Page last updated: 2024-09-05

antalarmin and yohimbine

antalarmin has been researched along with yohimbine in 4 studies

Compound Research Comparison

Studies
(antalarmin)
Trials
(antalarmin)
Recent Studies (post-2010)
(antalarmin)
Studies
(yohimbine)
Trials
(yohimbine)
Recent Studies (post-2010) (yohimbine)
1810765,893253532

Protein Interaction Comparison

ProteinTaxonomyantalarmin (IC50)yohimbine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0353
Cytochrome P450 2D6Homo sapiens (human)1.02
D(2) dopamine receptorHomo sapiens (human)2.06
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-2B adrenergic receptorHomo sapiens (human)0.0428
Alpha-2C adrenergic receptorHomo sapiens (human)0.0466
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.126
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-1D adrenergic receptorHomo sapiens (human)1.013
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.126
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.074
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)1.3
5-hydroxytryptamine receptor 6Homo sapiens (human)1.689

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Epstein, DH; Ghitza, UE; Gray, SM; Rice, KC; Shaham, Y1
Funk, D; Harding, S; Juzytsch, W; Lê, AD; Marinelli, PW; Rice, KC; Shaham, Y1
Coen, K; Funk, D; Lê, AD1
Bhat, S; Georgiou, P; Gould, TD; McCarthy, MM; Merchenthaler, IJ; Tracy, JK; Zanos, P1

Other Studies

4 other study(ies) available for antalarmin and yohimbine

ArticleYear
The anxiogenic drug yohimbine reinstates palatable food seeking in a rat relapse model: a role of CRF1 receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:10

    Topics: Adrenergic alpha-Antagonists; Animals; Anxiety; Behavior, Animal; Conditioning, Operant; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Extinction, Psychological; Food Preferences; Interpersonal Relations; Male; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Yohimbine

2006
The CRF1 receptor antagonist antalarmin attenuates yohimbine-induced increases in operant alcohol self-administration and reinstatement of alcohol seeking in rats.
    Psychopharmacology, 2007, Volume: 195, Issue:3

    Topics: Adrenergic alpha-Antagonists; Alcoholism; Animals; Behavior, Addictive; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Self Administration; Yohimbine

2007
The role of kappa opioid receptors in stress-induced reinstatement of alcohol seeking in rats.
    Brain and behavior, 2014, Volume: 4, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Behavior, Addictive; Behavior, Animal; Cues; Drug-Seeking Behavior; Ethanol; Male; Naltrexone; Narcotic Antagonists; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Receptors, Opioid, kappa; Self Administration; Stress, Physiological; Yohimbine

2014
Dopamine and Stress System Modulation of Sex Differences in Decision Making.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2018, Volume: 43, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Amygdala; Animals; Behavior, Animal; Decision Making; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Female; Male; Pyrimidines; Pyrroles; Quinpirole; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Receptors, Dopamine D2; Salicylamides; Sex Characteristics; Yohimbine

2018