apomorphine has been researched along with 4-butyrolactone in 77 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 60 (77.92) | 18.7374 |
1990's | 17 (22.08) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Roth, RH; Walters, JR | 2 |
Morgenroth, VH; Roth, RH; Walters, JR | 1 |
Persson, SA | 2 |
Cott, J; Engel, J | 1 |
Nowycky, MC; Roth, RH | 1 |
Andén, NE; Wachtel, H | 1 |
Engel, J; Liljequist, S | 1 |
Demarest, KT; Moore, KE | 1 |
Costentin, J; Marcais, H; Protais, P | 1 |
Algeri, S; Cattabeni, F; Di Giulio, AM; Galli, CL; Groppetti, A; Maggi, A; Ponzio, F | 1 |
Gianutsos, G; Moore, KE; Thornburg, JE | 1 |
Agnati, L; Everitt, BJ; Fuxe, K; Hökfelt, T; Ljungdahl, A; Perez de la Mora, M | 1 |
Baudry, M; Costentin, J; Marcais, H; Martres, MP; Protais, P; Schwartz, JC | 1 |
Kehr, W | 2 |
Ekman, A; Eriksson, E | 1 |
Carboni, E; Di Chiara, G; Tanda, G | 1 |
Harsing, LG; Vizi, ES | 1 |
Abraini, JH; Raharison, L; Rostain, JC | 1 |
Evans, DL; Figur, LM; Huff, RM; Lahti, RA; Moon, MW | 1 |
Brown, EE; Cumming, P; Damsma, G; Fibiger, HC | 1 |
De Vries, JB; Duran, R; Westerink, BH | 1 |
Coward, DM; Dixon, AK; Enz, A; Karobath, M; Shearman, G; Urwyler, S; White, TG | 1 |
Ali, SF; Gough, BJ; Holson, RR; Newport, GD; Scalzo, FM | 1 |
Jackson, DM; Ross, SB | 1 |
Giambalvo, CT | 1 |
de Vries, JB; Dijkstra, D; Grol, CJ; Horn, AS; Mulder, TB; Wiechers, JW | 1 |
Carlsson, A; Nissbrandt, H; Pileblad, E | 1 |
Salama, AI; Saller, CF | 1 |
Barton, AC; Demarest, KT; Moore, KE | 1 |
Carlsson, A; Johansson, AM; Magnusson, T; Svensson, K | 1 |
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Namba, Y | 1 |
Bean, AJ; Bunney, BS; Nestler, EJ; Roth, RH; Shepard, PD | 1 |
Galloway, MP; Roth, RH; Wolf, ME | 1 |
Andersson, B; Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, AM; Sanchez, D; Svensson, K; Wikström, H | 1 |
Kaneno, S; Takahashi, R; Watanabe, A | 1 |
Anderson, CM; Ely, TD; Kilts, CD; Nishita, JK | 1 |
DeWald, HA; Hawkins, ES; Heffner, TG; Meltzer, LT; Pugsley, TA; Reynolds, DM; Wise, LD | 1 |
Altar, CA; Kim, HS; Wood, PL | 1 |
Nomura, Y; Sekihara, S; Suda, H; Watanabe, H | 1 |
Fukuda, K; Kashihara, K; Otsuki, S; Sato, M | 1 |
Adler, CH; Bohmaker, K; Friedhoff, AJ; Goldstein, M; Helmer-Matyjek, E; Meller, E | 1 |
Andersson, B; Eriksson, E; Hjorth, S | 1 |
De Vries, JB; Dijkstra, D; Hazelhoff, B; Horn, AS; Mulder, TB | 1 |
Carlsson, A; Clark, D; Hjorth, S | 1 |
Spaan, SJ; van Es, TP; Westerink, BH | 1 |
Goldstein, M | 1 |
Jin, GZ; Li, JH; Wang, XL; Yu, LP | 1 |
Roth, RH | 1 |
Demarest, KT; Lawson-Wendling, KL; Moore, KE | 1 |
Fadda, F; Gessa, GL; Marcou, M; Mosca, E; Rossetti, Z | 1 |
De Vries, JB; Dijkstra, D; Horn, AS; Renkema, RJ; Tepper, PG; Van Oene, JC | 1 |
