amthamine has been researched along with histamine in 17 studies
Studies (amthamine) | Trials (amthamine) | Recent Studies (post-2010) (amthamine) | Studies (histamine) | Trials (histamine) | Recent Studies (post-2010) (histamine) |
---|---|---|---|---|---|
33 | 0 | 11 | 37,718 | 1,372 | 3,457 |
Protein | Taxonomy | amthamine (IC50) | histamine (IC50) |
---|---|---|---|
Histamine H1 receptor | Rattus norvegicus (Norway rat) | 0.1585 | |
Histamine H1 receptor | Homo sapiens (human) | 0.1585 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (29.41) | 18.2507 |
2000's | 5 (29.41) | 29.6817 |
2010's | 6 (35.29) | 24.3611 |
2020's | 1 (5.88) | 2.80 |
Authors | Studies |
---|---|
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Buschauer, A; Dove, S; Igel, P | 1 |
Eriks, JC; Sterk, GJ; Timmerman, H; van der Goot, H | 1 |
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H | 1 |
Eriks, JC; Timmerman, H; van der Goot, H | 1 |
D'Souza, T; Dryer, SE; Nowak, JZ; Sek, B | 1 |
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C | 1 |
Falus, A; László, V; Orsó, E; Schmitz, G; Szeberényi, JB | 1 |
Bugajski, AJ; Bugajski, J; Gadek-Michalska, A; Głód, R; Thor, P | 1 |
Eckman, JR; Wagner, MC; Wick, TM | 1 |
Jarajapu, YP; Knot, HJ; Oomen, C; Uteshev, VV | 1 |
Dartt, DA; Hayashi, C; Hayashi, D; Hodges, RR; Li, D; Shatos, M | 1 |
Dandekar, RD; Khan, MM | 1 |
Kang, JH; Kim, HJ; Kim, HM; Kim, YL; Lee, AY; Lee, CH; Lee, EJ; Lee, HJ; Park, MK | 1 |
Ali, AS; Ali, SA; Salim, S | 1 |
Alonso, N; Davio, C; Diaz Nebreda, A; Fernandez, N; Gutkind, JS; Monczor, F; Shayo, C | 1 |
Awane, H; Ezaki, M; Hishinuma, S; Inazuki, N; Michinaga, S; Mizuguchi, H; Shimizu, K; Sonoda, K | 1 |
17 other study(ies) available for amthamine and histamine
Article | Year |
---|---|
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Histamine H4 receptor agonists.
Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2010 |
Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4- and 5-(2-aminoethyl)thiazoles.
Topics: Animals; Atrial Function; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Guinea Pigs; Heart Atria; Histamine; Ileum; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles | 1992 |
In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine: comparisons with histamine and dimaprit.
Topics: Animals; Atrial Function; Dimaprit; Electric Stimulation; Guinea Pigs; Heart; Heart Atria; Histamine; Histamine Agonists; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Rabbits; Ranitidine; Thiazoles | 1993 |
New activation model for the histamine H2 receptor, explaining the activity of the different classes of histamine H2 receptor agonists.
Topics: Histamine; Kinetics; Models, Chemical; Quantum Theory; Receptors, Histamine H2; Stimulation, Chemical; Structure-Activity Relationship; Thiazoles | 1993 |
Does histamine stimulate cyclic AMP formation in the avian pineal gland via a novel (non-H1, non-H2, non-H3) histamine receptor subtype.
Topics: Animals; Benzothiazoles; Chickens; Cyclic AMP; Ducks; Histamine; Histamine Agonists; Histamine H2 Antagonists; Ion Channels; Male; Methylation; Phenoxypropanolamines; Pineal Gland; Piperidines; Receptors, Histamine; Stimulation, Chemical; Thiazoles | 1995 |
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles | 1999 |
Histamine and H2 agonist amthamine increase oxidative burst activity of human leukocytes determined by flow cytometry.
Topics: Flow Cytometry; Granulocytes; Histamine; Histamine Agonists; Humans; Leukocytes; Monocytes; Receptors, Histamine H1; Receptors, Histamine H2; Respiratory Burst; Thiazoles | 2000 |
Influence of cyclooxygenase inhibitors on the central histaminergic stimulations of hypothalamic - pituitary - adrenal axis.
Topics: Adrenocorticotropic Hormone; Animals; Corticosterone; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Drug Administration Schedule; Histamine; Histamine Agonists; Hypothalamo-Hypophyseal System; Indomethacin; Injections, Intraperitoneal; Injections, Intraventricular; Isoenzymes; Male; Membrane Proteins; Nitrobenzenes; Piroxicam; Pituitary-Adrenal System; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Sulfonamides; Thiazoles | 2003 |
Histamine increases sickle erythrocyte adherence to endothelium.
Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules | 2006 |
Histamine decreases myogenic tone in rat cerebral arteries by H2-receptor-mediated KV channel activation, independent of endothelium and cyclic AMP.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Animals; Benzenesulfonates; Calcium; Cerebral Arteries; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Oxadiazoles; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Potassium Chloride; Quinoxalines; Rats; Rats, Sprague-Dawley; Thiazoles; Vasoconstriction; Vasodilation | 2006 |
Role of histamine and its receptor subtypes in stimulation of conjunctival goblet cell secretion.
Topics: Animals; Blotting, Western; Cells, Cultured; Cimetidine; Conjunctiva; Conjunctivitis, Allergic; Dose-Response Relationship, Drug; Fluorescent Antibody Technique; Goblet Cells; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Indoles; Male; Methylhistamines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles | 2012 |
Involvement of histamine receptors in SAPK/JNK phosphorylation.
Topics: Animals; Betahistine; Female; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; MAP Kinase Signaling System; Methylhistamines; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphorylation; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Spleen; Tetradecanoylphorbol Acetate; Thiazoles; Tumor Necrosis Factor-alpha | 2012 |
Histamine receptor 2-mediated growth-differentiation factor-15 expression is involved in histamine-induced melanogenesis.
Topics: Cell Line, Tumor; Cell Proliferation; Chemotaxis; Cimetidine; Gene Expression; Gene Expression Regulation; Growth Differentiation Factor 15; Histamine; Histamine Agonists; Humans; Intramolecular Oxidoreductases; Melanins; Membrane Glycoproteins; Monophenol Monooxygenase; Oxidoreductases; Receptors, Histamine H2; Thiazoles | 2012 |
On the role of histamine receptors in regulating pigmentary responses in Oreochromis mossambicus melanophores.
Topics: Animals; Female; Histamine; Histamine Agonists; Histamine Antagonists; Male; Melanins; Melanophores; p-Methoxy-N-methylphenethylamine; Pigments, Biological; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tilapia | 2012 |
PI3K pathway is involved in ERK signaling cascade activation by histamine H2R agonist in HEK293T cells.
Topics: Cell Line; Cell Proliferation; Extracellular Signal-Regulated MAP Kinases; HEK293 Cells; Histamine; Histamine Agonists; Humans; MAP Kinase Signaling System; Phosphatidylinositol 3-Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Signal Transduction; Thiazoles; TOR Serine-Threonine Kinases | 2016 |
Selective histamine H
Topics: Angiopoietin-1; Animals; Blood-Brain Barrier; Brain Injuries, Traumatic; Dimaprit; Endothelial Cells; Evans Blue; Hedgehog Proteins; Histamine; Histamine Agonists; Male; Mice; Protective Factors; Ranitidine; Receptors, Histamine H2; RNA, Messenger; Thiazoles | 2022 |