arcaine and dizocilpine maleate

arcaine has been researched along with dizocilpine maleate in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (60.87)18.2507
2000's8 (34.78)29.6817
2010's1 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Donevan, SD; Jones, SM; Rogawski, MA1
Reynolds, IJ3
Canton, H; Colpaert, F; Lehmann, J1
Bagga, L; Derks, M; Doyle, KM; Purcell, WM1
Calligaro, DO; Monn, JA; O'Malley, PJ1
Berrino, L; Leyva, J; Maione, S; Pizzirusso, A; Rossi, F; Stella, L1
Baudry, M; Marvizón, JC1
Burns, MA; Palmer, AM1
Reynolds, IJ; Rothermund, KD1
Artemowicz, B; Lutostanska, A; Wiśniewski, K2
Carr, AJ; Davis, RS; Hamilton, AD; Reynolds, IJ; Sharma, TA1
Mo, LL; Sundström, E1
Gibson, DA; Harris, BR; Littleton, JM; Rogers, DT1
Littleton, JM; Mulholland, PJ; Nath, A; Prendergast, MA; Rogers, DT; Self, RL; Wilkins, LH1
Awe, SO; Harris, LC; Kulkarni, K; LeDay, AM; Ohia, SE; Opere, CA; Sharif, NA1
Bellé, NA; Dalmolin, GD; Fonini, G; Rocha, JB; Rubin, MA1
Bakalkin, G; Marinova, Z; Nakagawasai, O; Niijima, F; Sakurada, S; Sato, T; Satoh, S; Tadano, T; Takahashi, H; Tan-No, K; Terenius, L; Yakovleva, T1
Camera, K; Ceretta, AP; Mello, CF; Rubin, MA2
Carvalho, FB; Ferreira, J; Girardi, BA; Marisco, PC; Mello, CF; Oliveira, MS; Rubin, MA; Tonello, R1

Other Studies

23 other study(ies) available for arcaine and dizocilpine maleate

ArticleYear
Arcaine blocks N-methyl-D-aspartate receptor responses by an open channel mechanism: whole-cell and single-channel recording studies in cultured hippocampal neurons.
    Molecular pharmacology, 1992, Volume: 41, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Biguanides; Cations, Divalent; Cells, Cultured; Dizocilpine Maleate; gamma-Aminobutyric Acid; Glycine; Hippocampus; Ibotenic Acid; Ion Channels; Kainic Acid; Magnesium; Membrane Potentials; N-Methylaspartate; Neurons; Polyamines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1992
Interactions between zinc and spermidine on the N-methyl-D-aspartate receptor complex: clues to the mechanism of action of 1,10-bis(guanidino)decane and pentamidine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Biguanides; Binding Sites; Brain Chemistry; Diethyl Pyrocarbonate; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Guanidines; Pentamidine; Rats; Receptors, N-Methyl-D-Aspartate; Spermidine; Zinc

1992
Glutamate and glycine co-activate while polyamines merely modulate the NMDA receptor complex.
    Progress in neuro-psychopharmacology & biological psychiatry, 1991, Volume: 15, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Adrenergic alpha-Antagonists; Animals; Biguanides; Binding, Competitive; Biogenic Polyamines; Biotransformation; Brain; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; In Vitro Techniques; Kynurenic Acid; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine

1991
Arcaine uncovers dual interactions of polyamines with the N-methyl-D-aspartate receptor.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Animals; Biguanides; Binding, Competitive; Cations, Divalent; Dizocilpine Maleate; Drug Interactions; Kinetics; Polyamines; Rats; Receptors, N-Methyl-D-Aspartate; Tritium

1990
Arcaine is a competitive antagonist of the polyamine site on the NMDA receptor.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Biguanides; Binding, Competitive; Biogenic Polyamines; Dibenzocycloheptenes; Dizocilpine Maleate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spermidine

