arginine has been researched along with thiazoles in 92 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 22 (23.91) | 18.7374 |
1990's | 14 (15.22) | 18.2507 |
2000's | 29 (31.52) | 29.6817 |
2010's | 27 (29.35) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Makisumi, S; Mizusaki, K; Ohyama, S; Tsunematsu, H | 1 |
Carminati, R; Falchi, M; Guadagni, L; Lodi, R; Nebuloni, R | 1 |
Saigot, T | 1 |
Ripani, G; Trasatti, GA | 1 |
Axelrud-Cavadore, C; Coletti-Previero, MA | 1 |
de Nucci, G; Mitchell, JA; Vane, JR; Warner, TD | 1 |
Alary, J; Carrera, G; de Saint Blanquat, G; Faurie, M; Lamboeuf, Y; Roumec, C | 1 |
Halbach, G; Trost, W; Vogel, G | 1 |
Fairwell, T; Lovins, RE | 1 |
Sommavilla, B; Zanetti, R | 1 |
Hojima, Y; Moriwaki, C; Moriya, H; Todoki, N | 1 |
Kovaliv, IuD | 1 |
Caciacli, F; Ciancetta, S; Ciccarelli, R | 1 |
Faini, D; Pagella, PG; Turba, C | 2 |
Buzzi, S; Ghetti, C; Sala, G | 2 |
Raymond, N | 1 |
Dubini, F; Falchi, M | 1 |
Dubini, F; Falchi, M; Nebuloni, R | 1 |
Dubini, F; Falchi, M; Ferrario, F; Marcucci, A | 1 |
Carminati, R; Dubini, F; Falchi, M; Ferrario, F; Marcucci, A | 1 |
Bortolan-Gianese, P; Dubini, F; Falchi, M; Ferrario, F; Marcucci, A | 1 |
Fowler, M; Furfine, ES; Garvey, EP; Harmon, MF; Marshall, S; Oplinger, JA; Paith, JE; Sherman, PA; Tanoury, GJ | 1 |
Chang, K; Corbett, JA; Currie, MG; Hasan, KS; McDaniel, ML; Misko, TP; Moore, WM; Petrash, JM; Smith, SR; Tilton, RG | 1 |
Devissaguet, M; Ferreira, SH; Lesieur, D; Lorenzetti, BB; Tsouderos, Y | 1 |
Andrade-Gordon, P; Costanzo, MJ; Hecker, LR; Kauffman, JA; Krishnan, R; Lewis, JM; Maryanoff, BE; Schott, MR; Tulinsky, A; Yabut, SC; Zhang, HC | 1 |
Cendan, JC; Copeland, EM; Lind, DS; Souba, WW | 1 |
Lesage, AS; Leysen, JE; Peeters, L | 1 |
Conejo, L; Ortiz, JA; Palop, D; Sacristán, A | 1 |
Ischiropoulos, H; Thom, SR; Xu, YA | 1 |
Carson, M; Chattopadhyay, D; Costanzo, MJ; DeLucas, LJ; Maryanoff, B; Recacha, R | 1 |
Bouisson, M; Escrieut, C; Fehrentz, JA; Fourmy, AD; Gigoux, V; Gully, D; Maigret, B; Martinez, J; Moroder, L; Silvente-Poirot, S; Vaysse, N | 1 |
Hirasawa, Y; Ito, K; Kato, Y; Kita, Y; Motoyama, Y; Nishio, M; Seki, J; Yamanaka, T | 1 |
Ambler, J; Baettig, U; Brown, L; Brundish, D; Cockcroft, X; Dell, C; Furzer, A; Garman, S; Janus, D; Kane, PD; Mitchelson, A; Smith, G; Talbot, MD; Tweed, M; Walker, CV; Wills, N | 1 |
Chakraborty, T; Domann, E; Gerstel, B; Gröbe, L; Machesky, LM; Pistor, S; Sechi, AS; Wehland, J | 1 |
Bakala, H; Depreux, P; Fourmaintraux, E; Schwedler, SB; Striker, GE; Striker, LJ; Verbeke, P; Vilar, J; Weiss, MF | 1 |
Andrews, RC; Becherer, JD; Bickett, DM; Bubacz, DG; Conway, JG; Cowan, DJ; Gaul, M; Glennon, K; Lambert, MH; Leesnitzer, MA; McDougald, DL; Moss, ML; Musso, DL; Rabinowitz, MH; Rizzolio, MC | 1 |
Chough, E; Daley, J; Gupta, S; Keaney, JF; Oates, P; Ruderman, NB; Tornheim, K | 1 |
Abbasi, F; Chu, JW; Cooke, JP; Lamendola, C; McLaughlin, TL; Reaven, GM; Stühlinger, MC; Tsao, PS | 1 |
Beck-Sickinger, A; Demuth, H; Dimitrijević, M; Kovacević-Jovanović, V; Stanojević, S; von Hörsten, S; Vujić, V | 1 |
Eliseenkova, AV; Garbi, M; Goldfarb, M; Mohammadi, M; Olsen, SK; Ornitz, DM; Zampieri, N | 1 |
Hirasawa-Taniyama, Y; Ito, K; Kato, Y; Kita, Y; Mihara, K; Miyata, S; Mutoh, S; Nishio, M; Seki, J; Yamanaka, T | 1 |
Hollingdal, M; Juhl, CB; Lönnqvist, F; Prange, A; Pørksen, N; Schmitz, O | 1 |
LEVY, AL; LI, SO | 1 |
Furuichi, K; Hagiwara, M; Hosoya, T; Kimura, H; Koizumi, J; Koizumi, T; Krainer, AR; Muraki, M; Murray, MV; Ohkawara, B; Onogi, H; Shibuya, H; Sumi, K; Suzuki, M; Yomoda, J | 1 |
Bakija, AT; Kikelj, D; Krbavcic, A; Marinko, P; Mlinsek, G; Solmajer, T; Stegnar, M; Stojan, J | 1 |
Carlsson, K; Carlsson, U; Hammarström, P; Herland, A; Persson, E; Svensson, M; Wiréhn, J | 1 |
Jaiswal, TN; Koti, M; Mishra, SC; Tayade, C | 1 |
Abdel-Meguid, SS; Babine, RE; Bannister, TD; Bibbins, F; Celatka, CA; Deng, H; Gorga, J; Jin, L; Lazarova, TI; Lin, J; Meyers, HV; Nagafuji, P; Pandey, P; Quinn, J; Rynkiewicz, MJ; Strickler, JE | 1 |
Chen, CC; Huang, CJ; Huang, CL; Lee, JJ; Lu, YT; Tsai, PS | 1 |
Cherney, MM; James, MN; Lemieux, MJ; Mahuran, DJ; Mark, BL; Withers, SG | 1 |
Hassinger, JN; Iversen, PL; Lovejoy, CE; Moulton, HM; Nelson, MH; Wu, RP; Youngblood, DS | 1 |
