Page last updated: 2024-08-17

apomorphine and trifluoperazine

apomorphine has been researched along with trifluoperazine in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-199028 (87.50)18.7374
1990's1 (3.13)18.2507
2000's1 (3.13)29.6817
2010's2 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Florence, AT; Jenkins, AW; Loveless, AH1
Fowler, PJ; Kaiser, C; Macko, E; Sarau, H; Tedeschi, DH; Zirkle, CL1
Aghajanian, GK; Bunney, BS1
Aghajanian, GK; Cedarbaum, JM1
Clow, A; Jenner, P; Marsden, CD; Theodorou, A5
Andén, NE; Dahlström, A; Jackson, DM1
Andersen, H; Braestrup, C; Randrup, A1
Zetler, G2
Jeng, AY; Wennogle, LP; Wysowskyj, HE1
Jackson, DM; Jenkins, OF1
Clow, A; Jenner, P; Marsden, CD; Murugaiah, K; Theodorou, A1
Beliakov, AV; Matvienko, OA; Neduva, AA; Zharkovskiĭ, AM1
Lahti, RA; McAllister, B; Wozniak, J1
Thörner, R; Zetler, G1
Janssen, PA; Lenaerts, FM; Niemegeers, CJ; Schellekens, KH1
Morpurgo, C; Theobald, W1
Schelkunov, EL1
Clow, A; Jenner, P; Mann, S; Marsden, CD; Murugaiah, K; Theodorou, A1
Boyce, S; Jenner, P; Marsden, CD; Rupniak, NM1
Johnels, B1
De Ferrari, ME; Giannattasio, G; Spada, A1
Davis, JM; Schlemmer, RF1
Evans, DL; Figur, LM; Lahti, RA; Stratman, NC1
BHARGAVA, KP; CHANDRA, O1
Liang, JH; Lu, Y; Ye, XF; Zhang, P1

Reviews

1 review(s) available for apomorphine and trifluoperazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

31 other study(ies) available for apomorphine and trifluoperazine

ArticleYear
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Effect of formulation of intramuscular injections of phenothiazines on duration of activity.
    Journal of pharmaceutical sciences, 1976, Volume: 65, Issue:11

    Topics: Animals; Antipsychotic Agents; Apomorphine; Capsules; Chemistry, Pharmaceutical; Delayed-Action Preparations; Dogs; Emulsions; Female; Fluphenazine; Gels; Injections, Intramuscular; Male; Phenothiazines; Polyethylene Glycols; Solubility; Solutions; Suspensions; Time Factors; Trifluoperazine

1976
Pharmacological evaluation of clomacran, a new potent psychotropic agent.
    Arzneimittel-Forschung, 1977, Volume: 27, Issue:4

    Topics: Acridines; Adenylyl Cyclase Inhibitors; Animals; Antipsychotic Agents; Apomorphine; Autonomic Nervous System; Basal Ganglia Diseases; Behavior, Animal; Chlorpromazine; Chlorprothixene; Conditioning, Psychological; Corpus Striatum; Dogs; Dopamine; Female; Haplorhini; Hemodynamics; Humans; Lethal Dose 50; Macaca mulatta; Male; Mice; Motor Activity; Rage; Rats; Reaction Time; Stereotyped Behavior; Trifluoperazine

1977
Dopamine"autoreceptors": pharmacological characterization by microiontophoretic single cell recording studies.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 297, Issue:1

    Topics: Action Potentials; Animals; Apomorphine; Catecholamines; Clonidine; Dextroamphetamine; Feedback; Iontophoresis; Male; Piperoxan; Rats; Receptors, Dopamine; Sotalol; Substantia Nigra; Synaptic Transmission; Trifluoperazine

1977
Catecholamine receptors on locus coeruleus neurons: pharmacological characterization.
    European journal of pharmacology, 1977, Aug-15, Volume: 44, Issue:4