1990
Histamine release from mast cells by polyamines: an NMDA receptor-mediated event?
    Biochemical Society transactions, 1994, Volume: 22, Issue:4

    Topics: Animals; Biguanides; Dizocilpine Maleate; Histamine Release; In Vitro Techniques; Kinetics; Mast Cells; p-Methoxy-N-methylphenethylamine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermine

1994
beta-Amyloid (25-35) or substance P stimulates [3H]MK-801 binding to rat cortical membranes in the presence of glutamate and glycine.
    Journal of neurochemistry, 1993, Volume: 60, Issue:6

    Topics: Amino Acid Sequence; Amyloid beta-Peptides; Animals; Biguanides; Cell Membrane; Cerebral Cortex; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; Kinetics; Molecular Sequence Data; N-Methylaspartate; Peptide Fragments; Pipecolic Acids; Rats; Receptors, N-Methyl-D-Aspartate; Sequence Homology, Amino Acid; Substance P

1993
Evidence that arcaine increases the N-methyl-D-aspartate-induced cardiovascular effects into the periaqueductal gray area of anesthetized rats.
    Neuroscience letters, 1994, Jan-03, Volume: 165, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Anesthesia; Animals; Biguanides; Blood Pressure; Dizocilpine Maleate; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Male; N-Methylaspartate; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1994
[3H]dizocilpine association kinetics distinguish stimulatory and inhibitory polyamine sites of N-methyl-D-aspartate receptors.
    Journal of neurochemistry, 1994, Volume: 63, Issue:3

    Topics: Animals; Biguanides; Binding Sites; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; Kinetics; Male; Piperidines; Polyamines; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Tritium

1994
Preservation of redox, polyamine, and glycine modulatory domains of the N-methyl-D-aspartate receptor in Alzheimer's disease.
    Journal of neurochemistry, 1994, Volume: 62, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Analysis of Variance; Biguanides; Binding Sites; Brain; Cell Membrane; Cerebral Cortex; Dithionitrobenzoic Acid; Dizocilpine Maleate; Female; Frontal Lobe; Glycine; Humans; Male; Middle Aged; Organ Specificity; Oxidation-Reduction; Radioligand Assay; Receptors, N-Methyl-D-Aspartate; Spermidine; Temporal Lobe

1994
Characterization of the effects of polyamines on the modulation of the N-methyl-D-aspartate receptor by glycine.
    Neuropharmacology, 1995, Volume: 34, Issue:9

    Topics: Animals; Biguanides; Binding, Competitive; Dizocilpine Maleate; Dose-Response Relationship, Drug; Glycine; Polyamines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1995
The role of NMDA receptors in central action of angiotensin II.
    Acta physiologica Hungarica, 1996, Volume: 84, Issue:3

    Topics: Angiotensin II; Animals; Avoidance Learning; Biguanides; Brain; Conditioning, Psychological; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Memory; Motor Activity; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate

1996
The estimation of interactions between arginine-vasopressin (AVP) and NMDA receptors in memory and learning processes.
    Acta physiologica Hungarica, 1996, Volume: 84, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Arginine Vasopressin; Biguanides; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Learning; Male; Memory; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate

1996
Aromatic analogs of arcaine inhibit MK-801 binding to the NMDA receptor.
    Bioorganic & medicinal chemistry letters, 1998, Dec-15, Volume: 8, Issue:24

    Topics: Biguanides; Dizocilpine Maleate; Protein Binding; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

1998
Polyamine and redox modulation of [3H]MK-801 binding to N-methyl-D-aspartate receptors in the spinal cord and cerebral cortex.
    Pharmacology & toxicology, 2001, Volume: 88, Issue:6

    Topics: Animals; Biguanides; Cerebral Cortex; Dizocilpine Maleate; Hydrogen-Ion Concentration; Male; Neuroprotective Agents; Oxidation-Reduction; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine; Spinal Cord; Tritium