Bielawski, KP; Graczyk, A; Grinholc, M; Kawiak, A; Kurlenda, J | 1 |
Futaki, S; Jones, AT; Kosuge, M; Nakase, I; Takeuchi, T | 1 |
Bammler, TK; Hashioka, S; Jin, J; Kashima, DT; Klegeris, A; Li, J; Maguire, J; McGeer, PL; Pan, S; Zhang, J; Zhu, D | 1 |
Barter, PJ; Brown, BE; Davies, MJ; Nobécourt, E; Rye, KA; Yadav, S; Zeng, J | 1 |
Iwamoto, S; Katunuma, N; Marquez, VE; Nagahama, M; Nishizawa, M; Oda, M; Sakurai, J; Tsuge, H; Utsunomiya, H | 1 |
Gu, Z; He, B; Li, L; Luo, K; Nie, Y; Shi, S; Yang, J; Yang, Y; Zhu, R | 1 |
Drinkut, A; Falkenburger, BH; Gerhardt, E; Krenz, A; Schulz, JB | 1 |
El-Maradny, HA; Hikal, AH; Kamel, OA; Mortada, SA | 1 |
Hartog, JW; Voors, AA; Willemsen, S | 1 |
Heth, J; Hoff, JT; Hua, Y; Keep, RF; Muraszko, KM; Tang, L; Xi, G | 1 |
Adams-Deutsch, T; Heilig, M; Nair, SG; Navarre, BM; Pickens, CL; Shaham, Y | 1 |
Chen, CY; Liu, KN; Wang, HY; Wang, SS | 1 |
Ang, BU; Kirschner, RE; Nah, HD; Spivak, RM | 1 |
Chang, SH; Harocopos, GJ; Huang, AJ; Patel, DA; Thang, DH; Vora, SC | 1 |
Hänggi, D; Ogawa, T; Steiger, HJ | 1 |
Chiang, HJ; Dai, YH; Lee, HJ; Liu, BR | 1 |
Henderson, JP; Lv, H | 1 |
Bhende, S; Jadhav, N | 1 |
Komatsu, J; Kuwano, R; Matsunari, I; Ono, K; Samuraki, M; Shima, K; Yamada, M; Yanase, D | 1 |
Kamijo, S; Kawasaki, T | 1 |
Inoue, R; Ochi, M; Onoue, S; Yamada, S; Yamauchi, Y | 1 |
Cidral-Filho, FJ; Martins, DF; Mazzardo-Martins, L; Santos, AR; Stramosk, J | 1 |
Du, X; Fu, D; Huang, C; Liu, Y; Pei, D; Sun, H | 1 |
Banala, S; Overkleeft, HS; Piwowarska, NA; Süssmuth, RD | 1 |
Banerjee, S; Clayton, GM; Garavito, RM; Ghebreselasie, K; Hermanson, DJ; Marnett, LJ; Xu, S | 1 |
Aizawa, N; Homma, Y; Igawa, Y | 1 |
Ansell, JE; Bakhru, SH; Brown, K; Costin, JC; Dishy, V; Grosso, M; Laulicht, BE; Noveck, RJ; Steiner, SS | 1 |
Baneham, S; Cox, D; Kirby, BP; Moollan, A; O'Donnell, A; Ozgul, M; Pabari, RM; Ramtoola, Z | 1 |
Ashcroft, AE; Radford, SE; Raleigh, DP; Tu, LH; Wong, AG; Young, LM | 1 |
Cuker, A; Siegal, D | 1 |
Kaminskas, E; Reiffel, JA; Reilly, P; Sager, P; Sarich, T; Seltzer, J; Weitz, JI | 1 |
Antman, EM; Giugliano, RP; Ruff, CT | 1 |
Fanikos, J; Huisman, MV | 1 |
Ansell, JE; Bakhru, SH; Brown, K; Costin, JC; Dishy, V; Grosso, MA; Lanz, HJ; Laulicht, BE; Mercuri, MF; Noveck, RJ; Steiner, SS | 1 |
Bhagirath, VC; Eikelboom, JW; Monagle, S; Ng, KH | 1 |
Gkiatas, I; Korompilias, AV; Kostas-Agnantis, I; Papadopoulos, DV; Tsantes, AG; Ziara, P | 1 |
Ageno, W; Agnelli, G; Chan, NC; De Caterina, R; Diener, HC; Hylek, E; Lip, GYH; Raskob, GE; Siegal, DM; Verheugt, FWA; Weitz, JI | 1 |
Gemba, K; Kiura, K; Matsumura, T; Moritaka, T; Ohnoshi, T; Segawa, Y; Shibayama, T; Tabata, M; Takigawa, N; Ueoka, H | 1 |
Guo, D; Hou, L; Mao, P; Mo, L; Xiao, X; Yang, X | 1 |
7 review(s) available for arginine and thiazoles
Article | Year |
---|---|
Monitoring and reversal of direct oral anticoagulants.
Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Anticoagulants; Arginine; Blood Coagulation Factors; Blood Coagulation Tests; Dabigatran; Factor VIIa; Factor Xa; Factor Xa Inhibitors; Hemorrhage; Hemostasis; Humans; Partial Thromboplastin Time; Piperazines; Prothrombin; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Thiazoles; Thrombin Time | 2015 |
NOAC monitoring, reversal agents, and post-approval safety and effectiveness evaluation: A cardiac safety research consortium think tank.
Topics: Antibodies, Monoclonal, Humanized; Antidotes; Antithrombins; Arginine; Atrial Fibrillation; Congresses as Topic; Dabigatran; Drug Monitoring; Factor Xa; Factor Xa Inhibitors; Humans; Partial Thromboplastin Time; Piperazines; Product Surveillance, Postmarketing; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Stroke; Thiazoles; Thrombin Time; Venous Thromboembolism | 2016 |
Management of Bleeding With Non-Vitamin K Antagonist Oral Anticoagulants in the Era of Specific Reversal Agents.
Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Antithrombins; Arginine; Blood Coagulation Factors; Dabigatran; Factor VIIa; Factor Xa; Factor Xa Inhibitors; Hemorrhage; Hemostatics; Humans; Piperazines; Plasma; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Thiazoles | 2016 |
Idarucizumab and factor Xa reversal agents: role in hospital guidelines and protocols.