    Topics: Action Potentials; Animals; Apomorphine; Cerebral Ventricles; Clonidine; Dopamine; Epinephrine; gamma-Aminobutyric Acid; Iontophoresis; Isoproterenol; Male; Neurons; Nordefrin; Norepinephrine; Phenylephrine; Piperoxan; Rats; Receptors, Adrenergic; Sotalol; Trifluoperazine

1977
Striatal dopamine receptors become supersensitive while rats are geven trifluoperazine for six months.
    Nature, 1979, Mar-01, Volume: 278, Issue:5699

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Apomorphine; Corpus Striatum; Dopamine; Homovanillic Acid; Humans; Male; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Time Factors; Trifluoperazine

1979
A functional effect of dopamine in the nucleus accumbens and in some other dopamine-rich parts of the rat brain.
    Psychopharmacologia, 1975, Dec-31, Volume: 45, Issue:2

    Topics: Amphetamine; Amygdala; Animals; Apomorphine; Corpus Striatum; Dextroamphetamine; Dopamine; Dopamine Antagonists; Male; Motor Activity; Norepinephrine; Olfactory Bulb; Phenethylamines; Phenoxybenzamine; Pimozide; Rats; Receptors, Drug; Septal Nuclei; Septum Pellucidum; Trifluoperazine; Tyramine

1975
Apomorphine-induced stereotyped biting in the tortoise in relation to dopaminergic mechanisms.
    Brain, behavior and evolution, 1975, Volume: 11, Issue:5-6

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Behavior; Behavior, Animal; Brain; Dopamine; Haloperidol; Homovanillic Acid; Humans; Receptors, Drug; Stereotyped Behavior; Trifluoperazine; Turtles

1975
Antistereotypic effects of cholecystokinin octapeptide (CCK-8), ceruletide and related peptides on apomorphine-induced gnawing in sensitized mice.
    Neuropharmacology, 1985, Volume: 24, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Ceruletide; Dose-Response Relationship, Drug; Haloperidol; Humans; Irritants; Male; Mice; Scopolamine; Sincalide; Stereotyped Behavior; Thioxanthenes; Trifluoperazine

1985
Clonidine sensitizes mice for apomorphine-induced stereotypic gnawing: antagonism by neuroleptics and cholecystokinin-like peptides.
    European journal of pharmacology, 1985, May-20, Volume: 111, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Cholecystokinin; Clonidine; Haloperidol; Humans; Male; Mice; Oligopeptides; Stereotyped Behavior; Thioxanthenes; Trifluoperazine

1985
Profiling of inhibitors of protein kinase C.
    Advances in enzyme regulation, 1988, Volume: 27

    Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Enzyme Activation; Protein Kinase C; Tetrazoles; Trifluoperazine

1988
Bromocriptine enhances the behavioural effects of apomorphine and dopamine after systemic or intracerebral injection in rats.
    Neuropharmacology, 1986, Volume: 25, Issue:11

    Topics: Animals; Apomorphine; Behavior, Animal; Brain; Bromocriptine; Caudate Nucleus; Dopamine; Drug Interactions; Male; Nialamide; Nucleus Accumbens; Rats; Rats, Inbred Strains; Stereotyped Behavior; Trifluoperazine

1986
Effects of discontinuous drug administration on the development of dopamine receptor supersensitivity during chronic trifluoperazine or cis-flupenthixol administration to rats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Apomorphine; Corpus Striatum; Flupenthixol; Humans; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Thioxanthenes; Trifluoperazine

1985
[Adaptation to neuroleptic preparations and several ways of combatting it (experimental study)].
    Zhurnal nevropatologii i psikhiatrii imeni S.S. Korsakova (Moscow, Russia : 1952), 1985, Volume: 85, Issue:8

    Topics: Animals; Apomorphine; Catalepsy; Drug Therapy, Combination; Drug Tolerance; Haloperidol; Male; Mice; Schizophrenia, Paranoid; Trifluoperazine