2001
Radioligand binding studies reveal agmatine is a more selective antagonist for a polyamine-site on the NMDA receptor than arcaine or ifenprodil.
    Brain research, 2002, Oct-11, Volume: 952, Issue:1

    Topics: Agmatine; Animals; Biguanides; Binding Sites; Binding, Competitive; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermidine; Tritium

2002
Neurotoxic effects of the human immunodeficiency virus type-1 transcription factor Tat require function of a polyamine sensitive-site on the N-methyl-D-aspartate receptor.
    Brain research, 2002, Nov-08, Volume: 954, Issue:2

    Topics: Animals; ATPases Associated with Diverse Cellular Activities; Biguanides; Brain; Cerebellum; Cerebral Cortex; Culture Techniques; Dizocilpine Maleate; DNA-Binding Proteins; Excitatory Amino Acid Antagonists; Female; Hippocampus; HIV-1; Male; Neurons; Neurotoxins; Proteasome Endopeptidase Complex; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermidine

2002
Glucose-deprivation-induced [3H]D-aspartate release from isolated bovine and human retinae.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2003, Volume: 19, Issue:6

    Topics: Alanine; Animals; Biguanides; Calcium Channel Blockers; Cattle; D-Aspartic Acid; Diltiazem; Dizocilpine Maleate; Drug Synergism; Glucose; Glutamic Acid; Glycine; Humans; Kainic Acid; N-Methylaspartate; Nitrendipine; omega-Conotoxins; Perfusion; Piperidines; Polyamines; Receptors, Glutamate; Retina; Tritium; Verapamil

2003
Polyamines reduces lipid peroxidation induced by different pro-oxidant agents.
    Brain research, 2004, May-22, Volume: 1008, Issue:2

    Topics: Animals; Antioxidants; Biguanides; Biogenic Polyamines; Dizocilpine Maleate; Edetic Acid; Iron; Lipid Peroxidation; Nitroprusside; Oxidants; Quinolinic Acid; Rats; Rats, Wistar; Spermidine; Spermine; Thiobarbituric Acid Reactive Substances

2004
Pronociceptive role of dynorphins in uninjured animals: N-ethylmaleimide-induced nociceptive behavior mediated through inhibition of dynorphin degradation.
    Pain, 2005, Volume: 113, Issue:3

    Topics: Agmatine; Analysis of Variance; Animals; Behavior, Animal; Biguanides; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Dynorphins; Enkephalins; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; Immune Sera; Injections, Spinal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Narcotics; Nociceptin Receptor; Piperidines; Protein Precursors; Receptors, Opioid; Spinal Cord; Time Factors

2005
Systemic administration of polyaminergic agents modulate fear conditioning in rats.
    Psychopharmacology, 2007, Volume: 192, Issue:4

    Topics: Animals; Behavior, Animal; Biguanides; Conditioning, Classical; Dizocilpine Maleate; Fear; Injections, Intraperitoneal; Male; Memory; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermidine; Time Factors

2007
Arcaine and MK-801 make recall state-dependent in rats.
    Psychopharmacology, 2008, Volume: 201, Issue:3

    Topics: Animals; Avoidance Learning; Behavior, Animal; Biguanides; Buffers; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Administration Schedule; Excitatory Amino Acid Antagonists; Exploratory Behavior; Injections, Intraperitoneal; Male; Mental Recall; Neuroprotective Agents; Phosphates; Polyamines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Time Factors; Transfer, Psychology

2008
Spermidine decreases Na⁺,K⁺-ATPase activity through NMDA receptor and protein kinase G activation in the hippocampus of rats.
    European journal of pharmacology, 2012, Jun-05, Volume: 684, Issue:1-3

    Topics: Animals; Biguanides; Carbazoles; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dizocilpine Maleate; Enzyme Activation; Hippocampus; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Sodium-Potassium-Exchanging ATPase; Spermidine

2012