Page last updated: 2024-09-03

ar-c239 and oxymetazoline

ar-c239 has been researched along with oxymetazoline in 5 studies

Compound Research Comparison

Studies
(ar-c239)
Trials
(ar-c239)
Recent Studies (post-2010)
(ar-c239)
Studies
(oxymetazoline)
Trials
(oxymetazoline)
Recent Studies (post-2010) (oxymetazoline)
4505738128159

Protein Interaction Comparison

ProteinTaxonomyar-c239 (IC50)oxymetazoline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.578
Muscarinic acetylcholine receptor M4Homo sapiens (human)3.261
Muscarinic acetylcholine receptor M5Homo sapiens (human)1.332
Alpha-2A adrenergic receptorHomo sapiens (human)0.023
Cytochrome P450 2D6Homo sapiens (human)0.2
Alpha-2B adrenergic receptorHomo sapiens (human)1.273
Alpha-2C adrenergic receptorHomo sapiens (human)2.633
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0056
Alpha-1D adrenergic receptorHomo sapiens (human)2.844
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.285
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.578
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0056
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.056
5-hydroxytryptamine receptor 6Homo sapiens (human)1.67

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Musgrave, IF; Seifert, R1
Alburges, ME; Bylund, DB; Pundt, LL; Wamsley, JK1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Goepel, M; Michel, MC; RĂ¼bben, H; Wittmann, A1
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1

Other Studies

5 other study(ies) available for ar-c239 and oxymetazoline

ArticleYear
Alpha 2A-adrenoceptors mediate activation of non-selective cation channels via Gi-proteins in human erythroleukaemia (HEL) cells. No evidence for a functional role of imidazoline receptors in modulating calcium.
    Biochemical pharmacology, 1995, Jan-18, Volume: 49, Issue:2

    Topics: Binding, Competitive; Calcium; Cell Fractionation; GTP Phosphohydrolases; GTP-Binding Proteins; Humans; Imidazoline Receptors; Ion Channels; Isoquinolines; Leukemia, Erythroblastic, Acute; Oxymetazoline; Pertussis Toxin; Piperazines; Receptors, Adrenergic, alpha; Receptors, Drug; Tumor Cells, Cultured; Virulence Factors, Bordetella; Yohimbine

1995
Alpha 2-agonist binding sites in brain: [125I]para-iodoclonidine versus [3H]para-aminoclonidine.
    Brain research bulletin, 1993, Volume: 32, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding, Competitive; Brain; Clonidine; Iodine Radioisotopes; Isoquinolines; Male; Oxymetazoline; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Tritium

1993
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
    Neuroscience letters, 1996, May-24, Volume: 210, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine

1996
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
    Urological research, 1997, Volume: 25, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine

1997
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999