de Vries, JB; Horn, AS; van Oene, JC | 1 |
Dougherty, GG; Ellinwood, EH | 1 |
Dougherty, GG; Ellinwood, EH; Gonzalez, AE | 1 |
Bannon, MJ; Bunney, EB; Roth, RH; Skirboll, LR; Zigun, JR | 1 |
Haubrich, DR; Martin, GE; Williams, M | 2 |
Argiolas, A; Fadda, F; Gessa, GL; Marcou, M; Melis, MR; Porceddu, ML | 1 |
Spaan, SJ; Westerink, BH | 1 |
Bannon, MJ; Bunney, EB; Reinhard, JF; Roth, RH | 1 |
Conway, PG; Uretsky, NJ | 1 |
Clineschmidt, BV; Haubrich, DR; Jones, JH; Martin, GE; Williams, M; Yarbrough, GG | 1 |
Broxterman, HJ; Noach, EL; van Valkenburg, CF; Wijling, A | 1 |
de Vries, JB; Horn, AS; Sumners, C | 1 |
McMillen, BA | 1 |
Hirose, T; Kikuchi, T; Miwa, T; Morita, S; Oshiro, Y; Tottori, K; Uwahodo, Y | 1 |
Basham, DA; Bohmaker, K; Goldstein, M; Meller, E | 1 |
Bartoszyk, GD; Seyfried, CA | 1 |
Nagahama, M; Sakurai, J | 1 |
Carruba, MO; da Prada, M; Imhof, R; Nisoli, E; Scherschlicht, R; Tonello, C | 1 |
Caprathe, BW; Christoffersen, CL; Corbin, AE; Jaen, JC; Meltzer, LT; Ninteman, FW; Pugsley, TA; Serpa, KA; Shih, YH; Whetzel, SZ | 1 |
Bristow, LJ; Cook, GP; Gay, JC; Hutson, PH; Kulagowski, JJ; Landon, L; Murray, F; Saywell, KL; Young, L | 1 |
Kikuchi, T; Kurahashi, N; Nishi, T; Oshiro, Y; Sato, S; Tanaka, T; Tottori, K; Uwahodo, Y | 1 |
Carr, KD; Garcia-Espana, A; Goldstein, M; Haycock, JW; Lee, KY; Lew, JY; Meller, E | 1 |
3 review(s) available for apomorphine and 4-butyrolactone
Article | Year |
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Dopaminergic neurons - alteration in the sensitivity of tyrosine hydroxylase to inhibition by endovenous dopamine after cessation of impulse flow.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Haloperidol; Male; Neurons; Rats; Receptors, Adrenergic; Synapses; Synaptic Transmission; Tyrosine 3-Monooxygenase | 1976 |
Regulatory mechanisms of dopamine biosynthesis at the tyrosine hydroxylase step.
Topics: 4-Butyrolactone; Animals; Apomorphine; Bucladesine; Corpus Striatum; Dopamine; Enzyme Activation; Haloperidol; Phosphorylation; Receptors, Dopamine; Synapses; Synaptosomes; Tyrosine 3-Monooxygenase | 1984 |
CNS dopamine autoreceptors: distribution, pharmacology, and function.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Brain; Calmodulin; Dopamine; Dopamine Antagonists; Drug Tolerance; Electrophysiology; Homovanillic Acid; Limbic System; Mesencephalon; Methylation; Methyltyrosines; Neurons; Receptors, Dopamine; Stress, Physiological; Telencephalon; Tissue Distribution | 1984 |
74 other study(ies) available for apomorphine and 4-butyrolactone
Article | Year |
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Dopaminergic neurons--alteration in the kinetic properties of tyrosine hydroxylase after cessation of impulse flow.
