apomorphine has been researched along with metoclopramide in 96 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 73 (76.04) | 18.7374 |
1990's | 10 (10.42) | 18.2507 |
2000's | 8 (8.33) | 29.6817 |
2010's | 5 (5.21) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Lombardo, F; Obach, RS; Waters, NJ | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Colombo, M; Moragues, J; Prieto, J; Roberts, DJ; Salazar, W; Spickett, RG; Vega, A | 1 |
Sharman, DF | 1 |
Kebabian, JW; Kebabian, PR | 1 |
Beckett, PR; Berga, P; Roberts, DJ | 1 |
Elliott, PN; Huizing, G; Jenner, P; Marsden, CD; Miller, R | 1 |
Berry, MS; MacDonald, JF | 1 |
Colombo, M; Llupia, J; Roberts, DJ; Salazar, W | 1 |
Roufogalis, BD; Thornton, M; Wade, DN | 1 |
Dolphin, A; Jenner, P; Marsden, CD; Pycock, C; Tarsy, D | 1 |
Kojima, T; Koyama, Y; Marumo, H; Nakamura, N; Shiozaki, S | 1 |
Angrist, B; Gershon, S; Shopsin, B; Thompson, H | 1 |
Ahtee, L | 1 |
Marsden, CD; Pycock, C; Tarsy, D | 1 |
Cianchetti, C; Corsini, GU; Mangoni, A; Zompo, MD | 1 |
Destrade, C; Messier, C; Mrabet, O | 2 |
Imamura, M; Naitoh, T; Wassersug, RJ | 1 |
Heaton, JP; Varrin, SJ | 1 |
Awouters, FH; Megens, AA; Niemegeers, CJ | 1 |
Baldwin, BA; Ebenezer, IS; Forsling, ML; Parrott, RF | 1 |
Protais, P; Vasse, M | 1 |
Ljungberg, T | 1 |
el-Dardiry, SA; el-Hawash, SA; el-Khawass, EM; Ibrahim, EA; Shafik, RM | 1 |
Felício, LF; Nasello, AG; Palermo-Neto, J | 2 |
Ekker, M; Sourkes, TL | 1 |
Barone, FC; Fine, CF; Fowler, PJ; Grous, M; Lombardi, DM; Ormsbee, HS; Phyall, WB; Rush, JA | 1 |
Ståhle, L; Ungerstedt, U | 1 |
Hand, TH; Kasser, RJ; Wang, RY | 1 |
Hadley, MS; King, FD; McClelland, CM | 1 |
Starr, BS; Starr, MS | 1 |
Buyniski, JP; Crenshaw, RR; Gylys, JA; Nicolosi, WD; Wright, RN | 1 |
Kruk, ZL; Millar, J; Stamford, JA | 1 |
Cunningham, FJ; Howles, CM; Knight, PG | 1 |
Miner, WD; Sanger, GJ; Turner, DH | 1 |
Cubeddu, LX; Lovenberg, T; Suarez-Roca, H | 1 |
Andrews, PL; Hawthorn, J; Ostler, KJ | 1 |
Henke, PG; Ray, A; Sullivan, RM | 1 |
Frussa-Filho, R; Palermo-Neto, J | 1 |
Clopton, JK; Curtin, JC; Gordon, JH; Koller, WC | 1 |
Ozaki, L; Stern, N; Tuck, ML | 1 |
Molloy, AG; Waddington, JL | 1 |
Gerber, R; Gerhardt, S; Liebman, JM | 1 |
Hietala, J; Koulu, M; Scheinin, M; Syvälahti, E | 1 |
Fink, H; Morgenstern, R | 1 |
Bertagna, A; Godano, A; Goffi, S; Massara, F; Molinatti, GM; Tangolo, D | 1 |
Hackman, R; Neuvonen, PJ; Pentikainen, P; Vapaatalo, H | 1 |
Tuncer, M | 1 |
Andén, NE; Grabowska-Andén, M | 1 |
Bracha, HS; Davis, KL; Kendler, KS | 1 |
Anderson, RJ; Carp, JS | 1 |
Worms, P | 1 |
Azuma, H; Iwai, K; Kikuta, M; Liu, HJ; Oshino, N; Sato, K | 1 |
Morgan, M | 1 |
Dunn, AJ; Guild, AL | 1 |
Groĭsman, SD; Karevina, TG; Khokholia, VP | 1 |
Gershon, S; Lautin, A; Rotrosen, J; Stanley, M; Wazer, D | 1 |
Laville, C; Margarit, J | 1 |
Helmreich, I; Hertting, G; Reimann, W; Starke, K | 1 |
Chang, JP; Nahorniak, CS; Peter, RE; Sokolowska, M | 1 |
Bernardi, MM; Palermo-Neto, J; Saban, R | 1 |
Uppal, RP | 1 |
Bendesky, RJ; Hichens, M; King, SW; Mangel, AW; Martin, GE; Remy, DC; Robinson, JL; Taylor, DA; Williams, M; Yarbrough, GG | 1 |
Costall, B; Gunning, SJ; Naylor, RJ; Simpson, KH | 1 |
Dashputra, PG; Hemnani, TJ | 1 |
Benson, DI; Kuhn, CM; Meyerson, LR; Stanley, M; Virgilio, J; Wazer, D | 1 |
