanave, E; Garcia, C; Guillon, G; Maffrand, JP; Pascal, M; Raufaste, D; Serradeil-Le Gal, C | 1 |
Arban, R; Curcuruto, O; Dickinson, BA; Green, A; Griffante, C; Haslam, CP | 1 |
Albizu, L; Ansanay, H; Bazin, H; Durroux, T; Manning, M; Mouillac, B; Seyer, R; Teppaz, G | 1 |
Boutin, M; Le Fur, G; Maffrand, JP; Serradeil-Le Gal, C; Villanova, G | 1 |
Delisee, C; Dol, F; Garcia, C; Herbert, JM; Le Fur, G; Maffrand, JP; Marty, E; Raufaste, D; Schaeffer, P; Serradeil-Le Gal, C | 1 |
Garcia, C; Le Fur, G; Maffrand, JP; Marty, E; Raufaste, D; Serradeil-Le Gal, C | 2 |
Bourrié, B; Carayon, P; Casellas, P; Garcia, C; Le Fur, G; Maffrand, JP; Raufaste, D; Serradeil-Le Gal, C | 1 |
Christophe, B; Garcia, C; Guiraudou, P; Lacour, C; Le Fur, G; Maffrand, JP; Nisato, D; Serradeil-Le Gal, C; Villanova, G; Wagnon, J | 1 |
Burrell, LM; Buxton, BB; Chen, JR; Johnston, CI; Liu, JJ | 1 |
Bax, WA; Bos, E; Nisato, D; Saxena, PR; Stam, WB; Van der Graaf, PH | 1 |
Goncharevskaya, OA; Natochin, YV; Shakhmatova, EI | 1 |
Akerlund, M; Bossmar, T; Rasmussen, T | 1 |
Barthelmebs, M; Grima, M; Imbs, JL; Krieger, JP; Nisato, D | 1 |
Calò, G; Regoli, D; Rizzi, A; Traina, L | 1 |
Brouard, R; Brunner, HR; Burnier, M; Gerc, V; Hayoz, D; Lahmy, JP; Pechère-Bertschi, A; Weber, R | 1 |
Ishikawa, S; Saito, T | 1 |
Akerlund, M; Bossmar, T; Kostrzewska, A; Laudanski, T; Serradeil-Le Gal, C; Steinwall, M | 1 |
Koshio, H; Matsuhisa, A; Sakamoto, K; Tanaka, A; Taniguchi, N; Yatsu, T | 1 |
Saxena, PR; Stam, WB; Van der Graaf, PH | 1 |
Heinemann, A; Holzer, P; Horina, G; Pertl, C; Peskar, BA; Stauber, RE | 1 |
Brouard, R; Donat, F; Dreux, F; Fournie, D; Jang, H; Laporte, V; Lockwood, G; Pignol, R; Serradeil Le Gal, C | 1 |
Dayanithi, G; Gouzénes, L; Moos, FC; Richard, P; Sabatier, N | 1 |
Andres, M; Boccara, G; Breton, C; Colson, P; Derick, S; Grazzini, E; Guérineau, NC; Guillon, G; Raufaste, D; Rickwaert, F; Serradeil-le Gal, C | 1 |
Ayajiki, K; Fujioka, H; Okamura, T; Toda, N | 1 |
Chen, YL; Lai, FM; Shepherd, C; Spinelli, W | 1 |
Dayanithi, G; Gouzènes, L; Moos, FC | 1 |
Cros, G; Laurent, F; Méchaly, I; Portet, K; Serrano, J | 1 |
Brouard, R; DiBlasi, TP; Kilani, A; Leenhardt, AF; Rahman, M; Smith, MC; Thibonnier, M; Warner, K | 1 |
Lankhuizen, IM; Saxena, PR; Schoemaker, RG; van Veghel, R | 1 |
Ishii, N; Kusayama, T; Tahara, A; Tanaka, A; Taniguchi, N; Tomura, Y; Tsukada, J; Uchida, W; Yatsu, T | 1 |
Dapzol, J; Girod, V; Grélot, L; Maffrand, JP; Serradeil-Le Gal, C | 1 |
Chevaleyre, V; Desarménien, MG; Moos, FC | 1 |
Ji, X; Kurahashi, K; Murakami, S; Nishihashi, T; Trandafir, CC; Wang, A | 1 |
Streefkerk, JO; van Zwieten, PA | 1 |
Bankhead, P; Curtis, TM; Jeffries, O; Lozano, MM; McGahon, MK; McGeown, JG; Scholfield, CN | 1 |
Kamo, I; Kuno, M; Shintani, Y; Ueno, H | 1 |
Arban, R; Griffante, C; Perdonà, E | 1 |
Barr, LA; Carter, RL; Cheung, JY; Coleman, RC; Feldman, AM; Gao, E; Grisanti, LA; Houser, SR; Koch, WJ; Li, X; Makarewich, CA; Myers, VD; Song, J; Tilley, DG; Troupes, CD; Yu, D; Zhu, W | 1 |
Aman, NA; Hancock, M; Kang, SW; Kuenzel, WJ; Nagarajan, G | 1 |
Dehpour, AR; Doustimotlagh, AH; Javadi-Paydar, M; Javadian, N; Rahimi, N | 1 |
Best, C; Brydges, NM; Drake, AJ; Hall, J; Lewis, C; Rule, L; Thomas, KL; Watkin, H | 1 |
2 review(s) available for arginine vasopressin and relcovaptan
Article | Year |
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[Disorders of body water regulation and the therapy--vasopressin antagonists].