Topics: 4-Butyrolactone; Animals; Apomorphine; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Egtazic Acid; Female; Kinetics; Male; Median Eminence; Neurons; Olfactory Bulb; Piperazines; Pterins; Rats; Receptors, Adrenergic; Substantia Nigra; Synapses; Synaptic Transmission; Tyrosine 3-Monooxygenase | 1976 |
Dopaminergic neurons: an in vivo system for measuring drug interactions with presynaptic receptors.
Topics: 4-Butyrolactone; Action Potentials; Animals; Antipsychotic Agents; Apomorphine; Butyrophenones; Corpus Striatum; Dopamine; Drug Interactions; Male; Neurons; Phenothiazines; Rats; Receptors, Dopamine; Synaptic Transmission | 1976 |
The effect of LSD and 2-bromo LSD on the striatal DOPA accumulation after decarboxylase inhibition in rats.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Corpus Striatum; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Lysergic Acid Diethylamide; Male; Neural Pathways; Rats; Reserpine; Substantia Nigra; Time Factors | 1977 |
Suppression by GABAergic drugs of the locomotor stimulation induced by morphine, amphetamine, and apomorphine: evidence for both pre- and post-synaptic inhibition of catecholamine systems.
Topics: 4-Butyrolactone; Aminobutyrates; Aminooxyacetic Acid; Animals; Apomorphine; Brain; Clonidine; Corpus Striatum; Dextroamphetamine; Diencephalon; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Limbic System; Methyltyrosines; Mice; Morphine; Motor Activity; Naloxone; Norepinephrine; Reserpine; Tryptophan Hydroxylase; Tyrosine 3-Monooxygenase | 1977 |
Nonstriatal dopaminergic neurons: role of presynaptic receptors in the modulation of transmitter synthesis.
Topics: 4-Butyrolactone; Animals; Apomorphine; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Kinetics; Limbic System; Neurons; Rats; Receptors, Dopamine; Synapses; Tyrosine 3-Monooxygenase | 1977 |
Increase in the turnover of brain dopamine by stimulation of muscarinic receptors outside the dopamine nerve terminals.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Atropine; Atropine Derivatives; Brain; Corpus Striatum; Dopamine; Hydrazines; Male; Nerve Endings; Norepinephrine; Oxotremorine; Physostigmine; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1977 |
Effect of morphine on the accumulation of DOPA after decarboxylase inhibition in the rat.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Dihydroxyphenylalanine; DNA; Haloperidol; Male; Morphine; Naloxone; Rats; Receptors, Drug; Reserpine; Time Factors | 1979 |
Attenuation of the gamma-butyrolactone-induced increase in DOPA accumulation by chronic ethanol administration.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Corpus Striatum; Dihydroxyphenylalanine; Ethanol; Furans; Limbic System; Male; Rats | 1979 |
Comparison of dopamine synthesis regulation in the terminals of nigrostriatal, mesolimbic, tuberoinfundibular and tuberohypophyseal neurons.
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Benzyl Alcohols; Dihydroxyphenylalanine; Dopamine; Hydrazines; Hypothalamo-Hypophyseal System; Male; Median Eminence; Nialamide; Olfactory Bulb; Piribedil; Pituitary Gland, Posterior; Rats; Reserpine | 1979 |
Hypersensitivity of the climbing behaviour response to apomorphine induced by a short depression of dopaminergic neurone activity.
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Cycloheximide; Dopamine; Hydroxybutyrates; Male; Mice; Motor Activity; Neurons; Sodium Oxybate | 1979 |
Significance of dopamine metabolites in the evaluation of drugs acting on dopaminergic neurons.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Cocaine; Dextroamphetamine; Dopamine; Homovanillic Acid; Male; Methyltyrosines; Neurons; Nomifensine; Pargyline; Rats; Tyramine | 1978 |
Differential actions of dopamine agonists and antagonists on the gamma-butyrolactone-induced in mouse brain dopamine.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Dopamine; Drug Interactions; Furans; Haloperidol; Male; Mice; Pimozide; Piribedil; Receptors, Dopamine | 1976 |
Action of beta(4-chlorphenyl)GABA, gamma-hydroxybutyrolactone, and apomorphine on central dopamine neurons.
