Page last updated: 2024-09-05

antalarmin and cocaine

antalarmin has been researched along with cocaine in 8 studies

Compound Research Comparison

Studies
(antalarmin)
Trials
(antalarmin)
Recent Studies (post-2010)
(antalarmin)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
18107632,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyantalarmin (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (50.00)29.6817
2010's3 (37.50)24.3611
2020's1 (12.50)2.80

Authors

AuthorsStudies
Mello, NK; Mendelson, JH; Negus, SS; Rice, KC1
Boutrel, B; Koob, GF; O'Dell, LE; Specio, SE; Wee, S; Zorrilla, EP1
Chowen, JA; de Lecea, L; Frago, LM; Huitron-Resendiz, S; PaƱeda, C; Picetti, R; Roberts, AJ1
Blendy, JA; Briand, L; Cleck, JN; Ecke, L; Kreibich, AS; Rice, KC1
Baker, DA; Blacktop, JM; Ferda, N; Graf, EN; Lee, G; Mantsch, JR; Seubert, C1
Baker, DA; Lim, Y; Makky, K; Mantsch, JR; McReynolds, JR; Thao, M; Vranjkovic, O1
Cosme, CV; Gutman, AL; LaLumiere, RT1
Christian, RJ; Fuchs, RA; Galliou, JMC; Grogan, SR; Ibarra, CK; Qi, S; Ritchie, JL; Savenkova, MI; Walters, JL1

Other Studies

8 other study(ies) available for antalarmin and cocaine

ArticleYear
Effects of the CRF1 antagonist antalarmin on cocaine self-administration and discrimination in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 85, Issue:4

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Corticotropin-Releasing Hormone; Discrimination, Psychological; Female; Hypothalamo-Hypophyseal System; Macaca mulatta; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Self Administration

2006
CRF(1) receptor antagonists attenuate escalated cocaine self-administration in rats.
    Psychopharmacology, 2008, Volume: 196, Issue:3

    Topics: Animals; Behavior, Addictive; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Self Administration; Time Factors

2008
Neuropeptide S reinstates cocaine-seeking behavior and increases locomotor activity through corticotropin-releasing factor receptor 1 in mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Apr-01, Volume: 29, Issue:13

    Topics: Analysis of Variance; Animals; Anxiety; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Extinction, Psychological; Injections, Intraventricular; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Neuropeptides; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Self Administration

2009
Stress-induced potentiation of cocaine reward: a role for CRF R1 and CREB.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:12

    Topics: Animals; Cocaine; Conditioning, Classical; Cyclic AMP Response Element-Binding Protein; Dopamine Uptake Inhibitors; Mice; Mice, Knockout; Nucleus Accumbens; Phosphorylation; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Reward; Septum of Brain; Space Perception; Stress, Psychological; Swimming; Time Factors

2009
Augmented cocaine seeking in response to stress or CRF delivered into the ventral tegmental area following long-access self-administration is mediated by CRF receptor type 1 but not CRF receptor type 2.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Aug-03, Volume: 31, Issue:31

    Topics: Aminopyridines; Analysis of Variance; Animals; Behavior, Addictive; Behavior, Animal; Cocaine; Conditioning, Operant; Corticotropin-Releasing Hormone; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Extinction, Psychological; Flavonoids; Food Preferences; Glucosides; Male; Peptide Fragments; Peptides, Cyclic; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Self Administration; Stress, Psychological; Ventral Tegmental Area

2011
Beta-2 adrenergic receptors mediate stress-evoked reinstatement of cocaine-induced conditioned place preference and increases in CRF mRNA in the bed nucleus of the stria terminalis in mice.
    Psychopharmacology, 2014, Volume: 231, Issue:20

    Topics: Adrenergic beta-Agonists; Animals; Behavior, Addictive; Clenbuterol; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Corticotropin-Releasing Hormone; Dopamine Uptake Inhibitors; Extinction, Psychological; Male; Mice; Pyrimidines; Pyrroles; Receptors, Adrenergic, beta-2; Receptors, Corticotropin-Releasing Hormone; Recurrence; Reward; Self Administration; Septal Nuclei; Stress, Psychological

2014
The Dorsal Agranular Insular Cortex Regulates the Cued Reinstatement of Cocaine-Seeking, but not Food-Seeking, Behavior in Rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:10

    Topics: Analysis of Variance; Animals; Baclofen; Cerebral Cortex; Cocaine; Conditioning, Operant; Cues; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Extinction, Psychological; Food; GABA Agonists; Male; Microinjections; Muscimol; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration

2015
Basolateral amygdala corticotropin-releasing factor receptor type 1 regulates context-cocaine memory strength during reconsolidation in a sex-dependent manner.
    Neuropharmacology, 2021, 12-01, Volume: 200

    Topics: Animals; Basolateral Nuclear Complex; Cocaine; Cocaine-Related Disorders; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Female; Male; Memory; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2021