Page last updated: 2024-08-17

apomorphine and u-50488

apomorphine has been researched along with u-50488 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's3 (30.00)18.2507
2000's5 (50.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Lookingland, KJ; Manzanares, J; Moore, KE1
Ohno, M; Ueki, S; Yamamoto, T1
Funada, M; Misawa, M; Nagase, H; Narita, M; Suzuki, T1
Capasso, A; Sorrentino, L1
Ho, IK; Jang, CG; Lee, SY; Loh, HH; Ma, T; Park, Y1
Aru, GN; Bortolato, M; Fà, M; Frau, R; Gessa, GL; Manunta, M; Mereu, G; Orrù, M; Puddu, M1
Ito, S; Mori, T; Sawaguchi, T1
Charntikov, S; Halladay, LR; Herbert, MS; Marquez, EM; McDougall, SA1
Isotani, K; Miyatake, M; Mori, T; Narita, M; Suzuki, T; Tomiyasu, S; Tsukiyama, Y; Yoshizawa, K1

Other Studies

10 other study(ies) available for apomorphine and u-50488

ArticleYear
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Kappa-opioid-receptor-mediated regulation of alpha-melanocyte-stimulating hormone secretion and tuberohypophyseal dopaminergic neuronal activity.
    Neuroendocrinology, 1990, Volume: 52, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; 3,4-Dihydroxyphenylacetic Acid; alpha-MSH; Animals; Apomorphine; Dihydroxyphenylalanine; Dopamine; Hypothalamo-Hypophyseal System; Male; Neurons; Pituitary Gland; Propranolol; Pyrrolidines; Radioimmunoassay; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1990
Inhibitory effect of a selective kappa receptor agonist, U-50, 488H, on methamphetamine-elicited ipsilateral circling behavior in rats with unilateral nigral lesions.
    Psychopharmacology, 1989, Volume: 97, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Apomorphine; Male; Methamphetamine; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Stereotyped Behavior; Substantia Nigra; Time Factors

1989
Blockade of morphine reward through the activation of kappa-opioid receptors in mice.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; 3,4-Dihydroxyphenylacetic Acid; Analgesics; Animals; Apomorphine; Conditioning, Operant; Dopamine; Dynorphins; Homovanillic Acid; Injections, Subcutaneous; Limbic System; Male; Mice; Mice, Inbred Strains; Morphine; Motivation; Naltrexone; Peptide Fragments; Prosencephalon; Pyrrolidines; Receptors, Opioid, kappa; Reward

1993
Differential influence of D1 and D2 dopamine receptors on acute opiate withdrawal in guinea-pig isolated ileum.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Guinea Pigs; Haloperidol; Ileum; In Vitro Techniques; Male; Morphine; Muscle, Smooth; Pyrrolidines; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance Withdrawal Syndrome

1997
Differential effects of morphine, DPDPE, and U-50488 on apomorphine-induced climbing behavior in mu-opioid receptor knockout mice.
    Brain research. Molecular brain research, 2001, Oct-19, Volume: 94, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Apomorphine; Dopamine Agonists; Enkephalin, D-Penicillamine (2,5)-; Female; Male; Mice; Mice, Knockout; Morphine; Motor Activity; Receptors, Opioid, mu

2001
Kappa opioid receptor activation disrupts prepulse inhibition of the acoustic startle in rats.
    Biological psychiatry, 2005, Jun-15, Volume: 57, Issue:12

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acoustic Stimulation; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Antipsychotic Agents; Apomorphine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Excitatory Amino Acid Antagonists; Haloperidol; Inhibition, Psychological; Male; Naltrexone; Narcotic Antagonists; Rats; Receptors, Opioid, kappa; Reflex, Startle

2005
Differential effects of micro-opioid, delta-opioid and kappa-opioid receptor agonists on dopamine receptor agonist-induced climbing behavior in mice.
    Behavioural pharmacology, 2006, Volume: 17, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Apomorphine; Benzamides; Benzazepines; Dopamine Agonists; Male; Mice; Mice, Inbred Strains; Morphine; Motor Activity; Piperazines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tetrahydronaphthalenes

2006
Effects of dorsal striatal infusions of R(-)-propylnorapomorphine on kappa-opioid-mediated locomotor activity in the young rat: possible role of the indirect pathway.
    Neuroscience, 2008, Aug-26, Volume: 155, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Animals, Newborn; Apomorphine; Behavior, Animal; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Globus Pallidus; Motor Activity; Neural Pathways; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Subthalamic Nucleus

2008
Role of dopamine D2 and D3 receptors in mediating the U-50,488H discriminative cue: comparison with methamphetamine and cocaine.
    Addiction biology, 2012, Volume: 17, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Apomorphine; Cocaine; Discrimination Learning; Dopamine Agonists; Dopamine Uptake Inhibitors; Male; Methamphetamine; Rats; Rats, Inbred F344; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2012