apomorphine has been researched along with raclopride in 80 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (10.00) | 18.7374 |
1990's | 31 (38.75) | 18.2507 |
2000's | 26 (32.50) | 29.6817 |
2010's | 14 (17.50) | 24.3611 |
2020's | 1 (1.25) | 2.80 |
Authors | Studies |
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Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P | 1 |
Liu, C; Park, H; Urs, AN; Urs, NM; Wang, Q; Zimmerman, J | 1 |
Eaton, RC; Hull, EM; Loucks, JA; Lumley, LA; Markowski, VP; Moses, J | 1 |
Carlsson, A; Carlsson, ML; Svensson, A | 1 |
Hall, H; Halldin, C; Sedvall, G | 1 |
Ferre, S; Fredholm, BB; Fuxe, K; Johansson, B; von Euler, G | 1 |
Jaehnig, P; Jenner, P; Lange, KW; Löschmann, PA; Marsden, CD; Smith, LA | 1 |
Agerberth, B; Ferré, S; Fuxe, K; Mutt, V; von Euler, G; von Euler, M | 1 |
Bervoets, K; Mavridis, M; Millan, MJ | 1 |
Ross, SB | 1 |
Braff, DL; Geyer, MA; Keith, VA; Swerdlow, NR | 1 |
Cozzolino, A; Di Chiara, G; Fenu, S; Morelli, M | 1 |
Ahlenius, S; Ericson, EL; Högberg, K; Wijkström, A | 1 |
Bengtsson, S; de Paulis, T; Hall, H; Högberg, T; Johansson, L; Ogren, SO; Ström, P | 1 |
Crocker, AD; Overstreet, DH | 1 |
Allikmets, LKh; Kharro, IaE; Lang, AE; Vasar, EE | 1 |
Crocker, AD; Faunt, JE | 1 |
Cameron, DL; Crocker, AD | 1 |
Ljungberg, T | 1 |
Hall, H; Köhler, C; Magnusson, O; Ogren, SO; Sjöstrand, SE | 1 |
Andersen, PH; Nielsen, EB | 1 |
Karlsson-Boethius, G; Köhler, C | 1 |
Angeby-Möller, K; de Paulis, T; Hall, H; Johansson, L; Kumar, Y; Ogren, SO; Rämsby, S; Sällemark, M | 1 |
Hull, EM; Loucks, JA; Matuszewich, L; Moses, J; Watson, HL | 1 |
Conway, PC; Corbett, R; Dunn, RW; Hartman, H; Helsley, GC; Kerman, LL; Strupczewski, JT; Woods, AT | 1 |
Artigas, F; Ferré, S | 1 |
Glenthøj, B | 1 |
Crocker, AD; Double, KL | 1 |
Eaton, MJ; Gopalan, C; Kim, E; Lookingland, KJ; Moore, KE | 1 |
Fuxe, K; Hedlund, PB; Li, XM | 1 |
Agnati, LF; Fuxe, K; Hedlund, PB; Li, XM | 1 |
Day, JC; Fibiger, HC | 1 |
Korf, J; Vaalburg, W; van der Worp, H; Visser, GM; Wiegman, T; Zijlstra, S | 1 |
Day, J; Fibiger, HC | 1 |
Evans, DL; Figur, LM; Lahti, RA; Stratman, NC | 1 |
Carlsson, A; Haadsma-Svensson, SR; Smith, MW; Svensson, K; Waters, N | 1 |
Glenthøj, B; Hemmingsen, R; Holm, S; Laursen, H; Mogensen, J | 1 |
Chase, TN; Kapitzoglou-Logothetis, V; Marin, C; Parashos, SA; Peppe, A | 1 |
Navas, F; Norman, MH; Rigdon, GC; Thompson, JB | 1 |
Comoy, E; Lesourd, M; Protais, P | 1 |
Stoessl, AJ; Van Kampen, JM | 1 |
Artigas, F; Honrubia, MA; Martín-Ruiz, R; Mengod, G; Ugedo, L | 1 |
Calne, DB; de la Fuente-Fernández, R; Ruth, TJ; Schulzer, M; Sossi, V; Stoessl, AJ | 1 |
Calne, DB; de La Fuente-Fernández, R; Holden, JE; Lim, AS; Ruth, TJ; Sossi, V; Stoessl, AJ | 1 |
Cumming, P; Gillings, N; Gjedde, A; Hilton, J; Scheffel, U; Wong, DF | 1 |
Cumming, P; Dannals, RF; Gillings, N; Gjedde, A; Hilton, J; Scheffel, U; Wong, DF | 1 |
Calne, DB; de la Fuente-Fernández, R; Phillips, AG; Ruth, TJ; Sossi, V; Stoessl, AJ; Zamburlini, M | 1 |
Bucan, M; Fetsko, LA; Hranilovic, D; Wang, Y; Xu, R | 1 |