Topics: 4-Butyrolactone; Aminobutyrates; Animals; Apomorphine; Baclofen; Brain; Castration; Dopamine; Estrogens; Female; Furans; Neurons; Piribedil; Rats; Receptors, Dopamine; Sexual Behavior, Animal; Time Factors | 1977 |
Long-term changes in the sensitivity of pre-and postsynaptic dopamine receptors in mouse striatum evidenced by behavioural and biochemical studies.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dose-Response Relationship, Drug; Haloperidol; Homovanillic Acid; Hydroxydopamines; Male; Mice; Motor Activity; Piribedil; Receptors, Dopamine; Time Factors | 1977 |
3-Methoxytyramine as an indicator of impulse-induced dopamine release in rat brain in vivo.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Denervation; Dopamine; Haloperidol; Male; Methyltyrosines; Pargyline; Rats; Tyramine | 1976 |
Effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline on the prolactin suppression induced by a series of full and partial dopamine D2 receptor agonists in male rats.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Dopamine Agents; Ergolines; Levodopa; Male; Piperidines; Prolactin; Quinolines; Rats; Rats, Sprague-Dawley | 1992 |
Extracellular striatal concentrations of endogenous 3,4-dihydroxyphenylalanine in the absence of a decarboxylase inhibitor: a dynamic index of dopamine synthesis in vivo.
Topics: 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Carboxy-Lyases; Chromatography, High Pressure Liquid; Colorimetry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Extracellular Matrix; Haloperidol; Male; Methyltyrosines; Rats; Rats, Sprague-Dawley; Tetrodotoxin | 1992 |
Alpha 2-adrenoceptors are not involved in the regulation of striatal glutamate release: comparison to dopaminergic inhibition.
Topics: 4-Butyrolactone; Animals; Apomorphine; Berberine; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Drug Interactions; Glutamates; Glutamic Acid; Haloperidol; Hydrazines; Hydroxydopamines; Male; Oxidopamine; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Secretory Rate; Synaptic Transmission; Yohimbine | 1991 |
Long-term depression in striatal dopamine release monitored by in vivo voltammetry in free moving rats.
Topics: 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Cerebral Ventricles; Corpus Striatum; Dopamine; Electrochemistry; Injections, Intraventricular; Kinetics; Male; Methyltyrosines; Rats; Rats, Inbred Strains; Tyrosine 3-Monooxygenase | 1991 |
Pre- and postsynaptic dopaminergic activities of U-86170F.
Topics: 4-Butyrolactone; Administration, Oral; Aminoquinolines; Animals; Apomorphine; Dopamine Agents; Injections, Intraperitoneal; Male; Mice; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Synapses | 1991 |
Interstitial 3-methoxytyramine reflects striatal dopamine release: an in vivo microdialysis study.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Antidepressive Agents; Apomorphine; Bupropion; Corpus Striatum; Dialysis; Dopamine; Haloperidol; Homovanillic Acid; Kinetics; Male; Propiophenones; Rats; Rats, Inbred Strains; Tetrodotoxin | 1991 |
Use of microdialysis for monitoring tyrosine hydroxylase activity in the brain of conscious rats.
Topics: 1-Methyl-4-phenylpyridinium; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Brain; Chromatography, High Pressure Liquid; Consciousness; Dialysis; Dihydroxyphenylalanine; Haloperidol; Male; Methyltyrosines; Monitoring, Physiologic; Rats; Rats, Inbred Strains; Tyrosine 3-Monooxygenase | 1990 |
Partial dopamine-agonistic and atypical neuroleptic properties of the amino-ergolines SDZ 208-911 and SDZ 208-912.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Avoidance Learning; Behavior, Animal; Catalepsy; Dopamine; Dopamine Agents; Ergolines; Female; Male; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1990 |
Chronic prenatal haloperidol exposure: lack of effect on presynaptic dopamine autoreceptors.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain Chemistry; Caudate Nucleus; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Female; Haloperidol; Hydrazines; Nucleus Accumbens; Olfactory Bulb; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Dopamine; Synapses | 1989 |
Kinetic properties of the in vivo accumulation of 3H-(-)-N-n-propylnorapomorphine in mouse brain.