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Clinical Trials as Topic; Heart Failure; Hormone Antagonists; Humans; Hyponatremia; Inappropriate ADH Syndrome; Indoles; Liver Cirrhosis, Experimental; Pyrrolidines | 1997 |
Vasopressin receptor antagonists: pharmacological tools and potential therapeutic agents.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Drug Design; Heart Failure; Hormone Antagonists; Humans; Hypertension; Inappropriate ADH Syndrome; Indoles; Presynaptic Terminals; Pyrrolidines; Receptors, Vasopressin; Renal Artery; Sympathetic Nervous System; Synaptic Transmission; Tolvaptan; Vasoconstriction; Vasoconstrictor Agents | 2006 |
3 trial(s) available for arginine vasopressin and relcovaptan
Article | Year |
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Effects of SR 49059, a new orally active and specific vasopressin V1 receptor antagonist, on vasopressin-induced vasoconstriction in humans.
Topics: Administration, Oral; Adult; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcitonin Gene-Related Peptide; Double-Blind Method; Forearm; Hormone Antagonists; Humans; Indoles; Injections, Intra-Arterial; Injections, Intradermal; Male; Pyrrolidines; Radial Artery; Reference Values; Regional Blood Flow; Skin; Vasoconstriction | 1997 |
Safety, tolerability, and pharmacokinetics of SR 49059, a V1a vasopressin receptor antagonist, after repeated oral administration in healthy volunteers.
Topics: Administration, Oral; Adult; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Blood Platelets; Blood Pressure; Diuresis; Dose-Response Relationship, Drug; Double-Blind Method; Hormone Antagonists; Humans; Indoles; Male; Metabolic Clearance Rate; Placebos; Platelet Aggregation Inhibitors; Pyrrolidines; Regional Blood Flow; Skin; Vasopressins | 1998 |
Effects of the nonpeptide V(1) vasopressin receptor antagonist SR49059 in hypertensive patients.
Topics: Administration, Oral; Adult; Aldosterone; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Black People; Blood Volume; Cross-Over Studies; Double-Blind Method; Heart Rate; Hormone Antagonists; Humans; Hypertension; Indoles; Kidney Function Tests; Male; Platelet Aggregation; Pyrrolidines; Renin; Serum Albumin; Sodium; Treatment Outcome; White People | 1999 |
43 other study(ies) available for arginine vasopressin and relcovaptan
Article | Year |
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Molecular cloning, sequencing, and functional expression of a cDNA encoding the human V1a vasopressin receptor.
Topics: Amino Acid Sequence; Animals; Arginine Vasopressin; Base Sequence; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; DNA Probes; DNA, Complementary; Gene Expression; Humans; Inositol Phosphates; Kinetics; Liver; Molecular Sequence Data; Oligodeoxyribonucleotides; Pertussis Toxin; Rats; Receptors, Oxytocin; Receptors, Vasopressin; Recombinant Proteins; Sequence Homology, Amino Acid; Transfection; Virulence Factors, Bordetella | 1994 |
The human V3 pituitary vasopressin receptor: ligand binding profile and density-dependent signaling pathways.