Rotrosen, J; Stanley, M; Wazer, DE | 1 |
Bloxham, CA; Cross, AJ; Ferrier, IN | 1 |
Lang, WJ; Rechtman, MP; Woodman, OL | 1 |
Janssen, PA; Niemegeers, CJ; Wauquier, A | 1 |
Fang, VS | 1 |
Dubocovich, ML; Weiner, N | 1 |
Kim, HS; Liebman, J; Welch, JJ | 1 |
Alander, T; Andén, NE; Grabowska-Andén, M | 1 |
Gershon, S; Lautin, A; Rotorsen, J; Stanley, M; Wazer, D | 1 |
Conway, SB; Gietzen, DW; Hope, WG; Thompson-Reece, MA; Woolley, DE | 1 |
Farooqui, T; Harrold, MW; Matsumoto, K; Miller, DD; Sriburi, A; Uretsky, N | 1 |
Itoh, Z; Iwanaga, Y; Miyashita, N; Morikawa, K; Saito, T | 1 |
Frussa-Filho, R; Palermo-Neto, J; Vital, MB | 1 |
Mok, EY; Munro, AD | 1 |
Fang, X; Liu, YX; Minami, M; Wang, L; Yue, W; Zhang, F | 1 |
Lahlou, S | 1 |
JUSTIN-BESANCON, L; LAVILLE, C; THOMINET, M | 1 |
JUSTIN-BESANCON, L; LAVILLE, C | 1 |
BOISSIER, JR; FICHELLE-PAGNY, J; LWOFF, JM; SIMON, P | 1 |
Auff, E; Kotzailias, N; Sycha, T; Tribl, GG; Zeitlhofer, J | 1 |
Liu, ZT; Wang, L; Yang, ZH; Yue, W; Zhang, F | 1 |
Axelsson, P; Lövqvist, A; Thörn, SE; Wattwil, L; Wattwil, M | 1 |
Fukui, H; Iwachido, T; Miwa, E; Suyama, Y | 1 |
4 review(s) available for apomorphine and metoclopramide
Article | Year |
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DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Brain dopamine metabolism and behavioral problems of farm animals.
Topics: Animals; Animals, Domestic; Antipsychotic Agents; Apomorphine; Behavior; Brain; Dopamine; Guinea Pigs; Humans; Metoclopramide; Stereotyped Behavior; Swine | 1978 |
Control of intragastric pH and volume.
Topics: Anesthesia, General; Animals; Antacids; Apomorphine; Benzimidazoles; Child; Female; Gastric Acid; Gastric Emptying; Histamine H2 Antagonists; Humans; Hydrogen-Ion Concentration; Metoclopramide; Parasympatholytics; Pneumonia, Aspiration; Pregnancy; Premedication; Stomach; Suction | 1984 |
The benzamides: evidence for action at dopamine receptors--shortcomings of current models.
Topics: Animals; Apomorphine; Benzamides; Humans; Metoclopramide; Models, Biological; Receptors, Dopamine; Serotonin; Stereotyped Behavior | 1982 |
2 trial(s) available for apomorphine and metoclopramide
Article | Year |
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Apomorphine in idiopathic restless legs syndrome: an exploratory study.
Topics: Administration, Oral; Adult; Aged; Apomorphine; Dopamine Agonists; Dopamine Antagonists; Drug Therapy, Combination; Electromyography; Female; Humans; Male; Metoclopramide; Middle Aged; Naloxone; Narcotic Antagonists; Restless Legs Syndrome; Treatment Outcome | 2005 |
Betamethasone does not prevent nausea and vomiting induced by the dopamine-agonist apomorphine.
Topics: Adult; Apomorphine; Betamethasone; Dopamine Agonists; Dopamine Antagonists; Female; Glucocorticoids; Humans; Male; Metoclopramide; Nausea; Pain Measurement; Reference Values; Severity of Illness Index; Time Factors; Treatment Outcome; Vasopressins; Vomiting | 2006 |
90 other study(ies) available for apomorphine and metoclopramide
Article | Year |
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Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Synthesis and pharmacological properties of a series of antidopaminergic piperidyl benzamides.
