amphetamine has been researched along with piperidines in 146 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 71 (48.63) | 18.7374 |
1990's | 21 (14.38) | 18.2507 |
2000's | 24 (16.44) | 29.6817 |
2010's | 28 (19.18) | 24.3611 |
2020's | 2 (1.37) | 2.80 |
Authors | Studies |
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Borisenko, SA | 1 |
Barailler, J; Pacheco, H; Ramirez, A; Vial, H | 1 |
Costall, B; Fortune, DH; Naylor, RJ | 1 |
Denber, HC | 1 |
Ferris, RM; Tang, FL | 1 |
Iversen, SD; Morgan, MJ; Robbins, TW; Sahakian, BJ | 1 |
Debackere, M; Delbeke, FT | 1 |
Colpaert, FC; Lal, H; Niemegeers, C; Wauquier, A | 1 |
Boeck, V; Christensen, AV; Danneskiold-Samsoe, P; Hyttel, J; Langeland, J; Nielsen, IM; Pedersen, V; Svendsen, O | 1 |
Baran, L; Gancarczyk, L; Maj, J; Sowińska, H | 1 |
Baran, L; Maj, J; Palider, W | 1 |
Moffat, AC | 1 |
van Zwieten, PA | 1 |
Baker, JC; Day, WA; Fuller, RW; Molloy, BB; Perry, KW | 1 |
Awouters, FH; Megens, AA; Niemegeers, CJ | 1 |
Gessa, GL; Hmaidan, Y; Rossetti, ZL | 1 |
Hayakawa, K; Imaizumi, N; Ishikura, H; Kobayashi, H; Minogawa, E; Miyazaki, M; Takayama, N | 1 |
Awouters, F; Janssen, PA; Meert, TF; Megens, AA; Niemegeers, CJ; Schellekens, KH | 1 |
Goiny, M; Uvnäs-Moberg, K | 1 |
Nichols, NF; Schreur, PJ | 1 |
Smith, DF | 1 |
Bourat, G; Ducrot, R; Fournel, J; Garret, C; Julou, L | 1 |
Moore, KE; Thornburg, JE | 1 |
Rolinski, Z; Scheel-Krüger, J | 1 |
Absava, GI | 1 |
Hasselager, E; Scheel-Krüger, J | 1 |
Naumenko, EV | 1 |
Aceto, MD; Brown, TG; Harris, LS; Lesher, GY; Pearl, J | 1 |
Hite, G; Kuhn, WL; Pazdernik, TL; Portoghese, PS; Shafi'ee, A | 1 |
Lechat, P; Streichenberger, G | 1 |
Berstein, BM; Latimer, CN | 1 |
Vinar, O | 1 |
Reigle, TG; Rollins, DE; Rowland, CR; Wolf, HH | 1 |
Bouttier, D; Julou, L; Sigwald, J; Thomas, J | 1 |
Fog, R | 1 |
Dominic, JA; Moore, KE | 2 |
Muskens, AT; van Rossum, JM; Vree, TB | 1 |
Chiba, S; Nagawa, Y; Yui, T | 1 |
Sharov, PA; Shugina, TM; Vysotskaia, NB | 1 |
Patil, PN; Yamauchi, D | 1 |
Messini, M | 1 |
Carr, LA; Moore, KE | 1 |
Smirnov, GD; Vinogradova, VM | 1 |
Iakovlev, NN | 1 |
Costall, B; Naylor, RJ | 1 |
Allen, LE; Ferguson, HC; McKinney, GR | 1 |
Schuster, CR; Wilson, MC | 1 |
Bej, AJ; Tanner, NS; Wolters, RJ | 1 |
Bartolini, A; Domino, EF | 1 |
Ayhan, IH; Randrup, A | 1 |
Williams, CH | 1 |
Chrusciel, TL; Isbell, H | 1 |
Ferris, RM; Maxwell, RA; Tang, FL | 1 |
Hermans, G | 1 |
Stepanek, J | 1 |
Janssen, PA; Niemegeers, CJ; Verbruggen, FJ | 1 |
Barkov, N; Geller, A; Jarvik, ME | 1 |
Fish, B | 1 |
Schneider, C | 1 |
Kasé, Y; Nakanishi, M; Okada, T; Tsumagari, T | 1 |
Keuhnelian, AM; Sinsheimer, JE | 1 |
Funcke, AB; Harms, AF; Louwerse, WJ; Nauta, WT; Tersteege, HM | 1 |
Dandiya, PC; Gurbani, NK; Hrishi Keshavan, HJ | 1 |
Cenajek, D; Chodera, A; Mazurek, K | 1 |
Antonin, KH; Bieck, P; Feldtrauer, JJ; Grunenwald, C; Lauber, J; Paul, E; Waldmeier, PC | 1 |
Gueudet, C; Le Fur, G; Rinaldi-Carmona, M; Santucci, V; Soubrié, P | 1 |
Awouters, FH; Janssen, PA | 1 |
Jackson, A; Rupniak, NM | 1 |
Bervoets, K; Maurel-Remy, S; Millan, MJ | 1 |
Clark, D; Exner, M; Furmidge, LJ; Sonesson, C; Svensson, K | 1 |
Clapham, J; Kilpatrick, GJ | 1 |
Abreu, ME; Borosky, S; Clissold, DB; Erickson, RH; Hartman, T; Jones, BE; Karbon, EW; Mansbach, RS; Natalie, KJ; Pontecorvo, MJ | 1 |
Gerlach, J; Peacock, L | 1 |
Järbe, TU | 1 |
Frank, RA; Kehne, JH; Moran, PM; Moser, PC | 1 |
Bourin, M; Hascoet, M; Lombet, A; Payeur, R; Peglion, JL | 1 |
Vanover, KE | 1 |
Brown, D; Byrd, G; Feldman, DJ; Flannery, R; Frank, RA; Kehne, JH; Shah, S; Soni, S | 1 |
Hagan, J; Hatcher, JP; Lewis, VA; Reavill, C; Sanger, GJ | 1 |
Piercey, MF; Ray, CA; Walker, EL | 1 |
Carlsson, A; Carlsson, ML; Martin, P; Nilsson, M; Sorensen, SM; Waters, N; Waters, S | 1 |
Heron-Maxwell, CL; O'Neill, MF; Shaw, G | 1 |
Karoum, F; Masserano, JM; Wyatt, RJ | 1 |
Henry, BL; LaHoste, GJ; Marshall, JF | 1 |
Ichikawa, J; Kuroki, T; Meltzer, HY | 1 |
Rimmerman, N; Weiner, I; Zuckerman, L | 1 |
ARRIGONI-MARTELLI, E; GENOVESE, E; GOLDWURM, GF | 1 |
ARIENS, EJ; HURKMANS, JA; van der SCHOOT, J; van ROSSUM, J | 1 |
BRIMBLECOMBE, RW | 1 |
FITZLOFF, J; PLOTNIKOFF, NP | 1 |
HIDALGO, J; THOMPSON, CR | 1 |
DROOBY, AS | 1 |
SIEGLER, PE | 1 |
FELLNER, CH | 1 |
Chiou, LC; Gean, PW; Huang, YC; Wang, SJ | 1 |
Aujla, H; Beninger, RJ | 1 |
Caraballo, I; El Banoua, F; Fernandez-Espejo, E; Ferrer, B; Flores, JA; Galan-Rodriguez, B; Rodriguez de Fonseca, F | 1 |
Burton, P; Mechoulam, R; Parker, LA; Sorge, RE; Yakiwchuk, C | 1 |
Gessa, GL; Melis, M; Muntoni, AL; Perra, S; Pillolla, G; Pistis, M | 1 |
Ferguson, SM; Robinson, TE | 1 |
Marona-Lewicka, D; Nichols, DE; Thisted, RA | 1 |
Andersen, MB; Brandt-Christensen, M; Fink-Jensen, A; Gerlach, J; Werge, T | 1 |
Alonso, R; Avenet, P; Biton, B; Boulay, D; Coste, A; Cudennec, A; Dargazanli, G; Decobert, M; Depoortère, R; Desvignes, C; Estenne-Bouhtou, G; Françon, D; George, P; Griebel, G; Heaulme, M; Lanneau, C; Marabout, B; Oury-Donat, F; Perrault, G; Poncelet, M; Roger, P; Santucci, V; Scatton, B; Sevrin, M; Soubrié, P; Steinberg, R; Stemmelin, J; Terranova, JP; Vigé, X; Voltz, C | 1 |
Kruse, CG; McCreary, AC; Olijslagers, JE; Perlstein, B; Siarey, R; Wadman, WJ; Werkman, TR | 1 |
Akhtar, M; Ali, A; Pillai, KK; Uma Devi, P; Vohora, D | 1 |
de Boissezon, X; de Boysson, C; Démonet, JF; Peran, P | 1 |
Asgari, K; Bezzina, G; Body, S; Bradshaw, CM; Cheung, TH; Fone, KC; Glennon, JC; Szabadi, E | 1 |
Anderson, GT; Barido, R; Bonhaus, DW; Brann, MR; Brunmark, P; Davis, RE; Dyssegaard, A; Gardell, LR; Hacksell, U; Johnson, RW; Pounds, L; Tabatabaei, A; Vanover, KE; Veinbergs, I | 1 |
Fujiki, N; Honda, Y; Kodama, T; Nishino, S; Song, YH; Soya, A | 1 |
Di Marzo, V; Hasenöhrl, RU; Molleman, A; Thiemann, G | 1 |
Arad, M; Barak, S; Black, MD; Boulay, D; De Levie, A; Griebel, G; Pichat, P; Varty, GB; Weiner, I | 1 |
Davis, RJ; Degroot, A; Nomikos, GG; Tzavara, ET; Wade, MR | 1 |
Feldon, J; Singer, P; Yee, BK | 1 |
Advani, T; Cassano, T; Giuffrida, A; Hensler, JG; Seillier, A | 1 |
Gross, G; Jongen-Rêlo, AL; Schoemaker, H; Unger, L; van Gaalen, MM | 1 |
Hinchliffe, RM; Huszar, SL; Hutson, PH; Pachmerhiwala, R; Smith, SM; Uslaner, JM; Vardigan, JD | 1 |
Fan, X; Hess, EJ; Xu, M | 1 |