Geyer, MA; Lehmann-Masten, V; Ralph-Williams, RJ | 1 |
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH | 1 |
Garland, T; Rhodes, JS | 1 |
Fan, LW; Ho, IK; Loh, HH; Ma, T; Park, Y; Tien, LT | 1 |
Gazi, L; López-Giménez, JF; Rüdiger, MP; Strange, PG | 1 |
Gibney, BC; Lewis, MH; Presti, MF | 1 |
Antonini, A; Leenders, KL; Linazasoro, G; Maguire, RP | 1 |
Abi-Dargham, A; Cooper, TB; Erritzoe, D; Huang, Y; Hwang, DR; Kegeles, LS; Laruelle, M; Martinez, D; Narendran, R; Slifstein, M; Talbot, PS | 1 |
Ekelund, J; Guillin, O; Huang, Y; Hwang, DR; Hwang, Y; Laruelle, M; Martinez, D; Narendran, R; Scher, E; Slifstein, M | 1 |
Savel'ev, SA | 2 |
Hwang, DR; Hwang, Y; Laruelle, M; Martinez, D; Narendran, R; Reeder, S; Scher, E; Slifstein, M | 1 |
Ji, XQ; Jin, DZ; Liu, DZ; Tang, CP; Ye, Y; Zhang, LM; Zhu, J; Zhu, XZ | 1 |
Michaelides, M; Piyis, YK; Thanos, PK; Volkow, ND; Wang, GJ | 1 |
Bazinet, RP; Bhattacharjee, AK; Chang, L; Rapoport, SI; White, L | 1 |
Seeman, P | 1 |
Bang-Andersen, B; Bundgaard, C; Farde, L; Finnema, SJ; Gulyás, B; Halldin, C; Wikström, HV | 1 |
Eriksson, L; Farde, L; Gulyás, B; Halldin, C; Sjöholm, N; Varrone, A | 1 |
Jang, CG; Kim, HC; Lee, HK; Lee, SY; Yoo, JH | 1 |
Frankle, WG; Kendro, S; Laymon, CM; Lopresti, BJ; Martinez, D; Mason, NS; Mathis, CA; May, MA; Narendran, R; Velasquez, ND | 1 |
Ding, M; Dorff, P; Elmore, CS; Maier, D; Malmquist, J; Mrzljak, L; Peng, T; Ström, P; Tuke, D; Werkheiser, J; Widzowski, D; Zysk, J | 1 |
Kakiuchi, T; Nishiyama, S; Ohba, H; Tsukada, H | 1 |
Arakawa, R; Farde, L; Halldin, C; Ito, H; Kodaka, F; Miyoshi, M; Nakayama, K; Okumura, M; Otsuka, T; Suhara, T; Takahashi, H; Takano, H | 1 |
de Lima, MN; Dornelles, A; Garcia, VA; Presti-Torres, J; Roesler, R; Scalco, FS; Schröder, N | 1 |
Brantley, E; Karain, B; Shi, WX; Xu, D | 1 |
Farde, L; Fujie, S; Fujiwara, H; Halldin, C; Ito, H; Kimura, Y; Kodaka, F; Nakayama, K; Sasaki, T; Suhara, T; Takano, H | 1 |
Battaglia, G; Bucci, D; Consolazione, M; Lionetto, L; Maccari, S; Mairesse, J; Marrocco, J; Morley-Fletcher, S; Nicoletti, F; Ravasi, L; Simmaco, M | 1 |
Baladi, MG; France, CP; Newman, AH | 1 |
Gong, X; Liang, X; Liu, L; Wang, X; Zhang, W | 1 |
Andersen, AH; Forman, E; Gash, DM; Gerhardt, GA; Grondin, RC; Hardy, PA; Zhang, Z | 1 |
Antkiewicz-Michaluk, L; Czarnecka, A; Kamińska, K; Konieczny, J; Lenda, T | 1 |
Fujiwara, H; Higuchi, M; Ito, H; Kimura, Y; Kodaka, F; Kubota, M; Moriguchi, S; Nagashima, T; Okubo, Y; Suhara, T; Takahashi, H; Takahata, K; Takano, H | 1 |
3 trial(s) available for apomorphine and raclopride
Article | Year |
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Expectation and dopamine release: mechanism of the placebo effect in Parkinson's disease.
Topics: Aged; Antiparkinson Agents; Apomorphine; Corpus Striatum; Dopamine; Female; Humans; Male; Middle Aged; Parkinson Disease; Placebo Effect; Placebos; Raclopride; Synapses; Tomography, Emission-Computed | 2001 |
Dopamine release in human ventral striatum and expectation of reward.