Topics: Antibodies, Monoclonal, Humanized; Anticoagulants; Arginine; Clinical Protocols; Dabigatran; Emergency Treatment; Factor Xa; Factor Xa Inhibitors; Hemorrhage; Hospitals; Humans; Patient Selection; Piperazines; Practice Guidelines as Topic; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Surgical Procedures, Operative; Thiazoles | 2016 |
Clinical implications of reversal agents for direct oral anticoagulants.
Topics: Antibodies, Monoclonal, Humanized; Anticoagulants; Antithrombins; Arginine; Dabigatran; Factor Xa; Factor Xa Inhibitors; Hemorrhage; Humans; Piperazines; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Thiazoles; Venous Thromboembolism | 2017 |
The role of new oral anticoagulants in orthopaedics: an update of recent evidence.
Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Anticoagulants; Arginine; Blood Coagulation Tests; Dabigatran; Factor Xa; Hemorrhage; Humans; Orthopedic Procedures; Piperazines; Practice Guidelines as Topic; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Rivaroxaban; Thiazoles; Venous Thromboembolism | 2017 |
The Non-Vitamin K Antagonist Oral Anticoagulants in Heart Disease: Section V-Special Situations.
Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Anticoagulants; Arginine; Atrial Fibrillation; Benzamides; Biomarkers; Blood Coagulation; Clinical Trials as Topic; Dabigatran; Drug Administration Schedule; Factor Xa; Heart Diseases; Humans; Piperazines; Pyrazoles; Pyridines; Pyridones; Recombinant Proteins; Risk; Rivaroxaban; Stroke; Thiazoles; Thrombin; Venous Thromboembolism; Vitamin K; Warfarin | 2019 |
3 trial(s) available for arginine and thiazoles
Article | Year |
---|---|
Influence of rosiglitazone treatment on beta-cell function in type 2 diabetes: evidence of an increased ability of glucose to entrain high-frequency insulin pulsatility.
Topics: Arginine; Blood Glucose; Diabetes Mellitus, Type 2; Double-Blind Method; Entropy; Female; Glucose; Glucose Clamp Technique; Humans; Hypoglycemic Agents; Insulin; Islets of Langerhans; Male; Middle Aged; Rosiglitazone; Stimulation, Chemical; Thiazoles; Thiazolidinediones | 2003 |
Effect of desensitising paste containing 8% arginine and calcium carbonate on biofilm formation of Streptococcus mutans in vitro.
Topics: Adolescent; Adult; Anti-Bacterial Agents; Arginine; Bacterial Adhesion; Biofilms; Calcium Carbonate; Coloring Agents; Dental Prophylaxis; Dentifrices; Dentin; Dentin Desensitizing Agents; Fluorides; Humans; Imaging, Three-Dimensional; Lactic Acid; Microbial Viability; Microscopy, Electron, Scanning; Phosphates; Silicates; Streptococcus mutans; Tetrazolium Salts; Thiazoles; Time Factors; Young Adult | 2013 |
Single-dose ciraparantag safely and completely reverses anticoagulant effects of edoxaban.
Topics: Administration, Oral; Adult; Arginine; Blood Coagulation; Double-Blind Method; Drug Monitoring; Factor Xa Inhibitors; Humans; Injections, Intravenous; Male; North Carolina; Piperazines; Pyridines; Thiazoles; Whole Blood Coagulation Time | 2017 |
82 other study(ies) available for arginine and thiazoles
Article | Year |
---|---|
Kinetics of hydrolysis of phenylthiazolones of arginine, homoarginine, norarginine, and canaavanine by trypsin.
Topics: Arginine; Canavanine; Homoarginine; Hydrogen-Ion Concentration; Kinetics; Substrate Specificity; Thiazoles; Trypsin | 1979 |
[Antihepatotoxic activity of arginine thiazolidinecarboxylate in hepatitis induced by galactosamine in the rat].
Topics: Animals; Arginine; Chemical and Drug Induced Liver Injury; Female; Galactosamine; Rats; Thiazoles | 1979 |
[Value of tiadilon in hepatobiliary pathology].
Topics: Adult; Aged; Alcoholic Intoxication; Arginine; Asthenia; Dietary Fats; Female; Hepatitis, Viral, Human; Humans; Liver Diseases; Male; Middle Aged; Thiazoles; Thiazolidines | 1979 |
[Therapeutic effectiveness of thiazolidinecarboxylate of arginine in psychiatric patients with hepatic disorders of toxic origin (alcohol, drugs)].
Topics: Adult; Aged; Antidepressive Agents; Arginine; Carboxylic Acids; Chemical and Drug Induced Liver Injury; Drug Combinations; Female; Hepatitis, Alcoholic; Humans; Male; Mental Disorders; Middle Aged; Thiazoles; Tranquilizing Agents | 1979 |
Changes of substrate configuration during trypsin hydrolysis of arginine and lysine 2-phenyl-thiazol-5-ones.
Topics: Arginine; Kinetics; Lysine; Molecular Conformation; Optical Rotation; Protein Binding; Stereoisomerism; Thiazoles; Trypsin | 1975 |
Alkaline buffers release EDRF from bovine cultured aortic endothelial cells.
Topics: Animals; Arginine; Buffers; Cattle; Cells, Cultured; Cyclohexanones; Endothelium, Vascular; Epoprostenol; Hydrogen-Ion Concentration; Lipoprotein Lipase; Nitric Oxide; omega-N-Methylarginine; Platelet Activating Factor; Pyrimidinones; Thiazoles | 1991 |
Impairment of mitochondrial membrane by ethanol and protective effect of a thiazolidine compound in in vitro and in vivo experiments.
Topics: Animals; Arginine; Cell Membrane; Ethanol; Fatty Acids; Glutathione; Membrane Lipids; Microsomes, Liver; Rats; Thiazoles; Thiazolidines | 1990 |
[Protective action of silymarine in phalloidine intoxication in the mouse].
Topics: Animals; Arginine; Betaine; Female; Glycosides; Homocysteine; Lactones; Mice; Mycotoxins; Phalloidine; Silymarin; Structure-Activity Relationship; Thiazoles | 1974 |
Quantitative protein sequencing using mass spectrometry: mass spectral analysis of 2-anilino-5-thiazolinone derivatives of amino acids without prior conversion to the phenyl thiohydantoins.