Markou, A; Semenova, S | 1 |
Amantini, D; Antolini, M; Bifone, A; Cesari, N; Corsi, M; Gozzi, A; Martinelli, P; Massagrande, M; Montanari, D; Piccoli, L; Tessari, M; Turrini, G | 1 |
Fletcher, PJ; Higgins, GA; Noble, K; Rizos, Z | 1 |
Bonhaus, DW; McFarland, K; Price, DL | 2 |
Kõks, S; Matsui, T; Orav, L; Rünkorg, K; Vasar, E; Volke, V | 1 |
Pattij, T; Schetters, D; Schoffelmeer, AN; Stoop, N; Wiskerke, J | 1 |
Arnold, JC; Cain, ME; Gill, MJ | 1 |
Hammond, B; Hussain, I; Kew, JN; Stean, TO; Upton, N; Virley, DJ; Waters, KA | 1 |
Burton, CL; Fletcher, PJ | 1 |
Århem, P; Fuxe, K; Marcellino, D; Sahlholm, K | 1 |
Carroll, FI; McMahon, LR; Schulze, DR | 1 |
Barrot, M; Bockaert, J; Charnay, Y; Compan, V; Dusticier, N; Jean, A; Laurent, L; Neve, R; Nieoullon, A | 1 |
Singer, P; Yee, BK; Zhang, W | 1 |
Andersen, ML; Howell, LL; Murnane, KS; Rice, KC | 1 |
Hacksell, U; Hubbard, D; McFarland, K | 1 |
Antoniou, K; Chouliara, O; Galanopoulos, A; Naxakis, G; Papadopoulou-Daifoti, Z; Papahatjis, D; Polissidis, A | 1 |
Bouchard, C; Ducrot, C; Fortier, E; Gallo, A; Rompré, PP | 1 |
Ansari, MS; Conn, PJ; Daniels, JS; Emmitte, KA; Felts, AS; Jones, CK; Kessler, RM; Lindsley, CW; Niswender, CM; Rook, JM; Stauffer, SR; Tantawy, MN | 1 |
Bernard, P; Bizot, JC; David, S; Puech, A; Tassin, JP; Trovero, F | 1 |
Carlsson, A; Eriksson, E; Näslund, J; Studer, E; Westman, A | 1 |
Bunner, KD; Cheer, JF; Covey, DP; Garris, PA; Schuweiler, DR | 1 |
Clancy, PT; Lim, YW; Muelbl, MJ; Nawarawong, NN; Nettesheim, CE; Olsen, CM | 1 |
Brodney, MA; Davoren, JE; Edgerton, JR; Fortin, JP; Garnsey, M; Grimwood, S; Harris, AR; Jenkinson, S; Kenakin, T; Lazzaro, JT; Lee, CW; Lotarski, SM; Nottebaum, L; O'Neil, SV; Pettersen, B; Popiolek, M; Ramsey, S; Steyn, SJ; Thorn, CA; Webb, D; Zhang, L | 1 |
Coupal, M; Laird, J; Lindberg, M; Martino, G; Sandin, J; Santhakumar, V; Schroeder, P; Valiquette, M; Widzowski, D; Wood, MW | 1 |
Benade, V; Bhyrapuneni, G; Daripelli, S; Jayarajan, P; Nirogi, R; Tirumalasetty, C | 1 |
Arreguin-Campos, R; Caldara, M; Cleij, TJ; Diliën, H; Eersels, K; Heidt, B; Jimenez-Monroy, KL; Lowdon, JW; Rogosic, R; van Grinsven, B | 1 |
Belliard, S; Berrebi-Bertrand, I; Finance, O; Giret, M; Krief, S; Lecomte, JM; Ligneau, X; Nagmar, I; Perrin, D; Robert, P; Schwartz, JC; Uguen, M | 1 |
6 review(s) available for amphetamine and piperidines
Article | Year |
---|---|
[Psychopharmaca in modern medicine].
Topics: Amphetamine; Antidepressive Agents; Barbiturates; Butyrophenones; Chlordiazepoxide; Chlorprothixene; Diazepam; Dibenzazepines; Guaifenesin; Hallucinogens; Humans; Hypnotics and Sedatives; Imipramine; Lithium; Lysergic Acid Diethylamide; Methylphenidate; Monoamine Oxidase Inhibitors; Oxazepam; Phenmetrazine; Phenothiazines; Phytotherapy; Piperidines; Plants, Medicinal; Psilocybin; Psychopharmacology; Rauwolfia; Reserpine; Tranquilizing Agents; Xanthenes | 1968 |
[On the harmful effects of drugs. II].
Topics: Adrenergic beta-Antagonists; Allopurinol; Amphetamine; Animals; Anti-Bacterial Agents; Contraceptives, Oral; Digitalis Glycosides; Drug and Narcotic Control; Drug-Related Side Effects and Adverse Reactions; Ephedrine; Gonanes; Humans; Immunosuppressive Agents; Italy; Legislation, Drug; Methyldopa; Morpholines; Piperidines; Sympatholytics | 1970 |
[Physiological aspects of endurance during muscular activity].
Topics: Adenosine Triphosphate; Amphetamine; Brain; Fatigue; Humans; Mitochondria, Muscle; Muscles; Myocardium; Oxygen Consumption; Phosphocreatine; Physical Education and Training; Physical Exertion; Piperidines; Uracil; Vitamin B Complex | 1970 |
Dependence liability of "non-narcotic" drugs.
Topics: Alcohols; Amphetamine; Barbiturates; Benzazepines; Carbamates; Chloral Hydrate; Dronabinol; Ephedrine; Esters; Ethers, Cyclic; Glycols; Hallucinogens; Halogens; Herbicides; Humans; Indoles; Phenethylamines; Piperidines; Plant Extracts; Quinazolines; Substance-Related Disorders | 1970 |
CURRENT STATUS OF DRUG TREATMENT IN THE DEPRESSIVE STATE.
Topics: Amitriptyline; Amphetamine; Amphetamines; Antidepressive Agents; Aspartic Acid; Benactyzine; Classification; Deanol; Depression; Desipramine; Humans; Imipramine; Isocarboxazid; Methylphenidate; Monoamine Oxidase Inhibitors; Nialamide; Pargyline; Pharmacology; Phenelzine; Phenmetrazine; Piperidines; Sympathomimetics; Toxicology; Tranylcypromine | 1964 |
Pharmacotherapy of aphasia: myth or reality?
Topics: Amphetamine; Aphasia; Bromocriptine; Cholinesterase Inhibitors; Clinical Trials as Topic; Donepezil; Dopamine Agents; Fluoxetine; GABA Agonists; Humans; Indans; Neuroprotective Agents; Paroxetine; Physostigmine; Piperidines; Piracetam; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Stroke; Zolpidem | 2007 |
140 other study(ies) available for amphetamine and piperidines
Article | Year |
---|---|
[Mechanism of the analgesic effect of narcotic analgetics].
Topics: Amphetamine; Analgesics, Opioid; Animals; Fentanyl; Hypothalamus; Male; Morphine; Pentazocine; Piperidines; Rats; Self Stimulation; Septum Pellucidum | 1976 |
[Effects of levophacetoperane, pemoline, fenozolone, and centrophenoxine on catecholamines and serotonin uptake in various parts of the rat brain].
Topics: Amphetamine; Animals; Benzyl Alcohols; Binding, Competitive; Brain; Brain Chemistry; Catecholamines; Central Nervous System Stimulants; Cerebral Cortex; Corpus Striatum; Hypothalamus; In Vitro Techniques; Male; Meclofenoxate; Pemoline; Piperidines; Rats; Serotonin; Synaptosomes | 1978 |
Neuropharmacological studies on the neuroleptic potential of domperidone (R33812).
Topics: Amphetamine; Animals; Antipsychotic Agents; Benzimidazoles; Brain Chemistry; Haloperidol; Humans; Motor Activity; Piperidines; Rats; Stereotyped Behavior | 1979 |
The pharmacologic treatment of depression.
Topics: Amphetamine; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Deanol; Depression; Dose-Response Relationship, Drug; Humans; Lithium; Methylphenidate; Monoamine Oxidase Inhibitors; Phenmetrazine; Piperidines | 1979 |
Comparison of the effects of the isomers of amphetamine, methylphenidate and deoxypipradrol on the uptake of l-[3H]norepinephrine and [3H]dopamine by synaptic vesicles from rat whole brain, striatum and hypothalamus.
