Page last updated: 2024-09-03

arg-3-hyp-7-phe-bradykinin and endothelins

arg-3-hyp-7-phe-bradykinin has been researched along with endothelins in 2 studies

Compound Research Comparison

Studies (arg-3-hyp-7-phe-bradykinin)	Trials (arg-3-hyp-7-phe-bradykinin)	Recent Studies (post-2010) (arg-3-hyp-7-phe-bradykinin)	Studies (endothelins)	Trials (endothelins)	Recent Studies (post-2010) (endothelins)
52	2	3	10	0	3

Protein Interaction Comparison

Protein	Taxonomy	endothelins (IC50)
Endothelin receptor type B	Rattus norvegicus (Norway rat)	0.0016
Endothelin receptor type B	Homo sapiens (human)	0.0002
Endothelin-1 receptor	Homo sapiens (human)	0.0002
Endothelin-1 receptor	Sus scrofa (pig)	0.0002

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	1 (50.00)	29.6817
2010's	1 (50.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X	1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L	1

Other Studies

2 other study(ies) available for arg-3-hyp-7-phe-bradykinin and endothelins

Article	Year
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity. Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14 Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship	2008
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor. Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10 Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship	2013

Article

Year

Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.

Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008

Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.

Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013