Topics: Animals; Apomorphine; Benzamides; Catalepsy; Depression, Chemical; Dextroamphetamine; Dopamine; Female; Humans; Male; Metoclopramide; Mice; Piperidines; Rats; Stereotyped Behavior; Structure-Activity Relationship | 1977 |
Lergotrile and lisuride: in vivo dopaminergic agonists which do not stimulate the presynaptic dopamine autoreceptor.
Topics: Animals; Apomorphine; Corpus Striatum; Ergolines; In Vitro Techniques; Lisuride; Male; Metoclopramide; Rats; Receptors, Dopamine; Tyrosine 3-Monooxygenase | 1978 |
[Antagonism of pre- and postsynaptic dopamine receptors by clebopride and related orthopramides].
Topics: Animals; Apomorphine; Benzamides; Dopamine Antagonists; Drug Interactions; Metoclopramide; Mice; Piperidines; Sulpiride; Synapses | 1979 |
Substituted benzamides as cerebral dopamine antagonists in rodents.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Behavior, Animal; Benzamides; Brain; Catalepsy; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Male; Metoclopramide; Mice; Receptors, Dopamine; Sulpiride | 1977 |
Further identification of multiple responses mediated by dopamine in the CNS of Planorbis corneus.
Topics: Animals; Apomorphine; Central Nervous System; Dopamine; Evoked Potentials; Fluphenazine; Ganglia; Haloperidol; In Vitro Techniques; Lysergic Acid Diethylamide; Metoclopramide; Mollusca; Tubocurarine | 1978 |
[Comparison of antiapomorphinic activity of metoclopramide, sulpiride and clebopride in the rat and dog].
Topics: Administration, Oral; Animals; Apomorphine; Benzamides; Dogs; Injections, Intravenous; Metoclopramide; Piperidines; Rats; Sulpiride | 1978 |
Specificity of the dopamine sensitive adenylate cyclase for antipsychotic antagonists.
Topics: Adenylyl Cyclases; Animals; Apomorphine; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Activation; Haloperidol; Male; Metoclopramide; Rats; Sulpiride | 1976 |
Pharmacological evidence for cerebral dopamine receptor blockade by metoclopramide in rodents.
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Humans; Male; Metoclopramide; Mice; Mice, Inbred Strains; Motor Activity; Parkinson Disease; Pimozide; Rats; Receptors, Drug; Reserpine; Rotation; Stereotyped Behavior; Substantia Nigra | 1975 |
Pharmacological studies of caerulein. II. The possibility of mediation through the central nervous system.
Topics: Animals; Apomorphine; Atropine; Blood Pressure; Central Nervous System; Ceruletide; Chlorpromazine; Copper; Dogs; Female; Gallbladder; Gastrointestinal Motility; Male; Metoclopramide; Splanchnic Nerves; Sulfates; Vagotomy; Vomiting | 1975 |
Clinical studies with dopamine-receptor stimulants.
Topics: Adult; Apomorphine; Blood Pressure; Dopamine; Female; Hallucinations; Humans; Male; Metoclopramide; Middle Aged; Piperazines; Piribedil; Receptors, Drug; Schizophrenia; Schizophrenia, Paranoid; Schizophrenic Psychology; Stimulation, Chemical; Vomiting | 1975 |
Inhibition by apomorphine of the metoclopramide-induced catalepsy and increase in striatal homovanillic acid content.
Topics: Animals; Apomorphine; Body Temperature; Brain; Catalepsy; Corpus Striatum; Dopamine; Female; Homovanillic Acid; Humans; Metoclopramide; Norepinephrine; Phenylacetates; Rats; Stimulation, Chemical; Time Factors | 1975 |
Inhibition of circling behavior by neuroleptic drugs in mice with unilateral 6-hydroxydopamine lesions of the striatum.
Topics: Animals; Apomorphine; Basal Ganglia Diseases; Behavior; Biogenic Amines; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Chlorpromazine; Clozapine; Corpus Striatum; Dextroamphetamine; Diazepam; Dopamine; Haloperidol; Humans; Hydroxydopamines; Levodopa; Male; Metoclopramide; Mice; Motor Activity; Pentobarbital; Phenoxybenzamine; Pimozide; Promethazine; Stereotyped Behavior; Tranquilizing Agents | 1975 |
Therapeutical efficacy of a combination of apomorphine with sulpiride or metoclopramide in Parkinsonism.
Topics: Adult; Apomorphine; Drug Therapy, Combination; Haloperidol; Humans; Male; Metoclopramide; Parkinson Disease; Sleep; Sulpiride; Vomiting | 1976 |
Locomotor bias produced by intra-accumbens injection of dopamine agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dextroamphetamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Haloperidol; Injections; Male; Metoclopramide; Mice; Mice, Inbred BALB C; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior | 1992 |
Interspecific variation in the emetic response of anurans.