Topics: Amphetamine; Animals; Brain; Corpus Striatum; Desipramine; Dopamine; Energy Metabolism; Hypothalamus; In Vitro Techniques; Kinetics; Male; Methylphenidate; Norepinephrine; Piperidines; Rats; Reserpine; Stereoisomerism; Synaptic Vesicles; Temperature | 1979 |
The effects of psychomotor stimulants on stereotypy and locomotor activity in socially-deprived and control rats.
Topics: Amphetamine; Animals; Apomorphine; Brain Chemistry; Cocaine; Dopamine; Dose-Response Relationship, Drug; Female; Humans; Locomotion; Motor Activity; Norepinephrine; Piperidines; Rats; Social Isolation; Stereotyped Behavior | 1975 |
Isolation and detection of methylphenidate, phacetoperane and some other sympatomimetic central nervous stimulants with special reference to doping. I. Gas chromatographic detection procedure with electron capture detection for some secondary amines.
Topics: Amphetamine; Benzyl Alcohols; Chemical Phenomena; Chemistry; Chromatography, Gas; Hydrogen-Ion Concentration; Hydrolysis; Mass Spectrometry; Methylphenidate; Piperidines; Sympathomimetics; Temperature | 1975 |
Reversal by a central antiacetylcholine drug of pimozide-induced inhibition of mouse-jumping in amphetamine-dopa treated mice.
Topics: Acetylcholine; Amphetamine; Animals; Dexetimide; Levodopa; Male; Mice; Motor Activity; Pimozide; Piperidines; Time Factors | 1975 |
The pharmacology of a new potent, long acting neuroleptic, piflutixol.
Topics: Adenylyl Cyclases; Amphetamine; Anesthesia; Animals; Apomorphine; Arousal; Barbiturates; Behavior, Animal; Catalepsy; Dogs; Dopamine Antagonists; Escape Reaction; Ethanol; Female; Humans; Male; Methylphenidate; Mice; Motor Activity; Piperidines; Rabbits; Rats; Thioxanthenes; Tranquilizing Agents | 1977 |
The action of compound WA-335 on the central nervous system.
Topics: Amphetamine; Animals; Anthracenes; Antidepressive Agents, Tricyclic; Body Temperature; Brain; Brain Chemistry; Drug Synergism; Female; Humans; Male; Mice; Motor Activity; Piperidines; Rats; Receptors, Drug; Reserpine; Serotonin; Stereotyped Behavior | 1976 |
The effects of serotonergic and antiserotonergic drugs on the flexor reflex of spinal rat: a proposed model to evaluate the action on the central serotonin receptor.
Topics: 5-Hydroxytryptophan; Amphetamine; Animals; Anthracenes; Clonidine; Cyproheptadine; Decerebrate State; Fenfluramine; Hindlimb; Lysergic Acid Diethylamide; Male; Metergoline; Muscle Contraction; p-Chloroamphetamine; Piperidines; Rats; Reflex; Serotonin; Tryptophan | 1976 |
Use of SE-30 as a stationary phase for the gas-liquid chromatography of drugs.
Topics: Absorption; Amphetamine; Chromatography, Gas; Diphenhydramine; Methadone; Methods; Pharmaceutical Preparations; Piperidines; Silicone Elastomers | 1975 |
Interaction between centrally acting hypotensive drugs and tricyclic antidepressants.
Topics: Amphetamine; Animals; Antidepressive Agents, Tricyclic; Antihypertensive Agents; Benzimidazoles; Blood Pressure; Cats; Clonidine; Cocaine; Desipramine; Dioxanes; Drug Interactions; Ephedrine; Female; Male; Methyldopa; Piperidines; Reserpine | 1975 |
Biochemical pharmacology of some chlorinated 3-phenyl-piperidines in rats.
Topics: Amphetamine; Animals; Brain Chemistry; Desipramine; Half-Life; Hydroxyindoleacetic Acid; Male; Monoamine Oxidase Inhibitors; Piperidines; Rats; Serotonin; Time Factors | 1975 |
Behavioral disinhibition and depression in amphetaminized rats: a comparison of risperidone, ocaperidone and haloperidol.
Topics: Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Isoxazoles; Male; Motor Activity; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Risperidone | 1992 |
Marked inhibition of mesolimbic dopamine release: a common feature of ethanol, morphine, cocaine and amphetamine abstinence in rats.
Topics: Amphetamine; Animals; Cocaine; Corpus Striatum; Dizocilpine Maleate; Dopamine; Ethanol; Male; Morphine; Naloxone; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome | 1992 |
Determination of methamphetamine, amphetamine and piperidine in human urine by high-performance liquid chromatography with chemiluminescence detection.
Topics: Amphetamine; Chromatography, Gas; Chromatography, High Pressure Liquid; Humans; Luminescent Measurements; Methamphetamine; Piperidines | 1990 |
Pharmacology of risperidone (R 64 766), a new antipsychotic with serotonin-S2 and dopamine-D2 antagonistic properties.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Conditioning, Psychological; Dogs; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Haloperidol; Isoxazoles; Male; Motor Activity; Oxazoles; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Risperidone; Serotonin Antagonists | 1988 |
Effects of dopaminomimetics on the secretion of VIP-like immunoreactivity in conscious dogs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Apomorphine; Benzazepines; Dogs; Ergolines; Nitroglycerin; Pergolide; Piperidines; Prazosin; Receptors, Dopamine; Somatostatin; Vasoactive Intestinal Peptide | 1986 |
Two automated locomotor activity tests for dopamine autoreceptor agonists.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Drug Evaluation, Preclinical; Exploratory Behavior; Indoles; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
The stereoselectivity of serotonin uptake in brain tissue and blood platelets: the topography of the serotonin uptake area.
Topics: Alanine; Amphetamine; Aniline Compounds; Animals; Antidepressive Agents; Blood Platelets; Brain; Fluoxetine; Humans; Male; Methadone; Mianserin; Mirtazapine; Morpholines; Naphthalenes; Nefopam; Nomifensine; Paroxetine; Piperidines; Rabbits; Serotonin; Stereoisomerism; Tranylcypromine; Viloxazine; Zimeldine | 1986 |
Pharmacological study of pipotiazine (19.366 R.P.) and its undecylenic (19.551 R.P.) and palmitic (19.552 R.P.) esters.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dogs; Esters; Fluphenazine; Guinea Pigs; Humans; Lethal Dose 50; Mice; Motor Activity; Palmitic Acids; Phenothiazines; Piperidines; Rats; Respiration; Sleep; Species Specificity; Sulfonamides; Time Factors; Undecylenic Acids | 1973 |
The relative importance of dopaminergic and noradrenergic neuronal systems for the stimulation of locomotor activity induced by amphetamine and other drugs.
Topics: Amphetamine; Animals; Appetite; Carbon Radioisotopes; Diet; Disulfides; Dopamine; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Imidazoles; Male; Methylphenidate; Methyltyrosines; Mice; Motor Activity; Neurons; Norepinephrine; Phenmetrazine; Piperidines; Stimulation, Chemical; Thiazoles; Thiourea; Time Factors | 1973 |
The effect of dopamine and noradrenaline antagonists on amphetamine induced locomotor activity in mice and rats.
Topics: Adrenergic alpha-Antagonists; Amphetamine; Animals; Aza Compounds; Behavior, Animal; Depression, Chemical; Dopamine Antagonists; Dopamine beta-Hydroxylase; Ergotamine; Female; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Norepinephrine; Perphenazine; Phenoxybenzamine; Phenyl Ethers; Pimozide; Piperidines; Rats; Receptors, Drug; Spiro Compounds; Time Factors; Tranquilizing Agents; Trifluoperazine | 1973 |
[Effect of psychostimulants on membrane permeability for K42 in different areas of the rat brain].
Topics: Amphetamine; Animals; Brain; Caffeine; Cell Membrane Permeability; Cerebral Cortex; Diencephalon; Medulla Oblongata; Mesencephalon; Piperidines; Potassium; Potassium Isotopes; Rats | 1973 |
Studies of various amphetamines, apomorphine and clonidine on body temperature and brain 5-hydroxytryptamine metabolism in rats.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Body Temperature; Brain; Brain Chemistry; Carboxylic Acids; Chromatography, Ion Exchange; Clonidine; Fever; Hydroxyindoleacetic Acid; Male; Methylphenidate; Naphthyridines; Phenmetrazine; Piperidines; Rats; Serotonin; Spectrometry, Fluorescence; Temperature | 1974 |
Role of adrenergic and cholinergic structures in the control of the pituitary-adrenal system.
Topics: 17-Hydroxycorticosteroids; Acetylcholine; Adrenal Glands; Amphetamine; Animals; Electrocardiography; Electroencephalography; Epinephrine; Galantamine; Guinea Pigs; Imidazoles; Mesencephalon; Naphthalenes; Neostigmine; Piperidines; Pituitary Gland; Pituitary-Adrenal System | 1967 |
Pharmacologic studies with 7-benzyl-1-ethyl-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid.
Topics: Amphetamine; Animals; Catecholamines; Chlorine; Depression; Drug Antagonism; Drug Synergism; Humans; Methyltyrosines; Mice; Motor Activity; Movement Disorders; Naphthyridines; Norepinephrine; Phenoxybenzamine; Phenylalanine; Piperidines; Reserpine; Stimulation, Chemical | 1967 |
Stereochemical studies on medicinal agents. V. Synthesis, configuration, and pharmacological activity of pipradrol enantiomers.
