Page last updated: 2024-09-03

angiotensin ii, sar(1)-me-tyr(4)- and saralasin

angiotensin ii, sar(1)-me-tyr(4)- has been researched along with saralasin in 4 studies

Compound Research Comparison

Studies
(angiotensin ii, sar(1)-me-tyr(4)-)
Trials
(angiotensin ii, sar(1)-me-tyr(4)-)
Recent Studies (post-2010)
(angiotensin ii, sar(1)-me-tyr(4)-)
Studies
(saralasin)
Trials
(saralasin)
Recent Studies (post-2010) (saralasin)
25001,4971316
6001,4971316

Protein Interaction Comparison

ProteinTaxonomyangiotensin ii, sar(1)-me-tyr(4)- (IC50)saralasin (IC50)
Type-1A angiotensin II receptor Rattus norvegicus (Norway rat)0.0017
Type-1B angiotensin II receptorRattus norvegicus (Norway rat)0.0017
Type-1 angiotensin II receptorHomo sapiens (human)0.0006
Type-2 angiotensin II receptorHomo sapiens (human)0.0008

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's1 (25.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bovy, PR; McMahon, EG; Palomo, M; Trapani, AJ1
Franklin, KJ; Moore, GJ; Nystrom, DM1
Georgiev, V; Georgieva, D1
Alova, L; Georgiev, V; Stancheva, S; Velkova, M1

Other Studies

4 other study(ies) available for angiotensin ii, sar(1)-me-tyr(4)- and saralasin

ArticleYear
A carboxy-terminus truncated analogue of angiotensin II, [Sar1]angiotensin II-(1-7)-amide, provides an entry to a new class of angiotensin II antagonists.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:3

    Topics: Angiotensin II; Animals; Blood Pressure; In Vitro Techniques; Peptide Fragments; Rabbits; Rats; Saralasin; Structure-Activity Relationship; Vasoconstriction

1989
Structure dependence of angiotensin tachyphylaxis and the mechanisms of saralasin like and sarmesin like antagonism.
    Proceedings of the Western Pharmacology Society, 1985, Volume: 28

    Topics: Angiotensin II; Animals; Female; Rats; Saralasin; Structure-Activity Relationship; Tachyphylaxis

1985
The role of angiotensin II and of its receptor subtypes in the acetic acid-induced abdominal constriction test.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 62, Issue:2

    Topics: Acetic Acid; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Colic; Imidazoles; Losartan; Male; Mice; Mice, Inbred ICR; Pain; Pain Measurement; Pyridines; Receptors, Angiotensin; Saralasin

1999
The effects of peptide and nonpeptide antagonists of angiotensin II receptors on the noradrenaline uptake of different brain structures in rats with angiotensin II-induced increase of water intake.
    Acta physiologica et pharmacologica Bulgarica, 2003, Volume: 27, Issue:2-3

    Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Brain; Drinking Behavior; Imidazoles; Losartan; Male; Norepinephrine; Rats; Rats, Wistar; Saralasin; Tetrazoles

2003