Topics: Animals; Antimony; Anura; Apomorphine; Copper; Copper Sulfate; Emetics; Metoclopramide; Potassium; Species Specificity; Stress, Mechanical; Tartrates | 1991 |
Metoclopramide decreases apomorphine-induced yawning and penile erection.
Topics: Animals; Apomorphine; Male; Metoclopramide; Penile Erection; Rats; Rats, Inbred Strains; Receptors, Dopamine; Yawning | 1991 |
General pharmacology of the four gastrointestinal motility stimulants bethanechol, metoclopramide, trimebutine, and cisapride.
Topics: Animals; Apomorphine; Bethanechol Compounds; Cisapride; Conditioning, Operant; Diarrhea; Dogs; Gastric Emptying; Gastrointestinal Agents; Gastrointestinal Motility; Metoclopramide; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Species Specificity; Trimebutine; Vomiting | 1991 |
Hormonal effects of apomorphine and cholecystokinin in pigs: modification of the response to cholecystokinin by a dopamine antagonist (metoclopramide) and a kappa opioid agonist (PD117302).
Topics: Animals; Apomorphine; Cholecystokinin; Dopamine Antagonists; Feeding Behavior; Female; Hydrocortisone; Lypressin; Male; Metoclopramide; Pyrroles; Swine; Thiophenes | 1991 |
[Circling behavior produced by the unilateral intra-accumbens injection of dopaminergic agonist and two dopaminergic antagonists in mice].
Topics: Animals; Apomorphine; Behavior, Animal; Haloperidol; Male; Metoclopramide; Mice; Mice, Inbred BALB C; Motor Activity; Nucleus Accumbens; Septal Nuclei | 1989 |
Potentiation of apomorphine-induced stereotyped behaviour by acute treatment with dopamine depleting agents: a potential role for an increased stimulation of D1 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; alpha-Methyltyrosine; Amisulpride; Animals; Apomorphine; Corpus Striatum; Cyclic AMP; Dopamine Antagonists; Drug Synergism; In Vitro Techniques; Male; Methyltyrosines; Metoclopramide; Mice; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Sulpiride | 1989 |
Dopamine D-2 antagonists reverse apomorphine-induced decreased water intake in the rat: prediction of antipsychotic drugs with few extrapyramidal side-effects?
Topics: Animals; Antipsychotic Agents; Apomorphine; Domperidone; Dose-Response Relationship, Drug; Drinking Behavior; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1989 |
Synthesis of some 2-(3,4-dimethoxy-phenyl)-1,3-propanediamines as potential dopaminergic agents.
Topics: Animals; Apomorphine; Brain Chemistry; Chemical Phenomena; Chemistry; Diamines; Dopamine; Dopamine Agents; Membranes; Metoclopramide; Mitochondria; Monoamine Oxidase; Norepinephrine; Rats | 1989 |
Perinatal bromopride treatment: effects on motor activity and stereotyped behavior of offspring.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Female; Lactation; Male; Metoclopramide; Motor Activity; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Stereotyped Behavior; Time Factors | 1989 |
Differential effects of thioridazine, clozapine and metoclopramide on the induction of adrenomedullary enzymes by apomorphine.
Topics: Adrenal Medulla; Animals; Apomorphine; Clozapine; Corpus Striatum; Dibenzazepines; Enzyme Induction; Male; Metoclopramide; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Substantia Nigra; Thioridazine; Tyrosine 3-Monooxygenase | 1985 |
DA1 receptor mediates dopamine-induced relaxation of opossum lower esophageal sphincter in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Aporphines; Benzazepines; Deoxyepinephrine; Domperidone; Dopamine; Dose-Response Relationship, Drug; Esophagogastric Junction; Female; In Vitro Techniques; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Opossums; Receptors, Dopamine | 1986 |
Effects of neuroleptic drugs on the inhibition of exploratory behaviour induced by a low dose of apomorphine: implications for the identity of dopamine receptors.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Drug Interactions; Exploratory Behavior; Flupenthixol; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1986 |
Effects of acute thioridazine, metoclopramide and SCH 23390 on the basal activity of A9 and A10 dopamine cells.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Thioridazine | 1987 |
Substituted benzamides with conformationally restricted side chains. 2. Indolizidine derivatives as central dopamine receptor antagonists.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Chemical Phenomena; Chemistry; Gastrointestinal Motility; Indolizines; Male; Metoclopramide; Mice; Molecular Conformation; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Structure-Activity Relationship | 1988 |
Behavioural interactions involving D1 and D2 dopamine receptors in non-habituated mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Drug Interactions; Haloperidol; Male; Metoclopramide; Mice; Motor Activity; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1987 |
BMY-25801, an antiemetic agent free of D2-dopamine receptor antagonist properties.