Topics: Animals; Arachidonic Acid; Base Sequence; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; CHO Cells; Cricetinae; Cyclic AMP; DNA; Dose-Response Relationship, Drug; Female; Humans; Ligands; Pertussis Toxin; Phenotype; Phosphorylation; Pituitary Gland; Protein Binding; Protein Kinase C; Receptors, Vasopressin; Signal Transduction; Thymidine; Tritium; Type C Phospholipases; Virulence Factors, Bordetella | 1997 |
Mapping peptide-binding domains of the human V1a vasopressin receptor with a photoactivatable linear peptide antagonist.
Topics: Amino Acid Sequence; Animals; CHO Cells; Cricetinae; Endopeptidases; Glycosylation; Humans; Hydrolysis; Molecular Sequence Data; Mutagenesis, Site-Directed; Peptide Mapping; Peptides; Photoaffinity Labels; Precipitin Tests; Protein Binding; Receptors, Vasopressin; Recombinant Proteins | 1997 |
Pharmacological characterization of the human vasopressin receptor subtypes stably expressed in Chinese hamster ovary cells.
Topics: Animals; Benzazepines; Binding, Competitive; Calcium; CHO Cells; Cricetinae; Cyclic AMP; Humans; Indoles; Morpholines; Piperidines; Pyrrolidines; Quinolones; Receptors, Vasopressin; Spiro Compounds; Transfection; Tritium | 1998 |
Receptor binding of oxytocin and vasopressin antagonists and inhibitory effects on isolated myometrium from preterm and term pregnant women.
Topics: Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Cell Line; Cesarean Section; Female; Hormone Antagonists; Humans; Indoles; Morpholines; Myometrium; Obstetric Labor, Premature; Oxytocin; Pregnancy; Pyrrolidines; Receptors, Oxytocin; Spiro Compounds; Vasopressins | 1999 |
Conserved aromatic residues in the transmembrane region VI of the V1a vasopressin receptor differentiate agonist vs. antagonist ligand binding.
Topics: Amino Acid Sequence; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Binding Sites; Cell Membrane; Conserved Sequence; COS Cells; Humans; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Receptors, Vasopressin | 2000 |
Binding properties of a selective tritiated vasopressin V2 receptor antagonist, [H]-SR 121463.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Binding, Competitive; Cattle; CHO Cells; Cricetinae; Dogs; Haplorhini; Homeostasis; Humans; Kidney; Kinetics; Morpholines; Rabbits; Radioligand Assay; Rats; Spiro Compounds; Swine; Tritium; Vasopressins; Water-Electrolyte Balance | 2000 |
Selectivity of d[Cha4]AVP and SSR149415 at human vasopressin and oxytocin receptors: evidence that SSR149415 is a mixed vasopressin V1b/oxytocin receptor antagonist.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcium; CHO Cells; Cricetinae; Humans; Indoles; Pyrrolidines; Receptors, Oxytocin | 2005 |
Toward efficient drug screening by homogeneous assays based on the development of new fluorescent vasopressin and oxytocin receptor ligands.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Binding, Competitive; Chlorocebus aethiops; CHO Cells; COS Cells; Cricetinae; Cricetulus; Cyclic AMP; Fluoresceins; Fluorescence Polarization; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Ligands; Oligopeptides; Organometallic Compounds; Peptides, Cyclic; Quinolinium Compounds; Radioligand Assay; Receptors, Oxytocin; Receptors, Vasopressin | 2007 |
Effects of SR 49059, a non-peptide antagonist of vasopressin V1a receptors, on vasopressin-induced coronary vasoconstriction in conscious rabbits.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Coronary Vessels; Electrocardiography; Indoles; Male; Pyrrolidines; Rabbits; Stereoisomerism; Vasoconstriction | 1995 |
Effect of SR-49059, a vasopressin V1a antagonist, on human vascular smooth muscle cells.
Topics: Aorta; Arginine Vasopressin; Calcium; Cell Division; Cell Membrane; Cells, Cultured; Deamino Arginine Vasopressin; Dose-Response Relationship, Drug; Humans; Indoles; Iodine Radioisotopes; Kinetics; Muscle, Smooth, Vascular; Oxytocin; Piperidines; Pyrrolidines; Quinolones; Radioligand Assay; Receptors, Vasopressin; Vasopressins | 1995 |
Binding of [3H] SR 49059, a potent nonpeptide vasopressin V1a antagonist, to rat and human liver membranes.
