aminoimidazole carboxamide has been researched along with dorsomorphin in 59 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 23 (38.98) | 29.6817 |
2010's | 35 (59.32) | 24.3611 |
2020's | 1 (1.69) | 2.80 |
Authors | Studies |
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Chen, Y; Doebber, T; Fenyk-Melody, J; Fujii, N; Goodyear, LJ; Hirshman, MF; Li, Y; Moller, DE; Musi, N; Myers, R; Shen, X; Ventre, J; Wu, M; Zhou, G | 1 |
Ismail-Beigi, F; Jing, M | 1 |
Bauvy, C; Codogno, P; Dubbelhuis, PF; Helmond, MT; Houben-Weerts, JH; Meijer, AJ; Meley, D | 1 |
Bailey, SJ; Mountjoy, PD; Rutter, GA | 1 |
Fuchsel, L; Goldstein, BJ; Mahadev, K; Ouedraogo, R; Wu, X; Xu, SQ | 1 |
Barrow, JR; Brown, JD; Fillmore, N; Herway, ST; Kim, H; Thomson, DM; Winder, WW | 1 |
Han, Y; Li, C; Li, X; Pang, W; Shyy, JY; Xie, X; Zhu, Y | 1 |
Chakour, KS; Freund, GG; Guest, CB | 1 |
Blanco, EA; Clark, JH; Evans, AM; Hardie, DG; Lewis, TH; Mustard, KJ; Peers, C; Robertson, TP; Wyatt, CN | 1 |
Ashford, JW; Casadesus, G; Greco, SJ; Johnston, JM; Sarkar, S; Smith, MA; Su, B; Tezapsidis, N; Zhu, X | 1 |
Floride, E; Föller, M; Gu, S; Koka, S; Lang, F; Mahmud, H; Münzel, T; Schleicher, E; Schulz, E; Sopjani, M; Wang, K | 1 |
Chen, Z; DeFea, K; Fu, Y; Hsu, PH; Pan, S; Peng, IC; Shyy, JY; Su, MI; Sun, W; Tsai, MD; Zhu, Y | 1 |
Feng, LY; Li, J; Nan, FJ; Yu, LF; Zang, Y | 1 |
Greco, SJ; Johnston, JM; Sarkar, S; Tezapsidis, N | 1 |
Anthony, NM; Ceddia, RB; Gaidhu, MP | 1 |
Cotero, VE; Routh, VH | 1 |
Bustos, M; Lorente-Cebrián, S; Marti, A; Martinez, JA; Moreno-Aliaga, MJ | 1 |
Asakura, M; Asanuma, H; Fujita, M; Ito, S; Kim, J; Kitakaze, M; Komamura, K; Minamino, T; Mochizuki, N; Ogai, A; Sanada, S; Sasaki, H; Sugimachi, M; Takahama, H; Takashima, S; Wakeno, M | 1 |
Harhaji-Trajkovic, L; Isenovic, E; Janjetovic, K; Micic, D; Misirkic, M; Prica, M; Stevanovic, D; Sudar, E; Sumarac-Dumanovic, M; Trajkovic, V; Vucicevic, L | 1 |
Alway, SE; Butler, DC; Williamson, DL | 1 |
Chang, KC; Kim, HJ; Kim, YM; Lee, JH; Nizamutdinova, IT; Seo, HG | 1 |
Chikahisa, S; Fujiki, N; Kitaoka, K; Séi, H; Shimizu, N | 1 |
Bala, M; Buechler, C; Kopp, A; Neumeier, M; Schäffler, A; Sporrer, D; Stögbauer, F; Wanninger, J; Weber, M; Weigert, J; Wurm, S | 1 |
Auberger, P; Bénéteau, M; Chauvin, C; Jacquin, MA; Marchetti, S; Muñoz-Pinedo, C; Pende, M; Pradelli, LA; Ricci, JE | 1 |
Adamczyk, J; Gabryel, B; Labuzek, K; Liber, S; Okopień, B | 1 |
Barnett, D; Burger, C; O'Riordan, KJ; Osting, SM; Potter, WB; Roopra, A; Wagoner, M | 1 |
Belcher, JD; Geng, JG; Huo, Y; Slungaard, A; Tang, R; Viollet, B; Wang, H; Wang, J; Wu, C; Zhang, C; Zhang, W; Zhu, C | 1 |
Bradley, EA; Clark, MG; Eringa, EC; Korstjens, I; Musters, R; Rattigan, S; Sipkema, P; Stehouwer, CD; van Nieuw Amerongen, GP | 1 |
Davidson, SM; Gonçalves, LM; Mocanu, MM; Paiva, MA; Providência, LA; Yellon, DM | 1 |
Li, D; Ling, W; Ma, J; Xia, M; Zhang, Y | 1 |
Yang, SJ; Yu, L | 1 |
Gao, R; Li, J; Pu, Y; Qi, Y; Song, X; Wang, H; Xu, K; Zhang, X; Zhao, L | 1 |
Chen, CY; Chen, YL; Chuang, LM; Tsai, JS | 1 |
Chen, BL; Dong, YG; Liu, C; Ma, YD; Meng, RS; Wang, HN; Xiong, ZJ; Zeng, JY | 1 |
Gao, L; Guo, H; Sun, S; Zhang, X; Zhang, XJ; Zhao, JJ | 1 |
Davis, CC; Downs, SM; Ya, R | 1 |
Banerjee, A; Flynt, L; Ghosh, S; Mellema, M; Panettieri, RA; Shore, SA; Williams, E; Zhu, M | 1 |
Durante, W; Korthuis, RJ; Liu, XM; Peyton, KJ; Shebib, AR; Wang, H | 1 |
Fukui, T; Hasegawa, S; Narishima, R; Tanaka, S; Yamasaki, M; Yoshida, S | 1 |
Chen, MB; Gu, JH; Lu, PH; Shen, WX; Wu, XY; Yang, Y | 1 |
Denbow, DM; Siegel, PB; Xu, P | 1 |