Topics: Amphetamine; Animals; Anticonvulsants; Central Nervous System; Chemical Phenomena; Chemistry; Ephedrine; Infrared Rays; Methods; Mice; Motor Activity; Pipecolic Acids; Piperidines; Spectrum Analysis | 1968 |
[Application of sleep induced in the rat by sudden change in the environmental temperature to the study of antagonism between neurostimulants and hypnotics].
Topics: Amphetamine; Animals; Antidepressive Agents; Bemegride; Caffeine; Central Nervous System; Chloral Hydrate; Cocaine; Drug Antagonism; Environment; Hypnotics and Sedatives; Pentobarbital; Pentylenetetrazole; Piperidines; Pregnanediones; Rats; Secobarbital; Sleep; Strychnine; Temperature; Thiazoles | 1967 |
Behavioral facilitation: the interaction of imipramine and desipra- mine with amphetamine, alpha-pipradrol, methylphenidate, and thozalinone.
Topics: Amphetamine; Animals; Antidepressive Agents; Avoidance Learning; Behavior, Animal; Desipramine; Drug Synergism; Imipramine; Male; Methylphenidate; Oxazoles; Piperidines; Rats; Stimulation, Chemical | 1968 |
The importance of endogenous catecholamines in the activity of some CNS stimulants.
Topics: Amphetamine; Animals; Antidepressive Agents; Catecholamines; Central Nervous System; Ephedrine; Male; Mice; Pentylenetetrazole; Piperidines; Seizures; Sensory Receptor Cells; Sympathomimetics; Time Factors; Tremor | 1969 |
[Therapy of hypersomnia].
Topics: Amphetamine; Animals; Antidepressive Agents; Appetite Depressants; Bemegride; Caffeine; Cats; Central Nervous System Stimulants; Chlorphentermine; Desipramine; Electroencephalography; Ephedrine; Glycolates; Humans; Hydroxybutyrates; Imipramine; Mice; Narcolepsy; Pemoline; Phentermine; Piperidines; Rabbits; Rats; Sleep Wake Disorders; Strychnine; Sympathomimetics | 1967 |
Stereotyped and non-stereotyped behaviour in rats induced by various stimulant drugs.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Brain; Caffeine; Central Nervous System; Cocaine; Lysergic Acid Diethylamide; Male; Methamphetamine; Methylphenidate; Nikethamide; Pemoline; Phenmetrazine; Piperidines; Rats | 1969 |
Supersensitivity to the central stimulant actions of adrenergic drugs following discontinuation of a chronic diet of alpha-methyltyrosine.
Topics: Amphetamine; Animals; Brain Chemistry; Diet; Dopamine; Drug Tolerance; Ephedrine; Male; Methylphenidate; Methyltyrosines; Mice; Motor Activity; Norepinephrine; Piperidines | 1969 |
Some physico-chemical properties of amphetamine and related drugs.
Topics: Amphetamine; Antidepressive Agents; Benzphetamine; Chromatography, Gas; Dextroamphetamine; Ephedrine; Humans; Hydrogen-Ion Concentration; Kinetics; Phenmetrazine; Piperidines; Solubility | 1969 |
[Pharmacological studies on 2-methyl-4-amino-6-methoxy-s-triazine (CV399); with special reference to its central effects].
Topics: Amphetamine; Analgesics; Animals; Avoidance Learning; Behavior, Animal; Blood Pressure; Body Temperature; Brain Chemistry; Caffeine; Cats; Central Nervous System; Chlordiazepoxide; Chlorpromazine; Drug Synergism; Ethanol; Haplorhini; Indoleacetic Acids; Male; Meprobamate; Methylphenidate; Mice; Morphine; Motor Activity; Pentobarbital; Piperidines; Rats; Reserpine; Respiration; Salivation; Seizures; Serotonin; Triazines | 1970 |
[Importance of noradrenaline in the mechanism of action of psychotropic drugs].
Topics: Amphetamine; Animals; Antidepressive Agents; Brain Stem; Male; Motor Activity; Norepinephrine; Piperidines; Rats; Reserpine; Tranquilizing Agents; Trifluoperazine | 1968 |
Influence of the optical isomers of some centrally acting drugs on norepinephrine responses.
Topics: Amphetamine; Animals; Drug Synergism; In Vitro Techniques; Male; Morpholines; Norepinephrine; Oxazoles; Piperidines; Rats; Stereoisomerism; Vas Deferens | 1970 |
Release of norepinephrine and normetanephrine from cat brain by central nervous system stimulants.
Topics: Amphetamine; Animals; Brain; Caffeine; Cats; Chlorine; Cocaine; Dextroamphetamine; Ephedrine; Methylphenidate; Norepinephrine; Normetanephrine; Piperidines; Tritium | 1970 |
[The effect of catecholamines (piridrol and phenamine) on various synaptic systems of the cerebral cortex].
Topics: Amphetamine; Animals; Cerebral Cortex; Chlorpromazine; Depression, Chemical; Mesencephalon; Piperidines; Rabbits; Reticular Formation; Stimulation, Chemical; Sympathetic Nervous System; Synaptic Transmission | 1967 |
The relationship between the inhibition of dopamine uptake and the enhancement of amphetamine stereotypy.
Topics: Amantadine; Amphetamine; Animals; Behavior, Animal; Chlorpheniramine; Dopamine; Dopamine Antagonists; Drug Synergism; Histamine H1 Antagonists; Injections, Intraperitoneal; Male; Orphenadrine; Parasympatholytics; Parkinson Disease; Piperidines; Rats; Trihexyphenidyl | 1971 |
Behavior and brain contents of catecholamines in mice during chronic administration of methyldopa.
Topics: Aggression; Amphetamine; Animals; Behavior, Animal; Brain; Catecholamines; Dopamine; Drug Tolerance; Exploratory Behavior; Humans; Male; Methyldopa; Mice; Motor Activity; Norepinephrine; Piperidines | 1971 |
A survey of selected drugs on behavioral performance in ethanol-treated rats.
Topics: Amphetamine; Animals; Caffeine; Conditioning, Operant; Cyproheptadine; Drug Antagonism; Ethanol; Histamine H1 Antagonists; Imipramine; Male; Methylphenidate; Methyltyrosines; Pentylenetetrazole; Piperidines; Pyridines; Rats | 1971 |
The effects of chlorpromazine on psychomotor stimulant self-administration in the rhesus monkey.
Topics: Amphetamine; Animals; Behavior, Animal; Chlorpromazine; Cocaine; Drug Antagonism; Humans; Macaca; Methylphenidate; Phenmetrazine; Piperidines; Self Stimulation; Stimulation, Chemical; Substance-Related Disorders | 1972 |
Conformationally constrained analogs of mescaline.
Topics: Amphetamine; Animals; Behavior, Animal; Exploratory Behavior; Male; Mescaline; Methods; Methylphenidate; Mice; Molecular Conformation; Morpholines; Motor Activity; Piperidines | 1974 |
Effects of various psychotomimetic agents on the EEG and acetylcholine release from the cerebral cortex of brainstem transected cats.
Topics: Acetylcholine; Amphetamine; Animals; Blood Pressure; Brain Stem; Cats; Cerebral Cortex; Dronabinol; Drug Combinations; Electrodes, Implanted; Electroencephalography; Glycolates; Hallucinogens; Heart Rate; Isomerism; Lysergic Acid Diethylamide; Male; Pentobarbital; Phencyclidine; Piperidines; Pyrrolidines | 1972 |
Role of brain noradrenaline in morphine-induced stereotyped behaviour.
Topics: Acetamides; Amphetamine; Animals; Antihypertensive Agents; Behavior, Animal; Brain; Butyrophenones; Dopamine; Humans; Male; Methyltyrosines; Morphine Dependence; Norepinephrine; Phenoxybenzamine; Piperidines; Rats; Reserpine; Spiro Compounds; Thiocarbamates; Tranquilizing Agents | 1972 |
Monoamine oxidase. I. Specificity of some substrates and inhibitors.
Topics: Amines; Amphetamine; Animals; Benzyl Compounds; Brain; Cyclohexylamines; Fluorine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Mitochondria; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nerve Tissue Proteins; Oxidation-Reduction; Oximes; Phenethylamines; Phenylbutyrates; Phenylpropanolamine; Piperidines; Potentiometry; Swine; Tyramine | 1974 |
A comparison of the capacities of isomers of amphetamine, deoxypipradrol and methylphenidate to inhibit the uptake of tritiated catecholamines into rat cerebral cortex slices, synaptosomal preparations of rat cerebral cortex, hypothalamus and striatum and
Topics: Amphetamine; Animals; Aorta; Benzene Derivatives; Brain; Cerebral Cortex; Corpus Striatum; Depression, Chemical; Dopamine; Hypothalamus; Male; Methylphenidate; Norepinephrine; Piperidines; Rats; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship; Sympathetic Nervous System; Synaptosomes; Tritium | 1972 |
[Harmful effects of common drugs on the visual apparatus. Anorexigenic substances].
Topics: Amphetamine; Appetite Depressants; Cataract; Ephedrine; Eye Diseases; Humans; Morpholines; Piperidines; Pupil; Retinal Hemorrhage; Retinal Vessels; Thrombosis; Vision Disorders | 1972 |
[Alteration of the acid-base equilibrium by the anorectic diphemethoxidine in comparison with the effect of amphetamine and aminorex].