Topics: Antiparkinson Agents; Apomorphine; Dopamine; Dopamine Antagonists; Humans; Neostriatum; Nucleus Accumbens; Parkinson Disease; Raclopride; Reward; Tomography, Emission-Computed | 2002 |
Effect of risperidone on high-affinity state of dopamine D2 receptors: a PET study with agonist ligand [11C](R)-2-CH3O-N-n-propylnorapomorphine.
Topics: Adult; Apomorphine; Brain; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Ligands; Magnetic Resonance Imaging; Male; Positron-Emission Tomography; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Risperidone; Schizophrenia; Young Adult | 2011 |
77 other study(ies) available for apomorphine and raclopride
Article | Year |
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Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution | 1990 |
Structure-Functional-Selectivity Relationship Studies of Novel Apomorphine Analogs to Develop D1R/D2R Biased Ligands.
Topics: | 2020 |
Opposite influence of medial preoptic D1 and D2 receptors on genital reflexes: implications for copulation.
Topics: Animals; Apomorphine; Benzazepines; Copulation; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ejaculation; Male; Penile Erection; Penis; Preoptic Area; Raclopride; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Thiophenes | 1992 |
Differential locomotor interactions between dopamine D1/D2 receptor agonists and the NMDA antagonist dizocilpine in monoamine-depleted mice.
Topics: alpha-Methyltyrosine; Animals; Apomorphine; Benzazepines; Biogenic Monoamines; Bromocriptine; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Male; Methyltyrosines; Mice; Motor Activity; N-Methylaspartate; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Salicylamides; Tyrosine 3-Monooxygenase | 1992 |
Gpp(NH)p stimulates [3H]raclopride binding to homogenates from human putamen and accumbens.
Topics: Apomorphine; Binding, Competitive; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Nucleus Accumbens; Pergolide; Protein Binding; Putamen; Raclopride; Receptors, Dopamine; Salicylamides; Second Messenger Systems; Stimulation, Chemical | 1992 |
Stimulation of high-affinity adenosine A2 receptors decreases the affinity of dopamine D2 receptors in rat striatal membranes.
Topics: Adenosine; Animals; Apomorphine; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Dopamine; Dopamine Agents; Kinetics; Male; Phenethylamines; Phenylisopropyladenosine; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Purinergic; Salicylamides; Theophylline | 1991 |
Motor activity following the administration of selective D-1 and D-2 dopaminergic drugs to normal common marmosets.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Callithrix; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Female; Male; Motor Activity; Quinpirole; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Stereotyped Behavior | 1991 |
A trypsin inhibitor-like peptide PEC-60 reduces the affinity of dopamine D2 agonist binding sites in rat neostriatal membranes.
Topics: Animals; Apomorphine; Binding Sites; Corpus Striatum; Dopamine; Dopamine Antagonists; Kinetics; Membranes; Peptides; Raclopride; Rats; Salicylamides; Trypsin Inhibitors | 1991 |
The serotonin (5-HT)1A agonist, LY 165,163, induces contralateral rotation in unilateral substantia nigra-lesioned rats via dopamine receptors.
Topics: Alprenolol; Animals; Apomorphine; Benzazepines; Haloperidol; Male; Motor Activity; Oxidopamine; Piperazines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Serotonin Antagonists; Substantia Nigra | 1991 |
Synaptic concentration of dopamine in the mouse striatum in relationship to the kinetic properties of the dopamine receptors and uptake mechanism.
Topics: Aminoquinolines; Animals; Apomorphine; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Kinetics; Male; Mice; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Synapses; Synaptosomes; Tetrahydronaphthalenes | 1991 |
Effects of spiperone, raclopride, SCH 23390 and clozapine on apomorphine inhibition of sensorimotor gating of the startle response in the rat.
Topics: Analysis of Variance; Animals; Apomorphine; Benzazepines; Clozapine; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reflex, Startle; Salicylamides; Schizophrenia; Spiperone | 1991 |
Positive and negative interactions in the behavioural expression of D1 and D2 receptor stimulation in a model of Parkinsonism: role of priming.
Topics: Animals; Apomorphine; Behavior, Animal; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Hydroxydopamines; Male; Oxidopamine; Parkinson Disease; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Stereotyped Behavior | 1991 |
Behavioural and biochemical effects of subchronic treatment with raclopride in the rat: tolerance and brain monoamine receptor sensitivity.
Topics: Animals; Apomorphine; Brain; Dihydroxyphenylalanine; Dopamine Antagonists; Drug Tolerance; Male; Motor Activity; Raclopride; Rats; Rats, Inbred Strains; Reserpine; Salicylamides; Substance Withdrawal Syndrome; Time Factors | 1991 |
Potential antipsychotic agents 5. Synthesis and antidopaminergic properties of substituted 5,6-dimethoxysalicylamides and related compounds.
