Page last updated: 2024-09-05

ar-l 57 cl and ouabain

ar-l 57 cl has been researched along with ouabain in 5 studies

Compound Research Comparison

Studies
(ar-l 57 cl)
Trials
(ar-l 57 cl)
Recent Studies (post-2010)
(ar-l 57 cl)
Studies
(ouabain)
Trials
(ouabain)
Recent Studies (post-2010) (ouabain)
121016,35772747

Protein Interaction Comparison

ProteinTaxonomyar-l 57 cl (IC50)ouabain (IC50)
STAT3, partialHomo sapiens (human)1.154
Kruppel-like factor 5Homo sapiens (human)0.0832
Sodium/potassium-transporting ATPase subunit alpha-1 Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-1Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit alpha-1 Rattus norvegicus (Norway rat)4.3
Sodium/potassium-transporting ATPase subunit alpha-2Rattus norvegicus (Norway rat)0.17
Sodium/potassium-transporting ATPase subunit alpha-3 Rattus norvegicus (Norway rat)0.031
Sodium/potassium-transporting ATPase subunit beta-1 Rattus norvegicus (Norway rat)1.1263
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.1646
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 20.097
Sodium/potassium-transporting ATPase subunit alpha-3Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-2Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit alpha-2Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-3Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit gammaHomo sapiens (human)6
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.8
Sodium/potassium-transporting ATPase subunit alpha-4Homo sapiens (human)6
Sodium/potassium-transporting ATPase subunit beta-3Rattus norvegicus (Norway rat)0.0018
Sodium/potassium-transporting ATPase subunit alpha-4Rattus norvegicus (Norway rat)0.0031

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19905 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hayes, JS; Kauffman, RF; Robertson, DW; Wilson, HC; Wyss, VL1
van Meel, JC1
Baker, PF; Honerjäger, P; Reiter, M2
Hayes, JS1

Other Studies

5 other study(ies) available for ar-l 57 cl and ouabain

ArticleYear
Molecular basis for the in vitro and in vivo cardiotonic activities of AR-L100.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Animals; Carbachol; Cats; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Female; Heart; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Ouabain; Phosphodiesterase Inhibitors; Rubidium; Sodium-Potassium-Exchanging ATPase; Structure-Activity Relationship

1986
Comparison of some new positive inotropic agents in guinea pigs.
    Pharmacology, 1985, Volume: 31, Issue:1

    Topics: Aminopyridines; Amrinone; Animals; Blood Pressure; Cardiotonic Agents; Dose-Response Relationship, Drug; Enoximone; Guinea Pigs; Heart Rate; Hydralazine; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Ouabain; Vasodilation

1985
Effect of the cardioactive drug AR-L 57 on free intracellular calcium and ouabain-insensitive ion fluxes in the squid giant axon.
    Molecular pharmacology, 1981, Volume: 19, Issue:1

    Topics: Aequorin; Animals; Axonal Transport; Axons; Calcium; Cardiotonic Agents; Decapodiformes; Imidazoles; In Vitro Techniques; Intracellular Fluid; Ions; Membrane Potentials; Ouabain; Veratridine

1981
A simple technique for determining contractility, intraventricular pressure, and heart rate in the anesthetized guinea pig.
    Journal of pharmacological methods, 1982, Volume: 8, Issue:3

    Topics: Anesthesia; Animals; Guinea Pigs; Heart; Heart Rate; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Ouabain; Pressure; Time Factors

1982
Inhibition of the sodium pump in squid axons by the cardioactive drug AR-L 57.
    Molecular pharmacology, 1980, Volume: 17, Issue:3

    Topics: Animals; Axons; Biological Transport, Active; Cardiotonic Agents; Decapodiformes; Imidazoles; In Vitro Techniques; Ion Exchange; Ouabain; Potassium; Rubidium; Sodium; Time Factors

1980