Topics: Animals; Arginine Vasopressin; Binding, Competitive; Cell Membrane; Humans; Indoles; Kinetics; Liver; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin | 1994 |
Effect of a new, potent, non-peptide V1a vasopressin antagonist, SR 49059, on the binding and the mitogenic activity of vasopressin on Swiss 3T3 cells.
Topics: 3T3 Cells; Animals; Arginine Vasopressin; Binding Sites; Cell Division; DNA; Flow Cytometry; Indoles; Mice; Mitogens; Piperidines; Pyrrolidines; Quinolones; Receptors, Vasopressin | 1994 |
Biochemical and pharmacological properties of SR 49059, a new, potent, nonpeptide antagonist of rat and human vasopressin V1a receptors.
Topics: Animals; Arginine Vasopressin; Cattle; Cell Membrane; Humans; In Vitro Techniques; Indoles; Muscle Contraction; Piperidines; Platelet Aggregation; Pyrrolidines; Quinolones; Rats; Receptors, Vasopressin | 1993 |
Potent inhibitory effect of SR 49059, an orally active non-peptide vasopressin VIa receptor antagonist, on human arterial coronary bypass graft.
Topics: Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Hormone Antagonists; Humans; Indoles; Mammary Arteries; Muscle Contraction; Pyrrolidines | 1995 |
[Arg8]vasopressin-induced responses of the human isolated coronary artery: effects of non-peptide receptor antagonists.
Topics: Adolescent; Adult; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Child; Coronary Vessels; Endothelium, Vascular; Female; Humans; In Vitro Techniques; Indoles; Male; Middle Aged; Muscle, Smooth, Vascular; Piperidines; Potassium; Pyrrolidines; Quinolones; Vasoconstrictor Agents | 1995 |
Modulation of the effect of arginine-vasopressin on water and ion transport in the newt early distal tubule and frog urinary bladder by V1-antagonists.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Biological Transport; Hormone Antagonists; Indoles; Ions; Kidney Tubules, Distal; Naphthalenes; Osmolar Concentration; Permeability; Protein Kinase C; Pyrrolidines; Salamandridae; Urinary Bladder; Water | 1995 |
Effect of the non-peptide, vasopressin V1a receptor antagonist, SR 49059 and its enantiomer, SR 49770, on isolated human myometrium.
Topics: Arginine Vasopressin; Dysmenorrhea; Female; Hormone Antagonists; Humans; In Vitro Techniques; Indoles; Myometrium; Pyrrolidines; Vasoconstrictor Agents | 1996 |
Autoradiographic localization of vasopressin V1a receptors in the rat kidney using [3H]-SR 49059.
Topics: Animals; Arginine Vasopressin; Autoradiography; Hormone Antagonists; Humans; Indoles; Kidney; Kinetics; Liver; Male; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Tissue Distribution; Tritium | 1996 |
Vascular effects of [Arg8]vasopressin in the isolated perfused rat kidney.
Topics: Angiotensin II; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Enzyme Inhibitors; Hormone Antagonists; In Vitro Techniques; Indoles; Kidney; Male; Nitric Oxide; Norepinephrine; Perfusion; Prostaglandins; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Renal Agents; Vasoconstrictor Agents | 1996 |
Pharmacological characterization of a vasopressin V1 receptor in the isolated human gastric artery.
Topics: Aged; Aged, 80 and over; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Benzazepines; Humans; In Vitro Techniques; Indoles; Middle Aged; Muscle, Smooth, Vascular; Oxytocin; Piperidines; Pyrrolidines; Quinolones; Receptors, Vasopressin; Stomach; Vasoconstrictor Agents | 1997 |
Effects of the vasopressin V1a receptor antagonist, SR 49059, on the response of human uterine arteries to vasopressin and other vasoactive substances.
Topics: Adult; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Dinoprost; Dose-Response Relationship, Drug; Endothelin-1; Female; Humans; In Vitro Techniques; Indoles; Middle Aged; Norepinephrine; Pyrrolidines; Uterus; Vasoconstriction; Vasoconstrictor Agents | 1998 |
Nonpeptide arginine vasopressin antagonists for both V1A and V2 receptors: synthesis and pharmacological properties of 2-phenyl-4'-(2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-1-carbonyl) benzanilide derivatives.