Topics: Animals; Antipsychotic Agents; Apomorphine; Binding Sites; Chemical Phenomena; Chemistry; Dopamine Antagonists; Male; Raclopride; Rats; Rats, Inbred Strains; Salicylamides; Spiperone; Structure-Activity Relationship | 1990 |
Dopamine sensitivity in rats selectively bred for increases in cholinergic function.
Topics: Animals; Apomorphine; Autoradiography; Behavior, Animal; Body Temperature; Dopamine; Ergolines; Male; Parasympathetic Nervous System; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Stereotyped Behavior | 1991 |
[Adaptive changes in sigma and phencyclidine receptors during the long-term use of haloperidol and raclopride in rats].
Topics: Adaptation, Physiological; Animals; Apomorphine; Behavior, Animal; Drug Interactions; Haloperidol; Ketamine; Phenazocine; Phencyclidine; Raclopride; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Salicylamides; Time Factors; Tritium | 1989 |
Effects of adrenalectomy on responses mediated by dopamine D-1 and D-2 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenalectomy; Animals; Apomorphine; Behavior, Animal; Benzazepines; Body Temperature; Dopamine Agents; Ergolines; Male; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides | 1989 |
Localization of striatal dopamine receptor function by central injection of an irreversible receptor antagonist.
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine Antagonists; Male; Nucleus Accumbens; Quinolines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Septal Nuclei; Stereotyped Behavior | 1989 |
Attenuation of water intake and operant responding by dopamine D2 antagonists: raclopride provides important cues for understanding the functional mechanism of action.
Topics: Animals; Apomorphine; Conditioning, Operant; Cues; Dopamine Antagonists; Dose-Response Relationship, Drug; Drinking; Extrapyramidal Tracts; Male; Raclopride; Rats; Rats, Inbred Strains; Salicylamides | 1989 |
The selective dopamine D2 receptor antagonist raclopride discriminates between dopamine-mediated motor functions.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Behavior, Animal; Catalepsy; Dopamine; Emetics; Male; Motor Activity; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Stereotyped Behavior | 1986 |
The benzazepine, SCH 23390, inhibits 3H-NPA binding in mouse brain in vivo.
Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Male; Mice; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Spiperone | 1986 |
In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain.
Topics: Animals; Apomorphine; Binding, Competitive; Brain; Kinetics; Male; Organ Specificity; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Salicylamides; Spiperone; Stereoisomerism | 1988 |
Potential neuroleptic agents. 4. Chemistry, behavioral pharmacology, and inhibition of [3H]spiperone binding of 3,5-disubstituted N-[(1-ethyl-2-pyrrolidinyl)methyl]-6-methoxysalicylamides.
Topics: Animals; Apomorphine; Chemical Phenomena; Chemistry; Corpus Striatum; Haloperidol; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone; Stereotyped Behavior; Structure-Activity Relationship | 1986 |
Dopaminergic drugs in the medial preoptic area and nucleus accumbens: effects on motor activity, sexual motivation, and sexual performance.
Topics: Animals; Apomorphine; Benzazepines; Copulation; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Female; Male; Microinjections; Motivation; Motor Activity; Nucleus Accumbens; Preoptic Area; Quinolines; Raclopride; Rats; Salicylamides; Sexual Behavior, Animal | 1995 |
Effects of atypical antipsychotic agents on social behavior in rodents.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Catalepsy; Chlorpromazine; Clozapine; Diazepam; Haloperidol; Isoxazoles; Male; Mice; Mice, Inbred Strains; Piperidines; Raclopride; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Social Behavior | 1993 |
Dopamine D2 receptor-mediated regulation of serotonin extracellular concentration in the dorsal raphe nucleus of freely moving rats.
Topics: Animals; Apomorphine; Benzazepines; Dialysis; Dopamine D2 Receptor Antagonists; Ergolines; Extracellular Space; Hydroxyindoleacetic Acid; Male; Quinpirole; Raclopride; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Serotonin | 1993 |
Persistent vacuous chewing in rats following neuroleptic treatment: relationship to dopaminergic and cholinergic function.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Benzofurans; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Haloperidol; Male; Parasympathetic Nervous System; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Scopolamine; Stereotyped Behavior | 1993 |
Dopamine receptors in the substantia nigra are involved in the regulation of muscle tone.
Topics: Animals; Apomorphine; Benzazepines; Brain Mapping; Electromyography; Male; Muscles; Quinolines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Salicylamides; Substantia Nigra | 1995 |
Comparison of the effects of the dopamine D2 agonist quinelorane on tuberoinfundibular dopaminergic neuronal activity in male and female rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Female; Immune Sera; Male; Median Eminence; Neurons; Pituitary Gland; Prolactin; Quinolines; Raclopride; Rats; Receptors, Dopamine D2; Salicylamides; Sex Factors | 1993 |
Cholecystokinin receptor subtypes regulate dopamine D2 receptors in rat neostriatal membranes. Involvement of D1 receptors.