Topics: 4-Butyrolactone; Animals; Apomorphine; Benzazepines; Brain Chemistry; Corpus Striatum; Dextroamphetamine; Dopamine Agents; In Vitro Techniques; Male; Methylphenidate; Mice; Motor Activity; Olfactory Bulb; Reserpine; Synapses | 1989 |
Protein kinase C and dopamine release--III. Effect of dopamine depleting drugs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Benzazepines; Calcium-Calmodulin-Dependent Protein Kinases; Dopamine; Dopamine Agents; Elongation Factor 2 Kinase; Ergolines; Male; Methyltyrosines; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Quinpirole; Rats; Sulpiride | 1989 |
Further in vitro and in vivo studies with the putative presynaptic dopamine agonist N,N-dipropyl-7-hydroxy-2-aminotetralin.
Topics: 4-Butyrolactone; Animals; Apomorphine; Binding, Competitive; Corpus Striatum; Dopamine; In Vitro Techniques; Male; Motor Activity; Naphthalenes; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Spiperone; Substantia Nigra; Synaptosomes; Tetrahydronaphthalenes | 1987 |
Evidence for dopamine release and metabolism beyond the control of nerve impulses and dopamine receptors in rat substantia nigra.
Topics: 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Corpus Striatum; Dopamine; Haloperidol; Male; Methyltyrosines; Nerve Tissue Proteins; Pargyline; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Tropolone | 1985 |
3-Methoxytyramine accumulation: effects of typical neuroleptics and various atypical compounds.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Buspirone; Carbazoles; Chlorpromazine; Clozapine; Corpus Striatum; Dopamine; Dopamine Antagonists; Fluphenazine; Haloperidol; Male; Molindone; Pargyline; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Regression Analysis | 1986 |
Differential action of bromocriptine on nigrostriatal versus mesolimbic dopaminergic neurons.
Topics: 4-Butyrolactone; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Ergolines; Limbic System; Male; Nucleus Accumbens; Olfactory Bulb; Prolactin; Rats; Time Factors | 1987 |
(+)-AJ 76 and (+)-UH 232: central stimulants acting as preferential dopamine autoreceptor antagonists.
Topics: 4-Butyrolactone; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Brain; Male; Methyltyrosines; Motor Activity; Naphthalenes; Neurotransmitter Agents; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Tetrahydronaphthalenes | 1986 |
Relationship between receptor occupancy and response at striatal dopamine autoreceptors.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Homeostasis; Hydrazines; Levodopa; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
The effects of pertussis toxin on autoreceptor-mediated inhibition of dopamine synthesis in the rat striatum.
Topics: 4-Butyrolactone; Adenosine Diphosphate Ribose; Animals; Apomorphine; Chromatography, High Pressure Liquid; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; GTP-Binding Proteins; Hydrazines; Male; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Virulence Factors, Bordetella | 1988 |
Regulation of dopamine synthesis in the medial prefrontal cortex is mediated by release modulating autoreceptors: studies in vivo.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Feedback; Frontal Lobe; Hydrazines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
(+)-UH 232 and (+)-UH 242: novel stereoselective dopamine receptor antagonists with preferential action on autoreceptors.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Male; Motor Activity; Naphthalenes; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Serotonin; Stereoisomerism; Tetrahydronaphthalenes | 1986 |
Alteration of striatal dopaminergic functions implicated in methamphetamine-induced reverse tolerance in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Drug Tolerance; Homovanillic Acid; Male; Methamphetamine; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
Absence of synthesis-modulating nerve terminal autoreceptors on mesoamygdaloid and other mesolimbic dopamine neuronal populations.