Topics: Animals; Antiemetics; Apomorphine; Cisplatin; Cyclophosphamide; Dogs; Doxorubicin; Female; Ferrets; Male; Metoclopramide; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Reflex; Vomiting | 1988 |
Ascorbic acid does not modulate stimulated dopamine release: in vivo voltammetric data in the rat.
Topics: Animals; Apomorphine; Ascorbic Acid; Corpus Striatum; Dopamine; Electric Stimulation; In Vitro Techniques; Medial Forebrain Bundle; Metoclopramide; Neural Pathways; Rats; Rats, Inbred Strains; Substantia Nigra; Synaptic Transmission | 1985 |
Evidence that opioid peptides and dopamine participate in the suckling-induced release of prolactin in the ewe.
Topics: Animals; Apomorphine; Dopamine; Endorphins; Female; Lactation; Metoclopramide; Naloxone; Pituitary Gland, Anterior; Pregnancy; Prolactin; Sheep; Thyrotropin-Releasing Hormone | 1986 |
Evidence that 5-hydroxytryptamine3 receptors mediate cytotoxic drug and radiation-evoked emesis.
Topics: Animals; Antineoplastic Agents; Apomorphine; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Cyclophosphamide; Domperidone; Doxorubicin; Ferrets; Male; Metoclopramide; Receptors, Serotonin; Vomiting; Whole-Body Irradiation | 1987 |
Comparative dopamine-cholinergic mechanisms in the olfactory tubercle and the striatum: effects of metoclopramide.
Topics: Acetylcholine; Amphetamine; Animals; Apomorphine; Benzazepines; Corpus Striatum; Dopamine; Electric Stimulation; Male; Metoclopramide; Olfactory Bulb; Rabbits; Receptors, Dopamine; Reserpine | 1987 |
The role of the abdominal visceral innervation and 5-hydroxytryptamine M-receptors in vomiting induced by the cytotoxic drugs cyclophosphamide and cis-platin in the ferret.
Topics: Animals; Antiemetics; Apomorphine; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Carnivora; Cisplatin; Cyclophosphamide; Female; Ferrets; Male; Metoclopramide; Receptors, Serotonin; Splanchnic Nerves; Vagotomy; Vomiting | 1988 |
Effects of intra-amygdalar dopamine agonists and antagonists on gastric stress lesions in rats.
Topics: Amygdala; Animals; Apomorphine; Cold Temperature; Dopamine; Dopamine Antagonists; Haloperidol; Male; Metoclopramide; Rats; Rats, Inbred Strains; Restraint, Physical; Stomach Ulcer; Stress, Psychological | 1988 |
Effects of single and long-term metoclopramide administration on open field and stereotyped behavior of rats.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substance Withdrawal Syndrome | 1988 |
Dopaminergic supersensitivity after long-term bromopride treatment.
Topics: Animals; Apomorphine; Dopamine; Drug Administration Schedule; Female; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Sex Factors; Stereotyped Behavior | 1987 |
Chronic autoreceptor blockade and neuroleptic-induced dopamine receptor hypersensitivity.
Topics: Animals; Apomorphine; Dose-Response Relationship, Drug; Haloperidol; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Synapses | 1987 |
Evidence for dopaminergic binding sites in the human adrenal cortex.
Topics: Adrenal Cortex; Adult; Aged; Apomorphine; Binding, Competitive; Bromocriptine; Domperidone; Dopamine; Epinephrine; Female; Humans; Ketanserin; Male; Metoclopramide; Middle Aged; Receptors, Dopamine; Spiperone; Sulpiride; Time Factors | 1986 |
Sniffing, rearing and locomotor responses to the D-1 dopamine agonist R-SK&F 38393 and to apomorphine: differential interactions with the selective D-1 and D-2 antagonists SCH 23390 and metoclopramide.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Drug Interactions; Humans; Locomotion; Male; Metoclopramide; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Stereotyped Behavior | 1985 |
SCH 23390 dissociated from conventional neuroleptics in apomorphine climbing and primate acute dyskinesia models.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Benzimidazoles; Chlorpromazine; Chlorprothixene; Drug Synergism; Dyskinesia, Drug-Induced; Haloperidol; Male; Metoclopramide; Mice; Motor Activity; Saimiri; Stereotyped Behavior | 1985 |
Neuroendocrine aspects in monitoring of dopaminergic drugs in man.