Topics: Animals; Apomorphine; Cell Membrane; Dopamine Agents; Kinetics; Neostriatum; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Sincalide | 1994 |
Dopamine D1 receptors are involved in the modulation of D2 receptors induced by cholecystokinin receptor subtypes in rat neostriatal membranes.
Topics: Animals; Apomorphine; Benzazepines; Binding, Competitive; Dopamine; Dopamine Agonists; In Vitro Techniques; Kinetics; Male; Membranes; Neostriatum; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Sincalide | 1994 |
Dopaminergic regulation of septohippocampal cholinergic neurons.
Topics: Acetylcholine; Animals; Apomorphine; Benzazepines; Dextroamphetamine; Dialysis; Dopamine Agonists; Dopamine Antagonists; Ergolines; Hippocampus; Indoles; Male; Neurons; Phenanthridines; Quinpirole; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine; Salicylamides | 1994 |
Synthesis and in vivo distribution in the rat of a dopamine agonist: N-([11C]methyl)norapomorphine.
Topics: Animals; Apomorphine; Brain; Carbon Radioisotopes; Dopamine Agents; Kidney; Liver; Lung; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone | 1993 |
Dopaminergic regulation of cortical acetylcholine release: effects of dopamine receptor agonists.
Topics: Acetylcholine; Animals; Apomorphine; Benzazepines; Cerebral Cortex; Dialysis; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Indoles; Male; Nerve Endings; Oxazines; Phenanthridines; Quinpirole; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides | 1993 |
Dopamine D4 versus D2 receptor selectivity of dopamine receptor antagonists: possible therapeutic implications.
Topics: Animals; Apomorphine; Butyrophenones; Cell Line; Chlorpromazine; Clozapine; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Trifluoperazine | 1993 |
The dopamine D3-receptor: a postsynaptic receptor inhibitory on rat locomotor activity.
Topics: Aminoquinolines; Animals; Apomorphine; CHO Cells; Corpus Striatum; Cricetinae; Dextroamphetamine; Dopamine; Dopamine Antagonists; Drug Interactions; Indans; Male; Methyltyrosines; Models, Biological; Motor Activity; Nucleus Accumbens; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Fusion Proteins; Reserpine; Salicylamides; Spiperone; Stimulation, Chemical | 1993 |
Electrical sensitization of the meso-limbic dopaminergic system in rats: a pathogenetic model for schizophrenia.
Topics: Amphetamine; Animals; Apomorphine; Benzazepines; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Electric Stimulation; Electroencephalography; Habituation, Psychophysiologic; Haloperidol; Limbic System; Male; Models, Neurological; Motor Activity; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Salicylamides; Schizophrenia; Seizures; Stereotyped Behavior; Tegmentum Mesencephali; Time Factors | 1993 |
D1 and D2 dopamine receptor-mediated mechanisms and behavioral supersensitivity.
Topics: Animals; Apomorphine; Behavior, Animal; Benzazepines; Catalepsy; Dopamine D2 Receptor Antagonists; Haloperidol; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Salicylamides; Stereotyped Behavior; Up-Regulation | 1993 |
Synthesis and evaluation of heterocyclic carboxamides as potential antipsychotic agents.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Clozapine; Heterocyclic Compounds; Magnetic Resonance Spectroscopy; Mice; Molecular Structure; Piperazines; Raclopride; Receptors, Dopamine; Receptors, Serotonin; Risperidone; Salicylamides; Thiazoles | 1996 |
Similar pharmacological properties of 8-OH-DPAT and alnespirone (S 20499) at dopamine receptors: comparison with buspirone.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Apomorphine; Behavior, Animal; Benzazepines; Buspirone; Corpus Striatum; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Mice; Piperazines; Raclopride; Salicylamides; Serotonin; Serotonin Antagonists; Spiro Compounds; Tritium | 1998 |
Effects of oligonucleotide antisense to dopamine D(1A) receptor messenger RNA in a rodent model of levodopa-induced dyskinesia.
Topics: Animals; Antiparkinson Agents; Apomorphine; Autoradiography; Behavior, Animal; Cocaine; Denervation; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dyskinesia, Drug-Induced; Gene Expression; Levodopa; Male; Oligonucleotides, Antisense; Oxidopamine; Phenotype; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Rotation; Substantia Nigra; Sympatholytics; Tritium | 2000 |
Control of serotonergic neurons in rat brain by dopaminergic receptors outside the dorsal raphe nucleus.
