ar-c239 has been researched along with oxymetazoline in 5 studies
Studies (ar-c239) | Trials (ar-c239) | Recent Studies (post-2010) (ar-c239) | Studies (oxymetazoline) | Trials (oxymetazoline) | Recent Studies (post-2010) (oxymetazoline) |
---|---|---|---|---|---|
45 | 0 | 5 | 738 | 128 | 159 |
Protein | Taxonomy | ar-c239 (IC50) | oxymetazoline (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | 0.578 | |
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 3.261 | |
Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | 1.332 | |
Alpha-2A adrenergic receptor | Homo sapiens (human) | 0.023 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.2 | |
Alpha-2B adrenergic receptor | Homo sapiens (human) | 1.273 | |
Alpha-2C adrenergic receptor | Homo sapiens (human) | 2.633 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 0.0056 | |
Alpha-1D adrenergic receptor | Homo sapiens (human) | 2.844 | |
5-hydroxytryptamine receptor 2A | Homo sapiens (human) | 1.285 | |
5-hydroxytryptamine receptor 2C | Homo sapiens (human) | 0.578 | |
5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | 0.0056 | |
5-hydroxytryptamine receptor 2B | Homo sapiens (human) | 3.056 | |
5-hydroxytryptamine receptor 6 | Homo sapiens (human) | 1.67 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Musgrave, IF; Seifert, R | 1 |
Alburges, ME; Bylund, DB; Pundt, LL; Wamsley, JK | 1 |
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G | 1 |
Goepel, M; Michel, MC; RĂ¼bben, H; Wittmann, A | 1 |
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P | 1 |
5 other study(ies) available for ar-c239 and oxymetazoline
Article | Year |
---|---|
Alpha 2A-adrenoceptors mediate activation of non-selective cation channels via Gi-proteins in human erythroleukaemia (HEL) cells. No evidence for a functional role of imidazoline receptors in modulating calcium.
Topics: Binding, Competitive; Calcium; Cell Fractionation; GTP Phosphohydrolases; GTP-Binding Proteins; Humans; Imidazoline Receptors; Ion Channels; Isoquinolines; Leukemia, Erythroblastic, Acute; Oxymetazoline; Pertussis Toxin; Piperazines; Receptors, Adrenergic, alpha; Receptors, Drug; Tumor Cells, Cultured; Virulence Factors, Bordetella; Yohimbine | 1995 |
Alpha 2-agonist binding sites in brain: [125I]para-iodoclonidine versus [3H]para-aminoclonidine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding, Competitive; Brain; Clonidine; Iodine Radioisotopes; Isoquinolines; Male; Oxymetazoline; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Tritium | 1993 |
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine | 1996 |
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine | 1997 |
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine | 1999 |