Topics: 4-Butyrolactone; Amygdala; Animals; Apomorphine; Dihydroxyphenylalanine; Dopamine; Hydrazines; Limbic System; Male; Medial Forebrain Bundle; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
6- and 8-hydroxy-3,4-dihydro-3-(dipropylamino)-2H-1-benzopyrans. Dopamine agonists with autoreceptor selectivity.
Topics: 4-Butyrolactone; Animals; Apomorphine; Benzopyrans; Brain; Chromans; Dopamine; Haloperidol; In Vitro Techniques; Neurons; Rats; Receptors, Dopamine; Reserpine | 1988 |
Presynaptic inhibition of nigrostriatal dopamine release in the mouse: lack of cross tolerance between apomorphine, GBL and CGS 10746B.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Drug Tolerance; Efferent Pathways; Furans; Male; Mice; Substantia Nigra; Thiazepines | 1988 |
D-1 type of dopamine autoreceptors are not involved in the regulation of dopamine synthesis in the striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 4-Butyrolactone; Animals; Apomorphine; Benzazepines; Corpus Striatum; Dopamine; Male; Mice; Receptors, Dopamine | 1987 |
Haloperidol prevents the methamphetamine-induced apomorphine subsensitivity of dopamine metabolism in rat striatum.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Drug Combinations; Haloperidol; Male; Methamphetamine; Rats; Rats, Inbred Strains | 1987 |
Receptor reserve at striatal dopamine autoreceptors: implications for selectivity of dopamine agonists.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Indoles; Levodopa; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
Stereoselective inhibition of prolactin secretion by (-)-HW-165, a novel 3-PPP congener; further support for similarities between central DA autoreceptors and pituitary lactotroph DA receptors.
Topics: 4-Butyrolactone; Animals; Apomorphine; Depression, Chemical; Male; Phenanthrenes; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism | 1986 |
N-methyl,N-propargyl-2-aminotetralins:novel dopamine agonists with monoamine oxidase inhibiting properties.
Topics: 4-Butyrolactone; Alkynes; Animals; Apomorphine; Brain; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Female; Humans; In Vitro Techniques; Mice; Monoamine Oxidase Inhibitors; Motor Activity; Naphthalenes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Tetrahydronaphthalenes | 1985 |
(+)- and (-)-3-PPP exhibit different intrinsic activity at striatal dopamine autoreceptors controlling dopamine synthesis.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Isomerism; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter | 1984 |
Effects of drugs interfering with dopamine and noradrenaline biosynthesis on the endogenous 3,4-dihydroxyphenylalanine levels in rat brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Brain; Chlorpromazine; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dopamine; Female; Homovanillic Acid; Norepinephrine; Rats; Rats, Inbred Strains; Tissue Distribution; Tyrosine 3-Monooxygenase | 1982 |
[Effect of tetrahydroberberine on blockade of pre- and postsynaptic dopamine receptors (author's transl)].
Topics: 4-Butyrolactone; Animals; Apomorphine; Berberine; Berberine Alkaloids; Corpus Striatum; Hypnotics and Sedatives; Levodopa; Rats; Receptors, Dopamine | 1982 |
d-Amphetamine and gamma-butyrolactone alteration of dopamine synthesis in the terminals of nigrostriatal and mesolimbic neurons. Possible role of various autoreceptor sensitivities.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain Chemistry; Corpus Striatum; Dextroamphetamine; Dihydroxyphenylalanine; Dopamine; Furans; Haloperidol; Limbic System; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra | 1983 |
Evidence for dopamine autoreceptors in mesocortical dopamine neurons.