Topics: Alanine; Amino Acid Sequence; Amino Acids; Aniline Compounds; Animals; Arginine; Autoanalysis; Cattle; Chemical Phenomena; Chemistry; Drug Stability; Glutamates; Hydantoins; Lysine; Mass Spectrometry; Methods; Phenylalanine; Ribonucleases; Serine; Sulfides; Thiazoles; Thiocyanates; Threonine; Tyrosine | 1971 |
[On some aspects of the treatment of delirium tremens].
Topics: Arginine; Humans; Psychoses, Alcoholic; Sulfonic Acids; Thiazoles | 1970 |
A new sensitive assay method of kallikrein-like arginine-esterases.
Topics: Aldehydes; Arginine; Colorimetry; Endopeptidases; Hydrazines; Indicators and Reagents; Kallikreins; Ketones; Methods; Oxidation-Reduction; Thiazoles | 1971 |
[Synthesis of rhodanines on the basis of arginine].
Topics: Arginine; Thiazoles | 1968 |
Effect of arginine salt of thioproline (thiazolidine carboxylate) on cyclic nucleotides of cerebral tumour.
Topics: Arginine; Brain Chemistry; Brain Neoplasms; Cyclic AMP; Cyclic GMP; Humans; Thiazoles; Thiazolidines | 1980 |
Effect of arginine thiazolidinecarboxylate on allyl alcohol hepatotoxicity in the rat.
Topics: 1-Propanol; Alanine Transaminase; Alkaline Phosphatase; Animals; Arginine; Aspartate Aminotransferases; Chemical and Drug Induced Liver Injury; Kinetics; Propanols; Rats; Thiazoles; Thiazolidines | 1981 |
[Experiment comparative clinical study with three liver trophical substances on some alcoholic not cirrhotic liver disease (author's transl)].
Topics: Adult; Aged; Arginine; Cyclohexanecarboxylic Acids; Female; Humans; Liver Diseases, Alcoholic; Male; Middle Aged; Phosphatidylcholines; Thiazoles; Thiazolidines | 1980 |
[Further clinical observations on the treatment of noncirrhotic alcoholic liver disease].
Topics: Adult; Aged; Arginine; Cyclohexanecarboxylic Acids; Female; Humans; Liver Diseases, Alcoholic; Male; Middle Aged; Phosphatidylcholines; Thiazoles; Thiazolidines | 1980 |
[Value of the use of a new hepatotropic drug, arginine tidiacicate in gastroenterology. Results of a multicentric study].
Topics: Adult; Aged; Arginine; Female; Gastrointestinal Diseases; Humans; Liver Diseases; Male; Middle Aged; Thiazoles; Thiazolidines | 1981 |
Arginine thiazolidinecarboxylate 14C uptake by individual phospholipids isolated from rat liver microsomes.
Topics: Animals; Arginine; Carbon Radioisotopes; Male; Microsomes, Liver; Phospholipids; Rats; Thiazoles; Thiazolidines | 1981 |
[Tissue distribution of carbon-14 following oral administration of 14C-arginine thiazolidinecarboxylate in rats].
Topics: Animals; Arginine; Rats; Thiazoles; Thiazolidines; Tissue Distribution | 1981 |
[Protective effect of arginine thiazolidinecarboxylate on morphological and functional changes in the liver induced by chronic ethanol intoxication in the rat].
Topics: Animals; Arginine; Liver Diseases, Alcoholic; Rats; Thiazoles; Thiazolidines | 1980 |
[Normalizing effect of arginine thiazolidincarboxylate (ATCA) on hepatocytes in CCL4 poisoning in rats].
Topics: Animals; Arginine; Carbon Tetrachloride Poisoning; Chemical and Drug Induced Liver Injury; Male; Rats; Thiazoles; Thiazolidines | 1980 |
[Transmethylating activity of arginine thiazolidinecarboxylate (ATCA) in acute CCL4 poisoning and diet-induced steatosis in the rat].
Topics: Animals; Arginine; Carbon Tetrachloride Poisoning; Chemical and Drug Induced Liver Injury; Diet; Fatty Liver; Male; Methylation; Rats; Thiazoles; Thiazolidines | 1980 |
[Activity of arginine thiazolidin carboxylate on the acute poisoning by paracetamol in mice].
Topics: Acetaminophen; Animals; Arginine; Liver; Male; Mice; Thiazoles; Thiazolidines | 1980 |
Potent and selective inhibition of human nitric oxide synthases. Inhibition by non-amino acid isothioureas.
Topics: Amino Acid Oxidoreductases; Animals; Arginine; Endothelium, Vascular; Enzyme Induction; Humans; Isoenzymes; Isothiuronium; Kinetics; Mice; Models, Chemical; Neurons; Nitric Oxide Synthase; Species Specificity; Structure-Activity Relationship; Thiazoles; Thiourea | 1994 |
Prevention of diabetic vascular dysfunction by guanidines. Inhibition of nitric oxide synthase versus advanced glycation end-product formation.
Topics: Aldehyde Reductase; Amino Acid Oxidoreductases; Animals; Arginine; Benzothiazoles; Blood Pressure; Body Weight; Capillary Permeability; Citrulline; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Glycation End Products, Advanced; Guanidines; Imidazoles; Imidazolidines; Inositol; Iodine Radioisotopes; Male; Methylguanidine; Naphthalenes; Nitric Oxide Synthase; omega-N-Methylarginine; Phthalazines; Rats; Rats, Sprague-Dawley; Retina; Sciatic Nerve; Serum Albumin, Bovine; Sorbitol; Thiazoles; Uvea | 1993 |
S14080, a peripheral analgesic acting by release of an endogenous circulating opioid-like substance.
Topics: Adrenalectomy; Analgesics; Animals; Arginine; Dipyrone; Drug Tolerance; Edema; Endorphins; Fever; Hyperalgesia; Indomethacin; Male; Methylene Blue; Nitric Oxide; omega-N-Methylarginine; Pain Measurement; Rats; Rats, Wistar; Thiazoles; Yohimbine | 1995 |
Potent thrombin inhibitors that probe the S1 subsite: tripeptide transition state analogues based on a heterocycle-activated carbonyl group.
Topics: Amino Acid Sequence; Animals; Arginine; Binding Sites; Cattle; Crystallography, X-Ray; Guanidines; Humans; Molecular Sequence Data; Molecular Structure; Oligopeptides; Peptides; Pipecolic Acids; Protein Binding; Serine Proteinase Inhibitors; Sulfonamides; Thiazoles; Thrombin; Trypsin Inhibitors | 1996 |
Increased L-arginine transport in a nitric oxide-producing metastatic colon cancer cell line.
