Page last updated: 2024-09-04

angiotensin ii, asp(1)-val(5)- and losartan

angiotensin ii, asp(1)-val(5)- has been researched along with losartan in 4 studies

*Losartan: An antagonist of ANGIOTENSIN TYPE 1 RECEPTOR with antihypertensive activity due to the reduced pressor effect of ANGIOTENSIN II. [MeSH]

*Losartan: An antagonist of ANGIOTENSIN TYPE 1 RECEPTOR with antihypertensive activity due to the reduced pressor effect of ANGIOTENSIN II. [MeSH]

Compound Research Comparison

Studies
(angiotensin ii, asp(1)-val(5)-)
Trials
(angiotensin ii, asp(1)-val(5)-)
Recent Studies (post-2010)
(angiotensin ii, asp(1)-val(5)-)
Studies
(losartan)
Trials
(losartan)
Recent Studies (post-2010) (losartan)
20007,2311,2452,118

Protein Interaction Comparison

ProteinTaxonomyangiotensin ii, asp(1)-val(5)- (IC50)losartan (IC50)
Bile salt export pumpHomo sapiens (human)9.01
Cytochrome P450 2C9 Homo sapiens (human)2.882
Angiotensin-converting enzyme Homo sapiens (human)0.019
Atrial natriuretic peptide receptor 3Homo sapiens (human)0.0018
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.019
Type-1A angiotensin II receptor Rattus norvegicus (Norway rat)0.0247
Type-1B angiotensin II receptorRattus norvegicus (Norway rat)0.0234
Adenosine receptor A2aRattus norvegicus (Norway rat)0.0032
Type-1 angiotensin II receptorHomo sapiens (human)0.047
Type-1 angiotensin II receptorOryctolagus cuniculus (rabbit)0.025
Type-2 angiotensin II receptorRattus norvegicus (Norway rat)0.0118
Type-2 angiotensin II receptorHomo sapiens (human)0.019
Platelet glycoprotein VIHomo sapiens (human)4
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.1481
Type-1 angiotensin II receptorCavia porcellus (domestic guinea pig)0.018
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)0.2884

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Le Mevel, JC; Mabin, D; Pamantung, TF; Vaudry, H1
Coviello, A; Peral de Bruno, M1
Hymel, A; Imig, JD; Navar, LG; Zou, LX1
Breno, MC; Picarelli, ZP; Porto, CS1

Other Studies

4 other study(ies) available for angiotensin ii, asp(1)-val(5)- and losartan

ArticleYear
Intracerebroventricular administration of angiotensin II increases heart rate in the conscious trout.
    Brain research, 1994, Aug-22, Volume: 654, Issue:2

    Topics: Angiotensin II; Animals; Atropine; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Consciousness; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Injections, Intra-Arterial; Injections, Intraventricular; Losartan; Tetrazoles; Trout

1994
Effects of angiotensin II antagonists on the contractile and hydrosmotic effect of AT II and AT III in the toad (Bufo arenarum).
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1996, Volume: 165, Issue:7

    Topics: Analysis of Variance; Angiotensin II; Angiotensin III; Animals; Antihypertensive Agents; Aorta; Biphenyl Compounds; Bufo arenarum; Dose-Response Relationship, Drug; Drug Interactions; Female; Imidazoles; Losartan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Osmolar Concentration; Osmosis; Pyridines; Skin; Tetrazoles; Vasoconstrictor Agents

1996
Renal uptake of circulating angiotensin II in Val5-angiotensin II infused rats is mediated by AT1 receptor.
    American journal of hypertension, 1998, Volume: 11, Issue:5

    Topics: Angiotensin I; Angiotensin II; Animals; Antihypertensive Agents; Blood Pressure; Kidney; Losartan; Male; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Renin

1998
Angiotensin receptor in the heart of Bothrops jararaca snake.
    European journal of pharmacology, 2001, Apr-06, Volume: 417, Issue:1-2

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin Amide; Angiotensin II; Animals; Binding, Competitive; Bothrops; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Female; Imidazoles; Inositol Phosphates; Losartan; Male; Membranes; Myocardium; Pyridines; Receptors, Angiotensin; Saralasin; Tritium

2001