Topics: Animals; Apomorphine; Benzazepines; Corpus Striatum; In Situ Hybridization; Male; Microdialysis; Neurons; Quinpirole; Raclopride; Raphe Nuclei; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; RNA, Messenger; Serotonin; Tetrodotoxin | 2001 |
Apomorphine-induced changes in synaptic dopamine levels: positron emission tomography evidence for presynaptic inhibition.
Topics: Antiparkinson Agents; Apomorphine; Dopamine; Female; Functional Laterality; Humans; Male; Models, Biological; Parkinson Disease; Presynaptic Terminals; Raclopride; Synapses; Tomography, Emission-Computed | 2001 |
Specific binding of [(11)C]raclopride and N-[(3)H]propyl-norapomorphine to dopamine receptors in living mouse striatum: occupancy by endogenous dopamine and guanosine triphosphate-free G protein.
Topics: Animals; Apomorphine; Carbon Radioisotopes; Corpus Striatum; Dopamine; GTP-Binding Proteins; Kinetics; Male; Mice; Protein Binding; Raclopride; Receptors, Dopamine; Tritium | 2002 |
The competition between endogenous dopamine and radioligands for specific binding to dopamine receptors.
Topics: Aminoquinolines; Amphetamine; Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Kinetics; Male; Mice; Raclopride; Radioligand Assay; Receptors, Dopamine; Reserpine | 2002 |
Dopamine D2S and D2L receptors may differentially contribute to the actions of antipsychotic and psychotic agents in mice.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Clozapine; Dopamine Agonists; Dose-Response Relationship, Drug; Hallucinogens; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Parkinsonian Disorders; Protein Isoforms; Raclopride; Receptors, Dopamine D2 | 2002 |
Dopamine D1 rather than D2 receptor agonists disrupt prepulse inhibition of startle in mice.
Topics: Animals; Apomorphine; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Mice; Mice, Inbred C57BL; Mice, Knockout; Pergolide; Phenanthridines; Quinpirole; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Reflex, Startle | 2003 |
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes | 2003 |
Differential sensitivity to acute administration of Ritalin, apomorphine, SCH 23390, but not raclopride in mice selectively bred for hyperactive wheel-running behavior.
Topics: Animals; Animals, Outbred Strains; Apomorphine; Benzazepines; Breeding; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Hyperkinesis; Male; Methylphenidate; Mice; Motor Activity; Raclopride; Selection, Genetic; Species Specificity; Time Factors | 2003 |
Increased dopamine D2 receptor binding and enhanced apomorphine-induced locomotor activity in mu-opioid receptor knockout mice.
Topics: Analysis of Variance; Animals; Apomorphine; Autoradiography; Benzazepines; Binding Sites; Caudate Nucleus; Dopamine Agonists; Dopamine Antagonists; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nucleus Accumbens; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, mu; Time Factors; Tritium | 2003 |
Constitutive oligomerization of human D2 dopamine receptors expressed in Spodoptera frugiperda 9 (Sf9) and in HEK293 cells. Analysis using co-immunoprecipitation and time-resolved fluorescence resonance energy transfer.
Topics: Animals; Apomorphine; Base Sequence; Blotting, Western; Cell Membrane; Cells, Cultured; Dopamine Agonists; Dopamine Antagonists; Epitopes; Europium; Fluorescence Resonance Energy Transfer; Humans; Immunoglobulins; Ligands; Molecular Sequence Data; Precipitin Tests; Raclopride; Receptors, Dopamine D2; Recombinant Proteins; Spodoptera; Time Factors | 2003 |
Effects of intrastriatal administration of selective dopaminergic ligands on spontaneous stereotypy in mice.
Topics: Animals; Apomorphine; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Female; Injections; Locomotion; Male; Neostriatum; Peromyscus; Quinpirole; Raclopride; Receptors, Dopamine; Stereotyped Behavior | 2004 |
Pharmacological and PET studies in patient's with Parkinson's disease and a short duration-motor response: implications in the pathophysiology of motor complications.
Topics: Adult; Age of Onset; Aged; Apomorphine; Biological Transport; Corpus Striatum; Dihydroxyphenylalanine; Female; Fluorine Radioisotopes; Humans; Male; Middle Aged; Parkinson Disease; Raclopride; Reaction Time; Tomography, Emission-Computed; Tritium | 2004 |
In vivo vulnerability to competition by endogenous dopamine: comparison of the D2 receptor agonist radiotracer (-)-N-[11C]propyl-norapomorphine ([11C]NPA) with the D2 receptor antagonist radiotracer [11C]-raclopride.