Topics: Adenocarcinoma; Arginine; Biological Transport; Cell Division; Cell Membrane; Colonic Neoplasms; Coloring Agents; Dexamethasone; Glucocorticoids; Humans; Hydrogen-Ion Concentration; Kinetics; Lymphatic Metastasis; Nitric Oxide; Sodium; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Up-Regulation | 1996 |
Lubeluzole, a novel long-term neuroprotectant, inhibits the glutamate-activated nitric oxide synthase pathway.
Topics: Animals; Arginine; Cells, Cultured; Cyclic GMP; Glutamic Acid; Guanylate Cyclase; Hippocampus; Interferon-gamma; Lipopolysaccharides; Neuroprotective Agents; Nitric Oxide Synthase; Piperidines; Rats; Stereoisomerism; Thiazoles | 1996 |
Involvement of endogenous nitric oxide and sulfhydryl compounds in ebrotidine-induced gastroprotection.
Topics: Animals; Arginine; Benzenesulfonates; Ethanol; Ethylmaleimide; Gastric Mucosa; Histamine H2 Antagonists; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptic Ulcer; Rats; Rats, Sprague-Dawley; Specific Pathogen-Free Organisms; Sulfhydryl Compounds; Thiazoles | 1997 |
Vascular endothelial cells generate peroxynitrite in response to carbon monoxide exposure.
Topics: Animals; Arginine; Carbon Monoxide; Cattle; Cell Survival; Cells, Cultured; Chromium; Endothelium, Vascular; Nitrates; Nitric Oxide Synthase; Nitrites; Oxidants; Oxidation-Reduction; Oxygen Consumption; Sulfhydryl Compounds; Tetrazolium Salts; Thiazoles; Tyrosine | 1997 |
Structure of the RWJ-51084-bovine pancreatic beta-trypsin complex at 1.8 A.
Topics: Animals; Arginine; Benzothiazoles; Binding Sites; Cattle; Crystallography, X-Ray; Hydrogen Bonding; Models, Molecular; Molecular Sequence Data; Molecular Structure; Pancreas; Protein Folding; Protein Structure, Secondary; Serine Proteinase Inhibitors; Thiazoles; Thrombin; Trypsin; Trypsin Inhibitors | 1999 |
Arginine 197 of the cholecystokinin-A receptor binding site interacts with the sulfate of the peptide agonist cholecystokinin.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Arginine; Binding Sites; Cholecystokinin; Computer Simulation; COS Cells; Humans; Indoleacetic Acids; Inositol Phosphates; Iodine Radioisotopes; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Protein Conformation; Radioligand Assay; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Recombinant Proteins; Thiazoles; Transfection; Tritium | 1999 |
In vitro antiplatelet profile of FR171113, a novel non-peptide thrombin receptor antagonist.
Topics: Arginine; Aspirin; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Humans; Oligopeptides; Peptide Fragments; Pipecolic Acids; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Thrombin; Serine Endopeptidases; Sulfonamides; Thiazoles; Thiazolidines; Thrombin | 1999 |
The design and synthesis of thrombin inhibitors: analogues of MD805 containing non-polar surrogates for arginine at the P1 position.
Topics: Alanine; Antithrombins; Arginine; Chymotrypsin; Drug Design; Factor Xa Inhibitors; Fibrinolysin; Kallikreins; Models, Molecular; Molecular Structure; Pipecolic Acids; Serine Proteinase Inhibitors; Structure-Activity Relationship; Sulfonamides; Thiazoles; Thrombin; Trypsin | 2000 |
Mutations of arginine residues within the 146-KKRRK-150 motif of the ActA protein of Listeria monocytogenes abolish intracellular motility by interfering with the recruitment of the Arp2/3 complex.
Topics: Actin-Related Protein 2; Actin-Related Protein 3; Actins; Amino Acid Motifs; Amino Acid Sequence; Animals; Arginine; Bacterial Proteins; Biological Transport; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cell Membrane; Chromosomes, Bacterial; Cytoskeletal Proteins; Genes, Bacterial; Intracellular Fluid; Listeria monocytogenes; Membrane Proteins; Molecular Sequence Data; Mutagenesis, Site-Directed; Point Mutation; Sequence Deletion; Thiazoles; Thiazolidines | 2000 |
N-phenacylthiazolium bromide decreases renal and increases urinary advanced glycation end products excretion without ameliorating diabetic nephropathy in C57BL/6 mice.
Topics: Animals; Arginine; Collagen; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Female; Glomerular Mesangium; Glycation End Products, Advanced; Kidney; Kidney Glomerulus; Lysine; Mice; Mice, Inbred C57BL; Proteinuria; Thiazoles | 2001 |
Design of selective and soluble inhibitors of tumor necrosis factor-alpha converting enzyme (TACE).
Topics: ADAM Proteins; ADAM17 Protein; Animals; Arginine; Catalytic Domain; Cell Line; Exudates and Transudates; Female; Formamides; Guanidines; Humans; Leukocytes, Mononuclear; Lipopolysaccharides; Macrophage Activation; Male; Metalloendopeptidases; Mice; Models, Molecular; Molecular Mimicry; Pleurisy; Protease Inhibitors; Rats; Rats, Inbred Lew; Solubility; Structure-Activity Relationship; Thiazoles; Tumor Necrosis Factor-alpha | 2001 |
Hyperglycemia increases endothelial superoxide that impairs smooth muscle cell Na+-K+-ATPase activity.
Topics: Aldehyde Reductase; Animals; Aorta; Arginine; Benzothiazoles; Endothelium, Vascular; Enzyme Inhibitors; Free Radical Scavengers; Glucose; Hyperglycemia; In Vitro Techniques; Muscle, Smooth, Vascular; Phthalazines; Pyrogallol; Rabbits; Sodium-Potassium-Exchanging ATPase; Sorbitol; Superoxide Dismutase; Superoxides; Thiazoles | 2002 |
Relationship between insulin resistance and an endogenous nitric oxide synthase inhibitor.
Topics: Adult; Aged; Arginine; Cardiovascular Diseases; Cross-Sectional Studies; Enzyme Inhibitors; Female; Humans; Hypertension; Hypoglycemic Agents; Lipoproteins; Male; Metabolic Diseases; Metabolic Syndrome; Middle Aged; Nitric Oxide Synthase; Regression Analysis; Risk Factors; Rosiglitazone; Thiazoles; Thiazolidinediones; Vasodilator Agents | 2002 |
Effect of neuropeptide Y on inflammatory paw edema in the rat: involvement of peripheral NPY Y1 and Y5 receptors and interaction with dipeptidyl-peptidase IV (CD26).