Fuerst, J; Geibel, JP; Hufnagl, C; Jakab, M; Ketterl, N; Langelueddecke, C; Lehner, L; Ritter, M; Schmidt, S | 1 |
Ashrafian, H; Bellahcene, M; Carling, D; Casadei, B; Davies, JK; Ge, Y; Isackson, H; Oliveira, SM; Pinter, K; Redwood, C; Solis, RS; Walker, JW; Watkins, H; Yavari, A; Zhang, YH | 1 |
Alexandre, M; Diaz de Villalvilla, A; Gorelick, FS; Kolodecik, TR; Shugrue, CA; Thrower, EC; Young, LH | 1 |
Andrade, BM; Carvalho, DP; Cazarin, J; Zancan, P | 1 |
Cheng, S; Hao, J; Ji, G; Jiang, Z; Yang, Q; Zhang, Y; Zhao, X | 1 |
Chang, JW; Kim, JH; Kim, JS; Kim, SB; Lee, JH; Lee, SK; Park, JS | 1 |
Carson, JA; Gao, S; Puppa, MJ; Sato, S; Welle, SL; White, JP | 1 |
Alexeyev, MF; Creighton, JR; Jian, MY; Wolkowicz, PE; Zmijewski, JW | 1 |
Chen, M; Liu, R; Ma, Q; Nie, A; Ning, G; Wang, J; Wang, Z; Zhan, M | 1 |
Bai, A; Gu, Q; Guo, Y; Hong, K; Lu, N; Luo, F; Zhang, Y | 1 |
Alves, S; Blesbois, E; Froment, P; Grasseau, I; Métayer-Coustard, S; Nguyen, TM; Praud, C | 1 |
Aoyagi, M; Asano, K; Haneishi, A; Kanai, Y; Komatsu, Y; Moriizumi, M; Ono, M; Otsuka, H; Takagi, K; Tanaka, T; Tomita, K; Tsuchiya, Y; Tsukada, A; Yamada, K; Yanagisawa, Y; Yokouchi, H | 1 |
Egilmez, NK; Hao, J; Li, B; Li, Q; Rao, E; Suttles, J; Zhang, Y | 1 |
Cheng, XY; Huang, C; Li, J; Li, YY; Yao, HW | 1 |
Chen, H; Feger, M; Föller, M; Gaballa, MMS; Glosse, P; Hasan, AA; Hirche, F; Hocher, B; Lang, F; Mutig, K | 1 |
Liang, GY; Liu, DX; Wang, F; Yu, J; Zhang, DS | 1 |
Battson, ML; Cox-York, KA; Gentile, CL; Lee, DM; Sevits, KJ; Wei, Y | 1 |
Chen, D; Chen, H; Chen, X; He, J; Huang, Z; Luo, Y; Wen, W; Yu, B; Yu, J; Zheng, P | 1 |
59 other study(ies) available for aminoimidazole carboxamide and dorsomorphin
Article | Year |
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Role of AMP-activated protein kinase in mechanism of metformin action.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; CCAAT-Enhancer-Binding Proteins; Diabetes Mellitus, Type 2; DNA-Binding Proteins; Enzyme Activation; Fatty Acids; Gene Expression; Glucose; Hepatocytes; Humans; Hypoglycemic Agents; In Vitro Techniques; Male; Metformin; Multienzyme Complexes; Muscle, Skeletal; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; RNA, Messenger; Sterol Regulatory Element Binding Protein 1; Transcription Factors | 2001 |
Critical role of 5'-AMP-activated protein kinase in the stimulation of glucose transport in response to inhibition of oxidative phosphorylation.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinase Kinases; AMP-Activated Protein Kinases; Animals; Biological Transport; Cells, Cultured; Clone Cells; Drug Synergism; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Glucose; Glucose Transporter Type 1; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Multienzyme Complexes; Oxidative Phosphorylation; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Rats; Ribonucleotides; RNA, Small Interfering; Sodium Azide | 2007 |
AMP-activated protein kinase and the regulation of autophagic proteolysis.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Autophagy; HeLa Cells; Hepatocytes; HT29 Cells; Humans; Male; Multienzyme Complexes; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides | 2006 |
Inhibition by glucose or leptin of hypothalamic neurons expressing neuropeptide Y requires changes in AMP-activated protein kinase activity.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Glucose; Hypoglycemic Agents; Hypothalamus; Leptin; Membrane Potentials; Multienzyme Complexes; Neurons; Neuropeptide Y; Patch-Clamp Techniques; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides | 2007 |
