Page last updated: 2024-09-02

anatoxin a and physostigmine

anatoxin a has been researched along with physostigmine in 4 studies

Compound Research Comparison

Studies
(anatoxin a)
Trials
(anatoxin a)
Recent Studies (post-2010)
(anatoxin a)
Studies
(physostigmine)
Trials
(physostigmine)
Recent Studies (post-2010) (physostigmine)
52201266,230252331

Protein Interaction Comparison

ProteinTaxonomyanatoxin a (IC50)physostigmine (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.1666
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.3023
CholinesteraseHomo sapiens (human)0.3055
Cytochrome P450 2D6Homo sapiens (human)0.2
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.857
AcetylcholinesteraseMus musculus (house mouse)0.0269
AcetylcholinesteraseHomo sapiens (human)0.0853
Acetylcholinesterase Bos taurus (cattle)0.7197
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.857
Delta-type opioid receptorMus musculus (house mouse)1.1821
AcetylcholinesteraseGallus gallus (chicken)0.02
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0416
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.857
CholinesteraseEquus caballus (horse)0.4081
CholinesteraseMus musculus (house mouse)0.28
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.0189
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.018
Carboxylic ester hydrolase Equus caballus (horse)1.263

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's1 (25.00)18.2507
2000's0 (0.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beasley, VR; Carmichael, WW; Cook, WO; Dahlem, AM; Dellinger, JA; Harlin, KS1
Albuquerque, EX; Alkondon, M; Lindstrom, J; Maelicke, A; Peng, X; Pereira, EF; Reinhardt, S; Whiting, P1
Banerjee, S; Chattopadhyay, P; Ghosh, A; Pathak, MP; Singh, S; Veer, V1
Banerjee, S; Chattopadhyay, P; Ghosh, A; Gogoi, J; Pathak, MP; Veer, V1

Other Studies

4 other study(ies) available for anatoxin a and physostigmine

ArticleYear
Comparison of effects of anatoxin-a(s) and paraoxon, physostigmine and pyridostigmine on mouse brain cholinesterase activity.
    Toxicon : official journal of the International Society on Toxinology, 1988, Volume: 26, Issue:8

    Topics: Animals; Bacterial Toxins; Brain; Cholinesterase Inhibitors; Cholinesterases; Cyanobacteria Toxins; Lethal Dose 50; Male; Marine Toxins; Mice; Mice, Inbred BALB C; Microcystins; Paraoxon; Physostigmine; Pyridostigmine Bromide; Rats; Tropanes

1988
Physostigmine and galanthamine: probes for a novel binding site on the alpha 4 beta 2 subtype of neuronal nicotinic acetylcholine receptors stably expressed in fibroblast cells.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Bacterial Toxins; Binding Sites; Cells, Cultured; Chickens; Cyanobacteria Toxins; Dexamethasone; Dose-Response Relationship, Drug; Fibroblasts; Galantamine; Kinetics; Marine Toxins; Membrane Potentials; Microcystins; Molecular Probes; Neurons; Nicotine; Physostigmine; Receptors, Nicotinic; Recombinant Proteins; Tropanes

1994
Acute dermal irritation, sensitization, and acute toxicity studies of a transdermal patch for prophylaxis against ({+/-}) anatoxin-a poisoning.
    International journal of toxicology, 2013, Volume: 32, Issue:4

    Topics: Administration, Cutaneous; Animals; Cyanobacteria Toxins; Drug Evaluation, Preclinical; Female; Guidelines as Topic; Guinea Pigs; Male; Physostigmine; Pralidoxime Compounds; Rabbits; Rats; Skin; Skin Tests; Toxicity Tests, Acute; Transdermal Patch; Tropanes

2013
Protection by a transdermal patch containing eserine and pralidoxime chloride for prophylaxis against (±)-Anatoxin A poisoning in rats.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2014, Jun-02, Volume: 56

    Topics: Animals; Anti-Arrhythmia Agents; Anticonvulsants; Arrhythmias, Cardiac; Brain; Cyanobacteria Toxins; Male; Neuroprotective Agents; Physostigmine; Pralidoxime Compounds; Rats, Wistar; Seizures; Skin; Transdermal Patch; Tropanes

2014