Topics: Acid-Base Equilibrium; Amines; Amphetamine; Animals; Appetite Depressants; Blood Gas Analysis; Blood Pressure; Body Temperature; Dogs; Hydrogen-Ion Concentration; Lactates; Oxazoles; Piperidines; Potassium; Pulse; Respiration; Sodium; Time Factors | 1972 |
The influence of various neuroleptic drugs on shock avoidance responding in rats. 3. Amphetamine antagonism in the discriminated Sidman avoidance procedure.
Topics: Amphetamine; Animals; Avoidance Learning; Benzimidazoles; Butyrophenones; Chlorpromazine; Electroshock; Female; Haloperidol; Light; Piperidines; Rats; Sodium Chloride; Tranquilizing Agents | 1970 |
The behavioral effects of a new psychoactive drug (d-carbine) on a passive avoidance response and locomotion and its interaction with amphetamine.
Topics: Amphetamine; Animals; Antidepressive Agents; Avoidance Learning; Chlorpromazine; Drug Antagonism; Drug Synergism; Escape Reaction; Female; Imipramine; Indoles; Mice; Motor Activity; Piperidines | 1971 |
Drug use in psychiatric disorders of children.
Topics: Amphetamine; Anticonvulsants; Antidepressive Agents; Child; Child Behavior Disorders; Chlordiazepoxide; Diphenhydramine; Humans; Hypnotics and Sedatives; Meprobamate; Phytotherapy; Piperazines; Piperidines; Plants, Medicinal; Psychopharmacology; Psychotherapy; Rauwolfia; Time Factors | 1968 |
Behavioural effects of some morphine antagonists and hallucinogens in the rat.
Topics: Amphetamine; Analgesics; Anesthetics; Animals; Ataxia; Atropine; Azocines; Behavior, Animal; Cyclazocine; Levallorphan; Lysergic Acid Diethylamide; Male; Mescaline; Morphine; Motor Activity; Movement Disorders; Nalorphine; Narcotic Antagonists; Pentazocine; Phencyclidine; Piperidines; Psilocybin; Psychopharmacology; Rats | 1968 |
Pharmacological studies on 5-(3-(4-piperidino-4-carbamoyl-piperidino)-propyl)-10,11-dihydro-5(H)-dibenz-(b,f)-azepine (carpipramine) dihydrochloride, a new psychotropic agent.
Topics: Amphetamine; Analgesics; Animals; Anti-Inflammatory Agents; Anticonvulsants; Antidepressive Agents; Apomorphine; Benzazepines; Blood Pressure; Body Temperature; Conditioning, Classical; Depression, Chemical; Dogs; Drug Synergism; Electroshock; Female; Guinea Pigs; Imipramine; In Vitro Techniques; Locomotion; Male; Mice; Muscle Contraction; Muscle, Smooth; Nictitating Membrane; Piperidines; Rabbits; Rats; Reserpine; Sleep; Stimulation, Chemical; Time Factors; Tremorine | 1968 |
Near-infrared spectroscopy of amine salts.
Topics: Amines; Ammonium Chloride; Amphetamine; Butylamines; Cyclopentanes; Ephedrine; Ethylamines; Imidazoles; Infrared Rays; Mephentermine; Metaraminol; Phenethylamines; Phenmetrazine; Phenylpropanolamine; Piperidines; Propylamines; Solvents; Spectrum Analysis; Sympathomimetics | 1966 |
Pharmacology of hepzidine maleate: 4-[10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)oxy]-1-methylpiperidine hydrogen maleate (BS 7051).
Topics: Amphetamine; Animals; Antidepressive Agents; Antiemetics; Atropine; Behavior, Animal; Birds; Blood Pressure; Dogs; Gastrointestinal Motility; Guinea Pigs; Mice; Parasympatholytics; Phenothiazines; Piperidines; Rabbits; Rats; Reserpine; Serotonin Antagonists | 1967 |
Neurochemical effects of danitracen (WA-355): mechanism of action.
Topics: Amphetamine; Animals; Apomorphine; Brain Chemistry; Humans; Hydroxyindoleacetic Acid; Hyperkinesis; Norepinephrine; Piperidines; Rats; Serotonin | 1982 |
Interaction of parachlorophenylalanine, mianserine and danitracen with amphetamine.
Topics: Amphetamine; Animals; Fenclonine; Humans; Male; Mianserin; Piperidines; Rats; Serotonin Antagonists; Stereotyped Behavior | 1981 |
Urinary excretion of O-methylated catecholamines, tyramine and phenyl-ethylamine by volunteers treated with tranylcypromine and CGP 11305 A.
Topics: Adult; Amphetamine; Epinephrine; Female; Humans; Male; Metanephrine; Monoamine Oxidase Inhibitors; Normetanephrine; Phenethylamines; Piperidines; Tranylcypromine; Tyramine | 1983 |
The CB1 cannabinoid receptor antagonist SR 141716A affects A9 dopamine neuronal activity in the rat.
Topics: Amphetamine; Animals; Apomorphine; Dopamine; Dopamine Agents; Dopamine Agonists; Electrophysiology; Male; Mesencephalon; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant | 1995 |
Is it possible to predict the clinical effects of neuroleptics from animal data? Part V: From haloperidol and pipamperone to risperidone.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Butyrophenones; Dogs; Dopamine D2 Receptor Antagonists; Haloperidol; Humans; In Vitro Techniques; Isoxazoles; Lysergic Acid Diethylamide; Motor Activity; Neostriatum; Oxygen Consumption; Piperidines; Rats; Risperidone; Schizophrenia; Serotonin Antagonists; Species Specificity; Tryptamines | 1994 |
Non-specific inhibition of dopamine receptor agonist-induced behaviour by the tachykinin NK1 receptor antagonist CP-99,994 in guinea-pigs.
Topics: Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Dopamine Agonists; Grooming; Guinea Pigs; Haloperidol; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oxazines; Piperidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P | 1994 |
Blockade of phencyclidine-induced hyperlocomotion by clozapine and MDL 100,907 in rats reflects antagonism of 5-HT2A receptors.
Topics: Amphetamine; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Clozapine; Excitatory Amino Acid Antagonists; Fluorobenzenes; Male; Motor Activity; Phencyclidine; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists | 1995 |
Effects of the dopamine autoreceptor antagonist (-)-DS121 on the discriminative stimulus properties of d-amphetamine and cocaine.
Topics: Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Caffeine; Cocaine; Discrimination, Psychological; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Nitriles; Piperidines; Random Allocation; Rats; Rats, Sprague-Dawley; Stereoisomerism | 1995 |
Thioperamide, the selective histamine H3 receptor antagonist, attenuates stimulant-induced locomotor activity in the mouse.
Topics: Amphetamine; Animals; Apomorphine; Central Nervous System Stimulants; Cocaine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Mice; Motor Activity; Piperidines | 1994 |
NPC 16377, a potent and selective sigma-ligand. II. Behavioral and neuroprotective profile.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Avoidance Learning; Brain; Flavonoids; Hypoxia; Lethal Dose 50; Male; Mice; Motor Activity; Nervous System; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma | 1993 |
Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.
Topics: Administration, Oral; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Benzothiazoles; Cebus; Disease Models, Animal; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Dystonia; Ergolines; Female; Haloperidol; Lisuride; Male; Piperidines; Pramipexole; Quinpirole; Raclopride; Salicylamides; Thiazoles | 1993 |
Repeated testing within drug discrimination learning: time course studies with cocaine, amphetamine, and 3-PPP.
Topics: Amphetamine; Animals; Cocaine; Columbidae; Discrimination Learning; Dopamine Antagonists; Male; Piperidines; Time Factors | 1993 |
Reversal of amphetamine-induced behaviours by MDL 100,907, a selective 5-HT2A antagonist.
Topics: Amphetamine; Animals; Behavior, Animal; Brain; Central Nervous System Stimulants; Discrimination, Psychological; Fluorobenzenes; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Reflex, Startle; Reward; Self Stimulation; Serotonin Antagonists | 1996 |
Sigma ligand S14905 and locomotor activity in mice.
Topics: Amphetamine; Animals; Central Nervous System Stimulants; Cocaine; Dose-Response Relationship, Drug; Hydroxamic Acids; Indans; Male; Mice; Morphine; Motor Activity; Narcotics; Piperidines; Radioligand Assay; Receptors, sigma; Stimulation, Chemical | 1995 |
Effects of AMPA receptor positive modulators on amphetamine- and dizocilpine-induced locomotion.
Topics: Amphetamine; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Dioxoles; Dizocilpine Maleate; Dopamine Antagonists; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Haloperidol; Locomotion; Male; Mice; Piperidines; Receptors, AMPA | 1997 |
Mixed D2/5-HT2 antagonism differentially affects apomorphine- and amphetamine-induced stereotyped behavior.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Fluorobenzenes; Male; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Stereotyped Behavior | 1997 |
5-HT4 receptor antagonism does not affect motor and reward mechanisms in the rat.