1985
Apomorphine antagonism of the elevation of homovanillic acid induced by antipsychotic drugs.
    Life sciences. Pt. 1: Physiology and pharmacology, 1972, Jul-01, Volume: 11, Issue:13

    Topics: Amantadine; Animals; Apomorphine; Brain; Chlorpromazine; Dopamine; Dose-Response Relationship, Drug; Drug Antagonism; Haloperidol; Homovanillic Acid; Mice; Morphine; Phenylacetates; Receptors, Adrenergic; Structure-Activity Relationship; Synaptic Transmission; Thiothixene; Tranquilizing Agents; Trifluoperazine

1972
Drug-induced catalepsy as influenced by psychostimulants, apomorphine, L-dopa, and yohimbine.
    Pharmacology, 1973, Volume: 10, Issue:4

    Topics: Amphetamine; Animals; Apomorphine; Catalepsy; Dihydroxyphenylalanine; Hallucinogens; Haloperidol; Humans; Male; Mecamylamine; Mice; Mice, Inbred Strains; Nicotine; Paraoxon; Pempidine; Phenmetrazine; Pilocarpine; Sparteine; Tetrabenazine; Trifluoperazine; Yohimbine

1973
Is it possible to predict the clinical effects of neuroleptic drugs (major tranquillizers) from animal data? IV. An improved experimental design for measuring the inhibitory effects of neuroleptic drugs on amphetamine-or apomorphine-induced "Cheroing" and
    Arzneimittel-Forschung, 1967, Volume: 17, Issue:7

    Topics: Acepromazine; Amphetamine; Animals; Apomorphine; Behavior, Animal; Benperidol; Chlorpromazine; Chlorprothixene; Fluphenazine; Haloperidol; Male; Mastication; Methods; Motor Activity; Norepinephrine; Perphenazine; Phenothiazines; Prochlorperazine; Promazine; Rats; Thiazines; Thioridazine; Tranquilizing Agents; Trifluoperazine; Triflupromazine; Trimeprazine

1967
Influence of antiparkinson drugs and amphetamine on some pharmacological effects of phenothiazine derivatives used as neuroleptics.
    Psychopharmacologia, 1964, Sep-11, Volume: 6, Issue:3

    Topics: Amphetamine; Animals; Apomorphine; Avoidance Learning; Behavior, Animal; Body Temperature; Catalepsy; Chlorpromazine; Dextroamphetamine; Dogs; Humans; Mastication; Mice; Movement; Pentobarbital; Perphenazine; Rats; Scopolamine; Trifluoperazine; Trihexyphenidyl; Vomiting

1964
Adrenergic effect of chronic administration of neuroleptics.
    Nature, 1967, Jun-17, Volume: 214, Issue:5094

    Topics: Amphetamine; Animals; Apomorphine; Chlorpromazine; Feedback; Haloperidol; Perphenazine; Rats; Sympathetic Nervous System; Tetrabenazine; Tranquilizing Agents; Trifluoperazine

1967
Changes in rat striatal dopamine turnover and receptor activity during one years neuroleptic administration.
    European journal of pharmacology, 1980, May-02, Volume: 63, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Binding Sites; Corpus Striatum; Cyclic AMP; Dopamine; Homovanillic Acid; Male; Rats; Receptors, Dopamine; Spiperone; Thioridazine; Time Factors; Trifluoperazine

1980
Cerebral dopamine function in rats following withdrawal from one year of continuous neuroleptic administration.
    European journal of pharmacology, 1980, May-02, Volume: 63, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Antipsychotic Agents; Apomorphine; Binding Sites; Body Weight; Brain; Corpus Striatum; Dopamine; Homovanillic Acid; Humans; Male; Motor Activity; Mouth; Movement; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Substance Withdrawal Syndrome; Thioridazine; Time Factors; Trifluoperazine

