Page last updated: 2024-09-05

anordiol and mifepristone

anordiol has been researched along with mifepristone in 6 studies

Compound Research Comparison

Studies
(anordiol)
Trials
(anordiol)
Recent Studies (post-2010)
(anordiol)
Studies
(mifepristone)
Trials
(mifepristone)
Recent Studies (post-2010) (mifepristone)
23016,5365951,758

Protein Interaction Comparison

ProteinTaxonomyanordiol (IC50)mifepristone (IC50)
Glucocorticoid receptor Canis lupus familiaris (dog)0.0264
Bile salt export pumpHomo sapiens (human)2.02
Estrogen receptorHomo sapiens (human)4.311
Glucocorticoid receptorHomo sapiens (human)0.0249
Prostaglandin G/H synthase 1Ovis aries (sheep)0.0003
Progesterone receptorHomo sapiens (human)0.1347
Glucocorticoid receptorRattus norvegicus (Norway rat)0.774
Glucocorticoid receptorMus musculus (house mouse)0.0022
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0022
Mineralocorticoid receptor Homo sapiens (human)2.0938
Cytochrome P450 3A4Homo sapiens (human)9.5
Coagulation factor VIIHomo sapiens (human)0.0003
Androgen receptorHomo sapiens (human)0.2988
Cytochrome P450 2C8Homo sapiens (human)1.5
Cytochrome P450 2C9 Homo sapiens (human)4.9
Steroid 17-alpha-hydroxylase/17,20 lyase Rattus norvegicus (Norway rat)0.0016
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)0.555
Tissue factorHomo sapiens (human)0.0003
Androgen receptorRattus norvegicus (Norway rat)0.0083
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0014
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.0022
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0022
Prostaglandin G/H synthase 1Homo sapiens (human)0.0078
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0022
Substance-P receptorCavia porcellus (domestic guinea pig)0.0015
Mu-type opioid receptorHomo sapiens (human)2.457
Estrogen receptor betaHomo sapiens (human)1.528
Glucocorticoid receptorSus scrofa (pig)0.0153

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bardin, CW; Kaplan-Kraicer, R; Shalgi, R1
Bardin, CW; Chang, CC; Wang, WC2
Bardin, CW; Dao, B; Koide, SS; Marshall, A; Vanage, G1
Bardin, CW; Dao, B; Koide, SS; Li, XJ; Vanage, G1
Koide, SS; Li, XJ; Yu, H1

Other Studies

6 other study(ies) available for anordiol and mifepristone

ArticleYear
Anordiol and RU486 synergize to produce preimplantation pregnancy loss by increasing embryo transport (rat).
    Contraception, 1995, Volume: 51, Issue:2

    Topics: Abortion, Induced; Animals; Body Weight; Drug Synergism; Embryonic Development; Female; Fetus; Mifepristone; Norandrostanes; Ovum Transport; Pregnancy; Rats; Rats, Wistar

1995
Anordiol is more potent than anordrin for terminating pregnancy when administered with RU 486.
    Contraception, 1993, Volume: 47, Issue:6

    Topics: Abortifacient Agents, Steroidal; Abortion, Induced; Animals; Drug Interactions; Drug Synergism; Estradiol; Female; Mifepristone; Norandrostanes; Organ Size; Pregnancy; Progesterone; Rats; Rats, Sprague-Dawley; Uterus

1993
Postcoital use of anordrin and RU 486 for prevention of implantation in the rat.
    Contraception, 1993, Volume: 47, Issue:4

    Topics: Animals; Contraceptives, Oral, Synthetic; Contraceptives, Postcoital; Drug Combinations; Drug Synergism; Embryo Implantation; Estradiol; Female; Male; Mifepristone; Norandrostanes; Ovum; Progesterone; Rats; Rats, Sprague-Dawley; Time Factors

1993
Anti-implantation activity of antiestrogens and mifepristone.
    Contraception, 1996, Volume: 54, Issue:4

    Topics: Administration, Oral; Animals; Contraceptives, Postcoital; Embryo Implantation; Estradiol; Estrogen Antagonists; Female; Fulvestrant; Injections, Subcutaneous; Male; Mifepristone; Norandrostanes; Pregnancy; Rats; Rats, Sprague-Dawley; Tamoxifen; Uterus

1996
Comparative effectiveness of three antiprogestins alone and in combination with anordiol in terminating pregnancy in the rat.
    Contraception, 1997, Volume: 55, Issue:1

    Topics: Abortion, Induced; Administration, Oral; Animals; Cohort Studies; Contraceptives, Postcoital; Dose-Response Relationship, Drug; Drug Combinations; Drug Synergism; Estradiol; Estrenes; Female; Furans; Gonanes; Hormone Antagonists; Male; Mifepristone; Norandrostanes; Pregnancy; Progesterone; Rats; Rats, Sprague-Dawley

1997
Effect of mifepristone and antiestrogens on uterine PGF2 alpha and PGE2 concentrations in ovariectomized and pregnant rats.
    Prostaglandins, 1997, Volume: 53, Issue:3

    Topics: Abortifacient Agents, Steroidal; Animals; Contraceptives, Postcoital, Synthetic; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Drug Therapy, Combination; Embryonic Development; Estradiol; Estrogen Antagonists; Female; Fulvestrant; Mifepristone; Norandrostanes; Organ Size; Ovariectomy; Pregnancy; Rats; Rats, Sprague-Dawley; Tamoxifen; Uterus

1997