Topics: Amphetamine; Animals; Behavior, Animal; Cocaine; Dioxanes; Hyperkinesis; Male; Motor Activity; Nicotine; Piperidines; Rats; Rats, Sprague-Dawley; Self Stimulation; Serotonin Antagonists | 1998 |
The effects of (+)-UH232 and (-)-DS121 on local cerebral glucose utilization in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Autoradiography; Brain; Central Nervous System Stimulants; Dopamine Antagonists; Drug Combinations; Glucose; Male; Nitriles; Piperidines; Rats; Rats, Sprague-Dawley | 1999 |
The 5-HT2A receptor antagonist M100907 is more effective in counteracting NMDA antagonist- than dopamine agonist-induced hyperactivity in mice.
Topics: Amphetamine; Animals; Dizocilpine Maleate; Dopamine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Glutamic Acid; Haloperidol; Hyperkinesis; Male; Mice; Mice, Inbred Strains; Motor Activity; N-Methylaspartate; Piperazines; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists | 1999 |
5-HT2 receptor antagonism reduces hyperactivity induced by amphetamine, cocaine, and MK-801 but not D1 agonist C-APB.
Topics: Aminopyridines; Amphetamine; Animals; Benzazepines; Cocaine; Dizocilpine Maleate; Dopamine Agonists; Drug Interactions; Female; Fluorobenzenes; Indoles; Mice; Motor Activity; Piperidines; Ritanserin; Serotonin Antagonists | 1999 |
SR 141716A, a CB1 cannabinoid receptor antagonist, potentiates the locomotor stimulant effects of amphetamine and apomorphine.
Topics: Amphetamine; Animals; Apomorphine; Central Nervous System Stimulants; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Injections, Intraperitoneal; Male; Motor Activity; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Rimonabant | 1999 |
Dopamine D1 receptors synergize with D2, but not D3 or D4, receptors in the striatum without the involvement of action potentials.
Topics: Action Potentials; Amphetamine; Animals; Corpus Striatum; Dopamine Antagonists; Genes, fos; Indans; Indoles; Male; Piperidines; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor Cross-Talk; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Tetrodotoxin | 2000 |
5-HT 2A receptor stimulation by DOI, a 5-HT 2A/2C receptor agonist, potentiates amphetamine-induced dopamine release in rat medial prefrontal cortex and nucleus accumbens.
Topics: Amphetamine; Animals; Central Nervous System Stimulants; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; Indophenol; Male; Nucleus Accumbens; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2003 |
Latent inhibition in 35-day-old rats is not an "adult" latent inhibition: implications for neurodevelopmental models of schizophrenia.
Topics: Aging; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Central Nervous System Stimulants; Clozapine; Conditioning, Classical; Disease Models, Animal; Drinking Behavior; Fluorobenzenes; Male; Models, Neurological; Movement; Neural Inhibition; Piperidines; Rats; Rats, Wistar; Schizophrenia; Time Factors | 2003 |
[Effects of iproniazid on increased spontaneous motility due to central stimulants].
Topics: Amphetamine; Amphetamines; Central Nervous System Stimulants; Iproniazid; Methylphenidate; Movement Disorders; Niacin; Nicotinic Acids; Piperidines | 1958 |
Phenylisopropylamine derivatives, structure and action.
Topics: Amphetamine; Chlorpromazine; Dibucaine; Diethylpropion; Dihydroxyphenylalanine; Dopamine; Ephedrine; Epinephrine; Hydrazines; Imipramine; Iproniazid; Mephentermine; Methamphetamine; Methylphenidate; Movement; Nialamide; Phenelzine; Phenethylamines; Phenmetrazine; Phenylhydrazines; Piperidines; Reserpine; Tranylcypromine; Tryptophan; Tyramine | 1962 |
EFFECTS OF PSYCHOTROPIC DRUGS ON OPEN-FIELD BEHAVIOUR IN RATS.
Topics: Amphetamine; Amphetamines; Anesthetics; Animals; Behavior, Animal; Chlorpromazine; Indoles; Lysergic Acid Diethylamide; Mescaline; Pentobarbital; Phenelzine; Piperidines; Psychotropic Drugs; Rats; Research; Reserpine | 1963 |
EFFECT OF STIMULANTS ON ISOLATED RATS.
Topics: Amphetamine; Amphetamines; Animals; Avoidance Learning; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Hydrazines; Methylphenidate; Noise; Pharmacology; Piperidines; Rats; Research; Tranylcypromine | 1963 |
ANTAGONISM OF MORPHINE AND OF RESERPINE BY LEVOROTATORY AND DEXTROROTATORY ISOMERS OF 2,2-DIPHENYL-4-(2-PIPERIDYL)-1,3-DIOXOLANE HCL.
Topics: Amphetamine; Amphetamines; Biphenyl Compounds; Chemical Phenomena; Chemistry; Dioxolanes; Heterocyclic Compounds; Hexobarbital; Hot Temperature; Hyperesthesia; Mice; Morphine; Pharmacology; Piperidines; Quinones; Reaction Time; Research; Reserpine; Sleep | 1963 |
A RELIABLE TRUCE WITH ENURESIS.
Topics: Adolescent; Amphetamine; Amphetamines; Atropa belladonna; Bromides; Child; Enuresis; Humans; Imipramine; Meprobamate; Methantheline; Methylphenidate; Piperidines; Quaternary Ammonium Compounds; Reserpine; Sympathomimetics | 1964 |
EARLY RECOGNITION OF DEPRESSION.
Topics: Amitriptyline; Amphetamine; Amphetamines; Barbiturates; Benactyzine; Chlordiazepoxide; Deanol; Depression; Depressive Disorder; Diagnosis; Diazepam; Drug Therapy; Geriatrics; Humans; Imipramine; Meprobamate; Methylphenidate; Monoamine Oxidase Inhibitors; Phenmetrazine; Piperidines; Psychotherapy; Toxicology | 1964 |
Mediation of amphetamine-induced long-term depression of synaptic transmission by CB1 cannabinoid receptors in the rat amygdala.
Topics: Amphetamine; Amygdala; Animals; Arachidonic Acids; Benzoxazines; Calcium; Calcium Channels; Central Nervous System Stimulants; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; In Vitro Techniques; Ligands; Long-Term Synaptic Depression; Male; Morpholines; Naphthalenes; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synaptic Transmission | 2003 |
Intra-accumbens protein kinase C inhibitor NPC 15437 blocks amphetamine-produced conditioned place preference in rats.
Topics: Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Male; Motor Activity; Nucleus Accumbens; Piperidines; Protein Kinase C; Rats; Rats, Wistar; Reward; Space Perception; Time Factors | 2003 |
Experimental parkinsonism alters anandamide precursor synthesis, and functional deficits are improved by AM404: a modulator of endocannabinoid function.
Topics: Acyltransferases; Amidohydrolases; Amphetamine; Analysis of Variance; Animals; Antiparkinson Agents; Arachidonic Acids; Behavior, Animal; Brain Chemistry; Cell Count; Central Nervous System Stimulants; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Endocannabinoids; Functional Laterality; Male; Motor Activity; Oxidopamine; Parkinsonian Disorders; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Rotation; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Tyrosine 3-Monooxygenase | 2004 |
Effect of low doses of delta9-tetrahydrocannabinol and cannabidiol on the extinction of cocaine-induced and amphetamine-induced conditioned place preference learning in rats.
Topics: Amphetamine; Animals; Cannabidiol; Cocaine; Conditioning, Operant; Dronabinol; Extinction, Psychological; Learning; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant | 2004 |
Adolescent exposure to cannabinoids induces long-lasting changes in the response to drugs of abuse of rat midbrain dopamine neurons.
Topics: Action Potentials; Age Factors; Amphetamine; Analysis of Variance; Animals; Benzoxazines; Cannabinoids; Cocaine; Critical Period, Psychological; Dopamine; Dose-Response Relationship, Drug; Drug Tolerance; Electrophysiology; Illicit Drugs; Male; Morphine; Morpholines; Naphthalenes; Nerve Net; Neurons; Nucleus Accumbens; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Ventral Tegmental Area | 2004 |
Amphetamine-evoked gene expression in striatopallidal neurons: regulation by corticostriatal afferents and the ERK/MAPK signaling cascade.
Topics: Afferent Pathways; Amphetamine; Animals; Cell Count; Dioxoles; Enzyme Inhibitors; Gene Expression Regulation; Genes, Immediate-Early; Globus Pallidus; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; Motor Activity; Neostriatum; Neurons; Piperidines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; RNA, Messenger | 2004 |
Distinct temporal phases in the behavioral pharmacology of LSD: dopamine D2 receptor-mediated effects in the rat and implications for psychosis.
Topics: Amphetamine; Amphetamines; Animals; Apomorphine; Behavior, Animal; Cues; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluorobenzenes; Hallucinogens; Haloperidol; Indans; Injections, Intraperitoneal; Lysergic Acid Diethylamide; Male; Piperidines; Psychotic Disorders; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2005 |
The substituted (S)-3-phenylpiperidine (-)-OSU6162 reduces apomorphine- and amphetamine-induced behaviour in Cebus apella monkeys.
Topics: Amphetamine; Animals; Apomorphine; Cebus; Dose-Response Relationship, Drug; Male; Piperidines; Stereotyped Behavior | 2006 |
Neurochemical, electrophysiological and pharmacological profiles of the selective inhibitor of the glycine transporter-1 SSR504734, a potential new type of antipsychotic.