1980
Chronic continuous administration of neuroleptic drugs alters cerebral dopamine receptors and increases spontaneous dopaminergic action in the striatum.
    Nature, 1982, Apr-08, Volume: 296, Issue:5857

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Rats; Receptors, Dopamine; Spiperone; Trifluoperazine

1982
Interpretation of changes in apomorphine-induced stereotyped behaviour in rats receiving continuous administration of trifluorperazine for 15 months.
    Neuropharmacology, 1984, Volume: 23, Issue:8

    Topics: Animals; Antipsychotic Agents; Apomorphine; Humans; Male; Motor Activity; Rats; Rats, Inbred Strains; Stereotyped Behavior; Time Factors; Trifluoperazine

1984
Reserpine-induced rigidity in rats: drug effects on muscle tone from corpus striatum and nucleus accumbens.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Carbidopa; Corpus Striatum; Male; Muscle Rigidity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Reserpine; Septal Nuclei; Trifluoperazine

1983
A comparison of striatal and mesolimbic dopamine function in the rat during 6-month trifluoperazine administration.
    Psychopharmacology, 1980, Volume: 69, Issue:3

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Binding Sites; Corpus Striatum; Dopamine; Humans; Limbic System; Male; Rats; Spiperone; Stereotyped Behavior; Time Factors; Trifluoperazine

1980
Changes in cerebral dopamine function induced by a year's administration of trifluoperazine or thioridazine and their subsequent withdrawal.
    Advances in biochemical psychopharmacology, 1980, Volume: 24

    Topics: Adenylyl Cyclases; Animals; Apomorphine; Brain; Corpus Striatum; Dopamine; Dyskinesia, Drug-Induced; Humans; Male; Rats; Spiperone; Stereotyped Behavior; Substance Withdrawal Syndrome; Thioridazine; Time Factors; Trifluoperazine

1980
Dopamine-inhibited adenylate cyclase in female rat adenohypophysis.
    Life sciences, 1981, Apr-06, Volume: 28, Issue:14

    Topics: Adenylyl Cyclase Inhibitors; Animals; Apomorphine; Dopamine; Female; Kinetics; Lactation; Male; Norepinephrine; Pituitary Gland, Anterior; Pregnancy; Rats; Sex Factors; Sulpiride; Trifluoperazine

1981
Evidence for dopamine mediation of submissive gestures in the stumptail macaque monkey.
    Pharmacology, biochemistry, and behavior, 1981, Volume: 14 Suppl 1

    Topics: Amphetamine; Animals; Apomorphine; Dominance-Subordination; Female; Haloperidol; Macaca; Male; Methoxydimethyltryptamines; Pimozide; Receptors, Dopamine; Serotonin Antagonists; Social Dominance; Trifluoperazine

1981
Dopamine D4 versus D2 receptor selectivity of dopamine receptor antagonists: possible therapeutic implications.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Animals; Apomorphine; Butyrophenones; Cell Line; Chlorpromazine; Clozapine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Trifluoperazine

1993
ANTI-EMETIC ACTIVITY OF PHENOTHIAZINES IN RELATION TO THEIR CHEMICAL STRUCTURE.
    British journal of pharmacology and chemotherapy, 1963, Volume: 21

    Topics: Animals; Antiemetics; Antipsychotic Agents; Apomorphine; Chemistry, Pharmaceutical; Chlorpromazine; Dogs; Perphenazine; Pharmacology; Phenothiazines; Prochlorperazine; Research; Thioridazine; Tranquilizing Agents; Trifluoperazine

1963
Calmodulin inhibitor trifluoperazine attenuates the development and expression of morphine-induced conditioned place preference in rats.
    European journal of pharmacology, 2004, Feb-23, Volume: 486, Issue:3

    Topics: Animals; Apomorphine; Calcium Channel Blockers; Calmodulin; Conditioning, Psychological; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Morphine; Motor Activity; Narcotics; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Trifluoperazine; Verapamil

2004