Topics: Algorithms; Amphetamine; Animals; Apomorphine; Binding, Competitive; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Image Processing, Computer-Assisted; Magnetic Resonance Imaging; Male; Papio; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Tomography, Emission-Computed | 2004 |
Measurement of the proportion of D2 receptors configured in state of high affinity for agonists in vivo: a positron emission tomography study using [11C]N-propyl-norapomorphine and [11C]raclopride in baboons.
Topics: Animals; Apomorphine; Brain; Carbon Radioisotopes; Dopamine Agonists; Male; Papio; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2 | 2005 |
[Influence of local administration of apomorphine on citrulline extracellular level in the striatum: participation of the dopamine D1 and D2 receptors].
Topics: Animals; Apomorphine; Benzazepines; Chromatography, Liquid; Citrulline; Corpus Striatum; Dopamine D2 Receptor Antagonists; Male; Microdialysis; Nitric Oxide Synthase; Nitroarginine; Raclopride; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2005 |
Effects of local infusions of apomorphine on the extracellular citrulline level in the striatum: Involvement of D1 and D2 dopamine receptors.
Topics: Animals; Apomorphine; Benzazepines; Chromatography, High Pressure Liquid; Citrulline; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Enzyme Inhibitors; Extracellular Fluid; Male; Nitroarginine; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2006 |
Amphetamine-induced dopamine release: duration of action as assessed with the D2/3 receptor agonist radiotracer (-)-N-[(11)C]propyl-norapomorphine ([11C]NPA) in an anesthetized nonhuman primate.
Topics: Amphetamine; Animals; Apomorphine; Binding, Competitive; Carbon Isotopes; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Male; Papio; Positron-Emission Tomography; Raclopride; Time Factors | 2007 |
Behavioral recovery following sub-chronic paeoniflorin administration in the striatal 6-OHDA lesion rodent model of Parkinson's disease.
Topics: Animals; Apomorphine; Behavior, Animal; Benzazepines; Benzoates; Binding, Competitive; Bridged-Ring Compounds; Dopamine Agonists; Dopamine Antagonists; Glucosides; Hydroxydopamines; In Vitro Techniques; Male; Membranes; Microinjections; Monoterpenes; Neostriatum; Parkinson Disease, Secondary; Raclopride; Rats; Rats, Sprague-Dawley; Stereotyped Behavior | 2007 |
Food restriction markedly increases dopamine D2 receptor (D2R) in a rat model of obesity as assessed with in-vivo muPET imaging ([11C] raclopride) and in-vitro ([3H] spiperone) autoradiography.
Topics: Age Factors; Animals; Apomorphine; Appetite Regulation; Autoradiography; Brain; Disease Models, Animal; Dopamine; Dopamine Agonists; Eating; Food Deprivation; In Vitro Techniques; Male; Motor Activity; Obesity; Positron-Emission Tomography; Raclopride; Rats; Rats, Zucker; Receptors, Dopamine D2; Receptors, Leptin; Spiperone; Tritium | 2008 |
Imaging apomorphine stimulation of brain arachidonic acid signaling via D2-like receptors in unanesthetized rats.
Topics: Animals; Apomorphine; Arachidonic Acid; Autoradiography; Brain; Brain Mapping; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Group IV Phospholipases A2; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine D2; Signal Transduction | 2008 |
Dopamine D2High receptors measured ex vivo are elevated in amphetamine-sensitized animals.
Topics: Amphetamine; Animals; Apomorphine; Binding, Competitive; Central Nervous System Stimulants; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Protein Binding; Raclopride; Rats; Receptors, Dopamine D2; Tritium | 2009 |
Dopamine D(2/3) receptor occupancy of apomorphine in the nonhuman primate brain--a comparative PET study with [11C]raclopride and [11C]MNPA.
Topics: Animals; Apomorphine; Brain; Carbon Radioisotopes; Dopamine D2 Receptor Antagonists; Female; Macaca fascicularis; Positron-Emission Tomography; Protein Binding; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Tissue Distribution | 2009 |
Advancement in PET quantification using 3D-OP-OSEM point spread function reconstruction with the HRRT.
Topics: Algorithms; Animals; Apomorphine; Brain; Carbon Radioisotopes; Dopamine Agonists; Dopamine Antagonists; Fluorine Radioisotopes; Humans; Image Processing, Computer-Assisted; Macaca fascicularis; Models, Statistical; Phantoms, Imaging; Positron-Emission Tomography; Raclopride; Radiopharmaceuticals | 2009 |
GABA(A) receptors mediate the attenuating effects of a 5-HT(3) receptor antagonist on methamphetamine-induced behavioral sensitization in mice.