Topics: Anilides; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Biological Availability; Female; In Vitro Techniques; Indoles; Magnetic Resonance Spectroscopy; Pyrrolidines; Rabbits; Rats; Receptors, Oxytocin | 1998 |
Characterization of receptors mediating contraction of the rat isolated small mesenteric artery and aorta to arginine vasopressin and oxytocin.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Aorta; Arginine Vasopressin; Dose-Response Relationship, Drug; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Pyrrolidines; Quinolones; Rats; Rats, Wistar; Receptors, Oxytocin; Receptors, Vasopressin; Vasotocin | 1998 |
Lack of effect of a selective vasopressin V1A receptor antagonist SR 49,059, on potentiation by vasopressin of adrenoceptor-mediated pressor responses in the rat mesenteric arterial bed.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Blood Pressure; Drug Synergism; Hormone Antagonists; Indoles; Male; Mesenteric Arteries; Methoxamine; Perfusion; Pressoreceptors; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Vasoconstriction; Vasoconstrictor Agents | 1998 |
V1a- and V2-type vasopressin receptors mediate vasopressin-induced Ca2+ responses in isolated rat supraoptic neurones.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcium; Deamino Arginine Vasopressin; In Vitro Techniques; Indoles; Kinetics; Male; Morpholines; Neurons; Pyrrolidines; Rats; Rats, Wistar; Receptors, Vasopressin; Spiro Compounds; Supraoptic Nucleus; Transcription, Genetic; Vasoconstrictor Agents; Vasopressins | 1999 |
Vasopressin receptors in human adrenal medulla and pheochromocytoma.
Topics: Adrenal Gland Neoplasms; Adrenal Medulla; Adult; Arginine Vasopressin; Autoradiography; Calcium; Cell Membrane; Cells, Cultured; Exocytosis; Hormone Antagonists; Humans; Indoles; Middle Aged; Pheochromocytoma; Pyrrolidines; Receptors, Vasopressin; Reverse Transcriptase Polymerase Chain Reaction; Tumor Cells, Cultured | 1999 |
Mechanisms underlying arginine vasopressin-induced relaxation in monkey isolated coronary arteries.
Topics: Animals; Arginine; Arginine Vasopressin; Coronary Vessels; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Macaca; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Pyrrolidines; Receptors, Vasopressin; Vasodilation | 1999 |
Oxytocin and vasopressin constrict rat isolated uterine resistance arteries by activating vasopressin V1A receptors.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Drug Antagonism; Female; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Muscle, Smooth, Vascular; Oxytocin; Pyrrolidines; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Uterine Contraction; Uterus; Vascular Resistance; Vasoconstriction; Vasotocin | 1999 |
Vasopressin(4-9) fragment activates V1a-type vasopressin receptor in rat supraoptic neurones.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcium; Fluorescent Dyes; Fura-2; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Morpholines; Neurons; Peptide Fragments; Pyrrolidines; Rats; Rats, Wistar; Receptors, Vasopressin; Spiro Compounds; Supraoptic Nucleus | 1999 |
Vasopressin V2 (SR121463A) and V1a (SR49059) receptor antagonists both inhibit desmopressin vasorelaxing activity.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Aorta; Arginine Vasopressin; Deamino Arginine Vasopressin; Endothelium, Vascular; Hemostatics; Hormone Antagonists; Indoles; Male; Morpholines; Pyrrolidines; Rats; Rats, Wistar; Spiro Compounds | 1999 |
[Arg8]-vasopressin-induced responses on coronary and mesenteric arteries of rats with myocardial infarction: the effects of V1a- and V2-receptor antagonists.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Coronary Circulation; Coronary Vessels; Indoles; Ligation; Male; Mesenteric Arteries; Myocardial Infarction; Pyrrolidines; Rats; Rats, Wistar; Receptors, Vasopressin; Vasoconstrictor Agents | 2000 |
Effects of YM471, a nonpeptide AVP V(1A) and V(2) receptor antagonist, on human AVP receptor subtypes expressed in CHO cells and oxytocin receptors in human uterine smooth muscle cells.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Azepines; Binding, Competitive; Calcium; Cell Membrane; CHO Cells; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Female; Humans; Indoles; Morpholines; Muscle, Smooth; Oxytocin; Piperidines; Pyrrolidines; Radioligand Assay; Receptors, Oxytocin; Receptors, Vasopressin; Spiro Compounds; Tritium; Uterus | 2001 |
A nonpeptide vasopressin V(1a) receptor antagonist, SR 49059, does not prevent cisplatin-induced emesis in piglets.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Antiemetics; Antineoplastic Agents; Arginine Vasopressin; Cell Membrane; Cisplatin; Disease Models, Animal; Hormone Antagonists; Hypertension; Indoles; Liver; Pyrrolidines; Swine; Vomiting | 2001 |
Interplay between presynaptic and postsynaptic activities is required for dendritic plasticity and synaptogenesis in the supraoptic nucleus.