Topics: Acetylcholine; Action Potentials; Amphetamine; Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Benzamides; Brain Chemistry; Carbon Isotopes; Cells, Cultured; Cerebral Cortex; Circadian Rhythm; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Glycine; Glycine Plasma Membrane Transport Proteins; Hippocampus; Humans; In Vitro Techniques; Inhibitory Concentration 50; Male; Mice; Motor Activity; Neural Inhibition; Neurons; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Reflex, Startle | 2005 |
The role of 5-HT(2A) receptor antagonism in amphetamine-induced inhibition of A10 dopamine neurons in vitro.
Topics: Action Potentials; Amphetamine; Animals; Antipsychotic Agents; Benzodiazepines; Clozapine; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluorobenzenes; In Vitro Techniques; Male; Mesencephalon; Neural Inhibition; Neurons; Olanzapine; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT2 Receptor Antagonists; Sulpiride | 2005 |
Antipsychotic-like profile of thioperamide, a selective H3-receptor antagonist in mice.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Catalepsy; Dose-Response Relationship, Drug; Haloperidol; Histamine Agonists; Histamine Antagonists; Methylhistamines; Mice; Models, Animal; Motor Activity; Piperidines; Receptors, Histamine H3; Schizophrenia; Stereotyped Behavior; Time Factors | 2006 |
Effects of d-amphetamine and DOI (2,5-dimethoxy-4-iodoamphetamine) on timing behavior: interaction between D1 and 5-HT2A receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Amphetamines; Animals; Conditioning, Operant; Drug Interactions; Female; Fluorobenzenes; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists; Time Perception | 2006 |
ACP-103, a 5-hydroxytryptamine 2A receptor inverse agonist, improves the antipsychotic efficacy and side-effect profile of haloperidol and risperidone in experimental models.
Topics: Amphetamine; Amphetamines; Animals; Antipsychotic Agents; Behavior, Animal; Brain Chemistry; Catalepsy; Dizocilpine Maleate; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Haloperidol; Head Movements; Male; Mice; Mice, Inbred Strains; Motor Activity; Piperidines; Prolactin; Rats; Rats, Sprague-Dawley; Risperidone; Serotonin 5-HT2 Receptor Agonists; Serotonin Receptor Agonists; Urea | 2007 |
CSF histamine levels in rats reflect the central histamine neurotransmission.
Topics: Amphetamine; Animals; Benzhydryl Compounds; Brain; Central Nervous System Stimulants; Circadian Rhythm; Disorders of Excessive Somnolence; Food Deprivation; Histamine; Male; Modafinil; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Sleep; Sleep Deprivation; Synaptic Transmission; Wakefulness | 2008 |
The CB(1) cannabinoid receptor antagonist AM251 attenuates amphetamine-induced behavioural sensitization while causing monoamine changes in nucleus accumbens and hippocampus.
Topics: Amphetamine; Animals; Behavior, Animal; Biogenic Monoamines; Dopamine; Hippocampus; Hydroxyindoleacetic Acid; Male; Mice; Motor Activity; Nucleus Accumbens; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Serotonin | 2008 |
Procognitive and antipsychotic efficacy of glycine transport 1 inhibitors (GlyT1) in acute and neurodevelopmental models of schizophrenia: latent inhibition studies in the rat.
Topics: Aging; Amphetamine; Animals; Animals, Newborn; Antipsychotic Agents; Benzamides; Central Nervous System Stimulants; Cognition; Conditioning, Operant; Dizocilpine Maleate; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine Plasma Membrane Transport Proteins; Haloperidol; Male; Nitroarginine; Piperidines; Rats; Rats, Wistar; Reflex, Startle; Schizophrenia; Schizophrenic Psychology | 2009 |
CB1 receptor knockout mice are hyporesponsive to the behavior-stimulating actions of d-amphetamine: role of mGlu5 receptors.
Topics: Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Dizocilpine Maleate; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Hyperkinesis; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Motor Activity; Nucleus Accumbens; Piperidines; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Rimonabant | 2009 |
Interactions between the glycine transporter 1(GlyT1) inhibitor SSR504734 and psychoactive drugs in mouse motor behaviour.
Topics: Amphetamine; Animals; Benzamides; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine Plasma Membrane Transport Proteins; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phencyclidine; Pilot Projects; Piperidines; Psychotropic Drugs; Receptors, N-Methyl-D-Aspartate | 2009 |
Inhibition of fatty-acid amide hydrolase and CB1 receptor antagonism differentially affect behavioural responses in normal and PCP-treated rats.
Topics: Amidohydrolases; Amphetamine; Animals; Autoradiography; Behavior, Animal; Benzamides; Cannabinoid Receptor Modulators; Carbamates; Central Nervous System Stimulants; Cyclohexanols; Drug Administration Schedule; Drug Interactions; Enzyme Inhibitors; Guanosine 5'-O-(3-Thiotriphosphate); Hallucinogens; Interpersonal Relations; Male; Memory, Short-Term; Motor Activity; Neuropsychological Tests; Phencyclidine; Piperidines; Protein Binding; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Statistics, Nonparametric; Sulfur Isotopes; Time Factors | 2010 |
Amphetamine decreases behavioral inhibition by stimulation of dopamine D2, but not D3, receptors.
Topics: Amphetamine; Animals; Cell Line, Transformed; Central Nervous System Stimulants; Choice Behavior; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Humans; Indoles; Inhibition, Psychological; Male; Nitriles; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2009 |
Combined administration of an mGlu2/3 receptor agonist and a 5-HT 2A receptor antagonist markedly attenuate the psychomotor-activating and neurochemical effects of psychostimulants.
Topics: Amino Acids; Amphetamine; Animals; Antipsychotic Agents; Dizocilpine Maleate; Dopamine; Drug Synergism; Drug Therapy, Combination; Excitatory Amino Acid Agonists; Fluorobenzenes; Male; Motor Activity; Norepinephrine; Nucleus Accumbens; Piperidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists | 2009 |
D2 dopamine receptor subtype-mediated hyperactivity and amphetamine responses in a model of ADHD.
Topics: Amphetamine; Animals; Attention Deficit Disorder with Hyperactivity; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Extracellular Space; Indoles; Locomotion; Mice; Mice, Knockout; Mice, Mutant Strains; Piperidines; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4 | 2010 |
The alpha2 adrenergic receptor antagonist idazoxan, but not the serotonin-2A receptor antagonist M100907, partially attenuated reward deficits associated with nicotine, but not amphetamine, withdrawal in rats.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic Uptake Inhibitors; Amphetamine; Animals; Brain; Dihydro-beta-Erythroidine; Electrodes, Implanted; Fluorobenzenes; Ganglionic Stimulants; Idazoxan; Male; Nicotine; Piperidines; Rats; Rats, Wistar; Receptors, Nicotinic; Reward; Serotonin Antagonists; Substance Withdrawal Syndrome | 2010 |
Functional magnetic resonance imaging reveals different neural substrates for the effects of orexin-1 and orexin-2 receptor antagonists.
Topics: Activity Cycles; Aminopyridines; Amphetamine; Animals; Behavior, Animal; Brain Mapping; Dioxanes; Magnetic Resonance Imaging; Motivation; Orexin Receptors; Phenylurea Compounds; Piperidines; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward | 2011 |
Impulsive action induced by amphetamine, cocaine and MK801 is reduced by 5-HT(2C) receptor stimulation and 5-HT(2A) receptor blockade.
Topics: Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ethylamines; Excitatory Amino Acid Antagonists; Fluorobenzenes; Impulsive Behavior; Indoles; Male; Piperidines; Psychomotor Performance; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists | 2011 |
Pimavanserin, a 5-HT2A inverse agonist, reverses psychosis-like behaviors in a rodent model of Parkinson's disease.
Topics: Amphetamine; Amphetamines; Animals; Antipsychotic Agents; Behavior, Animal; Central Nervous System Stimulants; Disease Models, Animal; Dyskinesias; Fenfluramine; Fluorobenzenes; Hyperkinesis; Male; Motor Activity; Oxidopamine; Parkinson Disease; Piperidines; Psychotic Disorders; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Sensory Gating; Serotonin 5-HT2 Receptor Antagonists; Serotonin Agents; Serotonin Receptor Agonists; Substantia Nigra; Tyrosine 3-Monooxygenase; Urea | 2011 |
Rimonabant attenuates amphetamine sensitisation in a CCK2 receptor-dependent manner.
Topics: Amphetamine; Animals; Behavior, Animal; Cannabinoid Receptor Antagonists; Cannabinoid Receptor Modulators; Central Nervous System Stimulants; Male; Mice; Mice, Knockout; Motor Activity; Piperidines; Pyrazoles; Receptor, Cholecystokinin B; Rimonabant | 2012 |
Cannabinoid CB1 receptor activation mediates the opposing effects of amphetamine on impulsive action and impulsive choice.
Topics: Amphetamine; Animals; Behavior, Animal; Choice Behavior; Dronabinol; Drug Inverse Agonism; Impulsive Behavior; Piperidines; Pyrans; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Reward; Rimonabant | 2011 |
Impact of mGluR5 during amphetamine-induced hyperactivity and conditioned hyperactivity in differentially reared rats.
Topics: Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Hyperkinesis; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Social Isolation; Thiazoles | 2012 |
Effects of the selective 5-HT(7) receptor antagonist SB-269970 in animal models of psychosis and cognition.
Topics: Amphetamine; Animals; Animals, Outbred Strains; Cognition; Disease Models, Animal; Fluorobenzenes; Locomotion; Male; Phencyclidine; Phenols; Piperidines; Psychotic Disorders; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Recognition, Psychology; Serotonin Antagonists; Sulfonamides | 2012 |
Age and sex differences in impulsive action in rats: the role of dopamine and glutamate.