Adiponectin suppresses IkappaB kinase activation induced by tumor necrosis factor-alpha or high glucose in endothelial cells: role of cAMP and AMP kinase signaling.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adiponectin; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dideoxyadenosine; Endothelial Cells; Enzyme Inhibitors; Glucose; Humans; I-kappa B Kinase; I-kappa B Proteins; Multienzyme Complexes; NF-KappaB Inhibitor alpha; Peptide Fragments; Phosphorylation; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Ribonucleotides; RNA, Small Interfering; Signal Transduction; Tumor Necrosis Factor-alpha | 2007 |
AMP-activated protein kinase phosphorylates transcription factors of the CREB family.
Topics: Acetyl-CoA Carboxylase; Activating Transcription Factor 1; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Line; Cyclic AMP Response Element Modulator; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Induction; Genes, Reporter; Hexokinase; Humans; Liver; Luciferases; Male; Mice; Mice, Knockout; Multienzyme Complexes; Muscle, Skeletal; Phosphorylation; Promoter Regions, Genetic; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Recombinant Proteins; Ribonucleotides; Signal Transduction; Time Factors; Transfection | 2008 |
AMP-activated protein kinase promotes the differentiation of endothelial progenitor cells.
Topics: Acetyl-CoA Carboxylase; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Biomarkers; Cell Differentiation; Cells, Cultured; Cord Blood Stem Cell Transplantation; Endothelial Cells; Enzyme Activators; Enzyme Inhibitors; Fetal Blood; Fetal Stem Cells; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Lovastatin; Mice; Mice, Nude; Multienzyme Complexes; Neovascularization, Physiologic; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphorylation; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Ribonucleotides; Signal Transduction; Vascular Endothelial Growth Factor A | 2008 |
Macropinocytosis is decreased in diabetic mouse macrophages and is regulated by AMPK.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Culture Techniques; Cell Line, Tumor; Diabetes Mellitus, Type 2; Disease Models, Animal; Energy Metabolism; Glucose; Hyperglycemia; Immunity; Leptin; Macrophage Activation; Macrophages, Peritoneal; Mice; Pinocytosis; Pyrazoles; Pyrimidines; Ribonucleosides | 2008 |
AMP-activated protein kinase and hypoxic pulmonary vasoconstriction.
Topics: Acetyl-CoA Carboxylase; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Calcium; Dinoprost; Hypoxia; Male; Multienzyme Complexes; Phosphorylation; Potassium; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pulmonary Artery; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; Signal Transduction; Vasoconstriction | 2008 |
Leptin reduces Alzheimer's disease-related tau phosphorylation in neuronal cells.
Topics: Alzheimer Disease; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Cell Line, Tumor; Humans; Insulin; Leptin; Multienzyme Complexes; Neurons; Phosphorylation; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Ribonucleotides; Signal Transduction; tau Proteins | 2008 |
Regulation of erythrocyte survival by AMP-activated protein kinase.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Annexin A5; Calcium; Cell Size; Cytosol; Erythrocyte Aging; Erythrocyte Membrane; Erythrocytes; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Glucose; Humans; Ionomycin; Ionophores; Male; Mice; Mice, Mutant Strains; Phosphatidylserines; Pyrazoles; Pyrimidines; Ribonucleotides | 2009 |
AMP-activated protein kinase functionally phosphorylates endothelial nitric oxide synthase Ser633.
