Page last updated: 2024-09-05

anidulafungin and tacrolimus

anidulafungin has been researched along with tacrolimus in 6 studies

Compound Research Comparison

Studies
(anidulafungin)
Trials
(anidulafungin)
Recent Studies (post-2010)
(anidulafungin)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
5683333117,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomyanidulafungin (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (50.00)29.6817
2010's2 (33.33)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Alspaugh, JA; Fortwendel, JR; Juvvadi, PR; Perfect, BZ; Perfect, JR; Pinchai, N; Steinbach, WJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Damle, B; Dowell, JA; Henkel, T; Krause, D; Stogniew, M1
Burhenne, H; Burkhardt, O; Kaever, V; Kielstein, JT1
Abdorahimi, M; Ahmadikia, K; Badali, H; Gharehbolagh, SA; Khodavaisy, S; Mahmoudi, S; Meis, JF; Rezaie, S1

Reviews

1 review(s) available for anidulafungin and tacrolimus

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for anidulafungin and tacrolimus

ArticleYear
Lack of pharmacokinetic interaction between anidulafungin and tacrolimus.
    Journal of clinical pharmacology, 2007, Volume: 47, Issue:3

    Topics: Administration, Oral; Adolescent; Adult; Alanine Transaminase; Anidulafungin; Antifungal Agents; Area Under Curve; Aspartate Aminotransferases; Creatine Kinase; Dizziness; Drug Interactions; Echinocandins; Fatigue; Half-Life; Headache; Humans; Immunosuppressive Agents; Infusions, Intravenous; Male; Middle Aged; Nocturia; Peptides, Cyclic; Tacrolimus; Therapeutic Equivalency; Thrombophlebitis

2007

Other Studies

4 other study(ies) available for anidulafungin and tacrolimus

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Differential effects of inhibiting chitin and 1,3-{beta}-D-glucan synthesis in ras and calcineurin mutants of Aspergillus fumigatus.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:2

    Topics: Aminoglycosides; Antifungal Agents; Aspergillus fumigatus; beta-Glucans; Calcineurin; Caspofungin; Cell Wall; Chitin; Echinocandins; Fluorescent Dyes; Fungal Proteins; Genes, Fungal; Genes, ras; Lipopeptides; Microbial Sensitivity Tests; Microscopy, Fluorescence; Mutation; Signal Transduction

2009
Quantitative analysis of the antifungal drug anidulafungin by LC-online SPE-MS/MS in human plasma.
    Biomedical chromatography : BMC, 2012, Volume: 26, Issue:6

    Topics: Anidulafungin; Antifungal Agents; Chromatography, Liquid; Echinocandins; Humans; Reproducibility of Results; Sensitivity and Specificity; Solid Phase Extraction; Tacrolimus; Tandem Mass Spectrometry

2012
In vitro combination of antifungal drugs with tacrolimus (FK506) holds promise against clinical Candida species, including Candida auris.
    Medical mycology, 2023, Jul-06, Volume: 61, Issue:7

    Topics: Anidulafungin; Animals; Antifungal Agents; Candida; Candida auris; Candida glabrata; Candida parapsilosis; Caspofungin; Echinocandins; Fluconazole; Itraconazole; Microbial Sensitivity Tests; Tacrolimus

2023