Page last updated: 2024-08-24

amprenavir and brecanavir

amprenavir has been researched along with brecanavir in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's0 (0.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Carter, HL; Danger, D; Furfine, ES; Hanlon, MH; Kaldor, IW; Miller, JF; Porter, DJ; Samano, VA; Shu, AY; Spaltenstein, A1
Andrews, CW; Brieger, M; Furfine, ES; Hale, MR; Hanlon, MH; Hazen, RJ; Kaldor, I; McLean, EW; Miller, JF; Reynolds, D; Sammond, DM; Sherrill, RG; Spaltenstein, A; Tung, R; Turner, EM; Xu, RX1
Boone, L; Craig, C; Ferris, R; Furfine, E; Griffin, P; Hale, M; Hanlon, M; Harvey, R; Hazen, R; Kaldor, I; Miller, J; Ray, J; Samano, V; Spaltenstein, A; St Clair, M; Tung, R; Yates, P1
Babusis, D; Bhoopathy, S; Hidalgo, IJ; Phan, TK; Ray, AS; Rhodes, GR; Robinson, KL; Strab, R; Tong, L1
Boucher, MJ; Brynda, J; Craik, CS; Drąg, M; Grzymska, J; Hájek, M; Hradilek, M; Konvalinka, J; Kryštůfek, R; Madhani, HD; Majer, P; Řezáčová, P; Rut, W; Šácha, P; Starková, J; Tloušt'ová, E1

Other Studies

5 other study(ies) available for amprenavir and brecanavir

ArticleYear
Inhibition of wild-type and mutant human immunodeficiency virus type 1 proteases by GW0385 and other arylsulfonamides.
    Biochemistry, 2004, Nov-16, Volume: 43, Issue:45

    Topics: Amino Acid Substitution; Binding, Competitive; Carbamates; Chromatography, Affinity; Chromatography, Gel; Dextrans; Dimerization; Furans; HIV Protease; HIV Protease Inhibitors; HIV-1; Hydrolysis; Kinetics; Protein Binding; Saquinavir; Spectrometry, Fluorescence; Substrate Specificity; Sulfonamides

2004
Ultra-potent P1 modified arylsulfonamide HIV protease inhibitors: the discovery of GW0385.
    Bioorganic & medicinal chemistry letters, 2006, Apr-01, Volume: 16, Issue:7

    Topics: HIV Protease Inhibitors; Molecular Structure; Sulfonamides

2006
In vitro antiviral activity of the novel, tyrosyl-based human immunodeficiency virus (HIV) type 1 protease inhibitor brecanavir (GW640385) in combination with other antiretrovirals and against a panel of protease inhibitor-resistant HIV.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:9

    Topics: Algorithms; Anti-Retroviral Agents; Benzodioxoles; Blood Proteins; Carbamates; Cell Line; Drug Resistance, Viral; HeLa Cells; HIV Protease Inhibitors; HIV-1; Humans; Orosomucoid; Phenotype; Serum; Serum Albumin; Tyrosine

2007
Effects of human immunodeficiency virus protease inhibitors on the intestinal absorption of tenofovir disoproxil fumarate in vitro.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:10

    Topics: Adenine; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cell Line; Chromatography, High Pressure Liquid; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Drug Interactions; Epithelium; HIV Protease Inhibitors; Humans; Hydrolysis; Indicators and Reagents; Intestinal Absorption; Mass Spectrometry; Organophosphonates; Subcellular Fractions; Tenofovir

2007
Re-emerging Aspartic Protease Targets: Examining
    Journal of medicinal chemistry, 2021, 05-27, Volume: 64, Issue:10

    Topics: Antifungal Agents; Aspartic Acid Proteases; Binding Sites; Catalytic Domain; Cryptococcus neoformans; Crystallography, X-Ray; Drug Evaluation, Preclinical; Fungal Proteins; Fungi; HIV; HIV Protease; Molecular Dynamics Simulation; Recombinant Proteins; Structure-Activity Relationship; Substrate Specificity

2021