Topics: Acetyl-CoA Carboxylase; Adiponectin; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Atorvastatin; Cattle; Cells, Cultured; Chromatography, Liquid; Endothelial Cells; Enzyme Activation; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Mice; Mice, Inbred C57BL; Mice, Knockout; Mutation; Nanotechnology; Nitric Oxide; Nitric Oxide Synthase Type III; Phosphorylation; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Pyrazoles; Pyrimidines; Pyrroles; Ribonucleotides; RNA Interference; RNA, Small Interfering; Serine; Signal Transduction; Stress, Mechanical; Tandem Mass Spectrometry; Time Factors; Transfection | 2009 |
AMP-activated protein kinase is involved in neural stem cell growth suppression and cell cycle arrest by 5-aminoimidazole-4-carboxamide-1-beta-D-ribofuranoside and glucose deprivation by down-regulating phospho-retinoblastoma protein and cyclin D.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinase Kinases; Animals; Apoptosis; Astrocytes; Cell Differentiation; Cell Line, Transformed; Cyclin D; Cyclins; Enzyme Activation; G1 Phase; Glucose; Humans; Hypoglycemic Agents; Janus Kinases; Mice; Neurons; Poly(ADP-ribose) Polymerases; Protein Kinases; Pyrazoles; Pyrimidines; Resting Phase, Cell Cycle; Retinoblastoma Protein; Ribonucleotides; STAT3 Transcription Factor; Stem Cells; Sweetening Agents | 2009 |
Leptin regulates tau phosphorylation and amyloid through AMPK in neuronal cells.
Topics: Alzheimer Disease; Aminoimidazole Carboxamide; AMP-Activated Protein Kinase Kinases; Amyloid beta-Peptides; Animals; Cells, Cultured; Humans; Leptin; Neurons; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Pyrazoles; Pyrimidines; Rats; Ribonucleotides; tau Proteins | 2009 |
Regulation of visceral and subcutaneous adipocyte lipolysis by acute AICAR-induced AMPK activation.
Topics: Acetyl-CoA Carboxylase; Adipocytes; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Enzyme Inhibitors; Epinephrine; Hypoglycemic Agents; Intra-Abdominal Fat; Lipolysis; Male; Phosphorylation; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides; Sterol Esterase; Subcutaneous Fat | 2009 |
Insulin blunts the response of glucose-excited neurons in the ventrolateral-ventromedial hypothalamic nucleus to decreased glucose.
Topics: Aminoimidazole Carboxamide; Androstadienes; Animals; Flavonoids; Glucose; In Vitro Techniques; Insulin; Male; Microscopy, Interference; Neurons; Patch-Clamp Techniques; Phosphatidylinositol 3-Kinases; Potassium Channels, Inwardly Rectifying; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; Ventromedial Hypothalamic Nucleus; Wortmannin | 2009 |
Eicosapentaenoic acid stimulates AMP-activated protein kinase and increases visfatin secretion in cultured murine adipocytes.
Topics: Adipocytes; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cells, Cultured; Chromones; Eicosapentaenoic Acid; Enzyme Activation; Hypoglycemic Agents; Male; Mice; Morpholines; Nicotinamide Phosphoribosyltransferase; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Rats; Ribonucleotides | 2009 |
Metformin prevents progression of heart failure in dogs: role of AMP-activated protein kinase.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Apoptosis; Cardiotonic Agents; Cells, Cultured; Disease Progression; Dogs; Drug Evaluation, Preclinical; Fibrosis; Gene Expression Regulation; Heart Failure; Insulin Resistance; Metformin; Myocytes, Cardiac; Natriuretic Peptides; Nitric Oxide; Nitric Oxide Synthase Type III; Oxidative Stress; Phosphorylation; Protein Processing, Post-Translational; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides; Transforming Growth Factor beta1; Ultrasonography; Ventricular Dysfunction, Left | 2009 |
AMP-activated protein kinase-dependent and -independent mechanisms underlying in vitro antiglioma action of compound C.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Antineoplastic Agents; Antioxidants; Apoptosis; bcl-2-Associated X Protein; Caspases; Cell Cycle; Cell Death; Cell Division; Cell Line, Tumor; Enzyme Activation; G2 Phase; Glioma; Humans; Metformin; Pheochromocytoma; Proto-Oncogene Proteins c-bcl-2; Pyrazoles; Pyrimidines; Reactive Oxygen Species; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleotides | 2009 |
AMPK inhibits myoblast differentiation through a PGC-1alpha-dependent mechanism.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Differentiation; Cell Nucleus; Cells, Cultured; Cyclin-Dependent Kinase Inhibitor p21; Enzyme Inhibitors; Forkhead Box Protein O3; Forkhead Transcription Factors; Mice; Myoblasts, Skeletal; Phosphorylation; Pyrazoles; Pyrimidines; Ribonucleotides; RNA, Small Interfering; Signal Transduction; Transcription Factors | 2009 |
Carbon monoxide (from CORM-2) inhibits high glucose-induced ICAM-1 expression via AMP-activated protein kinase and PPAR-gamma activations in endothelial cells.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Anilides; Anti-Inflammatory Agents; Benzophenones; Carbon Monoxide; Cell Adhesion; Cells, Cultured; Chromans; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activation; Enzyme Activators; Glucose; Humans; Hypoglycemic Agents; Intercellular Adhesion Molecule-1; Organometallic Compounds; PPAR gamma; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Ribonucleotides; Signal Transduction; Thiazolidinediones; Time Factors; Transfection; Troglitazone; Tyrosine | 2009 |
Central AMPK contributes to sleep homeostasis in mice.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Brain; Calcium-Calmodulin-Dependent Protein Kinase Kinase; Carnitine O-Palmitoyltransferase; Central Nervous System Agents; Delta Rhythm; Enzyme Inhibitors; Homeostasis; Hypothalamus; Male; Mice; Mice, Inbred ICR; Phosphorylation; Pyrazoles; Pyrimidines; Ribonucleotides; RNA, Messenger; Sleep; Sleep Deprivation | 2009 |
Adiponectin downregulates galectin-3 whose cellular form is elevated whereas its soluble form is reduced in type 2 diabetic monocytes.