Topics: Aging; Amphetamine; Analysis of Variance; Animals; Animals, Newborn; Choice Behavior; Conditioning, Operant; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; Food Deprivation; Glutamic Acid; Impulsive Behavior; Male; Phenols; Piperidines; Pregnancy; Rats; Rats, Sprague-Dawley; Sex Characteristics; Water Deprivation | 2012 |
The dopamine stabilizers ACR16 and (-)-OSU6162 display nanomolar affinities at the σ-1 receptor.
Topics: Amphetamine; Animals; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; HEK293 Cells; Humans; Male; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor; Transfection; Tritium | 2013 |
Interactions between dopamine transporter and cannabinoid receptor ligands in rhesus monkeys.
Topics: Amphetamine; Animals; Cocaine; Discrimination Learning; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Dronabinol; Female; Haloperidol; Imipramine; Macaca mulatta; Male; Piperidines; Pyrazoles; Receptors, Cannabinoid; Rimonabant; Tropanes | 2012 |
Pimavanserin, a 5-HT2A receptor inverse agonist, reverses psychosis-like behaviors in a rodent model of Alzheimer's disease.
Topics: Alzheimer Disease; Amphetamine; Amphetamines; Animals; Antipsychotic Agents; Behavior, Animal; Disease Models, Animal; Drug Inverse Agonism; Male; Mice; Piperidines; Psychotic Disorders; Serotonin 5-HT2 Receptor Antagonists; Urea | 2012 |
The nucleus accumbens 5-HTR₄-CART pathway ties anorexia to hyperactivity.
Topics: Amphetamine; Animals; Anorexia; Cocaine; Hyperkinesis; Male; Mice; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Nucleus Accumbens; Piperidines; Propane; Real-Time Polymerase Chain Reaction; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Antagonists | 2012 |
SSR504734 enhances basal expression of prepulse inhibition but exacerbates the disruption of prepulse inhibition by apomorphine.
Topics: Amphetamine; Animals; Apomorphine; Benzamides; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Glycine; Glycine Plasma Membrane Transport Proteins; Male; Mice; Mice, Inbred C57BL; Piperidines; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Sensory Gating | 2013 |
Selective serotonin 2A receptor antagonism attenuates the effects of amphetamine on arousal and dopamine overflow in non-human primates.
Topics: Amphetamine; Animals; Arousal; Caudate Nucleus; Central Nervous System Stimulants; Circadian Rhythm; Dopamine; Dopamine Uptake Inhibitors; Female; Fluorobenzenes; Macaca mulatta; Microdialysis; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine; Serotonin 5-HT2 Receptor Antagonists; Sleep; Telemetry; Wakefulness | 2013 |
Behavioral effects of clozapine, pimavanserin, and quetiapine in rodent models of Parkinson's disease and Parkinson's disease psychosis: evaluation of therapeutic ratios.
Topics: Amphetamine; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Clozapine; Dopamine; Dose-Response Relationship, Drug; Male; Parkinsonian Disorders; Piperidines; Psychotic Disorders; Quetiapine Fumarate; Rats; Rats, Sprague-Dawley; Urea | 2013 |
Cannabinoids negatively modulate striatal glutamate and dopamine release and behavioural output of acute D-amphetamine.
Topics: Amphetamine; Animals; Benzoxazines; Cannabinoid Receptor Antagonists; Cannabinoids; Central Nervous System Stimulants; Corpus Striatum; Dopamine; Drug Therapy, Combination; Glutamic Acid; Male; Microdialysis; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Synaptic Transmission | 2014 |
Cannabinoids reward sensitivity in a neurodevelopmental animal model of schizophrenia: a brain stimulation reward study.
Topics: Amphetamine; Analysis of Variance; Animals; Animals, Newborn; Benzoxazines; Brain; Brain Injuries; Central Nervous System Stimulants; Conditioning, Operant; Disease Models, Animal; Dronabinol; Female; Hippocampus; Male; Morpholines; Motivation; Naphthalenes; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Reward; Schizophrenia; Self Administration; Time Factors | 2014 |
Relationship between in vivo receptor occupancy and efficacy of metabotropic glutamate receptor subtype 5 allosteric modulators with different in vitro binding profiles.
Topics: Allosteric Regulation; Amphetamine; Animals; Benzamides; Calcium; Cerebellum; Corpus Striatum; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Locomotion; Male; Maze Learning; Niacinamide; Piperidines; Positron-Emission Tomography; Radioligand Assay; Rats; Receptor, Metabotropic Glutamate 5; Structure-Activity Relationship; Thiazoles | 2015 |
The Combination of Marketed Antagonists of α1b-Adrenergic and 5-HT2A Receptors Inhibits Behavioral Sensitization and Preference to Alcohol in Mice: A Promising Approach for the Treatment of Alcohol Dependence.
Topics: Adrenergic alpha-1 Receptor Antagonists; Alcoholism; Amphetamine; Animals; Behavior, Animal; Cyproheptadine; Ethanol; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Piperidines; Prazosin; Receptor, Serotonin, 5-HT2A; Serotonin 5-HT2 Receptor Antagonists | 2016 |
The effects of the dopamine stabilizer (-)-OSU6162 on aggressive and sexual behavior in rodents.
Topics: Aggression; Amphetamine; Animals; Behavior, Animal; Dopamine Uptake Inhibitors; Exploratory Behavior; Female; Locomotion; Male; Mice; Piperidines; Propanolamines; Rats; Rats, Wistar; Receptors, Dopamine D2; Serotonin 5-HT1 Receptor Antagonists; Sexual Behavior, Animal | 2016 |
Amphetamine elevates nucleus accumbens dopamine via an action potential-dependent mechanism that is modulated by endocannabinoids.
Topics: Action Potentials; Amphetamine; Animals; Cannabinoid Receptor Antagonists; Dopamine; Dopamine Agents; Endocannabinoids; Male; Neurons; Nucleus Accumbens; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Rimonabant; Sodium Channel Blockers; Tetrodotoxin; Ventral Tegmental Area | 2016 |
Responses to drugs of abuse and non-drug rewards in leptin deficient ob/ob mice.
Topics: Amphetamine; Animals; Behavior, Animal; Central Nervous System Depressants; Cocaine; Conditioning, Operant; Disease Models, Animal; Dopamine Uptake Inhibitors; Ethanol; Exploratory Behavior; Feeding Behavior; Illicit Drugs; Leptin; Locomotion; Male; Mice; Motor Activity; Piperidines; Remifentanil; Taste | 2016 |
Design and Synthesis of γ- and δ-Lactam M
Topics: Allosteric Regulation; Amphetamine; Animals; Ataxia; Diarrhea; Dogs; Donepezil; Drug Design; Female; Humans; Indans; Isoindoles; Lactams; Male; Mice, Inbred C57BL; Microsomes, Liver; Oxazoles; Piperidines; Rats, Wistar; Receptor, Muscarinic M1; Scopolamine; Seizures; Structure-Activity Relationship; Sulfonamides; Thiadiazoles; Vomiting | 2017 |
Broad analgesic activity of a novel, selective M1 agonist.
Topics: Amphetamine; Analgesics; Animals; Benzimidazoles; Brain; Central Nervous System Stimulants; CHO Cells; Cognition; Cricetulus; Disease Models, Animal; Humans; Male; Mice, Inbred C57BL; Mice, Knockout; Molecular Structure; Motor Activity; Muscarinic Agonists; Nootropic Agents; Pain; Piperidines; Pyrrolidines; Random Allocation; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Transfection | 2017 |
Simultaneous monitoring of electroencephalographic characteristics in animals subjected to behavioral tests: a preclinical investigation.
Topics: Amphetamine; Animals; Brain; Central Nervous System Agents; Donepezil; Electrocorticography; Electrodes, Implanted; Exploratory Behavior; Indans; Male; Motor Activity; Neuropsychological Tests; Piperidines; Rats, Wistar; Recognition, Psychology; Scopolamine; Telemetry | 2017 |
A Molecularly Imprinted Polymer-based Dye Displacement Assay for the Rapid Visual Detection of Amphetamine in Urine.
Topics: Amphetamine; Amphetamines; Brompheniramine; Bupropion; Coloring Agents; Dose-Response Relationship, Drug; Electrochemical Techniques; False Positive Reactions; Humans; Ibuprofen; Limit of Detection; Molecular Imprinting; Molecularly Imprinted Polymers; Naproxen; Pheniramine; Piperidines; Polymers; Powders; Quetiapine Fumarate; Substance Abuse Detection; Urine | 2020 |
Pitolisant, a wake-promoting agent devoid of psychostimulant properties: Preclinical comparison with amphetamine, modafinil, and solriamfetol.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic Uptake Inhibitors; Amphetamine; Animals; Carbamates; Corpus Striatum; Disorders of Excessive Somnolence; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Evaluation, Preclinical; Drug Inverse Agonism; Feeding Behavior; Histamine Antagonists; Locomotion; Mice; Modafinil; Narcolepsy; Neostriatum; Norepinephrine Plasma Membrane Transport Proteins; Nucleus Accumbens; Phenylalanine; Piperidines; Receptors, Histamine H3; Sleep Apnea, Obstructive; Wakefulness-Promoting Agents | 2021 |