Page last updated: 2024-08-17

apomorphine and roxindole

apomorphine has been researched along with roxindole in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (66.67)18.2507
2000's2 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnickel, G; Böttcher, H; Eiermann, V; Haase, AF; Hausberg, HH; Seyfried, CA1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Audinot, V; Boutin, JA; Cussac, D; Maiofiss, L; Millan, MJ; Newman-Tancredi, A1
Bartoszyk, GD; Seyfried, CA1
Bartoszyk, GD; Harting, J; Minck, KO1
Kolodziejczyk, K; Maj, J; Rogóz, Z; Skuza, G1

Other Studies

6 other study(ies) available for apomorphine and roxindole

ArticleYear
Synthesis and dopaminergic activity of some 3-(1,2,3,6-tetrahydro-1-pyridylalkyl)indoles. A novel conformational model to explain structure-activity relationships.
    Journal of medicinal chemistry, 1992, Oct-30, Volume: 35, Issue:22

    Topics: Animals; Binding, Competitive; Corpus Striatum; Dopamine Agents; In Vitro Techniques; Indoles; Male; Models, Molecular; Molecular Conformation; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior; Structure-Activity Relationship

1992
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Differential actions of antiparkinson agents at multiple classes of monoaminergic receptor. I. A multivariate analysis of the binding profiles of 14 drugs at 21 native and cloned human receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:2

    Topics: Animals; Antiparkinson Agents; Binding Sites; Binding, Competitive; Cholinergic Antagonists; Cloning, Molecular; Cluster Analysis; Dopamine Agonists; Humans; Rats; Receptor, Muscarinic M1; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Histamine H1; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Serotonin

2002
Sensitivity of dopamine D2 receptors following long-term treatment with roxindole.
    European journal of pharmacology, 1994, May-12, Volume: 257, Issue:1-2

    Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Down-Regulation; Drug Interactions; Haloperidol; Indoles; Injections, Intraperitoneal; Male; Oxindoles; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior

1994
Roxindole: psychopharmacological profile of a dopamine D2 autoreceptor agonist.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Avoidance Learning; Azepines; Catalepsy; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Interactions; Indoles; Male; Mice; Motor Activity; Oxindoles; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior

1996
Roxindole, a potential antidepressant. I. Effect on the dopamine system.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:5

    Topics: Amphetamine; Analysis of Variance; Animals; Antidepressive Agents; Apomorphine; Dopamine Agonists; Drug Administration Schedule; Indoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Oxindoles; Pyridines; Rats; Rats, Wistar; Stereotyped Behavior

1996