Topics: Adiponectin; Adult; Aged; Aged, 80 and over; Aminoimidazole Carboxamide; Body Mass Index; Cells, Cultured; Cholesterol; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Galectin 3; Humans; Immunoblotting; Male; Metformin; Middle Aged; Monocytes; Oleic Acid; Palmitic Acid; Pyrazoles; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleotides; Solubility; Time Factors | 2009 |
Glycolysis inhibition sensitizes tumor cells to death receptors-induced apoptosis by AMP kinase activation leading to Mcl-1 block in translation.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Antibodies; Apoptosis; Blotting, Western; Deoxyglucose; Enzyme Activation; fas Receptor; Glucose; Glycolysis; HeLa Cells; Humans; Intracellular Signaling Peptides and Proteins; Jurkat Cells; Models, Biological; Myeloid Cell Leukemia Sequence 1 Protein; Protein Biosynthesis; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-bcl-2; Pyrazoles; Pyrimidines; Receptors, Death Domain; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleotides; RNA Interference; Sirolimus; TNF-Related Apoptosis-Inducing Ligand; TOR Serine-Threonine Kinases; U937 Cells | 2010 |
Metformin increases phagocytosis and acidifies lysosomal/endosomal compartments in AMPK-dependent manner in rat primary microglia.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Amyloid beta-Peptides; Animals; Cells, Cultured; Endosomes; Enzyme Activation; Hydrogen-Ion Concentration; Hypoglycemic Agents; Lipopolysaccharides; Lysosomes; Metformin; Microglia; Peptide Fragments; Phagocytosis; Phosphoproteins; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides | 2010 |
Metabolic regulation of neuronal plasticity by the energy sensor AMPK.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Antimetabolites; Blotting, Western; Deoxyglucose; Energy Metabolism; Enzyme Activation; Hippocampus; Hypoglycemic Agents; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Long-Term Potentiation; Metformin; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Neuronal Plasticity; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Ribonucleotides; Signal Transduction; TOR Serine-Threonine Kinases; Vidarabine | 2010 |
Acadesine inhibits tissue factor induction and thrombus formation by activating the phosphoinositide 3-kinase/Akt signaling pathway.
Topics: Adenosine A2 Receptor Antagonists; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Apolipoproteins E; Atherosclerosis; Blood Coagulation; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activation; Fibrinolytic Agents; Humans; Lipopolysaccharides; Macrophages; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monocytes; NF-kappa B; Phosphatidylinositol 3-Kinases; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyrazoles; Pyrimidines; Receptor, Adenosine A2A; Ribonucleosides; RNA, Messenger; Sepsis; Signal Transduction; Thromboplastin; Transcription Factor AP-1; Triazines; Triazoles; Up-Regulation; Venous Thrombosis | 2010 |
Activation of AMP-activated protein kinase by 5-aminoimidazole-4-carboxamide-1-beta-D-ribofuranoside in the muscle microcirculation increases nitric oxide synthesis and microvascular perfusion.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Arteries; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Hindlimb; Infusions, Intravenous; Microcirculation; Muscle, Skeletal; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase Type III; Nitroarginine; Phosphorylation; Pyrazoles; Pyrimidines; Rats; Regional Blood Flow; Ribonucleotides; S-Nitroso-N-Acetylpenicillamine; Serine; Threonine; Time Factors; Vascular Resistance; Vasodilation; Vasodilator Agents | 2010 |
Transitory activation of AMPK at reperfusion protects the ischaemic-reperfused rat myocardium against infarction.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Enzyme Activation; Heart; Hemodynamics; Hypoglycemic Agents; Infarction; Male; Metformin; Myocardial Reperfusion Injury; Myocardium; Phosphorylation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Ribonucleotides | 2010 |
Adenosine monophosphate activated protein kinase regulates ABCG1-mediated oxysterol efflux from endothelial cells and protects against hypercholesterolemia-induced endothelial dysfunction.