Topics: Amphetamine-Related Disorders; Analysis of Variance; Animals; Apomorphine; Autoradiography; Behavior, Animal; Benzazepines; Brain Mapping; Dopamine Agonists; Drug Interactions; Flunitrazepam; GABA Modulators; Male; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Protein Binding; Raclopride; Receptors, GABA-A; Serotonin Antagonists; Tritium; Tropanes | 2010 |
A comparative evaluation of the dopamine D(2/3) agonist radiotracer [11C](-)-N-propyl-norapomorphine and antagonist [11C]raclopride to measure amphetamine-induced dopamine release in the human striatum.
Topics: Adult; Amphetamine; Apomorphine; Carbon Radioisotopes; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Humans; Male; Middle Aged; Positron-Emission Tomography; Raclopride; Young Adult | 2010 |
D2 receptor occupancy in conscious rat brain is not significantly distinguished with [3H]-MNPA, [3H]-(+)-PHNO, and [3H]-raclopride.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Brain; CHO Cells; Cricetinae; Cricetulus; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Male; Oxazines; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, G-Protein-Coupled | 2010 |
Differential effects of stress on [¹¹C]raclopride and [¹¹C]MNPA binding to striatal D₂/D₃ dopamine receptors: a PET study in conscious monkeys.
Topics: Animals; Apomorphine; Brain; Carbon Radioisotopes; Hydrocortisone; Macaca mulatta; Male; Positron-Emission Tomography; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Stress, Physiological | 2011 |
Modulatory influence of dopamine receptors on consolidation of object recognition memory.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Apomorphine; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Quinpirole; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Recognition, Psychology; Retention, Psychology; Signal Transduction; Statistics, Nonparametric; Time Factors | 2011 |
Effects of L-DOPA on nigral dopamine neurons and local field potential: comparison with apomorphine and muscimol.
Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Electrophysiological Phenomena; Evoked Potentials; GABA Agonists; Levodopa; Male; Muscimol; Neurons; Parkinson Disease, Secondary; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Substantia Nigra | 2011 |
Test-retest reproducibility of dopamine D2/3 receptor binding in human brain measured by PET with [11C]MNPA and [11C]raclopride.
Topics: Adult; Apomorphine; Brain; Data Interpretation, Statistical; Humans; Male; Positron-Emission Tomography; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results | 2013 |
Early life stress causes refractoriness to haloperidol-induced catalepsy.
Topics: Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Catecholamines; Cerebral Cortex; Dopamine Agonists; Female; Globus Pallidus; Haloperidol; Male; Maternal Exposure; Maternal-Fetal Relations; Pregnancy; Proto-Oncogene Proteins c-fos; Raclopride; Rats; Receptors, Dopamine; Stress, Physiological; Subthalamic Nucleus; Ventral Thalamic Nuclei | 2013 |
Feeding condition and the relative contribution of different dopamine receptor subtypes to the discriminative stimulus effects of cocaine in rats.
Topics: Animals; Apomorphine; Benzamides; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Electroshock; Food Deprivation; Indoles; Lisuride; Male; Piperidines; Pyridines; Quinpirole; Raclopride; Rats, Sprague-Dawley; Reinforcement, Psychology | 2014 |
Relation between microPET imaging and rotational behavior in a parkinsonian rat model induced by medial forebrain bundle axotomy.
Topics: Animals; Apomorphine; Axotomy; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Functional Laterality; Male; Medial Forebrain Bundle; Parkinson Disease; Raclopride; Radionuclide Imaging; Rats; Rats, Wistar; Stereotyped Behavior; Substantia Nigra; Time Factors; Tyrosine 3-Monooxygenase | 2014 |
Pharmacologic MRI (phMRI) as a tool to differentiate Parkinson's disease-related from age-related changes in basal ganglia function.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Aging; Animals; Apomorphine; Basal Ganglia; Benzazepines; Diagnosis, Differential; Dopamine Agents; Female; Macaca mulatta; Magnetic Resonance Imaging; Motor Activity; Parkinson Disease, Secondary; Raclopride | 2015 |
The significance of rotational behavior and sensitivity of striatal dopamine receptors in hemiparkinsonian rats: A comparative study of lactacystin and 6-OHDA.
Topics: Acetylcysteine; Amphetamine; Animals; Apomorphine; Benzazepines; Central Nervous System Stimulants; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Functional Laterality; Male; Motor Activity; Oxidopamine; Parkinsonian Disorders; Pars Compacta; Raclopride; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Rotation | 2017 |
Affinity States of Striatal Dopamine D2 Receptors in Antipsychotic-Free Patients with Schizophrenia.
Topics: Adult; Antipsychotic Agents; Apomorphine; Brain Mapping; Corpus Striatum; Female; Humans; Male; Positron-Emission Tomography; Raclopride; Radioligand Assay; Radiopharmaceuticals; Receptors, Dopamine D2; Schizophrenia; Statistics as Topic; Young Adult | 2017 |