Topics: 4-Butyrolactone; Adrenergic Fibers; Animals; Apomorphine; Caudate Nucleus; Dihydroxyphenylalanine; Frontal Lobe; Haloperidol; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1984 |
In vivo dopamine autoreceptor selectivity appears to be critically dependent upon the aromatic hydroxyl position in a series of N,N-disubstituted 2-aminotetralins.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Dihydroxyphenylalanine; Female; Male; Mice; Motor Activity; Naphthalenes; Piribedil; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Structure-Activity Relationship; Tetrahydronaphthalenes | 1984 |
The effectiveness of yohimbine in blocking rat central dopamine autoreceptors in vivo.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Dopamine; Female; Haloperidol; Homovanillic Acid; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Tetrahydronaphthalenes; Yohimbine | 1984 |
Influence of gamma-butyrolactone on behavior due to dopaminergic drugs.
Topics: 4-Butyrolactone; Animals; Apomorphine; Dextroamphetamine; Dose-Response Relationship, Drug; Drug Interactions; Furans; Humans; Male; Methylphenidate; Rats; Rats, Inbred Strains; Stereotyped Behavior; Time Factors | 1983 |
gamma-Butyrolactone effects on behavior induced by dopamine agonists.
Topics: 4-Butyrolactone; Amphetamine; Animals; Apomorphine; Bicuculline; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Male; Methylphenidate; Rats; Receptors, Dopamine; Stereotyped Behavior | 1983 |
Presynaptic dopamine receptors: insensitivity to kainic acid and the development of supersensitivity following chronic haloperidol.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Haloperidol; Kainic Acid; Male; Pyrrolidines; Rats; Receptors, Dopamine | 1980 |
A pharmacological comparison of 6,7-dihydroxy-2-dimethylaminotetralin (TL-99) and N-n-propyl-3-(3-hydroxyphenyl)piperidine with (3-PPP) selected dopamine agonists.
Topics: 4-Butyrolactone; Animals; Apomorphine; Cell Membrane; Corpus Striatum; Female; Humans; Hydroxydopamines; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes | 1982 |
Delayed inhibition of dopamine synthesis by gamma-butyrolactone and baclofen: dopamine autoreceptor supersensitivity?
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Furans; Haloperidol; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors | 1982 |
On the significance of endogenous 3-methoxytyramine for the effects of centrally acting drugs on dopamine release in the rat brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Benztropine; Brain; Chlorpromazine; Dextroamphetamine; Dopamine; Female; Haloperidol; Homovanillic Acid; Kinetics; Morphine; Nomifensine; Oxotremorine; Rats; Rats, Inbred Strains; Reserpine | 1982 |
Unique response to antipsychotic drugs is due to absence of terminal autoreceptors in mesocortical dopamine neurones.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Brain; Brain Mapping; Dopamine; Dopamine Antagonists; Haloperidol; Male; Rats; Receptors, Dopamine | 1982 |
Role of striatal dopaminergic receptors in amphetamine-induced behavioral facilitation.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Amphetamine; Animals; Apomorphine; Behavior, Animal; Brain; Corpus Striatum; Homovanillic Acid; Humans; Male; Molindone; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior | 1982 |
Potent dopamine agonist activity of a novel ergoline, 6-ethyl-9-oxaergoline (EOE).
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Dopamine; Ergolines; Female; Humans; Hypothermia; Mice; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Stereotyped Behavior | 1982 |
Cross-tolerance of dopamine metabolism to baclofen, gamma-butyrolactone and HA-966 in the striatum and olfactory tubercle of the rat.