Topics: Apomorphine; Bromocriptine; Growth Hormone; Homovanillic Acid; Humans; Levodopa; Male; Metoclopramide; Monitoring, Physiologic; Neurosecretory Systems; Prolactin; Receptors, Dopamine; Schizophrenia; Selegiline; Time Factors | 1985 |
Sulpiride blocks postsynaptic dopamine receptors in the nucleus accumbens.
Topics: Animals; Apomorphine; Exploratory Behavior; Male; Metoclopramide; Motor Activity; Nucleus Accumbens; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride; Tiapamil Hydrochloride | 1985 |
Effect of metoclopramide, domperidone and apomorphine on GH secretion in children and adolescents.
Topics: Adolescent; Age Factors; Apomorphine; Child; Domperidone; Female; Growth Hormone; Humans; Male; Metoclopramide; Receptors, Dopamine | 1985 |
Inhibition of the apomorphine gnawing compulsion by amantadine.
Topics: Amantadine; Animals; Apomorphine; Behavior, Animal; Chlorpromazine; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Drug Synergism; Male; Metoclopramide; Rats | 1973 |
The interaction between metoclopramide and dopaminergic agonists at the level of sympathetic ganglion.
Topics: Action Potentials; Animals; Apomorphine; Cats; Dopamine; Drug Interactions; Ganglia, Sympathetic; Hexamethonium; Hexamethonium Compounds; Metoclopramide; Norepinephrine; Receptors, Dopamine | 1984 |
Drug effects on pre- and postsynaptic dopamine receptors.
Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dopamine; Humans; Male; Metoclopramide; Rats; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Synapses; Time Factors | 1980 |
Dopamine autoreceptor and postsynaptic receptor blocking potency of neuroleptics.
Topics: Animals; Antipsychotic Agents; Apomorphine; Fluphenazine; Haloperidol; Male; Metoclopramide; Mice; Molindone; Motor Activity; Receptors, Dopamine; Sulpiride; Synapses | 1982 |
Dopamine receptor-mediated depression of spinal monosynaptic transmission.
Topics: Action Potentials; Animals; Apomorphine; Cats; Ergolines; Female; Haloperidol; Lisuride; Male; Metoclopramide; Phentolamine; Receptors, Dopamine; Spinal Cord; Synapses; Synaptic Transmission | 1982 |
Behavioral pharmacology of the benzamides as compared to standard neuroleptics.
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Benzamides; Catalepsy; Humans; Male; Metoclopramide; Mice; Oxotremorine; Rats; Rats, Inbred Strains; Stereotyped Behavior; Sulpiride | 1982 |
[Suppressive effects of lisuride on the synthesis, release and metabolism of dopamine in rat brain].
Topics: Animals; Apomorphine; Brain; Depression, Chemical; Dihydroergotoxine; Dopamine; Ergolines; Female; Haloperidol; Histocytochemistry; Homovanillic Acid; Lisuride; Metoclopramide; Nucleus Accumbens; Olfactory Bulb; Rats; Sulpiride; Tyrosine 3-Monooxygenase | 1982 |
Dopamine involvement in ACTH-induced grooming behavior.
Topics: Adrenocorticotropic Hormone; Animals; Apomorphine; Behavior, Animal; Butaclamol; Catalepsy; Dopamine; Grooming; Humans; Injections, Intraventricular; Male; Metoclopramide; Mice; Pimozide | 1982 |
[Role of dopamine receptors in the mechanism of formation of stress-induced stomach lesions].
Topics: Animals; Apomorphine; Female; Gastrointestinal Hemorrhage; Humans; Levodopa; Male; Metoclopramide; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stomach Ulcer; Stress, Psychological; Sulpiride; Vagotomy | 1984 |
Discrimination of functionally heterogeneous receptor subpopulations: antipsychotic and antidopaminergic properties of metoclopramide [proceedings].
Topics: Animals; Apomorphine; Binding Sites; Humans; Metoclopramide; Rats; Receptors, Dopamine; Receptors, Neurotransmitter; Schizophrenia; Spiperone | 1981 |
[Pharmacodynamics of alizapride (author's transl)].
Topics: Animals; Antiemetics; Apomorphine; Behavior, Animal; Central Nervous System; Dogs; Ergoloid Mesylates; Guinea Pigs; Male; Metoclopramide; Mice; Mice, Inbred Strains; Pyrrolidines; Rabbits; Rats; Rats, Inbred Strains | 1982 |
Are presynaptic dopamine autoreceptors and postsynaptic dopamine receptors in the rabbit caudate nucleus pharmacologically different?