Topics: 3' Untranslated Regions; Acetylcholine; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; ATP Binding Cassette Transporter, Subfamily G, Member 1; ATP-Binding Cassette Transporters; Biological Transport; Cattle; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelial Cells; Endothelium, Vascular; Enzyme Activation; Enzyme Activators; Genes, Reporter; Humans; Hypercholesterolemia; Ketocholesterols; Male; Mice; Mice, Inbred C57BL; Nitric Oxide; Nitric Oxide Synthase Type III; Nitroprusside; Oxidative Stress; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Reactive Oxygen Species; Ribonucleotides; RNA Interference; RNA Processing, Post-Transcriptional; RNA Stability; RNA, Messenger; Transfection; Up-Regulation; Vasodilation; Vasodilator Agents | 2010 |
AMP-activated protein kinase mediates activity-dependent regulation of peroxisome proliferator-activated receptor gamma coactivator-1alpha and nuclear respiratory factor 1 expression in rat visual cortical neurons.
Topics: Adenosine Triphosphate; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Blindness; Cells, Cultured; Enzyme Activation; Female; Gene Expression Regulation; Male; Membrane Potentials; Mitochondria; Neurons; Nuclear Respiratory Factors; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Resveratrol; Ribonucleotides; RNA-Binding Proteins; RNA, Messenger; Stilbenes; Transcription Factors; Visual Cortex | 2010 |
A pharmacological activator of AMP-activated protein kinase protects hypoxic neurons in a concentration-dependent manner.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Death; Cell Hypoxia; Cell Survival; Cells, Cultured; Cerebral Cortex; Cytoskeletal Proteins; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Neurons; Pyrazoles; Pyrimidines; Rats; Ribonucleotides | 2010 |
Rosiglitazone inhibits monocyte/macrophage adhesion through de novo adiponectin production in human monocytes.
Topics: Adiponectin; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Blotting, Western; Cell Adhesion; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; Macrophages; Monocytes; PPAR gamma; Pyrazoles; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleotides; Rosiglitazone; Signal Transduction; Thiazolidinediones | 2010 |
Activation of AMPK inhibits cardiomyocyte hypertrophy by modulating of the FOXO1/MuRF1 signaling pathway in vitro.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cardiomegaly; Cells, Cultured; Enzyme Activation; Forkhead Transcription Factors; Gene Silencing; Muscle Proteins; Myocytes, Cardiac; Nerve Tissue Proteins; Phenylephrine; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; RNA, Small Interfering; Signal Transduction; Transfection; Tripartite Motif Proteins; Ubiquitin-Protein Ligases | 2010 |
AMPK enhances the expression of pancreatic duodenal homeobox-1 via PPARalpha, but not PPARgamma, in rat insulinoma cell line INS-1.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Blotting, Western; Cell Line, Tumor; Gene Expression Regulation; Homeodomain Proteins; Insulinoma; PPAR alpha; PPAR gamma; Pyrazoles; Pyrimidines; Rats; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleotides; RNA, Messenger; Trans-Activators | 2010 |
Role of AMPK throughout meiotic maturation in the mouse oocyte: evidence for promotion of polar body formation and suppression of premature activation.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Analysis of Variance; Animals; Cumulus Cells; Enzyme Activators; Enzyme Inhibitors; Female; Immunohistochemistry; Meiosis; Mice; Mice, Inbred C57BL; Oocytes; Pyrazoles; Pyrimidines; Ribonucleotides; Spindle Apparatus; Time Factors | 2010 |
Anti-inflammatory effects of thiazolidinediones in human airway smooth muscle cells.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Anilides; Anti-Inflammatory Agents; Antimetabolites; Asthma; Cells, Cultured; Chromans; Cytokines; Enzyme Activators; Enzyme Inhibitors; Gene Knockdown Techniques; Humans; Hypoglycemic Agents; Inflammation Mediators; Metformin; Myocytes, Smooth Muscle; PPAR gamma; Pyrazoles; Pyrimidines; Respiratory System; Ribonucleotides; Rosiglitazone; Thiazolidinediones; Troglitazone; Vidarabine | 2011 |
Activation of AMPK stimulates heme oxygenase-1 gene expression and human endothelial cell survival.
Topics: Adenylate Kinase; Aminoimidazole Carboxamide; Analysis of Variance; Animals; Blotting, Northern; Blotting, Western; Caspase 3; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Endothelial Cells; Heme Oxygenase-1; Humans; Promoter Regions, Genetic; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; RNA, Small Interfering; Time Factors | 2011 |
Leptin controls ketone body utilization in hypothalamic neuron.
Topics: Aminoimidazole Carboxamide; Animals; Cells, Cultured; Coenzyme A Ligases; Coenzyme A-Transferases; Enzyme Inhibitors; Hypoglycemic Agents; Hypothalamus; Ketone Bodies; Leptin; Male; Mice; Mice, Obese; Neurons; Pyrazoles; Pyrimidines; Receptors, Leptin; Ribonucleotides; RNA, Messenger; Time Factors; Up-Regulation | 2011 |
Activation of AMP-activated protein kinase is involved in vincristine-induced cell apoptosis in B16 melanoma cell.
