Page last updated: 2024-09-05

antalarmin and mifepristone

antalarmin has been researched along with mifepristone in 4 studies

Compound Research Comparison

Studies
(antalarmin)
Trials
(antalarmin)
Recent Studies (post-2010)
(antalarmin)
Studies
(mifepristone)
Trials
(mifepristone)
Recent Studies (post-2010) (mifepristone)
1810766,5365951,758

Protein Interaction Comparison

ProteinTaxonomyantalarmin (IC50)mifepristone (IC50)
Glucocorticoid receptor Canis lupus familiaris (dog)0.0264
Bile salt export pumpHomo sapiens (human)2.02
Estrogen receptorHomo sapiens (human)4.311
Glucocorticoid receptorHomo sapiens (human)0.0249
Prostaglandin G/H synthase 1Ovis aries (sheep)0.0003
Progesterone receptorHomo sapiens (human)0.1347
Glucocorticoid receptorRattus norvegicus (Norway rat)0.774
Glucocorticoid receptorMus musculus (house mouse)0.0022
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0022
Mineralocorticoid receptor Homo sapiens (human)2.0938
Cytochrome P450 3A4Homo sapiens (human)9.5
Coagulation factor VIIHomo sapiens (human)0.0003
Androgen receptorHomo sapiens (human)0.2988
Cytochrome P450 2C8Homo sapiens (human)1.5
Cytochrome P450 2C9 Homo sapiens (human)4.9
Steroid 17-alpha-hydroxylase/17,20 lyase Rattus norvegicus (Norway rat)0.0016
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)0.555
Tissue factorHomo sapiens (human)0.0003
Androgen receptorRattus norvegicus (Norway rat)0.0083
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0014
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.0022
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0022
Prostaglandin G/H synthase 1Homo sapiens (human)0.0078
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0022
Substance-P receptorCavia porcellus (domestic guinea pig)0.0015
Mu-type opioid receptorHomo sapiens (human)2.457
Estrogen receptor betaHomo sapiens (human)1.528
Glucocorticoid receptorSus scrofa (pig)0.0153

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abid Masood, M; Bazin, M; Bunnage, ME; Fancy, SA; Farrant, E; Morao, I; Peakman, T; Perez, M1
Fischbach, PS; Rice, KC; Savit, AZ; Verhoeven, RE; Wood, SK; Woods, JH1
Brown, BE; Choi, EH; Crumrine, D; Demerjian, M; Elias, PM; Feingold, KR; Mauro, T1
Li, JS; Mei, YY1

Other Studies

4 other study(ies) available for antalarmin and mifepristone

ArticleYear
Lead diversification. Application to existing drug molecules: mifepristone 1 and antalarmin 8.
    Bioorganic & medicinal chemistry letters, 2012, Jan-01, Volume: 22, Issue:1

    Topics: Biomimetics; Carbon; Chemistry, Pharmaceutical; Chlorine; Drug Design; Humans; Hydrogen; Inhibitory Concentration 50; Metalloporphyrins; Metals; Microsomes, Liver; Mifepristone; Models, Chemical; Oxygen; Pyrimidines; Pyrroles; Structure-Activity Relationship

2012
Facilitation of cardiac vagal activity by CRF-R1 antagonists during swim stress in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:12

    Topics: Animals; Bradycardia; Cholinergic Antagonists; Corticotropin-Releasing Hormone; Death, Sudden, Cardiac; Disease Models, Animal; Exercise Tolerance; Fatigue; Heart Rate; Hypothalamo-Hypophyseal System; Hypothermia, Induced; Male; Mifepristone; Peptide Fragments; Psychomotor Agitation; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Swimming; Vagus Nerve; Vagus Nerve Diseases

2006
Glucocorticoid blockade reverses psychological stress-induced abnormalities in epidermal structure and function.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2006, Volume: 291, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Epidermis; Female; Glucocorticoids; Mice; Mice, Hairless; Mifepristone; Pyrimidines; Pyrroles; Skin Diseases; Stress, Psychological

2006
Involvements of stress hormones in the restraint-induced conditioned place preference.
    Behavioural brain research, 2013, Nov-01, Volume: 256

    Topics: Animals; Association Learning; Conditioning, Operant; Corticosterone; Male; Mifepristone; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Stress, Physiological

2013