Topics: Acetylcholine; Animals; Apomorphine; Atropine; Carbachol; Caudate Nucleus; Choline; Dopamine; Electric Stimulation; Female; Male; Membrane Potentials; Metoclopramide; Molindone; Physostigmine; Rabbits; Receptors, Dopamine; Sulpiride; Synapses; Synaptic Transmission | 1982 |
Effects of catecholaminergic agonists and antagonists on serum gonadotropin concentrations and ovulation in goldfish: evidence for specificity of dopamine inhibition of gonadotropin secretion.
Topics: Animals; Apomorphine; Bromocriptine; Cyprinidae; Dopamine; Female; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins; Metoclopramide; Octopamine; Ovulation; Phentolamine; Pimozide; Propranolol | 1984 |
Kinetic analysis of central nervous system supersensitivity induced in rats by long-term haloperidol administration. I. pA2 determination.
Topics: Animals; Apomorphine; Brain; Dose-Response Relationship, Drug; Haloperidol; Humans; Kinetics; Male; Metoclopramide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior | 1984 |
Effect of metoclopramide pretreatment on apomorphine induced cage climbing behaviour.
Topics: Animals; Apomorphine; Humans; Male; Metoclopramide; Mice; Stereotyped Behavior | 1984 |
L-646,462, a cyproheptadine-related antagonist of dopamine and serotonin with selectivity for peripheral systems.
Topics: Animals; Apomorphine; Cyproheptadine; Domperidone; Dopamine Antagonists; Gastrointestinal Motility; Haloperidol; Homovanillic Acid; Male; Metoclopramide; Prolactin; Receptors, Serotonin; Serotonin Antagonists | 1984 |
A central site of action for benzamide facilitation of gastric emptying.
Topics: Animals; Apomorphine; Atropine; Benzamides; Female; Gastric Emptying; Guinea Pigs; Male; Metoclopramide; Prazosin; Propranolol | 1983 |
Potentiation of the psychotropic effect of chlorpromazine by metoclopramide.
Topics: Animals; Apomorphine; Behavior, Animal; Chlorpromazine; Drug Synergism; Male; Metoclopramide; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains | 1983 |
Lack of potency of metoclopramide's metabolites in various dopaminergic models.
Topics: Animals; Apomorphine; Dopamine; Fluphenazine; Haloperidol; Homovanillic Acid; Humans; Male; Metoclopramide; Prolactin; Rats; Rats, Inbred Strains; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes | 1983 |
Dopamine D1 receptors in human parathyroid gland: in vitro and in vivo studies.
Topics: Adult; Apomorphine; Flupenthixol; Humans; Male; Metoclopramide; Parathyroid Glands; Parathyroid Hormone; Prolactin; Receptors, Dopamine; Schizophrenia; Thioxanthenes | 1983 |
A comparison of the responses to some dopamine-receptor agonists and antagonists in the isolated perfused rat kidney.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Bromocriptine; Dopamine; Dopamine Antagonists; Female; In Vitro Techniques; Kidney; Male; Metoclopramide; Rats; Receptors, Dopamine; Regional Blood Flow; Vasodilation | 1980 |
Neuropharmacological comparison between domperidone and metoclopramide.
Topics: Animals; Antiemetics; Apomorphine; Brain; Dogs; Domperidone; Electroencephalography; Female; Humans; Male; Metoclopramide; Self Stimulation; Stereotyped Behavior | 1981 |
Pharmacological difference of L-dopa, apomorphine, and bromocriptine against metoclopramide.
Topics: Animals; Apomorphine; Bromocriptine; Levodopa; Male; Metoclopramide; Prolactin; Rats; Serotonin | 1981 |
Modulation of the stimulation-evoked release of [3H]dopamine in the rabbit retina.
Topics: Animals; Apomorphine; Calcium; Dopamine; Electric Stimulation; Flupenthixol; In Vitro Techniques; Metoclopramide; Rabbits; Retina; Stereoisomerism; Sulpiride; Tritium | 1981 |
Amphetamine-induced increases in dopaminergic single cell firing rate after haloperidol pretreatment. Correlation with extrapyramidal side effects.
Topics: Animals; Apomorphine; Brain; Clozapine; Dextroamphetamine; Dopamine; Drug Interactions; Extrapyramidal Tracts; Haloperidol; Male; Metoclopramide; Neurons; Rats; Substantia Nigra; Thioridazine | 1980 |
Metoclopramide and sulpiride as selective blocking agents of pre- and postsynaptic dopamine receptors.
Topics: Aminooxyacetic Acid; Animals; Apomorphine; Atropine; Corpus Striatum; Dopamine; Dopamine Antagonists; Male; Metoclopramide; Norepinephrine; Prazosin; Rats; Receptors, Dopamine; Rotation; Sulpiride | 1980 |
Chronic treatment with metoclopramide induces behavioral supersensitivity to apomorphine and enhances specific binding of 3H-spiroperidol to rat striata.