Topics: Animals; Arginine Vasopressin; Calcium; Dendrites; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Hormone Antagonists; In Vitro Techniques; Indoles; Microinjections; Morpholines; N-Methylaspartate; Neuronal Plasticity; Neurons; Oxytocin; Presynaptic Terminals; Pyrrolidines; Rats; Receptors, N-Methyl-D-Aspartate; Spiro Compounds; Supraoptic Nucleus; Synapses; Synaptic Transmission | 2002 |
Participation of vasopressin in the development of cerebral vasospasm in a rat model of subarachnoid haemorrhage.
Topics: Animals; Arginine Vasopressin; Basilar Artery; Disease Models, Animal; Female; Indoles; Pyrans; Pyrrolidines; Quinolones; Rats; Rats, Sprague-Dawley; Subarachnoid Hemorrhage; Vasospasm, Intracranial | 2004 |
cAMP/PKA-dependent increases in Ca Sparks, oscillations and SR Ca stores in retinal arteriolar myocytes after exposure to vasopressin.
Topics: Aniline Compounds; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arterioles; Caffeine; Calcium; Calcium Signaling; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fluorometry; Fura-2; Indoles; Microscopy, Confocal; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Pyrrolidines; Receptors, Vasopressin; Retinal Artery; Sarcoplasmic Reticulum; Swine; Vasoconstrictor Agents; Xanthenes | 2010 |
Role of vasopressin V(₁A) receptor in the urethral closure reflex in rats.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Dose-Response Relationship, Drug; Female; Hormone Antagonists; In Situ Hybridization; Indoles; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Reflex; Reverse Transcriptase Polymerase Chain Reaction; Urethra | 2011 |
Distinct receptor subtypes mediate arginine vasopressin-dependent ACTH release and intracellular calcium mobilization in rat pituitary cells.
Topics: Adrenocorticotropic Hormone; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcium; Cells, Cultured; Cyclic AMP; Drug Interactions; Female; Indoles; Oxytocin; Pituitary Gland, Anterior; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Time Factors; Vasotocin | 2012 |
β-adrenergic receptor-mediated cardiac contractility is inhibited via vasopressin type 1A-receptor-dependent signaling.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Calcium Signaling; Cardiomyopathy, Hypertrophic; Cats; Cell Line, Tumor; Colforsin; Cyclic AMP; G-Protein-Coupled Receptor Kinases; Genes, Reporter; GTP-Binding Protein alpha Subunits, Gq-G11; Heart Failure; HEK293 Cells; Humans; Indoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Mutagenesis, Site-Directed; Myocardial Contraction; Pyrrolidines; Receptors, Adrenergic, beta; Receptors, Vasopressin; Recombinant Fusion Proteins; Rolipram; Second Messenger Systems | 2014 |
Central effect of vasotocin 4 receptor (VT4R/V1aR) antagonists on the stress response and food intake in chicks given neuropeptide Y (NPY).
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Chickens; Corticosterone; Eating; Immobilization; Indoles; Injections, Intraventricular; Male; Neuropeptide Y; Pyrrolidines; Receptors, Vasopressin; Stress, Psychological | 2016 |
The modulatory effect of nitric oxide in pro- and anti-convulsive effects of vasopressin in PTZ-induced seizures threshold in mice.
Topics: Animals; Anticonvulsants; Antidiuretic Hormone Receptor Antagonists; Arginine; Arginine Vasopressin; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guanidines; Indoles; Male; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Pentylenetetrazole; Pyrrolidines; Receptors, Vasopressin; Seizures | 2016 |
Childhood stress impairs social function through AVP-dependent mechanisms.
Topics: Adult; Adverse Childhood Experiences; Aged; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Behavior, Animal; Borderline Personality Disorder; Disease Models, Animal; Female; Humans; Indoles; Male; Middle Aged; Neurophysins; Paraventricular Hypothalamic Nucleus; Protein Precursors; Pyrrolidines; Rats; Sexual Maturation; Social Behavior; Stress, Psychological; Supraoptic Nucleus; Vasopressins; Young Adult | 2019 |