Topics: Animals; Arginine; Cells, Cultured; Concanavalin A; Dipeptidyl Peptidase 4; Dose-Response Relationship, Drug; Edema; Hydrogen Peroxide; Inflammation; Isoleucine; Macrophages; Male; Neuropeptide Y; Peptide Fragments; Peptide YY; Rats; Rats, Wistar; Receptors, Neuropeptide Y; Thiazoles | 2002 |
Fibroblast growth factor (FGF) homologous factors share structural but not functional homology with FGFs.
Topics: Amino Acid Sequence; Animals; Arginine; Binding Sites; Cell Survival; Coloring Agents; Crystallography, X-Ray; DNA; DNA Mutational Analysis; Dose-Response Relationship, Drug; Fibroblast Growth Factors; Heparin; Humans; Mice; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Protein Binding; Protein Isoforms; Protein Structure, Secondary; Protein Structure, Tertiary; Recombinant Proteins; Sequence Homology, Amino Acid; Sodium Channels; Sulfates; Tetrazolium Salts; Thiazoles | 2003 |
Inhibition of arterial thrombosis by a protease-activated receptor 1 antagonist, FR171113, in the guinea pig.
Topics: Animals; Arginine; Benzamides; Bleeding Time; Blood Coagulation; Carotid Artery Thrombosis; Chlorides; Dose-Response Relationship, Drug; Ferric Compounds; Guinea Pigs; Heparin; Injections, Subcutaneous; Male; Pipecolic Acids; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptor, PAR-1; Receptors, Thrombin; Sulfonamides; Thiazoles; Thiazolidines | 2003 |
The 2-thio-5-thiazolidones of serine and arginine.
Topics: Arginine; Humans; Serine; Thiazoles | 1954 |
Manipulation of alternative splicing by a newly developed inhibitor of Clks.
Topics: Alternative Splicing; Animals; Arginine; Binding Sites; Cell Nucleus; COS Cells; Dose-Response Relationship, Drug; Enzyme Inhibitors; Globins; HeLa Cells; Humans; Microscopy, Fluorescence; Models, Chemical; Phosphorylation; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Recombinant Proteins; RNA, Messenger; Serine; Signal Transduction; Thiazoles; Time Factors; Xenopus; Xenopus laevis | 2004 |
Novel non-covalent thrombin inhibitors incorporating P(1) 4,5,6,7-tetrahydrobenzothiazole arginine side chain mimetics.
Topics: Arginine; Binding Sites; Biomimetic Materials; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Models, Molecular; Molecular Structure; Protein Binding; Structure-Activity Relationship; Substrate Specificity; Thiazoles; Thrombin; Trypsin | 2004 |
Activity, folding, misfolding, and aggregation in vitro of the naturally occurring human tissue factor mutant R200W.
Topics: Amyloid; Anilino Naphthalenesulfonates; Arginine; Benzothiazoles; Extracellular Space; Factor VIIa; Genetic Carrier Screening; Humans; Kinetics; Mutation; Nephelometry and Turbidimetry; Protein Binding; Protein Denaturation; Protein Folding; Spectrometry, Fluorescence; Substrate Specificity; Thiazoles; Thromboplastin; Tryptophan | 2005 |
L-arginine stimulates immune response in chickens immunized with intermediate plus strain of infectious bursal disease vaccine.
Topics: Adjuvants, Immunologic; Animals; Animals, Newborn; Antibody Formation; Arginine; Birnaviridae Infections; Cell Proliferation; Chick Embryo; Chickens; Electrophoresis, Agar Gel; Enzyme-Linked Immunosorbent Assay; Hemagglutination Inhibition Tests; Immunity, Cellular; Infectious bursal disease virus; Lethal Dose 50; Organ Size; Poultry Diseases; Tetrazolium Salts; Thiazoles; Tissue Culture Techniques | 2006 |
Synthesis, SAR exploration, and X-ray crystal structures of factor XIa inhibitors containing an alpha-ketothiazole arginine.
Topics: Amides; Arginine; Crystallography, X-Ray; Factor XIa; Models, Molecular; Molecular Structure; Structure-Activity Relationship; Thiazoles | 2006 |
Platonin attenuates LPS-induced CAT-2 and CAT-2B induction in stimulated murine macrophages.
Topics: Amino Acid Transport Systems, Basic; Animals; Arginine; Cell Line; Densitometry; Dose-Response Relationship, Drug; Lipopolysaccharides; Luminescent Measurements; Macrophages; Mice; Nitric Oxide; Nitric Oxide Synthase Type II; Reverse Transcriptase Polymerase Chain Reaction; Stimulation, Chemical; Thiazoles; Up-Regulation | 2006 |
Crystallographic structure of human beta-hexosaminidase A: interpretation of Tay-Sachs mutations and loss of GM2 ganglioside hydrolysis.
Topics: Acetylglucosamine; Amino Acid Substitution; Arginine; Aspartic Acid; beta-N-Acetylhexosaminidases; Binding Sites; Crystallography, X-Ray; Dimerization; Gangliosidoses, GM2; Glycine; Glycosylation; Hexosaminidase A; Humans; Hydrolysis; Models, Molecular; Mutation; Protein Conformation; Protein Subunits; Tay-Sachs Disease; Thiazoles | 2006 |
Cell-penetrating peptides as transporters for morpholino oligomers: effects of amino acid composition on intracellular delivery and cytotoxicity.
Topics: Aminocaproic Acid; Arginine; beta-Alanine; Biological Transport; Cell Line; Cell Survival; Culture Media; Hemolysis; Humans; Indicators and Reagents; Oligonucleotides, Antisense; Peptides; Propidium; RNA Splicing; Stereoisomerism; Tetrazolium Salts; Thiazoles | 2007 |
Photodynamic effect of protoporphyrin diarginate (PPArg2) on methicillin-resistant Staphylococcus aureus and human dermal fibroblasts.
Topics: Arginine; Dermis; Dose-Response Relationship, Drug; Drug Resistance, Bacterial; Fibroblasts; Humans; Light; Methicillin; Methicillin Resistance; Models, Biological; Photochemistry; Photosensitizing Agents; Protoporphyrins; Skin; Staphylococcus aureus; Tetrazolium Salts; Thiazoles | 2008 |
Cellular internalization and distribution of arginine-rich peptides as a function of extracellular peptide concentration, serum, and plasma membrane associated proteoglycans.
Topics: Animals; Apoptosis; Arginine; Blood Proteins; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Drug Screening Assays, Antitumor; Endocytosis; Flow Cytometry; HeLa Cells; Humans; Membrane Potentials; Microscopy, Confocal; Oligopeptides; Proteoglycans; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Transferrin | 2008 |
Prolyl endopeptidase is revealed following SILAC analysis to be a novel mediator of human microglial and THP-1 cell neurotoxicity.