Topics: Animals; Apomorphine; Behavior, Animal; Binding, Competitive; Body Weight; Butyrophenones; Corpus Striatum; Male; Metoclopramide; Rats; Spiperone; Time Factors | 1980 |
Dopaminergic stimulation of estrogen receptor binding in vivo: a reexamination.
Topics: Adrenalectomy; Animals; Apomorphine; Brain; Bromocriptine; Cell Membrane; Cell Nucleus; Ditiocarb; Dopamine; Estradiol; Female; Hypothalamus; Kinetics; Metoclopramide; Ovariectomy; Pituitary Gland, Anterior; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Estrogen | 1994 |
The interaction of ammonium, sulfonium, and sulfide analogues of metoclopramide with the dopamine D2 receptor.
Topics: Animals; Apomorphine; Benzamides; Brain; Drug Interactions; Metoclopramide; Mice; Quaternary Ammonium Compounds; Receptors, Dopamine D2; Structure-Activity Relationship; Sulfonium Compounds | 1993 |
Gastroprokinetic effect of a new benzamide derivative itopride and its action mechanisms in conscious dogs.
Topics: Animals; Antiemetics; Apomorphine; Benzamides; Benzyl Compounds; Dogs; Domperidone; Dopamine Antagonists; Female; Gastrointestinal Motility; Male; Metoclopramide; Vomiting | 1996 |
Monosialoganglioside increased the in vivo affinity of D2 receptors for apomorphine in supersensitive rats.
Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; G(M1) Ganglioside; Haloperidol; Kinetics; Metoclopramide; Rats; Receptors, Dopamine D2; Stereotyped Behavior; Substance Withdrawal Syndrome | 1998 |
Effects of dopaminergic drugs on locomotor activity in teleost fish of the genus Oreochromis (Cichlidae): involvement of the telencephalon.
Topics: Animals; Apomorphine; Chlorpromazine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Metoclopramide; Motor Activity; Nasal Mucosa; Telencephalon; Tilapia | 1998 |
[A new vomiting animal model--mink].
Topics: Animals; Antiemetics; Apomorphine; Cisplatin; Copper Sulfate; Disease Models, Animal; Male; Metoclopramide; Mink; Ondansetron; Vomiting | 2003 |
Enhanced hypotensive response to intravenous apomorphine in chronic spinalized, conscious rats: role of spinal dopamine D(1) and D(2) receptors.
Topics: Animals; Apomorphine; Benzazepines; Blood Pressure; Consciousness; Domperidone; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Hypotension; Injections, Spinal; Male; Metoclopramide; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Spinal Cord Injuries; Thoracic Vertebrae | 2003 |
[METOCLOPRAMIDE AND ITS HOMOLOGUES. INTRODUCTION TO THEIR BIOLOGICAL STUDY].
Topics: Animals; Antiemetics; Apomorphine; Central Nervous System; Chlorpromazine; Dogs; Lagomorpha; Metoclopramide; Mice; Pharmacology; Rabbits; Rats; Research; Toxicology | 1964 |
[ANTIEMETIC ACTION OF METOCLOPRAMIDE WITH RESPECT TO APOMORPHINE AND HYDERGINE].
Topics: Antiemetics; Apomorphine; Benzamides; Cardiovascular Agents; Chlorpromazine; Dihydroergotoxine; Diphenhydramine; Dogs; Ergoloid Mesylates; Ergot Alkaloids; Metoclopramide; Oxytocics; Pharmacology; Prochlorperazine; Research; Toxicology | 1964 |
[PSYCHOLEPTIC ACTION OF METOCLOPRAMIDE].
Topics: Acetylcholine; Antiemetics; Apomorphine; Barbiturates; Behavior, Animal; Blood Pressure; Blood Pressure Determination; Dogs; Epinephrine; Humans; Male; Metoclopramide; Mice; Norepinephrine; Pharmacology; Procainamide; Psychopharmacology; Rats; Research; Seminal Vesicles; Toxicology | 1964 |
Value of mink vomit model in study of anti-emetic drugs.
Topics: Animals; Antiemetics; Apomorphine; Cisplatin; Copper Sulfate; Disease Models, Animal; Enterochromaffin Cells; Immunohistochemistry; Male; Metoclopramide; Mink; Ondansetron; Random Allocation; Reproducibility of Results; Serotonin; Vomiting | 2006 |
Possible involvement of β₁ receptors in various emetogen-induced increases in salivary amylase activity in rats.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Amylases; Animals; Antiemetics; Apomorphine; Atenolol; Butoxamine; Cisplatin; Depression, Chemical; Emetics; Isoproterenol; Lithium Chloride; Male; Metoclopramide; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Saliva | 2011 |