Page last updated: 2024-09-05

antalarmin and cp 154526

antalarmin has been researched along with cp 154526 in 5 studies

Compound Research Comparison

Studies
(antalarmin)
Trials
(antalarmin)
Recent Studies (post-2010)
(antalarmin)
Studies
(cp 154526)
Trials
(cp 154526)
Recent Studies (post-2010) (cp 154526)
1810762005
181076129140

Protein Interaction Comparison

ProteinTaxonomyantalarmin (IC50)cp 154526 (IC50)
Corticotropin-releasing factor receptor 1Homo sapiens (human)0.0134

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aldrich, PE; Arvanitis, A; Bakthavatchalam, R; Beck, JP; Cheeseman, RS; Chidester, D; Chien, BM; Chorvat, RJ; Cocuzza, AJ; Curry, M; Fernandez, CH; Fitzgerald, LW; Gilligan, PJ; Hobbs, FW; Hodge, CN; Huang, SM; Klaczkiewicz, JD; Krenitsky, P; Rescinito, JP; Shen, HL; Wasserman, ZR; Wilde, RG; Wong, YN; Yarem, JA; Zaczek, R1
Chen, TK; Crowe, PD; Dyck, B; Grey, J; Grigoriadis, DE; Gross, RS; Guo, Z; Haddach, M; Kiankarimi, M; Lanier, M; Li, BF; Luo, Z; McCarthy, JR; Moorjani, M; Saunders, J; Sullivan, R; Tellew, JE; Williams, JP; Zamani-Kord, S; Zhang, X1
Gilligan, PJ; Robertson, DW; Zaczek, R1
Grigoriadis, DE; Heinrichs, SC; McCarthy, JR1
Houshyar, H; Hsin, LW; Jutkiewicz, EM; Rice, KC; Wood, SK; Woods, JH1

Reviews

2 review(s) available for antalarmin and cp 154526

ArticleYear
Corticotropin releasing factor (CRF) receptor modulators: progress and opportunities for new therapeutic agents.
    Journal of medicinal chemistry, 2000, May-04, Volume: 43, Issue:9

    Topics: Amino Acid Sequence; Animals; Humans; Molecular Sequence Data; Receptors, Corticotropin-Releasing Hormone; Stress, Physiological

2000
Recent advances with the CRF1 receptor: design of small molecule inhibitors, receptor subtypes and clinical indications.
    Current pharmaceutical design, 1999, Volume: 5, Issue:5

    Topics: Animals; Anxiety; Depression; Drug Design; Humans; Kinetics; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Seizures; Substance-Related Disorders

1999

Other Studies

3 other study(ies) available for antalarmin and cp 154526

ArticleYear
Synthesis, corticotropin-releasing factor receptor binding affinity, and pharmacokinetic properties of triazolo-, imidazo-, and pyrrolopyrimidines and -pyridines.
    Journal of medicinal chemistry, 1999, Mar-11, Volume: 42, Issue:5

    Topics: Administration, Oral; Animals; Biological Availability; Cell Line; Dogs; Humans; Mice; Pyridines; Pyrimidines; Rats; Receptors, Corticotropin-Releasing Hormone; Recombinant Proteins; Structure-Activity Relationship

1999
Design and synthesis of tricyclic imidazo[4,5-b]pyridin-2-ones as corticotropin-releasing factor-1 antagonists.
    Journal of medicinal chemistry, 2005, Aug-11, Volume: 48, Issue:16

    Topics: Administration, Oral; Adrenocorticotropic Hormone; Animals; Blood-Brain Barrier; CHO Cells; Corticotropin-Releasing Hormone; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Heterocyclic Compounds, 3-Ring; Humans; Imidazoles; Injections, Intravenous; Male; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stereoisomerism; Structure-Activity Relationship

2005
The effects of CRF antagonists, antalarmin, CP154,526, LWH234, and R121919, in the forced swim test and on swim-induced increases in adrenocorticotropin in rats.
    Psychopharmacology, 2005, Volume: 180, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Corticotropin-Releasing Hormone; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stress, Psychological; Swimming; Triazoles

2005