Topics: Analysis of Variance; Arginine; Carbon Isotopes; Cell Line; Computational Biology; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Humans; Interferon-gamma; L-Lactate Dehydrogenase; Lipopolysaccharides; Mass Spectrometry; Microglia; Monocytes; Neuroblastoma; Neurotoxins; Prolyl Oligopeptidases; Serine Endopeptidases; Tetrazolium Salts; Thiazoles | 2008 |
Effects of cross-link breakers, glycation inhibitors and insulin sensitisers on HDL function and the non-enzymatic glycation of apolipoprotein A-I.
Topics: Apolipoprotein A-I; Arginine; Cross-Linking Reagents; Glycosylation; Guanidines; Humans; Lipoproteins, HDL; Lysine; Metformin; Phosphatidylcholine-Sterol O-Acyltransferase; Pyridoxamine; Pyruvaldehyde; Thiazoles; Tryptophan | 2008 |
Structural basis of actin recognition and arginine ADP-ribosylation by Clostridium perfringens iota-toxin.
Topics: Actins; Adenosine Diphosphate; ADP Ribose Transferases; Animals; Arginine; Bacterial Toxins; Crystallography, X-Ray; Hydrolysis; Mutagenesis, Site-Directed; Protein Conformation; Rabbits; Ribose; Thiazoles | 2008 |
Preparation and gene delivery of alkaline amino acids-based cationic liposomes.
Topics: Amino Acids; Arginine; Cations; Cell Line; Cholesterol; Deoxyribonuclease I; Drug Carriers; Electrophoresis, Agar Gel; Gene Transfer Techniques; Genes, Reporter; Histidine; Humans; Light; Liposomes; Luciferases; Lysine; Microscopy, Electron, Transmission; Scattering, Radiation; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Tetrazolium Salts; Thiazoles; Transfection | 2008 |
Aggregate formation and toxicity by wild-type and R621C synphilin-1 in the nigrostriatal system of mice using adenoviral vectors.
Topics: Adenoviridae; Animals; Arginine; Benzothiazoles; Carrier Proteins; Corpus Striatum; Cysteine; Gene Expression; Genetic Vectors; Green Fluorescent Proteins; Intracellular Signaling Peptides and Proteins; Mice; Mice, Inbred C57BL; Mice, Transgenic; Mutation; Nerve Degeneration; Nerve Tissue Proteins; Substantia Nigra; Thiazoles; Tyrosine 3-Monooxygenase | 2009 |
Characterization of ternary complexes of meloxicam-HPbetaCD and PVP or L-arginine prepared by the spray-drying technique.
Topics: 2-Hydroxypropyl-beta-cyclodextrin; Anti-Inflammatory Agents, Non-Steroidal; Arginine; beta-Cyclodextrins; Calorimetry, Differential Scanning; Meloxicam; Pyrrolidinones; Solubility; Technology, Pharmaceutical; Thiazines; Thiazoles | 2008 |
Letter by Hartog et al. regarding article, "Advanced glycation end products accumulate in vascular smooth muscle and modify vascular but not ventricular properties in elderly hypertensive canines".
Topics: Animals; Arginine; Collagen; Cross-Linking Reagents; Dogs; Glycation End Products, Advanced; Hypertension; Lysine; Muscle, Smooth, Vascular; Thiazoles | 2009 |
Thrombin enhances glioma growth.
Topics: Animals; Anticoagulants; Arginine; Behavior, Animal; Brain Neoplasms; Bromodeoxyuridine; Cell Line, Tumor; Cell Proliferation; Enzyme-Linked Immunosorbent Assay; Functional Laterality; Glioma; Hemostatics; Male; Neoplasm Transplantation; Pipecolic Acids; Rats; Rats, Inbred F344; Sulfonamides; Tetrazolium Salts; Thiazoles; Thrombin; Time Factors | 2008 |
Effect of pharmacological manipulations of neuropeptide Y and corticotropin-releasing factor neurotransmission on incubation of conditioned fear.
Topics: Acoustic Stimulation; Animals; Arginine; Benzazepines; Conditioning, Operant; Corticotropin-Releasing Hormone; Fear; Male; Neuropeptide Y; Pyridazines; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Receptors, Neuropeptide Y; Synaptic Transmission; Thiazoles; Time Factors | 2009 |
L-Arginine reduces thioflavin T fluorescence but not fibrillation of bovine serum albumin.
Topics: Animals; Arginine; Benzothiazoles; Binding Sites; Cattle; Fluorescence; Microscopy, Electron, Transmission; Protein Binding; Protein Conformation; Serum Albumin, Bovine; Thiazoles | 2010 |
Dura in the pathogenesis of syndromic craniosynostosis: fibroblast growth factor receptor 2 mutations in dural cells promote osteogenic proliferation and differentiation of osteoblasts.
Topics: Acrocephalosyndactylia; Adenoviridae; Alkaline Phosphatase; Animals; Arginine; Biomarkers; Cell Differentiation; Cell Proliferation; Cells, Cultured; Coculture Techniques; Coloring Agents; Core Binding Factor Alpha 1 Subunit; Craniofacial Dysostosis; Craniosynostoses; Cysteine; Dura Mater; Genetic Vectors; Mice; Osteoblasts; Osteogenesis; Osteopontin; Phenylalanine; Point Mutation; Receptor, Fibroblast Growth Factor, Type 2; Syndrome; Tetrazolium Salts; Thiazoles | 2010 |
Granular and lattice deposits in corneal dystrophy caused by R124C mutation of TGFBIp.
Topics: Adult; Amyloid; Antibody Specificity; Arginine; Benzothiazoles; Cornea; Corneal Dystrophies, Hereditary; Corneal Stroma; Cysteine; Extracellular Matrix Proteins; Fluorescent Antibody Technique; Fluorescent Dyes; Genotype; Heterozygote; Humans; Male; Mutation; Penetrance; Staining and Labeling; Thiazoles; Transforming Growth Factor beta | 2010 |
Treatment of experimental cerebral vasospasm by protein transduction of heme oxygenase 1 (HO-1) conjugated to a residue of 11 arginines.
Topics: Animals; Arginine; Disease Models, Animal; Dose-Response Relationship, Drug; Heme Oxygenase-1; Male; Rats; Rats, Sprague-Dawley; Tetrazolium Salts; Thiazoles; Vasospasm, Intracranial | 2011 |
Gene transport and expression by arginine-rich cell-penetrating peptides in Paramecium.