Topics: Acetyl-CoA Carboxylase; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Cell Line; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Mechanistic Target of Rapamycin Complex 1; Melanoma, Experimental; Mice; Multiprotein Complexes; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proteins; Pyrazoles; Pyrimidines; Reactive Oxygen Species; Ribonucleotides; RNA Interference; Time Factors; TOR Serine-Threonine Kinases; Tumor Suppressor Protein p53; Vincristine | 2011 |
AICAR and Compound C regulate food intake independently of AMP-activated protein kinase in lines of chickens selected for high or low body weight.
Topics: Acetyl-CoA Carboxylase; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Body Weight; Chickens; Drinking; Eating; Energy Metabolism; Injections, Intraventricular; Phosphorylation; Pyrazoles; Pyrimidines; Ribonucleotides | 2011 |
Effect of the AMP-kinase modulators AICAR, metformin and compound C on insulin secretion of INS-1E rat insulinoma cells under standard cell culture conditions.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Apoptosis; Calcium; Cell Line, Tumor; Cell Proliferation; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulinoma; KATP Channels; Membrane Potentials; Metformin; Phosphorylation; Pyrazoles; Pyrimidines; Rats; Ribonucleotides | 2012 |
AMP-activated protein kinase phosphorylates cardiac troponin I and alters contractility of murine ventricular myocytes.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Calcium Signaling; Enzyme Activation; Enzyme Activators; Heart Ventricles; Humans; Male; Mice; Mice, Inbred C57BL; Myocardial Contraction; Myocytes, Cardiac; Myosins; Phosphorylation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Ribonucleotides; Serine; Time Factors; Troponin I; Two-Hybrid System Techniques; Ventricular Function, Left | 2012 |
Cerulein hyperstimulation decreases AMP-activated protein kinase levels at the site of maximal zymogen activation.
Topics: Amino Acid Sequence; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cells, Cultured; Ceruletide; Cyclic AMP-Dependent Protein Kinases; Enzyme Precursors; Gene Expression Regulation; Male; Metformin; Octoxynol; Pancreas; Phosphorylation; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Ribonucleotides; Sodium Dodecyl Sulfate | 2012 |
AMP-activated protein kinase upregulates glucose uptake in thyroid PCCL3 cells independent of thyrotropin.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cells, Cultured; Glucose; Glucose Transporter Type 1; Pyrazoles; Pyrimidines; Rats; Ribonucleotides; Thyroid Gland; Thyrotropin; Up-Regulation | 2012 |
Genistein suppresses LPS-induced inflammatory response through inhibiting NF-κB following AMP kinase activation in RAW 264.7 macrophages.
Topics: Adenylate Kinase; Aminoimidazole Carboxamide; Animals; Cell Line; Dose-Response Relationship, Drug; Genistein; Inflammation; Interleukin-6; Lipopolysaccharides; Macrophages; Mice; NF-kappa B; Phosphorylation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Ribonucleotides; Signal Transduction; Tumor Necrosis Factor-alpha | 2012 |
AMP-activated protein kinase inhibits TGF-β-, angiotensin II-, aldosterone-, high glucose-, and albumin-induced epithelial-mesenchymal transition.
Topics: Albumins; Aldosterone; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Angiotensin II; Cell Line; Epithelial-Mesenchymal Transition; Glucose; Heme Oxygenase-1; Humans; Metformin; NADPH Oxidase 4; NADPH Oxidases; Nephrosclerosis; Pyrazoles; Pyrimidines; Reactive Oxygen Species; Ribonucleosides; Thioredoxins; Transforming Growth Factor beta | 2013 |
Muscle mTORC1 suppression by IL-6 during cancer cachexia: a role for AMPK.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Blotting, Western; Cachexia; Interleukin-6; Mechanistic Target of Rapamycin Complex 1; Mice; Mice, Inbred C57BL; Multiprotein Complexes; Muscle Fibers, Skeletal; Muscle, Skeletal; Neoplasms, Experimental; Phosphorylation; Physical Conditioning, Animal; Proteins; Pyrazoles; Pyrimidines; Real-Time Polymerase Chain Reaction; Recombinant Proteins; RNA, Messenger; Signal Transduction; STAT3 Transcription Factor; TOR Serine-Threonine Kinases | 2013 |
Metformin-stimulated AMPK-α1 promotes microvascular repair in acute lung injury.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Membrane Permeability; Cell Movement; Cells, Cultured; Electric Impedance; Endothelial Cells; Endothelium, Vascular; Enzyme Activation; Gene Knockdown Techniques; In Vitro Techniques; Lipopolysaccharides; Lung; Male; Metformin; Microvessels; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Respiratory Distress Syndrome; Ribonucleotides; RNA, Small Interfering; Wound Healing | 2013 |
Adiponectin regulates ACTH secretion and the HPAA in an AMPK-dependent manner in pituitary corticotroph cells.