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Central Nervous System Depressants; Corpus Striatum; Dopamine; Drug Tolerance; Male; Olfactory Bulb; Pyrrolidinones; Rats | 1981 |
3-Methoxytyramine and normetanephrine as indicators of dopamine and noradrenaline release in mouse brain in vivo.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Bromocriptine; Dextroamphetamine; Dopamine; Kinetics; Lisuride; Male; Mice; Norepinephrine; Normetanephrine; Pargyline; Receptors, Dopamine | 1981 |
Pharmacological profiles of the putative dopamine autoreceptor agonists 3-PPP and TL-99.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Dogs; Dopamine; Female; Male; Mice; Motor Activity; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Tetrahydronaphthalenes | 1981 |
Behavioural and neurochemical studies on apomorphine-induced hypomotility in mice.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain Chemistry; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Motor Activity; Norepinephrine; Time Factors | 1981 |
On the mechanism of morphine action on rat striatal dopamine metabolsim.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Female; Haloperidol; In Vitro Techniques; Morphine; Naloxone; Rats | 1980 |
7-(4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butyloxy)-3,4-dihydro-2(1H)-quinolinone (OPC-14597), a new putative antipsychotic drug with both presynaptic dopamine autoreceptor agonistic activity and postsynaptic D2 receptor antagonistic activity.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Aripiprazole; Catalepsy; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxidopamine; Piperazines; Presynaptic Terminals; Quinolones; Radioligand Assay; Rats; Reserpine; Spiperone; Stereotyped Behavior; Synapses; Tritium | 1995 |
Evidence that striatal synthesis-inhibiting autoreceptors are dopamine D3 receptors.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine Agents; Dose-Response Relationship, Drug; Levodopa; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereoisomerism | 1993 |
Sensitivity of dopamine D2 receptors following long-term treatment with roxindole.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Down-Regulation; Drug Interactions; Haloperidol; Indoles; Injections, Intraperitoneal; Male; Oxindoles; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior | 1994 |
Effect of drugs acting on the central nervous system on the lethality in mice of Clostridium perfringens epsilon toxin.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Bacterial Toxins; Barbiturates; Brain; Brain Chemistry; Butyrophenones; Calcium-Binding Proteins; Catechol O-Methyltransferase; Catecholamines; Central Nervous System Agents; Clostridium perfringens; Diazepam; Iodine Radioisotopes; Male; Mice; Mice, Inbred Strains; Monoamine Oxidase; Phenothiazines; Reserpine; Type C Phospholipases | 1993 |
Neurochemical and behavioral evidence that Ro 41-9067 is a selective presynaptic dopamine receptor agonist.
Topics: 4-Butyrolactone; Adenylyl Cyclases; Amphetamine; Animals; Apomorphine; Biogenic Monoamines; Brain; Catalepsy; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Levodopa; Locomotion; Male; Motor Activity; Perfusion; Potassium; Quinolines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Serotonin; Stereotyped Behavior; Synapses; Tetrahydronaphthalenes; Time Factors; Tritium | 1993 |
Pharmacological profile of the dopamine partial agonist, (+/-)-PD 128483 and its enantiomers.
Topics: 4-Butyrolactone; Aminoquinolines; Amphetamine; Animals; Apomorphine; Avoidance Learning; Behavior, Animal; Cebus; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Male; Mice; Motor Activity; Neurons; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Saimiri; Serotonin; Stereoisomerism; Stereotyped Behavior; Stimulation, Chemical; Thiazoles | 1993 |
The behavioural and neurochemical profile of the putative dopamine D3 receptor agonist, (+)-PD 128907, in the rat.
Topics: 4-Butyrolactone; Animals; Apomorphine; Behavior, Animal; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Nucleus Accumbens; Oxazines; Rats; Rats, Sprague-Dawley | 1996 |
Novel antipsychotic agents with dopamine autoreceptor agonist properties: synthesis and pharmacology of 7-[4-(4-phenyl-1-piperazinyl)butoxy]-3,4-dihydro-2(1H)-quinolinone derivatives.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Aripiprazole; Brain; Catalepsy; Dihydroxyphenylalanine; Dopamine Agonists; Dopamine Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; Molecular Structure; Piperazines; Quinolones; Rats; Stereotyped Behavior; Structure-Activity Relationship | 1998 |
Increased site-specific phosphorylation of tyrosine hydroxylase accompanies stimulation of enzymatic activity induced by cessation of dopamine neuronal activity.
Topics: 4-Butyrolactone; Animals; Apomorphine; Binding Sites; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Enzyme Activation; GABA Modulators; Hydroxylation; In Vitro Techniques; Male; Neurons; Phosphorylation; Rats; Rats, Sprague-Dawley; Tyrosine; Tyrosine 3-Monooxygenase | 1999 |