Topics: Arginine; Biological Transport; Carrier Proteins; Cell Membrane; Cell Physiological Phenomena; Cell-Penetrating Peptides; DNA, Protozoan; Genes, Protozoan; Green Fluorescent Proteins; Microscopy, Fluorescence; Paramecium caudatum; Plasmids; Tetrazolium Salts; Thiazoles; Transfection | 2011 |
Yersinia high pathogenicity island genes modify the Escherichia coli primary metabolome independently of siderophore production.
Topics: Arginine; Bacterial Proteins; Chromatography, Liquid; Cluster Analysis; Escherichia coli; Gene Expression Regulation, Bacterial; Genes, Bacterial; Genomic Islands; Metabolome; Metabolomics; Phenols; Sequence Deletion; Siderophores; Thiazoles; Trans-Activators; Transcription Factors; Yersinia | 2011 |
Moringa coagulant as a stabilizer for amorphous solids: Part I.
Topics: Arginine; Calorimetry, Differential Scanning; Chemistry, Pharmaceutical; Coagulants; Crystallography, X-Ray; Drug Stability; Excipients; Felodipine; Hydrogen Bonding; Ibuprofen; Kinetics; Meloxicam; Microscopy; Models, Molecular; Molecular Structure; Moringa oleifera; Plant Proteins; Solubility; Spectroscopy, Fourier Transform Infrared; Technology, Pharmaceutical; Thiazines; Thiazoles; Transition Temperature; X-Ray Diffraction | 2012 |
Imaging findings of familial dementia with a tau R406W mutation.
Topics: Aged; Aniline Compounds; Arginine; Dementia; Fluorodeoxyglucose F18; Humans; Magnetic Resonance Imaging; Male; Mutation; Positron-Emission Tomography; tau Proteins; Thiazoles; Tryptophan | 2011 |
Inhibition of aggregation of amyloid β42 by arginine-containing small compounds.
Topics: Amyloid; Amyloid beta-Peptides; Arginine; Benzothiazoles; Coumarins; Dipeptides; Electrophoresis, Polyacrylamide Gel; Humans; Peptide Fragments; Polymerization; Protein Binding; Small Molecule Libraries; Solubility; Solutions; Thiazoles | 2012 |
Development of meloxicam salts with improved dissolution and pharmacokinetic behaviors in rats with impaired gastric motility.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Arginine; Gastrointestinal Motility; Male; Meloxicam; Muscarinic Antagonists; Pharmaceutical Vehicles; Propantheline; Rats; Rats, Sprague-Dawley; Salts; Solubility; Thiazines; Thiazoles | 2013 |
Glycogen synthase kinase 3-specific inhibitor AR-A014418 decreases neuropathic pain in mice: evidence for the mechanisms of action.
Topics: Analgesics; Animals; Arginine; Cytokines; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Hyperalgesia; Ligation; Male; Mice; Motor Activity; Neuralgia; Nitric Oxide; Pain Measurement; Parasympathetic Nervous System; Sciatic Neuropathy; Serotonin; Spinal Cord; Thiazoles; Urea | 2012 |
Arg-Thz is a minimal substrate for the N(α),N(α)-arginyl methyltransferase involved in the biosynthesis of plantazolicin.
Topics: Arginine; Azoles; Methyltransferases; Oligopeptides; Substrate Specificity; Thiazoles | 2013 |
Oxicams bind in a novel mode to the cyclooxygenase active site via a two-water-mediated H-bonding Network.
Topics: Amino Acid Substitution; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arginine; Binding Sites; Catalytic Domain; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Hydrogen Bonding; Leucine; Meloxicam; Mice; Mutation; Piroxicam; Protein Structure, Secondary; Serine; Thiazines; Thiazoles; Tyrosine; Water | 2014 |
Effects of L-arginine, mirabegron, and oxybutynin on the primary bladder afferent nerve activities synchronized with reflexic, rhythmic bladder contractions in the rat.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Arginine; Electric Stimulation; Female; Mandelic Acids; Mechanotransduction, Cellular; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neurons, Afferent; Nitric Oxide; Periodicity; Pressure; Rats, Sprague-Dawley; Reflex; Thiazoles; Time Factors; Urinary Bladder | 2015 |
Use of PER977 to reverse the anticoagulant effect of edoxaban.
Topics: Arginine; Blood Coagulation; Factor Xa Inhibitors; Heparin Antagonists; Humans; Piperazines; Pyridines; Thiazoles | 2014 |
Intranasal and intravenous administration of octa-arginine modified poly(lactic-co-glycolic acid) nanoparticles facilitates central nervous system delivery of loperamide.
Topics: Administration, Intranasal; Administration, Intravenous; Analgesics; Animals; Arginine; Cell Line; Central Nervous System; Coumarins; Dogs; Drug Delivery Systems; Female; Lactic Acid; Loperamide; Male; Mice, Inbred C57BL; Nanoconjugates; Nanoparticles; Particle Size; Polyesters; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Polymers; Thiazoles | 2015 |
Mutational analysis of the ability of resveratrol to inhibit amyloid formation by islet amyloid polypeptide: critical evaluation of the importance of aromatic-inhibitor and histidine-inhibitor interactions.
Topics: Amino Acid Sequence; Amino Acids, Aromatic; Amyloid; Arginine; Benzothiazoles; Catechin; DNA Mutational Analysis; Histidine; Humans; Islet Amyloid Polypeptide; Molecular Sequence Data; Mutant Proteins; Resveratrol; Spectrometry, Mass, Electrospray Ionization; Stilbenes; Structure-Activity Relationship; Thiazoles | 2015 |
[In vitro comparison of podophyllotoxin analogues; etoposide, teniposide and NK 611 using human lung cancer cell lines].
Topics: Adenocarcinoma; Antineoplastic Agents; Carcinoma, Small Cell; Carcinoma, Squamous Cell; Cell Division; Drug Resistance; Drug Screening Assays, Antitumor; Etoposide; Humans; Lung Neoplasms; Podophyllotoxin; Teniposide; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured | 1993 |
Preparation and characterization of teniposide PLGA nanoparticles and their uptake in human glioblastoma U87MG cells.
Topics: Acetone; Antineoplastic Agents; Calorimetry, Differential Scanning; Cell Line, Tumor; Cell Survival; Coumarins; Drug Carriers; Endocytosis; Fluorescent Dyes; Glioblastoma; Humans; Lactic Acid; Microscopy, Electron, Transmission; Nanoparticles; Particle Size; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Polyvinyl Alcohol; Teniposide; Thiazoles | 2012 |