Topics: Adiponectin; Adrenocorticotropic Hormone; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Calcium; Cell Line, Tumor; Corticotrophs; Corticotropin-Releasing Hormone; Gene Expression Regulation; Humans; Hypothalamo-Hypophyseal System; Male; Mice; Phosphorylation; Pituitary-Adrenal System; Primary Cell Culture; Pyrazoles; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Adiponectin; Receptors, Corticotropin-Releasing Hormone; Ribonucleotides | 2014 |
AMPK inhibition blocks ROS-NFκB signaling and attenuates endotoxemia-induced liver injury.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Chemical and Drug Induced Liver Injury; Endotoxemia; Gene Expression Regulation; Hypoglycemic Agents; I-kappa B Kinase; Lipopolysaccharides; Liver; Male; Mice; Mice, Inbred BALB C; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Reactive Oxygen Species; Ribonucleotides; Signal Transduction; Transcription Factor RelA; Tumor Necrosis Factor-alpha | 2014 |
Central role of 5'-AMP-activated protein kinase in chicken sperm functions.
Topics: Acrosome Reaction; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Survival; Chickens; Male; Metformin; Phosphorylation; Pyrazoles; Pyrimidines; Ribonucleotides; Semen Analysis; Spermatozoa | 2014 |
5-Aminoimidazole-4-carboxyamide-1-β-D-ribofranoside stimulates the rat enhancer of split- and hairy-related protein-2 gene via atypical protein kinase C lambda.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Basic Helix-Loop-Helix Transcription Factors; Calcium; Cycloheximide; Dactinomycin; Enzyme Activation; Gene Expression; HEK293 Cells; Homeodomain Proteins; Humans; Intracellular Signaling Peptides and Proteins; Isoenzymes; Liver; Phosphatidylinositol 3-Kinases; Phosphoenolpyruvate Carboxykinase (GTP); Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein Synthesis Inhibitors; Pyrazoles; Pyrimidines; Rats; Ribonucleosides; RNA Polymerase II; RNA, Messenger; Signal Transduction; Transcription, Genetic | 2016 |
AMPK-dependent and independent effects of AICAR and compound C on T-cell responses.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Calcium Signaling; Cell Death; Cells, Cultured; Cytokines; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Genotype; Immunologic Factors; Lymphocyte Activation; Mice, Knockout; Phenotype; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Ribonucleosides; T-Lymphocytes; TOR Serine-Threonine Kinases | 2016 |
AMP-activated protein kinase reduces inflammatory responses and cellular senescence in pulmonary emphysema.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Line; Cellular Senescence; Energy Metabolism; Female; Humans; Inflammation; Lipid Metabolism; Lung; Male; Mice; Mice, Inbred C57BL; Pancreatic Elastase; Pulmonary Disease, Chronic Obstructive; Pulmonary Emphysema; Pyrazoles; Pyrimidines; Respiratory Mucosa; Ribonucleotides; Smoking | 2017 |
AMP-activated kinase is a regulator of fibroblast growth factor 23 production.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cell Line, Tumor; Down-Regulation; Fibroblast Growth Factor-23; Fibroblast Growth Factors; Kidney; Mice; Mice, Knockout; ORAI1 Protein; Phosphates; Pyrazoles; Pyrimidines; Rats; Renal Elimination; Ribonucleotides; Up-Regulation | 2018 |
Role of Phosphorylated AMP-Activated Protein Kinase (AMPK) in Myocardial Insulin Resistance After Myocardial Ischemia-Reperfusion During Cardiopulmonary Bypass Surgery in Dogs.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Cardioplegic Solutions; Cardiopulmonary Bypass; China; Coronary Artery Disease; Dogs; Female; Glucose; Glucose Transporter Type 4; Heart Ventricles; Insulin Resistance; Ischemia; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardial Reperfusion Injury; Myocardium; Phosphorylation; Pyrazoles; Pyrimidines; Ribonucleotides | 2019 |
Monounsaturated fatty acids protect against palmitate-induced lipoapoptosis in human umbilical vein endothelial cells.
Topics: Adenylate Kinase; Aminoimidazole Carboxamide; Apoptosis; Cardiovascular Diseases; Cell Survival; Dietary Fats; Endothelium, Vascular; Fatty Acids, Monounsaturated; Human Umbilical Vein Endothelial Cells; Humans; Palmitic Acid; Pyrazoles; Pyrimidines; Ribonucleotides | 2019 |
miR-22-3p regulates muscle fiber-type conversion through inhibiting AMPK/SIRT1/PGC-1α pathway.
Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinase Kinases; Animals; Cell Line; Gene Expression Regulation; Mice; MicroRNAs; Myoblasts; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Protein Kinases; Pyrazoles; Pyrimidines; Ribonucleotides; Sirtuin 1 | 2021 |